Works by Gratteri, Paola

Results: 53

Exploration of Aromatic Hydrazides as Inhibitors of Human Carbonic Anhydrases.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 4, p. 1, doi. 10.1002/ardp.202400963

By:

Menendez, German Benito;
Giovannuzzi, Simone;
Bonardi, Alessandro;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Exploring aliphatic sulfonamides as multiclass inhibitors of the carbonic anhydrases from the pathogen bacterium Vibrio cholerae.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400814

By:

Paoletti, Niccolò;
Giovannuzzi, Simone;
Bonardi, Alessandro;
De Luca, Viviana;
Capasso, Clemente;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2023, v. 356, n. 11, p. 1, doi. 10.1002/ardp.202300309

By:

Ommi, Ojaswitha;
Paoletti, Niccolò;
Bonardi, Alessandro;
Gratteri, Paola;
Bhalerao, Harshada Anil;
Sau, Shashikanta;
Nanduri, Srinivas;
Mohammed, Arifuddin;
Kalia, Nitin Pal;
Sonti, Rajesh;
Supuran, Claudiu T.;
Yaddanapudi, Venkata Madhavi

Publication type:

Article

Novel benzenesulfonamide‐bearing pyrazoles and 1,2,4‐thiadiazoles as selective carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100241

By:

Kumar, Rajiv;
Kumar, Amit;
Ram, Sita;
Angeli, Andrea;
Bonardi, Alessandro;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.;
Sharma, Pawan K.

Publication type:

Article

Induction of a Four‐Way Junction Structure in the DNA Palindromic Hexanucleotide 5′‐d(CGTACG)‐3′ by a Mononuclear Platinum Complex.

Published in:

Angewandte Chemie International Edition, 2019, v. 58, n. 28, p. 9378, doi. 10.1002/anie.201814532

By:

van Rixel, Vincent H. S.;
Busemann, Anja;
Wissingh, Mathijs F.;
Hopkins, Samantha L.;
Siewert, Bianka;
van de Griend, Corjan;
Siegler, Maxime A.;
Marzo, Tiziano;
Papi, Francesco;
Ferraroni, Marta;
Gratteri, Paola;
Bazzicalupi, Carla;
Messori, Luigi;
Bonnet, Sylvestre

Publication type:

Article

Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N -((4-Sulfamoylphenyl)carbamothioyl) Amides.

Published in:

Molecules, 2023, v. 28, n. 10, p. 4020, doi. 10.3390/molecules28104020

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Paoletti, Niccolò;
Aspatwar, Ashok;
Parkkila, Seppo;
Gratteri, Paola;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Sensing Zn2+ in Aqueous Solution with a Fluorescent Scorpiand Macrocyclic Ligand Decorated with an Anthracene Bearing Tail.

Published in:

Molecules, 2020, v. 25, n. 6, p. 1355, doi. 10.3390/molecules25061355

By:

Savastano, Matteo;
Fiaschi, Matteo;
Ferraro, Giovanni;
Gratteri, Paola;
Mariani, Palma;
Bianchi, Antonio;
Bazzicalupi, Carla

Publication type:

Article

Solid State and Solution Study on the Formation of Inorganic Anion Complexes with a Series of Tetrazine-Based Ligands.

Published in:

Molecules, 2019, v. 24, n. 12, p. 2247, doi. 10.3390/molecules24122247

By:

Savastano, Matteo;
García-Gallarín, Celeste;
Giorgi, Claudia;
Gratteri, Paola;
López de la Torre, Maria Dolores;
Bazzicalupi, Carla;
Bianchi, Antonio;
Melguizo, Manuel

Publication type:

Article

Tales of the Unexpected: The Case of Zirconium(IV) Complexes with Desferrioxamine.

Published in:

Molecules, 2019, v. 24, n. 11, p. 2098, doi. 10.3390/molecules24112098

By:

Savastano, Matteo;
Bazzicalupi, Carla;
Ferraro, Giovanni;
Fratini, Emiliano;
Gratteri, Paola;
Bianchi, Antonio

Publication type:

Article

Cation, Anion and Ion-Pair Complexes with a G-3 Poly(ethylene imine) Dendrimer in Aqueous Solution.

Published in:

Molecules, 2017, v. 22, n. 5, p. 816, doi. 10.3390/molecules22050816

By:

Savastano, Matteo;
Bazzicalupi, Carla;
Giorgi, Claudia;
Gratteri, Paola;
Bianchi, Antonio

Publication type:

Article

Optimization by experimental design of the adsorptive stripping voltammetric parameters in the determination of cinoxacin.

Published in:

Electroanalysis, 1995, v. 7, n. 12, p. 1161, doi. 10.1002/elan.1140071212

By:

Gratteri, Paola;
Furlanetto, Sandra;
Pinzauti, Sergio;
Leardi, Riccardo;
Corti, Piero

Publication type:

Article

Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements.

Published in:

Phytochemical Analysis, 2018, v. 29, n. 3, p. 233, doi. 10.1002/pca.2737

By:

Diuzheva, Alina;
Carradori, Simone;
Andruch, Vasil;
Locatelli, Marcello;
De Luca, Elisa;
Tiecco, Matteo;
Germani, Raimondo;
Menghini, Luigi;
Nocentini, Alessio;
Gratteri, Paola;
Campestre, Cristina

Publication type:

Article

A Series of Thiadiazolyl‐Benzenesulfonamides Incorporating an Aromatic Tail as Isoform‐Selective, Potent Carbonic Anhydrase II/XII Inhibitors.

Published in:

ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200056

By:

Banoglu, Erden;
Ercanlı, Taner;
Gür Maz, Tuğçe;
Vullo, Daniela;
Bonardi, Alessandro;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors.

Published in:

ChemMedChem, 2020, v. 15, n. 21, p. 2052, doi. 10.1002/cmdc.202000500

By:

Clima, Lilia;
Craciun, Bogdan Florin;
Angeli, Andrea;
Petreni, Andrea;
Bonardi, Alessandro;
Nocentini, Alessio;
Carta, Fabrizio;
Gratteri, Paola;
Pinteala, Mariana;
Supuran, Claudiu T.

Publication type:

Article

Natural Polyphenols Selectively Inhibit β‐Carbonic Anhydrase from the Dandruff‐Producing Fungus <italic>Malassezia globosa</italic>: Activity and Modeling Studies.

Published in:

ChemMedChem, 2018, v. 13, n. 8, p. 816, doi. 10.1002/cmdc.201800015

By:

Nocentini, Alessio;
Bua, Silvia;
Del Prete, Sonia;
Heravi, Yeganeh Entezari;
Saboury, Ali A.;
Karioti, Anastasia;
Bilia, Anna Rita;
Capasso, Clemente;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Solution NMR Structure of a Ligand/Hybrid-2-G-Quadruplex Complex Reveals Rearrangements that Affect Ligand Binding.

Published in:

Angewandte Chemie International Edition, 2017, v. 56, n. 25, p. 7102, doi. 10.1002/anie.201702135

By:

Wirmer‐Bartoschek, Julia;
Bendel, Lars Erik;
Jonker, Hendrik R. A.;
Grün, J. Tassilo;
Papi, Francesco;
Bazzicalupi, Carla;
Messori, Luigi;
Gratteri, Paola;
Schwalbe, Harald

Publication type:

Article

Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation.

Published in:

Angewandte Chemie International Edition, 2016, v. 55, n. 13, p. 4256, doi. 10.1002/anie.201511999

By:

Bazzicalupi, Carla;
Ferraroni, Marta;
Papi, Francesco;
Massai, Lara;
Bertrand, Benoît;
Messori, Luigi;
Gratteri, Paola;
Casini, Angela

Publication type:

Article

Effect of structure levels on surface-enhanced Raman scattering of human telomeric G-quadruplexes in diluted and crowded media.

Published in:

Analytical & Bioanalytical Chemistry, 2019, v. 411, n. 20, p. 5197, doi. 10.1007/s00216-019-01894-z

By:

Papi, Francesco;
Kenđel, Adriana;
Ratkaj, Marina;
Piantanida, Ivo;
Gratteri, Paola;
Bazzicalupi, Carla;
Miljanić, Snežana

Publication type:

Article

Assessment of human telomeric G-quadruplex structures using surface-enhanced Raman spectroscopy.

Published in:

Analytical & Bioanalytical Chemistry, 2017, v. 409, n. 9, p. 2285, doi. 10.1007/s00216-016-0172-y

By:

Miljanić, Snežana;
Ratkaj, Marina;
Matković, Marija;
Piantanida, Ivo;
Gratteri, Paola;
Bazzicalupi, Carla

Publication type:

Article

Modeling and Biological Investigations of an Unusual Behavior of Novel Synthesized Acridine-Based Polyamine Ligands in the Binding of Double Helix and G-Quadruplex DNA.

Published in:

ChemMedChem, 2010, v. 5, n. 12, p. 1995, doi. 10.1002/cmdc.201000332

By:

Bazzicalupi, Carla;
Chioccioli, Matteo;
Sissi, Claudia;
Porcù, Elena;
Bonaccini, Claudia;
Pivetta, Claudia;
Bencini, Andrea;
Giorgi, Claudia;
Valtancoli, Barbara;
Melani, Fabrizio;
Gratteri, Paola

Publication type:

Article

Central Nicotinic Receptors: Structure, Function, Ligands, and Therapeutic Potential.

Published in:

ChemMedChem, 2007, v. 2, n. 6, p. 746, doi. 10.1002/cmdc.200600207

By:

Romanelli, M. Novella;
Gratteri, Paola;
Guandalini, Luca;
Martini, Elisabetta;
Bonaccini, Claudia;
Gualtieri, Fulvio

Publication type:

Article

Induction of a Four‐Way Junction Structure in the DNA Palindromic Hexanucleotide 5′‐d(CGTACG)‐3′ by a Mononuclear Platinum Complex.

Published in:

Angewandte Chemie, 2019, v. 131, n. 28, p. 9478, doi. 10.1002/ange.201814532

By:

van Rixel, Vincent H. S.;
Busemann, Anja;
Wissingh, Mathijs F.;
Hopkins, Samantha L.;
Siewert, Bianka;
van de Griend, Corjan;
Siegler, Maxime A.;
Marzo, Tiziano;
Papi, Francesco;
Ferraroni, Marta;
Gratteri, Paola;
Bazzicalupi, Carla;
Messori, Luigi;
Bonnet, Sylvestre

Publication type:

Article

Solution NMR Structure of a Ligand/Hybrid-2-G-Quadruplex Complex Reveals Rearrangements that Affect Ligand Binding.

Published in:

Angewandte Chemie, 2017, v. 129, n. 25, p. 7208, doi. 10.1002/ange.201702135

By:

Wirmer ‐ Bartoschek, Julia;
Bendel, Lars Erik;
Jonker, Hendrik R. A.;
Grün, J. Tassilo;
Papi, Francesco;
Bazzicalupi, Carla;
Messori, Luigi;
Gratteri, Paola;
Schwalbe, Harald

Publication type:

Article

Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation.

Published in:

Angewandte Chemie, 2016, v. 128, n. 13, p. 4328, doi. 10.1002/ange.201511999

By:

Bazzicalupi, Carla;
Ferraroni, Marta;
Papi, Francesco;
Massai, Lara;
Bertrand, Benoît;
Messori, Luigi;
Gratteri, Paola;
Casini, Angela

Publication type:

Article

Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 5, p. 2584, doi. 10.3390/ijms25052584

By:

Bua, Silvia;
Bonardi, Alessandro;
Mük, Georgiana Ramona;
Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Leveraging SARS-CoV-2 Main Protease (M pro) for COVID-19 Mitigation with Selenium-Based Inhibitors.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 2, p. 971, doi. 10.3390/ijms25020971

By:

De Luca, Viviana;
Angeli, Andrea;
Nocentini, Alessio;
Gratteri, Paola;
Pratesi, Silvia;
Tanini, Damiano;
Carginale, Vincenzo;
Capperucci, Antonella;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Probing the Efficiency of 13-Pyridylalkyl Berberine Derivatives to Human Telomeric G-Quadruplexes Binding: Spectroscopic, Solid State and In Silico Analysis.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14061, doi. 10.3390/ijms232214061

By:

Bazzicalupi, Carla;
Bonardi, Alessandro;
Biver, Tarita;
Ferraroni, Marta;
Papi, Francesco;
Savastano, Matteo;
Lombardi, Paolo;
Gratteri, Paola

Publication type:

Article

Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 21, p. 11583, doi. 10.3390/ijms222111583

By:

Grande, Rossella;
Carradori, Simone;
Puca, Valentina;
Vitale, Irene;
Angeli, Andrea;
Nocentini, Alessio;
Bonardi, Alessandro;
Gratteri, Paola;
Lanuti, Paola;
Bologna, Giuseppina;
Simeone, Pasquale;
Capasso, Clemente;
De Luca, Viviana;
Supuran, Claudiu T.

Publication type:

Article

Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 7, p. 2621, doi. 10.3390/ijms21072621

By:

Hargunani, Priya;
Tadge, Nikhil;
Ceruso, Mariangela;
Leitans, Janis;
Kazaks, Andris;
Tars, Kaspars;
Gratteri, Paola;
Supuran, Claudiu T.;
Nocentini, Alessio;
Toraskar, Mrunmayee P.

Publication type:

Article

Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484

By:

Abdelrahman, Mohamed A.;
Eldehna, Wagdy M.;
Nocentini, Alessio;
Bua, Silvia;
Al-Rashood, Sara T.;
Hassan, Ghada S.;
Bonardi, Alessandro;
Almehizia, Abdulrahman A.;
Alkahtani, Hamad M.;
Alharbi, Amal;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

β3-Adrenoreceptor Activity Limits Apigenin Efficacy in Ewing Sarcoma Cells: A Dual Approach to Prevent Cell Survival.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2149, doi. 10.3390/ijms20092149

By:

Pasha, Amada;
Vignoli, Marina;
Subbiani, Angela;
Nocentini, Alessio;
Selleri, Silvia;
Gratteri, Paola;
Dabraio, Annalisa;
Casini, Tommaso;
Filippi, Luca;
Fotzi, Ilaria;
Favre, Claudio;
Calvani, Maura

Publication type:

Article

Total Syntheses of Casuarine and Its 6- O-α-Glucoside: Complementary Inhibition towards Glycoside Hydrolases of the GH31 and GH37 Families.

Published in:

Chemistry - A European Journal, 2009, v. 15, n. 7, p. 1627, doi. 10.1002/chem.200801578

By:

Cardona, Francesca;
Parmeggiani, Camilla;
Faggi, Enrico;
Bonaccini, Claudia;
Gratteri, Paola;
Sim, Lyann;
Gloster, Tracey M.;
Roberts, Shirley;
Davies, Gideon J.;
Rose, David R.;
Goti, Andrea

Publication type:

Article

DNA Binding by a New Metallointercalator that Contains a Proflavine Group Bearing a Hanging Chelating Unit.

Published in:

Chemistry - A European Journal, 2008, v. 14, n. 1, p. 184, doi. 10.1002/chem.200601855

By:

Bazzicalupi, Carla;
Bencini, Andrea;
Bianchi, Antonio;
Biver, Tarita;
Boggioni, Alessia;
Bonacchi, Sara;
Danesi, Andrea;
Giorgi, Claudia;
Gratteri, Paola;
Ingraín, Antonio Marchal;
Secco, Fernando;
Sissi, Claudia;
Valtancoli, Barbara;
Venturini, Marcella

Publication type:

Article

The crystal structure of human telomeric DNA complexed with berberine: an interesting case of stacked ligand to G-tetrad ratio higher than 1:1.

Published in:

Nucleic Acids Research, 2013, v. 41, n. 1, p. 632, doi. 10.1093/nar/gks1001

By:

Bazzicalupi, Carla;
Ferraroni, Marta;
Bilia, Anna Rita;
Scheggi, Francesca;
Gratteri, Paola

Publication type:

Article

[Au(9-methylcaffein-8-ylidene)<sub>2</sub>]<sup>+</sup>/DNA Tel23 System: Solution, Computational, and Biological Studies.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 55, p. 13784, doi. 10.1002/chem.201702854

By:

Papi, Francesco;
Bazzicalupi, Carla;
Ferraroni, Marta;
Massai, Lara;
Bertrand, Benoît;
Gratteri, Paola;
Colangelo, Donato;
Messori, Luigi

Publication type:

Article

Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 2, p. 188, doi. 10.3390/ph16020188

By:

Ialongo, Davide;
Messore, Antonella;
Madia, Valentina Noemi;
Tudino, Valeria;
Nocentini, Alessio;
Gratteri, Paola;
Giovannuzzi, Simone;
Supuran, Claudiu T.;
Nicolai, Alice;
Scarpa, Susanna;
Taurone, Samanta;
Camarda, Michele;
Artico, Marco;
Papa, Veronica;
Saccoliti, Francesco;
Scipione, Luigi;
Di Santo, Roberto;
Costi, Roberta

Publication type:

Article

Insights into docking and scoring neuronal α4β2 nicotinic receptor agonists using molecular dynamics simulations and QM/MM calculations.

Published in:

Journal of Computational Chemistry, 2009, v. 30, n. 15, p. 2443, doi. 10.1002/jcc.21251

By:

SGRIGNANI, JACOPO;
BONACCINI, CLAUDIA;
GRAZIOSO, GIOVANNI;
CHIOCCIOLI, MATTEO;
CAVALLI, ANDREA;
GRATTERI, PAOLA

Publication type:

Article

Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.

Published in:

Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527

By:

Sbravati, Davide;
Bonardi, Alessandro;
Bua, Silvia;
Angeli, Andrea;
Ferraroni, Marta;
Nocentini, Alessio;
Casnati, Alessandro;
Gratteri, Paola;
Sansone, Francesco;
Supuran, Claudiu T.

Publication type:

Article

Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide‐Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.

Published in:

Chemistry - A European Journal, 2019, v. 25, n. 5, p. 1188, doi. 10.1002/chem.201805039

By:

Nocentini, Alessio;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies.

Published in:

Chemistry - A European Journal, 2018, v. 24, n. 31, p. 7840, doi. 10.1002/chem.201800941

By:

Nocentini, Alessio;
Carta, Fabrizio;
Tanc, Muhammet;
Selleri, Silvia;
Supuran, Claudiu T.;
Bazzicalupi, Carla;
Gratteri, Paola

Publication type:

Article

Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide–hydantoin hybrids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2335927

By:

Abdoli, Morteza;
Bonardi, Alessandro;
Gratteri, Paola;
Supuran, Claudiu T.;
Žalubovskis, Raivis

Publication type:

Article

Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2202360

By:

Giovannuzzi, Simone;
Bonardi, Alessandro;
Gratteri, Paola;
Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407

By:

Badawi, Waleed A.;
Rashed, Mahmoud;
Nocentini, Alessio;
Bonardi, Alessandro;
Abd-Alhaseeb, Mohammad M.;
Al-Rashood, Sara T.;
Veerakanellore, Giri Babu;
Majrashi, Taghreed A.;
Elkaeed, Eslam B.;
Elgendy, Bahaa;
Gratteri, Paola;
Supuran, Claudiu T.;
Eldehna, Wagdy M.;
Elagawany, Mohamed

Publication type:

Article

Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2191165

By:

Astrain-Redin, Nora;
Paoletti, Niccolò;
Plano, Daniel;
Bonardi, Alessandro;
Gratteri, Paola;
Angeli, Andrea;
Sanmartin, Carmen;
Supuran, Claudiu T.

Publication type:

Article

The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 930, doi. 10.1080/14756366.2022.2053526

By:

Bonardi, Alessandro;
Bua, Silvia;
Combs, Jacob;
Lomelino, Carrie;
Andring, Jacob;
Osman, Sameh Mohamed;
Toti, Alessandra;
Di Cesare Mannelli, Lorenzo;
Gratteri, Paola;
Ghelardini, Carla;
McKenna, Robert;
Nocentini, Alessio;
Supuran, Claudiu T.

Publication type:

Article

Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 487, doi. 10.1080/14756366.2021.2020773

By:

Nocentini, Alessio;
Bonardi, Alessandro;
Pratesi, Simone;
Gratteri, Paola;
Dani, Carlo;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs – a joint docking/molecular dynamics study.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 469, doi. 10.1080/14756366.2020.1862102

By:

Bonardi, Alessandro;
Nocentini, Alessio;
Osman, Sameh Mohamed;
Alasmary, Fatmah Ali;
Almutairi, Tahani Mazyad;
Abdullah, Dalal Saied;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1891, doi. 10.1080/14756366.2020.1828401

By:

Guglielmi, Paolo;
Rotondi, Giulia;
Secci, Daniela;
Angeli, Andrea;
Chimenti, Paola;
Nocentini, Alessio;
Bonardi, Alessandro;
Gratteri, Paola;
Carradori, Simone;
Supuran, Claudiu T.

Publication type:

Article

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1011, doi. 10.1080/14756366.2020.1752201

By:

Pustenko, Aleksandrs;
Nocentini, Alessio;
Gratteri, Paola;
Bonardi, Alessandro;
Vozny, Igor;
Žalubovskis, Raivis;
Supuran, Claudiu T.

Publication type:

Article

Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1164, doi. 10.1080/14756366.2019.1626375

By:

Nocentini, Alessio;
Osman, Sameh M.;
Rodrigues, Igor A.;
Cardoso, Veronica S.;
Alasmary, Fatmah Ali S.;
AlOthman, Zeid;
Vermelho, Alane B.;
Gratteri, Paola;
Supuran, Claudiu T.

Publication type:

Article