Works matching AU Gratteri, Paola
Results: 51
Induction of a Four‐Way Junction Structure in the DNA Palindromic Hexanucleotide 5′‐d(CGTACG)‐3′ by a Mononuclear Platinum Complex.
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- Angewandte Chemie, 2019, v. 131, n. 28, p. 9478, doi. 10.1002/ange.201814532
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Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide–hydantoin hybrids.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2335927
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Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2202360
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Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407
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Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2191165
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The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 930, doi. 10.1080/14756366.2022.2053526
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Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 487, doi. 10.1080/14756366.2021.2020773
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Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs – a joint docking/molecular dynamics study.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 469, doi. 10.1080/14756366.2020.1862102
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Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1891, doi. 10.1080/14756366.2020.1828401
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The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1011, doi. 10.1080/14756366.2020.1752201
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Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1164, doi. 10.1080/14756366.2019.1626375
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Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1453, doi. 10.1080/14756366.2018.1512597
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Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1064, doi. 10.1080/14756366.2017.1355307
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Central Nicotinic Receptors: Structure, Function, Ligands, and Therapeutic Potential.
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- ChemMedChem, 2007, v. 2, n. 6, p. 746, doi. 10.1002/cmdc.200600207
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Effect of structure levels on surface-enhanced Raman scattering of human telomeric G-quadruplexes in diluted and crowded media.
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- Analytical & Bioanalytical Chemistry, 2019, v. 411, n. 20, p. 5197, doi. 10.1007/s00216-019-01894-z
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Optimization by experimental design of the adsorptive stripping voltammetric parameters in the determination of cinoxacin.
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- Electroanalysis, 1995, v. 7, n. 12, p. 1161, doi. 10.1002/elan.1140071212
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Solution and Solid-State Analysis of Binding of 13-Substituted Berberine Analogues to Human Telomeric G-quadruplexes.
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- Chemistry - An Asian Journal, 2016, v. 11, n. 7, p. 1107, doi. 10.1002/asia.201600116
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Induction of a Four‐Way Junction Structure in the DNA Palindromic Hexanucleotide 5′‐d(CGTACG)‐3′ by a Mononuclear Platinum Complex.
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- Angewandte Chemie International Edition, 2019, v. 58, n. 28, p. 9378, doi. 10.1002/anie.201814532
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A Series of Thiadiazolyl‐Benzenesulfonamides Incorporating an Aromatic Tail as Isoform‐Selective, Potent Carbonic Anhydrase II/XII Inhibitors.
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- ChemMedChem, 2022, v. 17, n. 10, p. 1, doi. 10.1002/cmdc.202200056
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Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors.
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- ChemMedChem, 2020, v. 15, n. 21, p. 2052, doi. 10.1002/cmdc.202000500
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Natural Polyphenols Selectively Inhibit β‐Carbonic Anhydrase from the Dandruff‐Producing Fungus <italic>Malassezia globosa</italic>: Activity and Modeling Studies.
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- ChemMedChem, 2018, v. 13, n. 8, p. 816, doi. 10.1002/cmdc.201800015
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Modeling and Biological Investigations of an Unusual Behavior of Novel Synthesized Acridine-Based Polyamine Ligands in the Binding of Double Helix and G-Quadruplex DNA.
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- ChemMedChem, 2010, v. 5, n. 12, p. 1995, doi. 10.1002/cmdc.201000332
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Insights into docking and scoring neuronal α4β2 nicotinic receptor agonists using molecular dynamics simulations and QM/MM calculations.
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- Journal of Computational Chemistry, 2009, v. 30, n. 15, p. 2443, doi. 10.1002/jcc.21251
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Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 5, p. 2584, doi. 10.3390/ijms25052584
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Leveraging SARS-CoV-2 Main Protease (M pro) for COVID-19 Mitigation with Selenium-Based Inhibitors.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 2, p. 971, doi. 10.3390/ijms25020971
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Probing the Efficiency of 13-Pyridylalkyl Berberine Derivatives to Human Telomeric G-Quadruplexes Binding: Spectroscopic, Solid State and In Silico Analysis.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 22, p. 14061, doi. 10.3390/ijms232214061
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Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 21, p. 11583, doi. 10.3390/ijms222111583
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Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 7, p. 2621, doi. 10.3390/ijms21072621
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Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484
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β3-Adrenoreceptor Activity Limits Apigenin Efficacy in Ewing Sarcoma Cells: A Dual Approach to Prevent Cell Survival.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2149, doi. 10.3390/ijms20092149
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Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N -((4-Sulfamoylphenyl)carbamothioyl) Amides.
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- Molecules, 2023, v. 28, n. 10, p. 4020, doi. 10.3390/molecules28104020
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Sensing Zn2+ in Aqueous Solution with a Fluorescent Scorpiand Macrocyclic Ligand Decorated with an Anthracene Bearing Tail.
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- Molecules, 2020, v. 25, n. 6, p. 1355, doi. 10.3390/molecules25061355
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Solid State and Solution Study on the Formation of Inorganic Anion Complexes with a Series of Tetrazine-Based Ligands.
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- Molecules, 2019, v. 24, n. 12, p. 2247, doi. 10.3390/molecules24122247
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Tales of the Unexpected: The Case of Zirconium(IV) Complexes with Desferrioxamine.
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- Molecules, 2019, v. 24, n. 11, p. 2098, doi. 10.3390/molecules24112098
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Cation, Anion and Ion-Pair Complexes with a G-3 Poly(ethylene imine) Dendrimer in Aqueous Solution.
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- Molecules, 2017, v. 22, n. 5, p. 816, doi. 10.3390/molecules22050816
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Pyrrolyl and Indolyl α-γ-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 2, p. 188, doi. 10.3390/ph16020188
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Assessment of human telomeric G-quadruplex structures using surface-enhanced Raman spectroscopy.
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- Analytical & Bioanalytical Chemistry, 2017, v. 409, n. 9, p. 2285, doi. 10.1007/s00216-016-0172-y
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- Article
Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.
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- Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527
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Phosphorus versus Sulfur: Discovery of Benzenephosphonamidates as Versatile Sulfonamide‐Mimic Chemotypes Acting as Carbonic Anhydrase Inhibitors.
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- Chemistry - A European Journal, 2019, v. 25, n. 5, p. 1188, doi. 10.1002/chem.201805039
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Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies.
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- Chemistry - A European Journal, 2018, v. 24, n. 31, p. 7840, doi. 10.1002/chem.201800941
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Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors.
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- Archiv der Pharmazie, 2023, v. 356, n. 11, p. 1, doi. 10.1002/ardp.202300309
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Novel benzenesulfonamide‐bearing pyrazoles and 1,2,4‐thiadiazoles as selective carbonic anhydrase inhibitors.
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- Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100241
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Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements.
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- Phytochemical Analysis, 2018, v. 29, n. 3, p. 233, doi. 10.1002/pca.2737
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[Au(9-methylcaffein-8-ylidene)<sub>2</sub>]<sup>+</sup>/DNA Tel23 System: Solution, Computational, and Biological Studies.
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- Chemistry - A European Journal, 2017, v. 23, n. 55, p. 13784, doi. 10.1002/chem.201702854
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Solution NMR Structure of a Ligand/Hybrid-2-G-Quadruplex Complex Reveals Rearrangements that Affect Ligand Binding.
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- Angewandte Chemie, 2017, v. 129, n. 25, p. 7208, doi. 10.1002/ange.201702135
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Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation.
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- Angewandte Chemie, 2016, v. 128, n. 13, p. 4328, doi. 10.1002/ange.201511999
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The crystal structure of human telomeric DNA complexed with berberine: an interesting case of stacked ligand to G-tetrad ratio higher than 1:1.
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- Nucleic Acids Research, 2013, v. 41, n. 1, p. 632, doi. 10.1093/nar/gks1001
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Total Syntheses of Casuarine and Its 6- O-α-Glucoside: Complementary Inhibition towards Glycoside Hydrolases of the GH31 and GH37 Families.
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- Chemistry - A European Journal, 2009, v. 15, n. 7, p. 1627, doi. 10.1002/chem.200801578
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DNA Binding by a New Metallointercalator that Contains a Proflavine Group Bearing a Hanging Chelating Unit.
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- Chemistry - A European Journal, 2008, v. 14, n. 1, p. 184, doi. 10.1002/chem.200601855
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Solution NMR Structure of a Ligand/Hybrid-2-G-Quadruplex Complex Reveals Rearrangements that Affect Ligand Binding.
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- Angewandte Chemie International Edition, 2017, v. 56, n. 25, p. 7102, doi. 10.1002/anie.201702135
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