Works matching AU Ghorab, Mostafa M.
Results: 44
Synthesis, DFT calculations, and anti-proliferative evaluation of pyrimidine and selenadiazolopyrimidine derivatives as dual Topoisomerase II and HSP90 inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2198163
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Novel sulphonamide-bearing methoxyquinazolinone derivatives as anticancer and apoptosis inducers: synthesis, biological evaluation and in silico studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 86, doi. 10.1080/14756366.2021.1983807
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Synthesis of some quinazolinones inspired from the natural alkaloid L-norephedrine as EGFR inhibitors and radiosensitizers.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 218, doi. 10.1080/14756366.2020.1854243
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Novel sulfonamide benzoquinazolinones as dual EGFR/HER2 inhibitors, apoptosis inducers and radiosensitizers.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1030, doi. 10.1080/14756366.2019.1609469
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Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1565, doi. 10.1080/14756366.2018.1513927
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Benzo[g]quinazolin-based scaffold derivatives as dual EGFR/HER2 inhibitors.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 67, doi. 10.1080/14756366.2017.1389922
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VEGFR-2 inhibitors and apoptosis inducers: synthesis and molecular design of new benzo [g] quinazolin bearing benzenesulfonamide moiety.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 893, doi. 10.1080/14756366.2017.1334650
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Synthesis and biological evaluation of novel 2-phenylquinazoline-4-amine derivatives: identification of 6-phenyl-8H-benzo[g]quinazolino[4,3-b]quinazolin-8-one as a highly potent inducer of NAD(P)H quinone oxidoreductase 1.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 34, doi. 10.3109/14756366.2016.1163343
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Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel 2-phenylquinazolin-4-amine derivatives.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1612, doi. 10.3109/14756366.2016.1158714
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NAD(P)H: quinone oxidoreductase 1 inducer activity of novel 4-aminoquinazoline derivatives.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1369, doi. 10.3109/14756366.2015.1135913
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Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel cyanoenone and enone benzenesulfonamides.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 6, p. 840, doi. 10.3109/14756366.2013.858146
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Design, synthesis and molecular docking of novel N,N-dimethylbenzenesulfonamide derivatives as potential antiproliferative agents.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 5, p. 619, doi. 10.3109/14756366.2013.833197
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Chemistry of 2-cyanomethylene-4-thiazolidinone.
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- Journal of Sulfur Chemistry, 2017, v. 38, n. 3, p. 314, doi. 10.1080/17415993.2016.1263304
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Novel Thiophenes, Thienopyrimidines, and Triazolothienopyrimidines for the Evaluation of Anticancer and Augmentation Effects of γ-Radiation.
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- Archiv der Pharmazie, 2010, v. 343, n. 7, p. 404, doi. 10.1002/ardp.200900150
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Antimicrobial and anticancer activity of some novel fluorinated thiourea derivatives carrying sulfonamide moieties: synthesis, biological evaluation and molecular docking.
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- Chemistry Central Journal, 2017, v. 11, p. 1, doi. 10.1186/s13065-017-0258-4
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Novel iodoquinazolinones bearing sulfonamide moiety as potential antioxidants and neuroprotectors.
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- Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-42239-2
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Novel iodoquinazolinones bearing sulfonamide moiety as potential antioxidants and neuroprotectors.
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- Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-42239-2
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NAD(P)H:quinone oxidoreductase 1 inducer activity of some novel anilinoquinazoline derivatives.
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- Drug Design, Development & Therapy, 2016, v. 10, p. 2515, doi. 10.2147/DDDT.S105423
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Crystal structure of the co-crystalline adduct 4-((4,4-dimethyl-2,6-dioxocyclohexylidene) methylamino)-N-(4,6-dimethylpyrimidin-2-yl) benzenesulfonamide - acetic acid (1/1), C<sub>21</sub>H<sub>24</sub>N<sub>4</sub>O<sub>4</sub>S ⋅ C<sub>2</sub>H<sub>4</sub>O<sub>2</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2017, v. 232, n. 3, p. 417, doi. 10.1515/ncrs-2016-0295
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Crystal Structure of 4-(2-chloroacetamido)pyridinium chloride monohydrate, C<sub>7</sub>H<sub>10</sub>Cl<sub>2</sub>N<sub>2</sub>O<sub>2</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2017, v. 232, n. 1, p. 91, doi. 10.1515/ncrs-2016-0164
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Crystal structure of 4-((4,4-dimethyl-2, 6-dioxocyclohexylidine)methylamino)- N-(3,4-dimethylisoxazol-5-yl)benzenesulfonamide, C<sub>20</sub>H<sub>23</sub>N<sub>3</sub>O<sub>5</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 4, p. 1117, doi. 10.1515/ncrs-2016-0082
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Crystal structure of ethyl-5-amino-1-(2,4-dinitrophenyl)-1 H-pyrazole-4-carboxylate, C<sub>12</sub>H<sub>11</sub>N<sub>5</sub>O<sub>6</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 699, doi. 10.1515/ncrs-2015-0239
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Crystal structure of 2-((2-chloropyridin-3-ylamino)methylene)malononitrile, C<sub>9</sub>H<sub>5</sub>ClN<sub>4</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 711, doi. 10.1515/ncrs-2015-0242
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Crystal structure of ( Z)-4-(4-oxopent-2-en-2-ylamino)benzenesulfonamide, C<sub>11</sub>H<sub>14</sub>N<sub>2</sub>O<sub>3</sub>S.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 867, doi. 10.1515/ncrs-2015-0297
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Crystal structure of 2-((dimethylamino)methylene)-5,5-Dimethylcyclohexane-1,3-dione, C<sub>11</sub>H<sub>17</sub>NO<sub>2</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 903, doi. 10.1515/ncrs-2016-0002
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Crystal structure of (E)-1-(3,4-dimethoxyphenyl)-3-(dimethylamino)prop-2-en-1-one, C<sub>13</sub>H<sub>17</sub>NO<sub>3</sub>.
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- Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 2, p. 437, doi. 10.1515/ncrs-2015-0121
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Synthesis, Antimicrobial, and Antibiofilm Activities of Some Novel 7-Methoxyquinoline Derivatives Bearing Sulfonamide Moiety against Urinary Tract Infection-Causing Pathogenic Microbes.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 10, p. 8933, doi. 10.3390/ijms24108933
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Cytotoxicity of Newly Synthesized Quinazoline–Sulfonamide Derivatives in Human Leukemia Cell Lines and Their Effect on Hematopoiesis in Zebrafish Embryos.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 9, p. 4720, doi. 10.3390/ijms23094720
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Synthesis, Characterization and Anti-Breast Cancer Activity of New 4-Aminoantipyrine-Based Heterocycles.
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- International Journal of Molecular Sciences, 2014, v. 15, n. 5, p. 7539, doi. 10.3390/ijms15057539
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Synthesis and Anti-Breast Cancer Evaluation of Novel N-(Guanidinyl)benzenesulfonamides.
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- International Journal of Molecular Sciences, 2014, v. 15, n. 4, p. 5582, doi. 10.3390/ijms15045582
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The Antiproliferative and Apoptotic Effects of a Novel Quinazoline Carrying Substituted-Sulfonamides: In Vitro and Molecular Docking Study.
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- Molecules, 2022, v. 27, n. 3, p. 981, doi. 10.3390/molecules27030981
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In-Vitro Anticancer Evaluation of Some Novel Thioureido-Benzensulfonamide Derivatives.
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- Molecules, 2016, v. 21, n. 4, p. 409, doi. 10.3390/molecules21040409
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Design, Synthesis and Anticancer Evaluation of Novel Quinazoline-Sulfonamide Hybrids.
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- Molecules, 2016, v. 21, n. 2, p. 189, doi. 10.3390/molecules21020189
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Utility of methyl 2-isothiocyanatobenzoate in the synthesis of some new quinazoline derivatives as potential anticancer and radiosensitizing agents.
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- Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 12, p. 719
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Novel quinolines bearing a biologically active trimethoxyphenyl moiety as a new class of antitumor agents.
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- Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 9, p. 527, doi. 10.1055/s-0031-1296239
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Design and synthesis of some novel hydrazide, 1,2 - dihydropyridine, chromene derivatives carrying biologically active sulfone moieties with potential anticancer activity.
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- Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 9, p. 521, doi. 10.1055/s-0031-1296238
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Synthesis of Certain New Thieno[2,3-d] pyrimidines as Potential Antitumor and Radioprotective Agents.
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- Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2006, v. 56, n. 7, p. 553
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Novel Synthesis of Pyrrolo[2,3-d] pyrimidines Bearing Sulfonamide Moieties as Potential Antitumor and Radioprotective Agents.
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- Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2006, v. 56, n. 4, p. 301
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Novel N-(Substituted) Thioacetamide Quinazolinone Benzenesulfonamides as Antimicrobial Agents.
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- International Journal of Nanomedicine, 2020, v. 15, p. 3161, doi. 10.2147/IJN.S241433
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Dapson in heterocyclic chemistry, part VIII: synthesis, molecular docking and anticancer activity of some novel sulfonylbiscompounds carrying biologically active 1,3-dihydropyridine, chromene and chromenopyridine moieties.
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- Chemistry Central Journal, 2012, v. 6, n. 1, p. 64, doi. 10.1186/1752-153X-6-64
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Novel Quinazoline Derivatives Bearing a Sulfapyridine Moiety as Anticancer and Radiosensitizing Agents.
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- Journal of Heterocyclic Chemistry, 2014, v. 51, p. E255, doi. 10.1002/jhet.1830
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Synthesis and antitumor activity of some novel hydrazide, 1,2-dihydropyridine, chromene, and benzochromene derivatives.
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- Journal of Heterocyclic Chemistry, 2012, v. 49, n. 2, p. 272, doi. 10.1002/jhet.829
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Design and synthesis of some novel quinoline derivatives as anticancer and radiosensitizing agents targeting VEGFR tyrosine kinase.
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- Journal of Heterocyclic Chemistry, 2011, v. 48, n. 6, p. 1269, doi. 10.1002/jhet.749
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In vitro cytotoxic evaluation of some new heterocyclic sulfonamide derivatives.
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- Journal of Heterocyclic Chemistry, 2011, v. 48, n. 3, p. 563, doi. 10.1002/jhet.619
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