Works by Gentilucci, Luca
Results: 34
Conjecturing about Small-Molecule Agonists and Antagonists of α4β1 Integrin: From Mechanistic Insight to Potential Therapeutic Applications.
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- Biomedicines, 2024, v. 12, n. 2, p. 316, doi. 10.3390/biomedicines12020316
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- Article
Design of α/β-Hybrid Peptide Ligands of α4β1 Integrin Equipped with a Linkable Side Chain for Chemoselective Biofunctionalization of Microstructured Materials.
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- Biomedicines, 2021, v. 9, n. 11, p. 1737, doi. 10.3390/biomedicines9111737
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- Article
Pursuing Orally Bioavailable Hepcidin Analogues via Cyclic N -Methylated Mini-Hepcidins.
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- Biomedicines, 2021, v. 9, n. 2, p. 164, doi. 10.3390/biomedicines9020164
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- Article
Integrin-Targeting Peptides for the Design of Functional Cell-Responsive Biomaterials.
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- Biomedicines, 2020, v. 8, n. 9, p. 307, doi. 10.3390/biomedicines8090307
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- Article
Integrin-Targeting Dye-Doped PEG-Shell/Silica-Core Nanoparticles Mimicking the Proapoptotic Smac/DIABLO Protein.
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- Nanomaterials (2079-4991), 2020, v. 10, n. 6, p. 1211, doi. 10.3390/nano10061211
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- Article
Controlling Cyclopeptide Backbone Conformation with β/α-Hybrid Peptide-Heterocycle Scaffolds.
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- European Journal of Organic Chemistry, 2016, v. 2016, n. 19, p. 3243, doi. 10.1002/ejoc.201600448
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- Article
Preparation of Non-Toxic Fluorescent Peptide-Coated Silica/PEG Nanoparticles from Peptide-Block Copolymer Conjugates.
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- Micro (2673-8023), 2022, v. 2, n. 2, p. 240, doi. 10.3390/micro2020016
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- Article
Leukocyte Integrin Antagonists as a Novel Option to Treat Dry Age-Related Macular Degeneration.
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- Frontiers in Pharmacology, 2021, v. 11, p. N.PAG, doi. 10.3389/fphar.2020.617836
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- Article
Functional Selectivity and Antinociceptive Effects of a Novel KOPr Agonist.
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- Frontiers in Pharmacology, 2020, p. 1, doi. 10.3389/fphar.2020.00188
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- Article
Development of Isoxazoline-Containing Peptidomimetics as Dual α<sub>v</sub>β<sub>3</sub> and α<sub>5</sub>β<sub>1</sub> Integrin Ligands.
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- ChemMedChem, 2011, v. 6, n. 12, p. 2264, doi. 10.1002/cmdc.201100372
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- Article
The Inverse Type II β-Turn on D-Trp-Phe, a Pharmacophoric Motif for MOR Agonists.
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- ChemMedChem, 2011, v. 6, n. 9, p. 1640, doi. 10.1002/cmdc.201100169
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- Article
Synthesis and Conformational Analysis of Cyclotetrapeptide Mimetic β-Turn Templates and Validation as 3D Scaffolds.
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- ChemMedChem, 2009, v. 4, n. 4, p. 517, doi. 10.1002/cmdc.200800407
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- Article
Design, Pharmacological Characterization, and Molecular Docking of Minimalist Peptidomimetic Antagonists of α 4 β 1 Integrin.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 11, p. 9588, doi. 10.3390/ijms24119588
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- Article
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 20, p. 12700, doi. 10.3390/ijms232012700
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- Article
Highly Regio- and Diastereoselective Palladium-Catalyzed Allylic Substitution. Synthesis of 3-(2-Aminobutylidene)- 4-arylazetidin-2-ones.
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- Advanced Synthesis & Catalysis, 2005, v. 347, n. 6, p. 833, doi. 10.1002/adsc.200404385
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- Article
Design of κ-Opioid Receptor Agonists for the Development of Potential Treatments of Pain with Reduced Side Effects.
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- Molecules, 2023, v. 28, n. 1, p. 346, doi. 10.3390/molecules28010346
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- Article
Synthesis and Antiproliferative Activity against Cancer Cells of Indole-Aryl-Amide Derivatives.
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- Molecules, 2023, v. 28, n. 1, p. 265, doi. 10.3390/molecules28010265
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- Article
PacDOCK: A Web Server for Positional Distance-Based and Interaction-Based Analysis of Docking Results.
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- Molecules, 2022, v. 27, n. 20, p. 6884, doi. 10.3390/molecules27206884
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- Article
Pharmacological Characterization of µ-Opioid Receptor Agonists with Biased G Protein or β-Arrestin Signaling, and Computational Study of Conformational Changes during Receptor Activation.
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- Molecules, 2021, v. 26, n. 1, p. 13, doi. 10.3390/molecules26010013
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- Article
Asymmetric Synthesis of Alkyl Aziridine-2-Carboxylates from Chiral 3′-Benzyloxy-aminoimides.
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- Angewandte Chemie International Edition, 1996, v. 35, n. 16, p. 1848, doi. 10.1002/anie.199618481
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- Article
Linker Hydrophilicity Modulates the Anticancer Activity of RGD–Cryptophycin Conjugates.
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- Chemistry - A European Journal, 2021, v. 27, n. 3, p. 1015, doi. 10.1002/chem.202003471
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- Article
DS-70, a novel and potent α<sub>4</sub> integrin antagonist, is an effective treatment for experimental allergic conjunctivitis in guinea pigs.
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- 2018
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- journal article
Investigation of the interaction between the atypical agonist c[YpwFG] and MOR.
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- FEBS Journal, 2008, v. 275, n. 9, p. 2315, doi. 10.1111/j.1742-4658.2008.06386.x
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- Article
Synthesis and Analysis of the Conformational Preferences of 5-Aminomethyloxazolidine-2,4-dione Scaffolds: First Examples of β<sup>2</sup>- and β<sup>2, 2</sup>-Homo-Freidinger Lactam Analogues.
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- Chemistry - A European Journal, 2014, v. 20, n. 41, p. 13390, doi. 10.1002/chem.201402519
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- Article
Integrin Ligands with α/β-Hybrid Peptide Structure: Design, Bioactivity, and Conformational Aspects.
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- Medicinal Research Reviews, 2016, v. 36, n. 3, p. 389, doi. 10.1002/med.21383
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- Article
Easy preparation of dehydroalanine building blocks equipped with oxazolidin-2-one chiral auxiliaries, and applications to the stereoselective synthesis of substituted tryptophans.
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- Amino Acids, 2014, v. 46, n. 12, p. 2823, doi. 10.1007/s00726-014-1839-3
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- Article
A straightforward route to enantiopure 2-substituted-3,4-dehydro-β-proline via ring closing metathesis.
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- Amino Acids, 2011, v. 41, n. 3, p. 575, doi. 10.1007/s00726-011-0921-3
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- Article
Selective detection of α4β1 integrin (VLA‐4)‐expressing cells using peptide‐functionalized nanostructured materials mimicking endothelial surfaces adjacent to inflammatory sites.
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- Peptide Science, 2018, v. 110, n. 5, p. N.PAG, doi. 10.1002/bip.23081
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- Article
A Straightforward Method for the Synthesis of Alkylidene and Arylidene Malonates Through Proline-Catalyzed Knoevenagel Condensation.
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- Synthetic Communications, 2003, v. 33, n. 9, p. 1587, doi. 10.1081/SCC-120018782
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- Article
Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic.
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- Biopolymers, 2016, v. 106, n. 3, p. 309, doi. 10.1002/bip.22846
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- Article
5-aminomethyloxazolidine-2,4-dione hybrid α/β-dipeptide scaffolds as inductors of constrained conformations: Applications to the synthesis of integrin antagonists.
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- Biopolymers, 2015, v. 104, n. 5, p. 636, doi. 10.1002/bip.22704
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- Article
Convenient Synthesis of the Antibiotic Linezolid via an Oxazolidine-2,4-dione Intermediate Derived from the Chiral Building Block Isoserine.
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- European Journal of Organic Chemistry, 2014, v. 2014, n. 34, p. 7614, doi. 10.1002/ejoc.201402888
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- Article
Synthesis of Constrained Peptidomimetics Containing 2-Oxo-1,3-oxazolidine-4-carboxylic Acids.
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- European Journal of Organic Chemistry, 2011, v. 2011, n. 25, p. 4925, doi. 10.1002/ejoc.201100346
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- Article
Peptides inhibiting the assembly of monomeric human l‐lactate dehydrogenase into catalytically active homotetramer decrease the synthesis of lactate in cultured cells.
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- Protein Science: A Publication of the Protein Society, 2024, v. 33, n. 10, p. 1, doi. 10.1002/pro.5161
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- Article