Works matching AU Gennari, Cesare
Results: 77
RGD Cyclopeptide Equipped with a Lysine‐Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency.
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- Chemistry - A European Journal, 2023, v. 29, n. 19, p. 1, doi. 10.1002/chem.202203768
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Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.
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- Angewandte Chemie, 2020, v. 132, n. 10, p. 4205, doi. 10.1002/ange.201916394
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Amine‐Carbamate Self‐Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads.
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- ChemBioChem, 2024, v. 25, n. 8, p. 1, doi. 10.1002/cbic.202400174
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Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery.
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- ChemistryOpen, 2019, v. 8, n. 6, p. 737, doi. 10.1002/open.201900110
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Insights into the Binding of Cyclic RGD Peptidomimetics to α<sub>5</sub>β<sub>1</sub> Integrin by using Live-Cell NMR And Computational Studies.
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- ChemistryOpen, 2017, v. 6, n. 1, p. 128, doi. 10.1002/open.201600112
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Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting α<sub>v</sub>β<sub>3</sub> Integrin and VEGF Receptors.
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- ChemistryOpen, 2015, v. 4, n. 5, p. 633, doi. 10.1002/open.201500062
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PhthalaPhos: Chiral Supramolecular Ligands for Enantioselective Rhodium-Catalyzed Hydrogenation Reactions.
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- Angewandte Chemie International Edition, 2010, v. 49, n. 37, p. 6633, doi. 10.1002/anie.201002958
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Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker.
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- Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1320524
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Metallaphotoredox C−O and C−N Cross‐Coupling Using Donor‐Acceptor Cyanoarene Photocatalysts.
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- ChemCatChem, 2022, v. 14, n. 23, p. 1, doi. 10.1002/cctc.202200990
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Use of the Trost Ligand in the Ruthenium-Catalyzed Asymmetric Hydrogenation of Ketones.
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- ChemCatChem, 2017, v. 9, n. 16, p. 3125, doi. 10.1002/cctc.201700545
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Synthesis of [Bis(hexamethylene)cyclopentadienone]iron Tricarbonyl and its Application to the Catalytic Reduction of C=O Bonds.
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- ChemCatChem, 2017, v. 9, n. 8, p. 1461, doi. 10.1002/cctc.201601591
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Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols.
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- ChemCatChem, 2016, v. 8, n. 22, p. 3431, doi. 10.1002/cctc.201600972
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Inside Cover: Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols (ChemCatChem 22/2016).
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- ChemCatChem, 2016, v. 8, n. 22, p. 3419, doi. 10.1002/cctc.201601402
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Celebrating Franco Cozzi's 70 th Birthday.
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- European Journal of Organic Chemistry, 2021, v. 2021, n. 29, p. 4216, doi. 10.1002/ejoc.202100745
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Functionalized 2‐Hydroxybenzaldehyde‐PEG Modules as Portable Tags for the Engagement of Protein Lysine ϵ‐Amino Groups.
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- European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1763, doi. 10.1002/ejoc.202100160
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Recent Catalytic Applications of (Cyclopentadienone)iron Complexes.
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- European Journal of Organic Chemistry, 2020, v. 2020, n. 22, p. 3192, doi. 10.1002/ejoc.201901925
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Improving C=N Bond Reductions with (Cyclopentadienone)iron Complexes: Scope and Limitations.
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- European Journal of Organic Chemistry, 2019, v. 2019, n. 4, p. 647, doi. 10.1002/ejoc.201801348
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Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and α<sub>V</sub>β<sub>3</sub>‐Integrin Ligands for Tumor Targeting.
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- European Journal of Organic Chemistry, 2018, v. 2018, n. 23, p. 2902, doi. 10.1002/ejoc.201800447
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- Article
Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.
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- Angewandte Chemie International Edition, 2020, v. 59, n. 10, p. 4176, doi. 10.1002/anie.201916394
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- Article
Discovery of a New Efficient Chiral Ligand for Copper-Catalyzed Enantioselective Michael Additions by High-Throughput Screening of a Parallel Library.
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- Chemistry - A European Journal, 2001, v. 7, n. 12, p. 2628, doi. 10.1002/1521-3765(20010618)7:12<2628::AID-CHEM26280>3.0.CO;2-7
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Hydrogen-Bonding Donor/Acceptor Scales in β-Sulfonamidopeptides.
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- Chemistry - A European Journal, 1998, v. 4, n. 10, p. 1924, doi. 10.1002/(SICI)1521-3765(19981002)4:10<1924::AID-CHEM1924>3.0.CO;2-P
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Conformational Studies of Chiral Vinylogous Sulfonamidopeptides.
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- Chemistry - A European Journal, 1996, v. 2, n. 6, p. 644, doi. 10.1002/chem.19960020608
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- Article
Advanced Pyrrolidine‐Carbamate Self‐Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release.
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- ChemMedChem, 2022, v. 17, n. 15, p. 1, doi. 10.1002/cmdc.202200279
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Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin α<sub>V</sub>β<sub>3</sub>.
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- ChemMedChem, 2019, v. 14, n. 9, p. 938, doi. 10.1002/cmdc.201900049
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Development and Biochemical Characterization of Self-Immolative Linker Containing GnRH-III-Drug Conjugates.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 9, p. 5071, doi. 10.3390/ijms23095071
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A Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts.
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- Advanced Synthesis & Catalysis, 2016, v. 358, n. 16, p. 2589, doi. 10.1002/adsc.201600348
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Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process.
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- Advanced Synthesis & Catalysis, 2016, v. 358, n. 4, p. 515, doi. 10.1002/adsc.201500933
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Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source.
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- Advanced Synthesis & Catalysis, 2015, v. 357, n. 10, p. 2223, doi. 10.1002/adsc.201500359
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Semisynthesis of Taxol: A Highly Enantio- and Diastereoselective Synthesis of the Side Chain and a New Method for Ester Formation at C13 Using Thioesters.
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- Angewandte Chemie International Edition, 1996, v. 35, n. 15, p. 1723, doi. 10.1002/anie.199617231
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Synthetic Receptors Based on Vinylogous Sulfonyl Peptides.
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- Angewandte Chemie International Edition, 1995, v. 34, n. 16, p. 1765, doi. 10.1002/anie.199517651
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Solid-Phase Synthesis of Vinylogous Sulfonyl Peptides.
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- Angewandte Chemie International Edition, 1995, v. 34, n. 16, p. 1763, doi. 10.1002/anie.199517631
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Synthesis of Sulfonamido-Pseudopeptides: New Chiral Unnatural Oligomers.
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- Angewandte Chemie International Edition, 1994, v. 33, n. 20, p. 2067, doi. 10.1002/anie.199420671
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Computer-Assisted Design of Chiral Boron Enolates: A Novel, Highly Enantioselective Aldol Reaction for Thioacetates and Thiopropionates.
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- Angewandte Chemie International Edition, 1993, v. 32, n. 11, p. 1618, doi. 10.1002/anie.199316181
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Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake.
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- Chemistry - A European Journal, 2020, v. 26, n. 33, p. 7492, doi. 10.1002/chem.202001115
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Frontispiece: Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.
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- Chemistry - A European Journal, 2019, v. 25, n. 65, p. N.PAG, doi. 10.1002/chem.201986561
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Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.
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- Chemistry - A European Journal, 2019, v. 25, n. 65, p. 14740, doi. 10.1002/chem.201903127
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- Article
The Importance of Detail: How Differences in Ligand Structures Determine Distinct Functional Responses in Integrin α<sub>v</sub>β<sub>3</sub>.
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- Chemistry - A European Journal, 2019, v. 25, n. 23, p. 5959, doi. 10.1002/chem.201900169
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- Article
Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin‐Targeted Conjugate.
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- Chemistry - A European Journal, 2019, v. 25, n. 7, p. 1696, doi. 10.1002/chem.201805447
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- Article
PhthalaPhos: Chiral Supramolecular Ligands for Enantioselective Rhodium-Catalyzed Hydrogenation Reactions.
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- Angewandte Chemie, 2010, v. 122, n. 37, p. 6783, doi. 10.1002/ange.201002958
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- Article
A Practical Approach to the Resolution of Racemic N-Benzyl α-Amino Acids by Liquid–Liquid Extraction with a Lipophilic Chiral Salen–Cobalt(III) ComplexWe thank the European Commission for financial support (IHP Network grant “Enantioselective Recognition: Towards the Separation of Racemates” HPRN-CT-2001-00182) and for postdoctoral fellowships to J.-P.C. and T.B.R. We would also like to thank “Merck Research Laboratories” (Merck's Academic Development Program Award to C.G.) for financial support. Salen=N,N′-bis(salicylidene)ethylenediamine dianion.
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- Angewandte Chemie, 2006, v. 118, n. 15, p. 2509, doi. 10.1002/ange.200504116
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A Formal Total Synthesis of Eleutherobin Through an Unprecedented Kinetically Controlled Ring-Closing-Metathesis Reaction of a Densely Functionalized Diene.
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- Angewandte Chemie, 2005, v. 117, n. 4, p. 594, doi. 10.1002/ange.200461767
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Riding the Wave of Monodentate Ligand Revival: From the A/B Concept to Noncovalent Interactions.
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- Chemical Record, 2016, v. 16, n. 6, p. 2544, doi. 10.1002/tcr.201600087
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Investigating the Interaction of Cyclic RGD Peptidomimetics with α<sub>V</sub>β<sub>6</sub> Integrin by Biochemical and Molecular Docking Studies.
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- Cancers, 2017, v. 9, n. 10, p. 128, doi. 10.3390/cancers9100128
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Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α<sub>V</sub>β<sub>3</sub>.
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- Chemistry - A European Journal, 2017, v. 23, n. 58, p. n/a, doi. 10.1002/chem.201703093
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Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α<sub>V</sub>β<sub>3</sub>.
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- Chemistry - A European Journal, 2017, v. 23, n. 58, p. 14410, doi. 10.1002/chem.201703093
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- Article
Tumor Targeting with an isoDGR-Drug Conjugate.
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- Chemistry - A European Journal, 2017, v. 23, n. 33, p. 7910, doi. 10.1002/chem.201701844
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- Article
Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts.
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- Chemistry - A European Journal, 2016, v. 22, n. 28, p. 9528, doi. 10.1002/chem.201601501
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- Article
Synthesis and Biological Evaluation of RGD Peptidomimetic-Paclitaxel Conjugates Bearing Lysosomally Cleavable Linkers.
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- Chemistry - A European Journal, 2015, v. 21, n. 18, p. 6921, doi. 10.1002/chem.201500158
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- Article
Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists.
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- Chemistry - A European Journal, 2015, v. 21, n. 16, p. 6265, doi. 10.1002/chem.201406567
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Cyclic isoDGR Peptidomimetics as Low-Nanomolar α<sub>v</sub>β<sub>3</sub> Integrin Ligands.
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- Chemistry - A European Journal, 2013, v. 19, n. 11, p. 3563, doi. 10.1002/chem.201204639
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