Works matching AU Gütschow, Michael

Results: 106

En Route to New Therapeutic Options for Iron Overload Diseases: Matriptase-2 as a Target for Kunitz-Type Inhibitors.

Published in:

ChemBioChem, 2016, v. 17, n. 7, p. 595, doi. 10.1002/cbic.201500651

By:

Beckmann, Anna‐Madeleine;
Maurer, Eva;
Lülsdorff, Verena;
Wilms, Annika;
Furtmann, Norbert;
Bajorath, Jürgen;
Gütschow, Michael;
Stirnberg, Marit

Publication type:

Article

Cover Picture: En Route to New Therapeutic Options for Iron Overload Diseases: Matriptase-2 as a Target for Kunitz-Type Inhibitors (ChemBioChem 7/2016).

Published in:

ChemBioChem, 2016, v. 17, n. 7, p. 523, doi. 10.1002/cbic.201600126

By:

Beckmann, Anna‐Madeleine;
Maurer, Eva;
Lülsdorff, Verena;
Wilms, Annika;
Furtmann, Norbert;
Bajorath, Jürgen;
Gütschow, Michael;
Stirnberg, Marit

Publication type:

Article

Inhibitors of Matriptase-2 Based on the Trypsin Inhibitor SFTI-1.

Published in:

ChemBioChem, 2015, v. 16, n. 11, p. 1601, doi. 10.1002/cbic.201500200

By:

Gitlin, Agata;
Dębowski, Dawid;
Karna, Natalia;
Łęgowska, Anna;
Stirnberg, Marit;
Gütschow, Michael;
Rolka, Krzysztof

Publication type:

Article

A Coumarin-Labeled Vinyl Sulfone as Tripeptidomimetic Activity-Based Probe for Cysteine Cathepsins.

Published in:

ChemBioChem, 2014, v. 15, n. 7, p. 955, doi. 10.1002/cbic.201300806

By:

Mertens, Matthias D.;
Schmitz, Janina;
Horn, Martin;
Furtmann, Norbert;
Bajorath, Jürgen;
Mareš, Michael;
Gütschow, Michael

Publication type:

Article

CPS49-induced neurotoxicity does not cause limb patterning anomalies in developing chicken embryos.

Published in:

Journal of Anatomy, 2018, v. 232, n. 4, p. 568, doi. 10.1111/joa.12712

By:

Mahony, Chris;
McMenemy, Scott;
Rafipay, Alexandra J.;
Beedie, Shaunna-Leigh;
Fraga, Lucas Rosa;
Gütschow, Michael;
Figg, William D.;
Erskine, Lynda;
Vargesson, Neil

Publication type:

Article

Design, Synthesis, and Evaluation of BCL‐2 Targeting PROTACs.

Published in:

Chemistry - A European Journal, 2024, v. 30, n. 45, p. 1, doi. 10.1002/chem.202400430

By:

Bricelj, Aleša;
Dora Ng, Yuen Lam;
Gobec, Martina;
Kuchta, Robert;
Hu, Wanyi;
Javornik, Špela;
Rožič, Miha;
Gütschow, Michael;
Zheng, Guangrong;
Krönke, Jan;
Steinebach, Christian;
Sosič, Izidor

Publication type:

Article

Two Tags in One Probe: Combining Fluorescence‐ and Biotin‐based Detection of the Trypanosomal Cysteine Protease Rhodesain.

Published in:

Chemistry - A European Journal, 2022, v. 28, n. 62, p. 1, doi. 10.1002/chem.202201636

By:

Lemke, Carina;
Jílková, Adéla;
Ferber, Dominic;
Braune, Annett;
On, Anja;
Johe, Patrick;
Zíková, Alena;
Schirmeister, Tanja;
Mareš, Michael;
Horn, Martin;
Gütschow, Michael

Publication type:

Article

Die Hauptprotease von SARS‐CoV‐2 als Zielstruktur: Von der Etablierung eines Hochdurchsatz‐Screenings zum Design maßgeschneiderter Inhibitoren.

Published in:

Angewandte Chemie, 2021, v. 133, n. 18, p. 10515, doi. 10.1002/ange.202016961

By:

Breidenbach, Julian;
Lemke, Carina;
Pillaiyar, Thanigaimalai;
Schäkel, Laura;
Al Hamwi, Ghazl;
Diett, Miriam;
Gedschold, Robin;
Geiger, Nina;
Lopez, Vittoria;
Mirza, Salahuddin;
Namasivayam, Vigneshwaran;
Schiedel, Anke C.;
Sylvester, Katharina;
Thimm, Dominik;
Vielmuth, Christin;
Phuong Vu, Lan;
Zyulina, Maria;
Bodem, Jochen;
Gütschow, Michael;
Müller, Christa E.

Publication type:

Article

Synthesis and Crystal Structure of Benzyl [(1S)-1-(5-amino-1,3,4-oxadiazol-2-yl)-2-phenylethyl]carbamate.

Published in:

Crystals (2073-4352), 2012, v. 2, n. 3, p. 1201, doi. 10.3390/cryst2031201

By:

Löser, Reik;
Nieger, Martin;
Gütschow, Michael

Publication type:

Article

Proteomic profiling reveals CDK6 upregulation as a targetable resistance mechanism for lenalidomide in multiple myeloma.

Published in:

Nature Communications, 2022, v. 13, n. 1, p. 1, doi. 10.1038/s41467-022-28515-1

By:

Ng, Yuen Lam Dora;
Ramberger, Evelyn;
Bohl, Stephan R.;
Dolnik, Anna;
Steinebach, Christian;
Conrad, Theresia;
Müller, Sina;
Popp, Oliver;
Kull, Miriam;
Haji, Mohamed;
Gütschow, Michael;
Döhner, Hartmut;
Walther, Wolfgang;
Keller, Ulrich;
Bullinger, Lars;
Mertins, Philipp;
Krönke, Jan

Publication type:

Article

Design and Synthesis of Multi-Functional Ligands through Hantzsch Reaction: Targeting Ca 2+ Channels, Activating Nrf2 and Possessing Cathepsin S Inhibitory, and Antioxidant Properties.

Published in:

Pharmaceutics, 2024, v. 16, n. 1, p. 121, doi. 10.3390/pharmaceutics16010121

By:

Pachón-Angona, Irene;
Bernard, Paul J.;
Simakov, Alexey;
Maj, Maciej;
Jozwiak, Krzysztof;
Novotna, Anna;
Lemke, Carina;
Gütschow, Michael;
Martin, Helene;
Oset-Gasque, María-Jesús;
Contelles, José-Marco;
Ismaili, Lhassane

Publication type:

Article

Solubility Enhanced Formulation Approaches to Overcome Oral Delivery Obstacles of PROTACs.

Published in:

Pharmaceutics, 2023, v. 15, n. 1, p. 156, doi. 10.3390/pharmaceutics15010156

By:

Pöstges, Florian;
Kayser, Kevin;
Appelhaus, Jan;
Monschke, Marius;
Gütschow, Michael;
Steinebach, Christian;
Wagner, Karl G.

Publication type:

Article

Solubility and Stability Enhanced Oral Formulations for the Anti-Infective Corallopyronin A.

Published in:

Pharmaceutics, 2020, v. 12, n. 11, p. 1105, doi. 10.3390/pharmaceutics12111105

By:

Krome, Anna K.;
Becker, Tim;
Kehraus, Stefan;
Schiefer, Andrea;
Steinebach, Christian;
Aden, Tilman;
Frohberger, Stefan J.;
López Mármol, Álvaro;
Kapote, Dnyaneshwar;
Jansen, Rolf;
Chaverra-Muñoz, Lillibeth;
Hübner, Marc P.;
Pfarr, Kenneth;
Hesterkamp, Thomas;
Stadler, Marc;
Gütschow, Michael;
König, Gabriele M.;
Hoerauf, Achim;
Wagner, Karl G.

Publication type:

Article

A Short Peptide Inhibitor as an Activity-Based Probe for Matriptase-2.

Published in:

Pharmaceuticals (14248247), 2018, v. 11, n. 2, p. 49, doi. 10.3390/ph11020049

By:

Mangold, Martin;
Gütschow, Michael;
Stirnberg, Marit

Publication type:

Article

Convergent Synthesis of Two Fluorescent Ebselen-Coumarin Heterodimers.

Published in:

Pharmaceuticals (14248247), 2016, v. 9, n. 3, p. 43, doi. 10.3390/ph9030043

By:

Küppers, Jim;
Schulz-Fincke, Anna Christina;
Palus, Jerzy;
Giurg, Mirosław;
Skar˙zewski, Jacek;
Gütschow, Michael

Publication type:

Article

3,1-Benzothiazines, 1,4-Benzodioxines and 1,4-Benzoxazines as Inhibitors of Matriptase-2: Outcome of a Focused Screening Approach.

Published in:

Pharmaceuticals (14248247), 2016, v. 9, n. 1, p. 2, doi. 10.3390/ph9010002

By:

Roydeva, Polya G.;
Beckmann, Anna-Madeleine;
Stirnberg, Marit;
Cesar, Jožko;
Kikelj, Danijel;
Ilaš, Janez;
Gütschow, Michael

Publication type:

Article

Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile.

Published in:

FEBS Journal, 2009, v. 276, n. 8, p. 2292, doi. 10.1111/j.1742-4658.2009.06957.x

By:

Pietsch, Markus;
Christian, Leonie;
Inhester, Therese;
Petzold, Susanne;
Gütschow, Michael

Publication type:

Article

The intact Kunitz domain protects the amyloid precursor protein from being processed by matriptase-2.

Published in:

Biological Chemistry, 2016, v. 397, n. 8, p. 777, doi. 10.1515/hsz-2015-0263

By:

Beckmann, Anna-Madeleine;
Glebov, Konstantin;
Walter, Jochen;
Merkel, Olaf;
Mangold, Martin;
Schmidt, Frederike;
Becker-Pauly, Christoph;
Gütschow, Michael;
Stirnberg, Marit

Publication type:

Article

Cell surface serine protease matriptase-2 suppresses fetuin-A/AHSG-mediated induction of hepcidin.

Published in:

Biological Chemistry, 2015, v. 396, n. 1, p. 81, doi. 10.1515/hsz-2014-0120

By:

Stirnberg, Marit;
Maurer, Eva;
Arenz, Katharina;
Babler, Anne;
Jahnen-Dechent, Willi;
Gütschow, Michael

Publication type:

Article

Matriptase-2 (TMPRSS6) is directly up-regulated by hypoxia inducible factor-1: identification of a hypoxia-responsive element in the TMPRSS6 promoter region.

Published in:

Biological Chemistry, 2012, v. 393, n. 6, p. 535, doi. 10.1515/hsz-2011-0221

By:

Maurer, Eva;
Gütschow, Michael;
Stirnberg, Marit

Publication type:

Article

Synthesis and preliminary radiopharmacological characterisation of an 11C‐labelled azadipeptide nitrile as potential PET tracer for imaging of cysteine cathepsins.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2019, v. 62, n. 8, p. 448, doi. 10.1002/jlcr.3729

By:

Laube, Markus;
Frizler, Maxim;
Wodtke, Robert;
Neuber, Christin;
Belter, Birgit;
Kniess, Torsten;
Bachmann, Michael;
Gütschow, Michael;
Pietzsch, Jens;
Löser, Reik

Publication type:

Article

Synthesis of 2H- and 13C-labelled sunitinib and its primary metabolite.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2009, v. 52, n. 9, p. 360, doi. 10.1002/jlcr.1608

By:

Elsinghorst, Paul W.;
Gütschow, Michael

Publication type:

Article

Synthesis of a Fluorescent-Labeled Bisbenzamidine Containing the Central (6,7-Dimethoxy-4-coumaryl)Alanine Building Block.

Published in:

Heteroatom Chemistry, 2015, v. 26, n. 5, p. 367, doi. 10.1002/hc.21269

By:

Häußler, Daniela;
Gütschow, Michael

Publication type:

Article

Highly potent inhibitors of cathepsin K with a differently positioned cyanohydrazide warhead: structural analysis of binding mode to mature and zymogen-like enzymes.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 515, doi. 10.1080/14756366.2021.2024527

By:

Benýšek, Jakub;
Buša, Michal;
Rubešová, Petra;
Fanfrlík, Jindřich;
Lepšík, Martin;
Brynda, Jiří;
Matoušková, Zuzana;
Bartz, Ulrike;
Horn, Martin;
Gütschow, Michael;
Mareš, Michael

Publication type:

Article

Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2′ site binding inhibitor.

Published in:

Acta Crystallographica: Section F, Structural Biology Communications, 2018, v. 74, n. 8, p. 480, doi. 10.1107/S2053230X1800537X

By:

Hochscherf, Jennifer;
Pietsch, Markus;
Tieu, William;
Kuan, Kevin;
Abell, Andrew D.;
Gütschow, Michael;
Niefind, Karsten

Publication type:

Article

Identification of novel disulfide adducts between the thiol containing leaving group of the nerve agent VX and cysteine containing tripeptides derived from human serum albumin.

Published in:

Drug Testing & Analysis, 2017, v. 9, n. 8, p. 1192, doi. 10.1002/dta.2144

By:

Kranawetvogl, Andreas;
Küppers, Jim;
Gütschow, Michael;
Worek, Franz;
Thiermann, Horst;
Elsinghorst, Paul W.;
John, Harald

Publication type:

Article

Azadipeptide Nitriles: Highly Potent and Proteolytically Stable Inhibitors of Papain-Like Cysteine Proteases.

Published in:

Angewandte Chemie International Edition, 2008, v. 47, n. 23, p. 4331, doi. 10.1002/anie.200705858

By:

Löser, Reik;
Frizler, Maxim;
Schilling, Klaus;
Gütschow, Michael

Publication type:

Article

Cell Type-Specific Anti-Viral Effects of Novel SARS-CoV-2 Main Protease Inhibitors.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 3972, doi. 10.3390/ijms24043972

By:

Geiger, Nina;
Diesendorf, Viktoria;
Roll, Valeria;
König, Eva-Maria;
Obernolte, Helena;
Sewald, Katherina;
Breidenbach, Julian;
Pillaiyar, Thanigaimalai;
Gütschow, Michael;
Müller, Christa E.;
Bodem, Jochen

Publication type:

Article

Cell-permeable high-affinity tracers for Gq proteins provide structural insights, reveal distinct binding kinetics and identify small molecule inhibitors.

Published in:

2020

By:

Kuschak, Markus;
Namasivayam, Vigneshwaran;
Rafehi, Muhammad;
Voss, Jan H.;
Garg, Jaspal;
Schlegel, Jonathan G.;
Abdelrahman, Aliaa;
Kehraus, Stefan;
Reher, Raphael;
Küppers, Jim;
Sylvester, Katharina;
Hinz, Sonja;
Matthey, Michaela;
Wenzel, Daniela;
Fleischmann, Bernd K.;
Pfeifer, Alexander;
Inoue, Asuka;
Gütschow, Michael;
König, Gabriele M.;
Müller, Christa E.

Publication type:

journal article

Polyketide Skeletons from the Marine Alga-Derived Fungus Coniothyrium cereale.

Published in:

European Journal of Organic Chemistry, 2012, v. 2012, n. 31, p. 6197, doi. 10.1002/ejoc.201200700

By:

Elsebai, Mahmoud Fahmi;
Nazir, Mamona;
Kehraus, Stefan;
Egereva, Ekaterina;
Ioset, Karine Ndjoko;
Marcourt, Laurence;
Jeannerat, Damien;
Gütschow, Michael;
Wolfender, Jean-Luc;
König, Gabriele M.

Publication type:

Article

Targeting the Main Protease of SARS‐CoV‐2: From the Establishment of High Throughput Screening to the Design of Tailored Inhibitors.

Published in:

Angewandte Chemie International Edition, 2021, v. 60, n. 18, p. 10423, doi. 10.1002/anie.202016961

By:

Breidenbach, Julian;
Lemke, Carina;
Pillaiyar, Thanigaimalai;
Schäkel, Laura;
Al Hamwi, Ghazl;
Diett, Miriam;
Gedschold, Robin;
Geiger, Nina;
Lopez, Vittoria;
Mirza, Salahuddin;
Namasivayam, Vigneshwaran;
Schiedel, Anke C.;
Sylvester, Katharina;
Thimm, Dominik;
Vielmuth, Christin;
Phuong Vu, Lan;
Zyulina, Maria;
Bodem, Jochen;
Gütschow, Michael;
Müller, Christa E.

Publication type:

Article

RECENT DEVELOPMENTS IN HYDANTOIN CHEMISTRY. A REVIEW.

Published in:

Organic Preparations & Procedures International, 2004, v. 36, n. 5, p. 391, doi. 10.1080/00304940409356627

By:

Meusel, Manuela;
Gütschow, Michael

Publication type:

Article

Tetrahydroimidazo[1,2‐a]pyrazine Derivatives: Synthesis and Evaluation as Gαq‐Protein Ligands.

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 55, p. 12615, doi. 10.1002/chem.202001446

By:

Küppers, Jim;
Benkel, Tobias;
Annala, Suvi;
Kimura, Kenichi;
Reinelt, Lisa;
Fleischmann, Bernd K.;
Kostenis, Evi;
Gütschow, Michael

Publication type:

Article

A Fluorescent-Labeled Phosphono Bisbenzguanidine As an Activity-Based Probe for Matriptase.

Published in:

Chemistry - A European Journal, 2017, v. 23, n. 22, p. 5205, doi. 10.1002/chem.201700319

By:

Häußler, Daniela;
Schulz ‐ Fincke, Anna ‐ Christina;
Beckmann, Anna ‐ Madeleine;
Keils, Aline;
Gilberg, Erik;
Mangold, Martin;
Bajorath, Jürgen;
Stirnberg, Marit;
Steinmetzer, Torsten;
Gütschow, Michael

Publication type:

Article

New Peptolides from the Cyanobacterium Nostoc insulare as Selective and Potent Inhibitors of Human Leukocyte Elastase.

Published in:

ChemBioChem, 2008, v. 9, n. 16, p. 2692, doi. 10.1002/cbic.200800415

By:

Mehner, Christian;
Müller, Daniela;
Kehraus, Stefan;
Hautmann, Stephanie;
Gütschow, Michael;
König, Gabriele M.

Publication type:

Article

Synthesis and Evaluation of Two Coumarin-Type.

Published in:

Chirality, 2013, v. 25, n. 12, p. 957, doi. 10.1002/chir.22240

By:

Mertens, Matthias D.;
Gütschow, Michael

Publication type:

Article

Michael Adducts of Palmitoylascorbic Acid: Effects on the Oxidative Burst of Neutrophils and the Production of Tumor Necrosis Factor-Alpha in Monocytes.

Published in:

Pharmacology, 2002, v. 66, n. 3, p. 162, doi. 10.1159/000063799

By:

Gütschow, Michael;
Hauschildt, Sunna;
Benard, Stefan;
Reichl, Sabine;
Witt, Uta G.;
Eger, Kurt;
Arnhold, Jürgen

Publication type:

Article

Preclinical Evaluation of a Novel Series of Polyfluorinated Thalidomide Analogs in Drug-Resistant Multiple Myeloma.

Published in:

Biomolecules (2218-273X), 2024, v. 14, n. 6, p. 725, doi. 10.3390/biom14060725

By:

Barton, Blaire E.;
Collins, Matthew K.;
Chau, Cindy H.;
Choo-Wosoba, Hyoyoung;
Venzon, David J.;
Steinebach, Christian;
Garchitorena, Kathleen M.;
Shah, Bhruga;
Sarin, Eric L.;
Gütschow, Michael;
Figg, William D.

Publication type:

Article

Calcium-sensing receptors signal constitutive macropinocytosis and facilitate the uptake of NOD2 ligands in macrophages.

Published in:

Nature Communications, 2016, v. 7, n. 4, p. 11284, doi. 10.1038/ncomms11284

By:

Canton, Johnathan;
Schlam, Daniel;
Breuer, Christian;
Gütschow, Michael;
Glogauer, Michael;
Grinstein, Sergio

Publication type:

Article

Synthesis, Structural Characterization, and Antiangiogenic Activity of Polyfluorinated Benzamides.

Published in:

ChemMedChem, 2018, v. 13, n. 19, p. 2080, doi. 10.1002/cmdc.201800263

By:

Steinebach, Christian;
Ambrożak, Agnieszka;
Dosa, Stefan;
Beedie, Shaunna L.;
Strope, Jonathan D.;
Schnakenburg, Gregor;
Figg, William D.;
Gütschow, Michael

Publication type:

Article

ω‐Phthalimidoalkyl Aryl Ureas as Potent and Selective Inhibitors of Cholesterol Esterase.

Published in:

ChemMedChem, 2018, v. 13, n. 17, p. 1833, doi. 10.1002/cmdc.201800388

By:

Dato, Florian M.;
Sheikh, Miriam;
Uhl, Rocky Z.;
Schüller, Alexandra W.;
Steinkrüger, Michaela;
Koch, Peter;
Neudörfl, Jörg‐Martin;
Gütschow, Michael;
Goldfuss, Bernd;
Pietsch, Markus

Publication type:

Article

Synthesis and Antiangiogenic Properties of Tetrafluorophthalimido and Tetrafluorobenzamido Barbituric Acids.

Published in:

ChemMedChem, 2016, v. 11, n. 23, p. 2621, doi. 10.1002/cmdc.201600496

By:

Ambrożak, Agnieszka;
Steinebach, Christian;
Gardner, Erin R.;
Beedie, Shaunna L.;
Schnakenburg, Gregor;
Figg, William D.;
Gütschow, Michael

Publication type:

Article

A Bisbenzamidine Phosphonate as a Janus-faced Inhibitor for Trypsin-like Serine Proteases.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1641, doi. 10.1002/cmdc.201500319

By:

Häußler, Daniela;
Scheidt, Tamara;
Stirnberg, Marit;
Steinmetzer, Torsten;
Gütschow, Michael

Publication type:

Article

Active Site Mapping of Human Cathepsin F with Dipeptide Nitrile Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 8, p. 1365, doi. 10.1002/cmdc.201500151

By:

Schmitz, Janina;
Furtmann, Norbert;
Ponert, Moritz;
Frizler, Maxim;
Löser, Reik;
Bartz, Ulrike;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Synthesis and Radiopharmacological Characterisation of a Fluorine-18-Labelled Azadipeptide Nitrile as a Potential PET Tracer for in vivo Imaging of Cysteine Cathepsins.

Published in:

ChemMedChem, 2013, v. 8, n. 8, p. 1330, doi. 10.1002/cmdc.201300135

By:

Löser, Reik;
Bergmann, Ralf;
Frizler, Maxim;
Mosch, Birgit;
Dombrowski, Lilli;
Kuchar, Manuela;
Steinbach, Jörg;
Gütschow, Michael;
Pietzsch, Jens

Publication type:

Article

Inside Cover: Synthesis and Radiopharmacological Characterisation of a Fluorine-18-Labelled Azadipeptide Nitrile as a Potential PET Tracer for in vivo Imaging of Cysteine Cathepsins (ChemMedChem 8/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 8, p. 1230, doi. 10.1002/cmdc.201390031

By:

Löser, Reik;
Bergmann, Ralf;
Frizler, Maxim;
Mosch, Birgit;
Dombrowski, Lilli;
Kuchar, Manuela;
Steinbach, Jörg;
Gütschow, Michael;
Pietzsch, Jens

Publication type:

Article

Inside Cover: Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants (ChemMedChem 1/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 2, doi. 10.1002/cmdc.201190061

By:

Maurer, Eva;
Sisay, Mihiret T.;
Stirnberg, Marit;
Steinmetzer, Torsten;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Insights into Matriptase-2 Substrate Binding and Inhibition Mechanisms by Analyzing Active-Site-Mutated Variants.

Published in:

ChemMedChem, 2012, v. 7, n. 1, p. 68, doi. 10.1002/cmdc.201100350

By:

Maurer, Eva;
Sisay, Mihiret T.;
Stirnberg, Marit;
Steinmetzer, Torsten;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Inhibition of Human Leukocyte Elastase by Brunsvicamides A-C: Cyanobacterial Cyclic Peptides.

Published in:

ChemMedChem, 2009, v. 4, n. 9, p. 1425, doi. 10.1002/cmdc.200900139

By:

Sisay, Mihiret T.;
Hautmann, Stephanie;
Mehner, Christian;
König, Gabriele M.;
Bajorath, Jürgen;
Gütschow, Michael

Publication type:

Article

Hit Expansion through Computational Selectivity Searching.

Published in:

ChemMedChem, 2009, v. 4, n. 1, p. 52, doi. 10.1002/cmdc.200800304

By:

Stumpfe, Dagmar;
Frizler, Maxim;
Sisay, Mihiret T.;
Batista, José;
Vogt, Ingo;
Gütschow, Michael;
Bajorath, Jürgen

Publication type:

Article