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Editorial: The GABAA receptor: a target of pharmacologically active molecules.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1440937
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- Article
Probes for the heterogeneity of muscimol binding sites in rat brain.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1368527
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- Article
Vascular effects of midazolam, flumazenil, and a novel imidazobenzodiazepine MP-III-058 on isolated rat aorta.
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- Canadian Journal of Physiology & Pharmacology, 2024, v. 102, n. 3, p. 206, doi. 10.1139/cjpp-2023-0285
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- Article
GABA<sub>A</sub> receptor-mediated seizure liabilities: a mixed-methods screening approach.
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- Cell Biology & Toxicology, 2023, v. 39, n. 6, p. 2793, doi. 10.1007/s10565-023-09803-y
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- Article
Pregnenolone sulfate analogues differentially modulate GABA<sub>A</sub> receptor closed/desensitised states.
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- British Journal of Pharmacology, 2023, v. 180, n. 19, p. 2482, doi. 10.1111/bph.16143
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- Article
Navigating the complex landscape of benzodiazepine- and Z-drug diversity: insights from comprehensive FDA adverse event reporting system analysis and beyond.
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- Frontiers in Psychiatry, 2023, p. 01, doi. 10.3389/fpsyt.2023.1188101
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- Article
Search for Novel Therapies for Essential Tremor Based on Positive Modulation of α6-Containing GABAA Receptors.
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- Tremor & Other Hyperkinetic Movements, 2023, v. 13, p. 1, doi. 10.5334/tohm.796
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- Article
Cys-loop receptors on cannabinoids: All high?
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- Frontiers in Physiology, 2022, v. 13, p. 1, doi. 10.3389/fphys.2022.1044575
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- Article
β subunits of GABA<sub>A</sub> receptors form proton-gated chloride channels: Insights into the molecular basis.
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- Communications Biology, 2022, v. 5, n. 1, p. 1, doi. 10.1038/s42003-022-03720-2
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- Article
Unravelling the Turn‐On Fluorescence Mechanism of a Fluorescein‐Based Probe in GABA<sub>A</sub> Receptors.
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- Angewandte Chemie, 2022, v. 134, n. 30, p. 1, doi. 10.1002/ange.202205198
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- Article
Rücktitelbild: Unravelling the Turn‐On Fluorescence Mechanism of a Fluorescein‐Based Probe in GABA<sub>A</sub> Receptors (Angew. Chem. 30/2022).
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- Angewandte Chemie, 2022, v. 134, n. 30, p. 1, doi. 10.1002/ange.202205198
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- Article
Unravelling the Turn‐On Fluorescence Mechanism of a Fluorescein‐Based Probe in GABA<sub>A</sub> Receptors.
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- Angewandte Chemie International Edition, 2022, v. 61, n. 30, p. 1, doi. 10.1002/anie.202205198
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- Article
Back Cover: Unravelling the Turn‐On Fluorescence Mechanism of a Fluorescein‐Based Probe in GABA<sub>A</sub> Receptors (Angew. Chem. Int. Ed. 30/2022).
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- Angewandte Chemie International Edition, 2022, v. 61, n. 30, p. 1, doi. 10.1002/anie.202205198
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- Article
Tricyclic antipsychotics and antidepressants can inhibit α5‐containing GABA<sub>A</sub> receptors by two distinct mechanisms.
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- British Journal of Pharmacology, 2022, v. 179, n. 14, p. 3675, doi. 10.1111/bph.15807
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- Article
A de novo missense variant in GABRA4 alters receptor function in an epileptic and neurodevelopmental phenotype.
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- Epilepsia (Series 4), 2022, v. 63, n. 4, p. e35, doi. 10.1111/epi.17188
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- Article
Structure-Guided Computational Methods Predict Multiple Distinct Binding Modes for Pyrazoloquinolinones in GABA<sub>A</sub> Receptors.
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- Frontiers in Neuroscience, 2021, v. 14, p. N.PAG, doi. 10.3389/fnins.2020.611953
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- Article
Molecular basis of mood and cognitive adverse events elucidated via a combination of pharmacovigilance data mining and functional enrichment analysis.
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- Archives of Toxicology, 2020, v. 94, n. 8, p. 2829, doi. 10.1007/s00204-020-02788-1
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- Article
Allosteric GABAA Receptor Modulators—A Review on the Most Recent Heterocyclic Chemotypes and Their Synthetic Accessibility †.
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- Molecules, 2020, v. 25, n. 4, p. 999, doi. 10.3390/molecules25040999
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- Article
A novel de novo variant of GABRA1 causes increased sensitivity for GABA in vitro.
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- Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-59323-6
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- Article
GABAA Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain—Can the Promiscuity Code Be Cracked?
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- International Journal of Molecular Sciences, 2020, v. 21, n. 1, p. 334, doi. 10.3390/ijms21010334
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- Article
Phenotypic variability of GABRA1‐related epilepsy in monozygotic twins.
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- Annals of Clinical & Translational Neurology, 2019, v. 6, n. 11, p. 2317, doi. 10.1002/acn3.50895
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- Article
Trigeminal neuropathic pain development and maintenance in rats are suppressed by a positive modulator of α6 GABA<sub>A</sub> receptors.
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- 2019
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- journal article
Cerebellar α<sub>6</sub> -subunit-containing GABA<sub>A</sub> receptors: a novel therapeutic target for disrupted prepulse inhibition in neuropsychiatric disorders.
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- 2018
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- journal article
Negative allosteric modulation of alpha 5-containing GABAA receptors engenders antidepressant-like effects and selectively prevents age-associated hyperactivity in tau-depositing mice.
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- Psychopharmacology, 2018, v. 235, n. 4, p. 1151, doi. 10.1007/s00213-018-4832-9
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- Article
Towards functional selectivity for α6β3γ2 GABA<sub>A</sub> receptors: a series of novel pyrazoloquinolinones.
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- 2018
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- journal article
Targeting the GABA<sub>A</sub> Receptor α4 Subunit in Airway Smooth Muscle to Alleviate Bronchoconstriction.
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- American Journal of Respiratory Cell & Molecular Biology, 2016, v. 54, n. 4, p. E1, doi. 10.1165/rcmb.2015-0176oc
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- Article
Targeting the γ-Aminobutyric Acid A Receptor a4 Subunit in Airway Smooth Muscle to Alleviate Bronchoconstriction.
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- American Journal of Respiratory Cell & Molecular Biology, 2016, v. 54, n. 4, p. 546, doi. 10.1165/rcmb.2015-0176OC
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- Article
GABA<sub>A</sub> receptor subtypes: structural variety raises hope for new therapy concepts.
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- Neuroforum, 2015, v. 21, n. 4, p. 97, doi. 10.1515/s13295-015-0016-9
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- Article
Functional characterization of ivermectin binding sites in α1β2γ2L GABA(A) receptors.
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- Frontiers in Molecular Neuroscience, 2015, p. 1, doi. 10.3389/fnmol.2015.00055
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- Article
A Pentasymmetric Open Channel Blocker for Cys-Loop Receptor Channels.
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- PLoS ONE, 2014, v. 9, n. 9, p. 1, doi. 10.1371/journal.pone.0106688
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- Article
Unexpected Properties of δ-Containing GABA Receptors in Response to Ligands Interacting with the α+ β− Site.
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- Neurochemical Research, 2014, v. 39, n. 6, p. 1057, doi. 10.1007/s11064-013-1156-3
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- Article
Comparing the high affinity benzodiazepine binding site with the homologous "CGS 9895" site in GABA‐A receptors (1059.1).
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- FASEB Journal, 2014, v. 28, p. N.PAG, doi. 10.1096/fasebj.28.1_supplement.1059.1
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- Article
Experiment‐guided virtual screening provides new high affinity ligands for the benzodiazepine site on GABA‐A receptors (654.4).
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- FASEB Journal, 2014, v. 28, p. N.PAG, doi. 10.1096/fasebj.28.1_supplement.654.4
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- Article
Molecular analysis of the site for 2-arachidonylglycerol (2- AG) on the β<sub>2</sub> subunit of GABA<sub>A</sub> receptors.
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- Journal of Neurochemistry, 2013, v. 126, n. 1, p. 29, doi. 10.1111/jnc.12270
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Identification of novel positive allosteric modulators and null modulators at the GABA<sub>A</sub> receptor α+β− interface.
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- British Journal of Pharmacology, 2013, v. 169, n. 2, p. 371, doi. 10.1111/bph.12151
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Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface.
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- 2013
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- journal article
Subtype selectivity of α+β− site ligands of GABA<sub>A</sub> receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors.
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- British Journal of Pharmacology, 2013, v. 169, n. 2, p. 384, doi. 10.1111/bph.12153
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- Article
Subtype selectivity of α+β- site ligands of GABAA receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors.
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- 2013
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- journal article
A novel GABA(A) receptor pharmacology: drugs interacting with the α(+) β(-) interface.
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- 2012
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- journal article
A novel GABA<sub>A</sub> receptor pharmacology: drugs interacting with the α<sup>+</sup>β<sup>-</sup> interface.
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- British Journal of Pharmacology, 2012, v. 166, n. 2, p. 476, doi. 10.1111/j.1476-5381.2011.01779.x
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- Article
Diazepam-bound GABA<sub>A</sub> receptor models identify new benzodiazepine binding-site ligands.
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- Nature Chemical Biology, 2012, v. 8, n. 5, p. 455, doi. 10.1038/nchembio.917
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- Article
The GABA<sub>A</sub> Receptor α + β Interface: A Novel Target for Subtype Selective Drugs.
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- Journal of Neuroscience, 2011, v. 31, n. 3, p. 870, doi. 10.1523/JNEUROSCI.5012-10.2011
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Identification of amino acid residues important for assembly of GABA<sub>A</sub> receptor α1 and γ2 subunits.
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- Journal of Neurochemistry, 2006, v. 96, n. 4, p. 983, doi. 10.1111/j.1471-4159.2005.03626.x
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Raman and infrared vibrational spectra, normal coordinate analysis and ab initio calculations of 1,1,2,2-tetrachlorodisilane and ab initio calculations of hexachlorodisilane.
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- Journal of Raman Spectroscopy, 1997, v. 28, n. 8, p. 589, doi. 10.1002/(SICI)1097-4555(199708)28:8<589::AID-JRS135>3.0.CO;2-G
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- Article