Works matching AU Elkaeed, Eslam B.

Results: 147

Construction of Te-ZnO@S-g-C3N4 Heterojunction Nanocomposites for the Efficient Removal of Methylene Blue, Antifungal Activity, and Adsorption of Cr(VI) Ion.

Published in:

Adsorption Science & Technology, 2023, v. 2023, p. 1, doi. 10.1155/2023/6736182

By:

Aroosh, Komal;
Javed, Mohsin;
Hussain, Nadia;
Alhujaily, Ahmad;
Iqbal, Shahid;
Alotaibi, Mohammed T.;
Faizan, Muhammad;
Khan, Muhammad Shuaib;
Bahadur, Ali;
Qayyum, Muhammad Abdul;
Awwad, Nasser S.;
Jazaa, Yosef;
Al-Fawzan, Foziah F.;
Elkaeed, Eslam B.;
Kooh, Muhammad Raziq Rahimi

Publication type:

Article

Comparative Evaluation of Various Extraction Techniques for Secondary Metabolites from Bombax ceiba L. Flowering Plants along with In Vitro Anti-Diabetic Performance.

Published in:

Bioengineering (Basel), 2022, v. 9, n. 10, p. N.PAG, doi. 10.3390/bioengineering9100486

By:

Yasien, Sara;
Iqbal, Muhammad Muntazir;
Javed, Mohsin;
Alnuwaiser, Maha Abdallah;
Iqbal, Shahid;
Mahmood, Qaiser;
Elkaeed, Eslam B.;
Dera, Ayed A.;
Alrbyawi, Hamad;
Pashameah, Rami Adel;
Alzahrani, Eman;
Farouk, Abd-ElAziem

Publication type:

Article

Combined Computational and Experimental Studies of Anabasine Encapsulation by Beta-Cyclodextrin.

Published in:

Plants (2223-7747), 2022, v. 11, n. 17, p. 2283, doi. 10.3390/plants11172283

By:

Muldakhmetov, Zeinolla;
Fazylov, Serik;
Nurkenov, Oral;
Gazaliev, Arstan;
Sarsenbekova, Akmaral;
Pustolaikina, Irina;
Nurmaganbetov, Zhangeldy;
Seilkhanov, Olzhas;
Alsfouk, Aisha A.;
Elkaeed, Eslam B.;
Eissa, Ibrahim H.;
Metwaly, Ahmed M.

Publication type:

Article

Isolation and In Silico Inhibitory Potential against SARS-CoV-2 RNA Polymerase of the Rare Kaempferol 3- O -(6″- O -acetyl)-Glucoside from Calligonum tetrapterum.

Published in:

Plants (2223-7747), 2022, v. 11, n. 15, p. 2072, doi. 10.3390/plants11152072

By:

Suleimen, Yerlan M.;
Jose, Rani A.;
Mamytbekova, Gulnur K.;
Suleimen, Raigul N.;
Ishmuratova, Margarita Y.;
Dehaen, Wim;
Alsfouk, Bshra A.;
Elkaeed, Eslam B.;
Eissa, Ibrahim H.;
Metwaly, Ahmed M.

Publication type:

Article

The Computational Preventive Potential of the Rare Flavonoid, Patuletin, Isolated from Tagetes patula , against SARS-CoV-2.

Published in:

Plants (2223-7747), 2022, v. 11, n. 14, p. N.PAG, doi. 10.3390/plants11141886

By:

Metwaly, Ahmed M.;
Elkaeed, Eslam B.;
Alsfouk, Bshra A.;
Saleh, Abdulrahman M.;
Mostafa, Ahmad E.;
Eissa, Ibrahim H.

Publication type:

Article

Combined In Silico and Experimental Investigations of Resveratrol Encapsulation by Beta-Cyclodextrin.

Published in:

Plants (2223-7747), 2022, v. 11, n. 13, p. 1678, doi. 10.3390/plants11131678

By:

Iskineyeva, Ainara;
Fazylov, Serik;
Bakirova, Ryszhan;
Sarsenbekova, Akmaral;
Pustolaikina, Irina;
Seilkhanov, Olzhas;
Alsfouk, Aisha A.;
Elkaeed, Eslam B.;
Eissa, Ibrahim H.;
Metwaly, Ahmed M.

Publication type:

Article

A Theobromine Derivative with Anticancer Properties Targeting VEGFR‐2: Semisynthesis, in silico and in vitro Studies.

Published in:

ChemistryOpen, 2023, v. 12, n. 10, p. 1, doi. 10.1002/open.202300066

By:

Eissa, Ibrahim H.;
Yousef, Reda G.;
Elkady, Hazem;
Elkaeed, Eslam B.;
Alsfouk, Aisha A.;
Husein, Dalal Z.;
Ibrahim, Ibrahim M.;
Radwan, Mohamed M.;
Metwaly, Ahmed M.

Publication type:

Article

The Discovery of Potential SARS-CoV-2 Natural Inhibitors among 4924 African Metabolites Targeting the Papain-like Protease: A Multi-Phase In Silico Approach.

Published in:

Metabolites (2218-1989), 2022, v. 12, n. 11, p. 1122, doi. 10.3390/metabo12111122

By:

Elkaeed, Eslam B.;
Khalifa, Mohamed M.;
Alsfouk, Bshra A.;
Alsfouk, Aisha A.;
El-Attar, Abdul-Aziz M. M.;
Eissa, Ibrahim H.;
Metwaly, Ahmed M.

Publication type:

Article

A New Anticancer Semisynthetic Theobromine Derivative Targeting EGFR Protein: CADDD Study.

Published in:

Life (2075-1729), 2023, v. 13, n. 1, p. 191, doi. 10.3390/life13010191

By:

Eissa, Ibrahim H.;
Yousef, Reda G.;
Elkady, Hazem;
Alsfouk, Aisha A.;
Alsfouk, Bshra A.;
Husein, Dalal Z.;
Ibrahim, Ibrahim M.;
Elkaeed, Eslam B.;
Metwaly, Ahmed M.

Publication type:

Article

Discovery of Potential SARS-CoV-2 Papain-like Protease Natural Inhibitors Employing a Multi-Phase In Silico Approach.

Published in:

Life (2075-1729), 2022, v. 12, n. 9, p. 1407, doi. 10.3390/life12091407

By:

Elkaeed, Eslam B.;
Metwaly, Ahmed M.;
Alesawy, Mohamed S.;
Saleh, Abdulrahman M.;
Alsfouk, Aisha A.;
Eissa, Ibrahim H.

Publication type:

Article

Isolation, Crystal Structure, and In Silico Aromatase Inhibition Activity of Ergosta-5, 22-dien-3β-ol from the Fungus Gyromitra esculenta.

Published in:

Journal of Chemistry, 2021, p. 1, doi. 10.1155/2021/5529786

By:

Suleimen, Yerlan Melsuly;
Metwaly, Ahmed M.;
Mostafa, Ahmad E.;
Elkaeed, Eslam B.;
Liu, Hong-Wei;
Basnet, Buddha Bahadur;
Suleimen, Raigul Nurbekkyzy;
Ishmuratova, Margarita Yulayevna;
Turdybekov, Koblandy Muboryakovich;
Van Heсke, Kristof

Publication type:

Article

Comprehensive In Silico Screening of the Antiviral Potentialities of a New Humulene Glucoside from Asteriscus hierochunticus against SARS-CoV-2.

Published in:

Journal of Chemistry, 2021, p. 1, doi. 10.1155/2021/5541876

By:

Imieje, Vincent O.;
Zaki, Ahmed A.;
Metwaly, Ahmed M.;
Mostafa, Ahmad E.;
Elkaeed, Eslam B.;
Falodun, Abiodun

Publication type:

Article

Isolation and In Silico Anti-COVID-19 Main Protease (Mpro) Activities of Flavonoids and a Sesquiterpene Lactone from Artemisia sublessingiana.

Published in:

Journal of Chemistry, 2021, p. 1, doi. 10.1155/2021/5547013

By:

Jalmakhanbetova, Roza I.;
Suleimen, Yerlan M.;
Oyama, Masayoshi;
Elkaeed, Eslam B.;
Eissa, Ibrahim. H.;
Suleimen, Raigul N.;
Metwaly, Ahmed M.;
Ishmuratova, Margarita Yu.

Publication type:

Article

Synthesis and Molecular Docking of Some Grossgemin Amino Derivatives as Tubulin Inhibitors Targeting Colchicine Binding Site.

Published in:

Journal of Chemistry, 2021, p. 1, doi. 10.1155/2021/5586515

By:

Jalmakhanbetova, R. I.;
Elkaeed, Eslam B.;
Eissa, Ibrahim H.;
Metwaly, Ahmed M.;
Suleimen, Ye. M.

Publication type:

Article

In Vitro and In Silico Cytotoxic and Antibacterial Activities of a Diterpene from Cousinia alata Schrenk.

Published in:

Journal of Chemistry, 2021, p. 1, doi. 10.1155/2021/5542455

By:

Zhanzhaxina, Almira;
Suleimen, Yerlan;
Metwaly, Ahmed M.;
Eissa, Ibrahim H.;
Elkaeed, Eslam B.;
Suleimen, Raigul;
Ishmuratova, Margarita;
Akatan, Kydyrmolla;
Luyten, Walter

Publication type:

Article

Discovery of potential FDA-approved SARS-CoV-2 Papain-like protease inhibitors: A multi-phase in silico approach.

Published in:

Journal of Chemical Research, 2024, v. 48, n. 6, p. 1, doi. 10.1177/17475198241298547

By:

Metwaly, Ahmed M;
Elkaeed, Eslam B;
Khalifa, Mohamed M;
Alsfouk, Aisha A;
Amin, Fatma G;
Ibrahim, Ibrahim M;
Eissa, Ibrahim H

Publication type:

Article

Computer-aided drug discovery of natural antiviral metabolites as potential SARS-CoV-2 helicase inhibitors.

Published in:

Journal of Chemical Research, 2024, v. 48, n. 1, p. 1, doi. 10.1177/17475198231221253

By:

Elkaeed, Eslam B;
Eissa, Ibrahim H;
Saleh, Abdulrahman M;
Alsfouk, Bshra A;
Metwaly, Ahmed M

Publication type:

Article

Chromium (III) Ions Were Extracted from Wastewater Effluent Using a Synergistic Green Membrane with a BinaryCombination of D2EHPA and Kerosene.

Published in:

Catalysts (2073-4344), 2022, v. 12, n. 10, p. 1220, doi. 10.3390/catal12101220

By:

Sarfraz, Sadaf;
Abid, Akmal Javed;
Javed, Mohsin;
Iqbal, Shahid;
Aljazzar, Samar O.;
Zahra, Manzar;
Alrbyawi, Hamad;
Elkaeed, Eslam B.;
Somaily, H. H.;
Pashameah, Rami Adel;
Alzahrani, Eman;
Farouk, Abd-ElAziem

Publication type:

Article

Optimization of Deposition Conditions of SrZrS3 Perovskite Thin Films Grown by Chemical Bath Deposition.

Published in:

Journal of Electronic Materials, 2024, v. 53, n. 3, p. 1551, doi. 10.1007/s11664-023-10825-9

By:

Fatima, Areej;
Iqbal, Shahid;
Fazal, Tanzeela;
Ismail, Bushra;
Shah, Mazloom;
Ayub, Ambreen;
Mahmood, Qaiser;
Awwad, Nasser S.;
Ibrahium, Hala A.;
Al-Fawzan, Foziah F.;
Elkaeed, Eslam B.

Publication type:

Article

Synthesis of novel biodegradable starch-PMA and Ag@starch-PMA polymer composite for boosting charge separation ability and superior photocatalytic performance.

Published in:

Journal of Materials Science: Materials in Electronics, 2023, v. 34, n. 21, p. 1, doi. 10.1007/s10854-023-10997-4

By:

Amjad, Muhammad;
Mohyuddin, Ayesha;
Javed, Mohsin;
Iqbal, Shahid;
Liaquat, Rabia;
Alotaibi, Mohammed T.;
Ulfat, Wajad;
Althobiti, Randa A.;
Alzahrani, Eman;
Farouk, Abd-ElAziem;
Al-Anazy, Murefah Mana;
Elkaeed, Eslam B.

Publication type:

Article

Novel 2-(5-Aryl-4,5-Dihydropyrazol-1-yl)thiazol-4-One as EGFR Inhibitors: Synthesis, Biological Assessment and Molecular Docking Insights.

Published in:

Drug Design, Development & Therapy, 2022, v. 16, p. 1457, doi. 10.2147/DDDT.S356988

By:

Al-Warhi, Tarfah;
El Kerdawy, Ahmed M;
Said, Mohamed A;
Albohy, Amgad;
Elsayed, Zainab M;
Aljaeed, Nada;
Elkaeed, Eslam B;
Eldehna, Wagdy M;
Abdel-Aziz, Hatem A;
Abdelmoaz, Miral A

Publication type:

Article

New Series of VEGFR-2 Inhibitors and Apoptosis Enhancers: Design, Synthesis and Biological Evaluation.

Published in:

Drug Design, Development & Therapy, 2022, v. 16, p. 587, doi. 10.2147/DDDT.S344750

By:

Abdallah, Abdallah E;
Mabrouk, Reda R;
Elnagar, Mohamed R;
Farrag, Amel Mostafa;
Kalaba, Mohamed H;
Sharaf, Mohamed H;
El-Fakharany, Esmail M;
Bakhotmah, Dina Abed;
Elkaeed, Eslam B;
Ward, Maged Mohammed Saleh Al

Publication type:

Article

A Systematic Review of the Global Intervention for SARS-CoV-2 Combating: From Drugs Repurposing to Molnupiravir Approval.

Published in:

Drug Design, Development & Therapy, 2022, v. 16, p. 685, doi. 10.2147/DDDT.S354841

By:

Ashour, Nada A;
Elmaaty, Ayman Abo;
Sarhan, Amany A;
Elkaeed, Eslam B;
Moussa, Ahmed M;
Erfan, Ibrahim Ali;
Al-Karmalawy, Ahmed A

Publication type:

Article

Chemical activation and magnetization of onion waste derived carbon for arsenic removal.

Published in:

Arabian Journal of Chemistry, 2023, v. 16, n. 10, p. N.PAG, doi. 10.1016/j.arabjc.2023.105118

By:

Bibi, Fozia;
Hussain, Rafaqat;
Iqbal, Naseem;
Saeed, Shaukat;
Waseem, Muhammad;
Elkaeed, Eslam B.;
Al-Anazy, Murefah Mana;
Haq, Sirajul

Publication type:

Article

Synthesis, molecular docking and ADMET studies of bis-benzimidazole-based thiadiazole derivatives as potent inhibitors, in vitro α-amylase and α-glucosidase.

Published in:

Arabian Journal of Chemistry, 2023, v. 16, n. 7, p. N.PAG, doi. 10.1016/j.arabjc.2023.104847

By:

Khan, Shoaib;
Iqbal, Shahid;
Rehman, Wajid;
Hussain, Nadia;
Hussain, Rafaqat;
Shah, Mazloom;
Ali, Farhan;
Fouda, Ahmed M.;
Khan, Yousaf;
Dera, Ayed A.;
Issa Alahmdi, Mohammed;
Bahadur, Ali;
Al-ghulikah, Hanan A.;
Elkaeed, Eslam B.

Publication type:

Article

Computational modeling of Hg/Ni ions separation via MOF/LDH nanocomposite: Machine learning based modeling.

Published in:

Arabian Journal of Chemistry, 2022, v. 15, n. 12, p. N.PAG, doi. 10.1016/j.arabjc.2022.104261

By:

Ibrahim, Munjed M.;
Alnuwaiser, Maha Abdallah;
Elkaeed, Eslam B.;
Kotb, Hossam;
Alshehri, Sameer;
Abourehab, Mohammed A.S.

Publication type:

Article

Quantification of multi-class pesticides in stomach contents and milk by gas chromatography–mass spectrometry with liquid extraction method.

Published in:

Arabian Journal of Chemistry, 2022, v. 15, n. 7, p. N.PAG, doi. 10.1016/j.arabjc.2022.103937

By:

Yasien, Sara;
Iqbal, Muhammad Muntazir;
Javed, Mohsin;
Iqbal, Shahid;
Ahmad, Zahoor;
Tamam, Nissren;
Nadeem, Sohail;
Elkaeed, Eslam B.;
Alzhrani, Rami M.;
Awwad, Nasser S.;
Ibrahium, Hala A.;
Hakami, Rabab A.

Publication type:

Article

Antileishmanial Derivatives of Humulene from Asteriscus hierochunticus with in silico Tubulin Inhibition Potential.

Published in:

Records of Natural Products, 2022, v. 16, n. 2, p. 150, doi. 10.25135/rnp.253.21.01.1945

By:

Imieje, Vincent O.;
Zaki, Ahmed A.;
Metwaly, Ahmed M.;
Eissa, Ibrahim. H.;
Elkaeed, Eslam B.;
Ali, Zulfiqar;
Khan, Ikhlas A.;
Falodun, Abiodun

Publication type:

Article

Computer-Assisted Drug Discovery of a Novel Theobromine Derivative as an EGFR Protein-Targeted Apoptosis Inducer.

Published in:

Evolutionary Bioinformatics, 2023, p. 1, doi. 10.1177/11769343231217916

By:

Eissa, Ibrahim H;
Yousef, Reda G;
Elkaeed, Eslam B;
Alsfouk, Aisha A;
Husein, Dalal Z;
Ibrahim, Ibrahim M;
El-Mahdy, Hesham A;
Elkady, Hazem;
Metwaly, Ahmed M

Publication type:

Article

Computer-Assisted Drug Discovery of a Novel Theobromine Derivative as an EGFR Protein-Targeted Apoptosis Inducer.

Published in:

Evolutionary Bioinformatics, 2023, v. 19, p. 1, doi. 10.1177/11769343231217916

By:

Eissa, Ibrahim H.;
Yousef, Reda G.;
Elkaeed, Eslam B.;
Alsfouk, Aisha A.;
Husein, Dalal Z.;
Ibrahim, Ibrahim M.;
El-Mahdy, Hesham A.;
Elkady, Hazem;
Metwaly, Ahmed M.

Publication type:

Article

Novel Thiazolidine‐2,4‐Dione Derivatives as Potential VEGFR‐2 Inhibitors: Synthesis, Biological Testing, and in Silico Studies.

Published in:

ChemistrySelect, 2024, v. 9, n. 11, p. 1, doi. 10.1002/slct.202303095

By:

Eissa, Ibrahim;
Elkady, Hazem;
Taghour, Mohammed S.;
Elwan, Alaa;
Dahab, Mohammed A.;
Hagras, Mohamed;
Elkaeed, Eslam B.;
Alsfouk, Bshra A.;
Ibrahim, Ibrahim M.;
Husein, Dalal Z.;
Hafez, Elsayed E.;
Mansour, Hanem M.;
Metwaly, Ahmed;
Mahdy, Hazem A.

Publication type:

Article

Discovery of Anti‐Breast Cancer Thiophene Sulfonamide Derivatives: Design, Synthesis, Molecular Docking against EGFR, MM‐PBSA, MD Simulations, ADME/Tox, and in vitro Studies.

Published in:

ChemistrySelect, 2023, v. 8, n. 27, p. 1, doi. 10.1002/slct.202301596

By:

Patel, Ashish K.;
Shah, Ujashkumar A;
Soni, Jigar Y.;
Metwaly, Ahmed M.;
Elkaeed, Eslam B.;
Eissa, Ibrahim H.;
Teli, Divya M.;
Patel, Purvesh R.;
Patel, Bhavin H.;
Valand, Nikunj;
Patel, Manish B.

Publication type:

Article

Synergistic Influences of Doping Techniques and Well‐Defined Heterointerface Formation to Improve the Photocatalytic Ability of the S‐ZnO/GO Nanocomposite.

Published in:

ChemistrySelect, 2022, v. 7, n. 29, p. 1, doi. 10.1002/slct.202201913

By:

Javed, Mohsin;
Qamar, Muhammad Azam;
Iqbal, Shahid;
Aljazzar, Samar O.;
Iqbal, Sadia;
Khan, Humaira;
Abourehab, Mohammed A. S.;
Elkaeed, Eslam B.;
Alharthi, Abdulrahman I.;
Awwad, Nasser S.;
Ibrahium, Hala A.

Publication type:

Article

A multidisciplinary approach to the antioxidant and hepatoprotective activities of Arbutus pavarii Pampan fruit; in vitro and in Vivo biological evaluations, and in silico investigations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2023.2293639

By:

Elshibani, Fatma A.;
Alamami, Abdullah D.;
Mohammed, Hamdoon A.;
Rasheed, Rabab Ahmed;
El Sabban, Radwa M.;
Yehia, Mohamed A.;
Abdel Mageed, Sherif S.;
Majrashi, Taghreed A.;
Elkaeed, Eslam B.;
El Hassab, Mahmoud A.;
Eldehna, Wagdy M.;
El-Ashrey, Mohamed K.

Publication type:

Article

Comparative metabolic study of the chloroform fraction of three Cystoseira species based on UPLC/ESI/MS analysis and biological activities.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2023.2292482

By:

Aly, Shaza H.;
Elissawy, Ahmed M.;
El Hassab, Mahmoud A.;
Majrashi, Taghreed A.;
Hassan, Fatma E.;
Elkaeed, Eslam B.;
Eldehna, Wagdy M.;
Singab, Abdel Nasser B.

Publication type:

Article

Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2278022

By:

Haffez, Hesham;
Elsayed, Nosaiba A.;
Ahmed, Marwa F.;
Fatahala, Samar S.;
Khaleel, Eman F.;
Badi, Rehab Mustafa;
Elkaeed, Eslam B.;
El Hassab, Mahmoud A.;
Hammad, Sherif F.;
Eldehna, Wagdy M.;
Masurier, Nicolas;
El-Haggar, Radwan

Publication type:

Article

Design, synthesis, docking, MD simulations, and anti-proliferative evaluation of thieno[2,3-d]pyrimidine derivatives as new EGFR inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2220579

By:

Sobh, Eman A.;
Dahab, Mohammed A.;
Elkaeed, Eslam B.;
Alsfouk, Aisha A.;
Ibrahim, Ibrahim M.;
Metwaly, Ahmed M.;
Eissa, Ibrahim H.

Publication type:

Article

Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2203389

By:

Shaldam, Moataz A.;
Almahli, Hadia;
Angeli, Andrea;
Badi, Rehab Mustafa;
Khaleel, Eman F.;
Zain-Alabdeen, Abdelrahman I.;
Elsayed, Zainab M.;
Elkaeed, Eslam B.;
Salem, Rofaida;
Supuran, Claudiu T.;
Eldehna, Wagdy M.;
Tawfik, Haytham O.

Publication type:

Article

Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407

By:

Badawi, Waleed A.;
Rashed, Mahmoud;
Nocentini, Alessio;
Bonardi, Alessandro;
Abd-Alhaseeb, Mohammad M.;
Al-Rashood, Sara T.;
Veerakanellore, Giri Babu;
Majrashi, Taghreed A.;
Elkaeed, Eslam B.;
Elgendy, Bahaa;
Gratteri, Paola;
Supuran, Claudiu T.;
Eldehna, Wagdy M.;
Elagawany, Mohamed

Publication type:

Article

Topo II inhibition and DNA intercalation by new phthalazine-based derivatives as potent anticancer agents: design, synthesis, anti-proliferative, docking, and in vivo studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 299, doi. 10.1080/14756366.2021.2007905

By:

Khalifa, Mohamed M.;
Al-Karmalawy, Ahmed A.;
Elkaeed, Eslam B.;
Nafie, Mohamed S.;
Tantawy, Mohamed A.;
Eissa, Ibrahim H.;
Mahdy, Hazem A.

Publication type:

Article

Synthesis, biological evaluation, and molecular docking of new series of antitumor and apoptosis inducers designed as VEGFR-2 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 573, doi. 10.1080/14756366.2021.2017911

By:

Abdallah, Abdallah E.;
Mabrouk, Reda R.;
Saleh Al Ward, Maged Mohammed;
Eissa, Sally I.;
Elkaeed, Eslam B.;
Mehany, Ahmed B. M.;
Abo-Saif, Mariam A.;
El-Feky, Ola A.;
Alesawy, Mohamed S.;
El-Zahabi, Mohamed Ayman

Publication type:

Article

Synthesis, biological evaluation, and in silico studies of new CDK2 inhibitors based on pyrazolo[3,4-d]pyrimidine and pyrazolo[4,3-e][1,2/4]triazolo[1/5-c]pyrimidine scaffold with apoptotic activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1957, doi. 10.1080/14756366.2022.2086866

By:

Mandour, Asmaa A.;
Nassar, Ibrahim F.;
Abdel Aal, Mohammed T.;
Shahin, Mahmoud A. E.;
El-Sayed, Wael A.;
Hegazy, Maghawry;
Yehia, Amr Mohamed;
Ismail, Ahmed;
Hagras, Mohamed;
Elkaeed, Eslam B.;
Refaat, Hanan M.;
Ismail, Nasser S. M.

Publication type:

Article

New quinoline and isatin derivatives as apoptotic VEGFR-2 inhibitors: design, synthesis, anti-proliferative activity, docking, ADMET, toxicity, and MD simulation studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2191, doi. 10.1080/14756366.2022.2110869

By:

Elkaeed, Eslam B.;
Taghour, Mohammed S.;
Mahdy, Hazem A.;
Eldehna, Wagdy M.;
El-Deeb, Nehal M.;
Kenawy, Ahmed M.;
Alsfouk, Bshra A.;
Dahab, Mohammed A.;
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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 403, doi. 10.1080/14756366.2021.2015343

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Elkady, Hazem;
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Ismail, Ahmed;
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Eissa, Ibrahim H.;
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Khalifa, Mohamed M.

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Multi-stage structure-based virtual screening approach towards identification of potential SARS-CoV-2 NSP13 helicase inhibitors.

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 563, doi. 10.1080/14756366.2021.2022659

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El Hassab, Mahmoud A.;
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Abou-Seri, Sahar M.

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1227, doi. 10.1080/14756366.2022.2062337

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Eldehna, Wagdy M.;
Maklad, Raed M.;
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Kerdawy, Ahmed M. El

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1389, doi. 10.1080/14756366.2022.2070744

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Yousef, Reda G.;
Ibrahim, Albaraa;
Khalifa, Mohamed M.;
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Metwaly, Ahmed M.;
Eissa, Ibrahim H.

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2283, doi. 10.1080/14756366.2022.2112575

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Gaber, Ahmed A.;
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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1053, doi. 10.1080/14756366.2022.2062752

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Elzahabi, Heba S. A.;
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Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1903, doi. 10.1080/14756366.2022.2085693

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Taghour, Mohammed S.;
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Kenawy, Ahmed M.;
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Eissa, Ibrahim. H.

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