Works by El-Gamal, Mohammed I.

Results: 36

An overview of the latest outlook of sulfamate derivatives as anticancer candidates (2020–2024).

Published in:

Archiv der Pharmazie, 2024, v. 357, n. 10, p. 1, doi. 10.1002/ardp.202400331

By:

Mustafa, Esra M.;
Shahin, Afnan I.;
Alrashed, Aishah S.;
Bahaaddin, Aesheh H.;
Alajmi, Aljawhra A.;
Hashem, Omar;
Anbar, Hanan S.;
El‐Gamal, Mohammed I.

Publication type:

Article

Design and synthesis of novel anti-urease imidazothiazole derivatives with promising antibacterial activity against Helicobacter pylori.

Published in:

PLoS ONE, 2023, v. 18, n. 6, p. 1, doi. 10.1371/journal.pone.0286684

By:

Shahin, Afnan I.;
Zaib, Sumera;
Zaraei, Seyed-Omar;
Kedia, Reena A.;
Anbar, Hanan S.;
Younas, Muhammad Tayyab;
Al-Tel, Taleb H.;
Khoder, Ghalia;
El-Gamal, Mohammed I.

Publication type:

Article

Recent advances with alkaline phosphatase isoenzymes and their inhibitors.

Published in:

Archiv der Pharmazie, 2020, v. 353, n. 5, p. 1, doi. 10.1002/ardp.202000011

By:

Zaher, Dana M.;
El‐Gamal, Mohammed I.;
Omar, Hany A.;
Aljareh, Sarah N.;
Al‐Shamma, Salma A.;
Ali, Aya J.;
Zaib, Sumera;
Iqbal, Jamshed

Publication type:

Article

Synthesis of New Tricyclic and Tetracyclic Fused Coumarin Sulfonate Derivatives and Their Inhibitory Effects on LPS-Induced Nitric Oxide and PGE<sub>2</sub> Productions in RAW 264.7 Macrophages: Part 2.

Published in:

Archiv der Pharmazie, 2016, v. 349, n. 11, p. 853, doi. 10.1002/ardp.201600243

By:

El ‐ Gamal, Mohammed I.;
Lee, Woo ‐ Seok;
Shin, Ji ‐ Sun;
Oh, Chang ‐ Hyun;
Lee, Kyung ‐ Tae;
Choi, Jungseung;
Myoung, Nohsun;
Baek, Daejin

Publication type:

Article

Cell-Based Biological Evaluation of a New Bisamide FMS Kinase Inhibitor Possessing Pyrrolo[3,2- c]pyridine Scaffold.

Published in:

Archiv der Pharmazie, 2014, v. 347, n. 9, p. 635, doi. 10.1002/ardp.201400051

By:

El ‐ Gamal, Mohammed I.;
Abdel ‐ Maksoud, Mohammed S.;
El ‐ Din, Mahmoud M. Gamal;
Yoo, Kyung Ho;
Baek, Daejin;
Oh, Chang ‐ Hyun

Publication type:

Article

Design, Synthesis, and Antiproliferative Activity of 3,4-Diarylpyrazole-1-carboxamide Derivatives Against Melanoma Cell Line.

Published in:

Archiv der Pharmazie, 2011, v. 344, n. 11, p. 745, doi. 10.1002/ardp.201000375

By:

El-Gamal, Mohammed I.;
Choi, Hong Seok;
Cho, Hae-Guk;
Hong, Jun Hee;
Yoo, Kyung Ho;
Oh, Chang-Hyun

Publication type:

Article

Synthesis of 1 H-Pyrazole-1-carboxamide Derivatives and Their Antiproliferative Activity against Melanoma Cell Line.

Published in:

Archiv der Pharmazie, 2011, v. 344, n. 3, p. 197, doi. 10.1002/ardp.201000057

By:

El-Gamal, Mohammed I.;
Sim, Tae Bo;
Hong, Jun Hee;
Cho, Jung-Hyuck;
Yoo, Kyung Ho;
Oh, Chang-Hyun

Publication type:

Article

Mechanistic/mammalian target of rapamycin: Recent pathological aspects and inhibitors.

Published in:

Medicinal Research Reviews, 2019, v. 39, n. 2, p. 631, doi. 10.1002/med.21535

By:

Abdel‐Maksoud, Mohammed S.;
El‐Gamal, Mohammed I.;
Benhalilou, Dalia Reyane;
Ashraf, Sandy;
Mohammed, Shatha Abdulghaffar;
Oh, Chang‐Hyun

Publication type:

Article

Evaluation of Substituted Pyrazole-Based Kinase Inhibitors in One Decade (2011–2020): Current Status and Future Prospects.

Published in:

Molecules, 2022, v. 27, n. 1, p. 1, doi. 10.3390/molecules27010330

By:

El-Gamal, Mohammed I.;
Zaraei, Seyed-Omar;
Madkour, Moustafa M.;
Anbar, Hanan S.

Publication type:

Article

A Review of HER4 (ErbB4) Kinase, Its Impact on Cancer, and Its Inhibitors.

Published in:

Molecules, 2021, v. 26, n. 23, p. 7376, doi. 10.3390/molecules26237376

By:

El-Gamal, Mohammed I.;
Mewafi, Nada H.;
Abdelmotteleb, Nada E.;
Emara, Minnatullah A.;
Tarazi, Hamadeh;
Sbenati, Rawan M.;
Madkour, Moustafa M.;
Zaraei, Seyed-Omar;
Shahin, Afnan I.;
Anbar, Hanan S.

Publication type:

Article

Evaluation of the Inhibitory Effects of Pyridylpyrazole Derivatives on LPS-Induced PGE 2 Productions and Nitric Oxide in Murine RAW 264.7 Macrophages.

Published in:

Molecules, 2021, v. 26, n. 21, p. 6489, doi. 10.3390/molecules26216489

By:

Gamal El-Din, Mahmoud M.;
El-Gamal, Mohammed I.;
Kwon, Young-Do;
Kim, Su-Yeon;
Han, Hee-Soo;
Park, Sang-Eun;
Oh, Chang-Hyun;
Lee, Kyung-Tae;
Kim, Hee-Kwon

Publication type:

Article

Synthesis of New Triarylpyrazole Derivatives Possessing Terminal Sulfonamide Moiety and Their Inhibitory Effects on PGE2 and Nitric Oxide Productions in Lipopolysaccharide-Induced RAW 264.7 Macrophages.

Published in:

Molecules, 2018, v. 23, n. 10, p. 2556, doi. 10.3390/molecules23102556

By:

Abdel-Maksoud, Mohammed S.;
El-Gamal, Mohammed I.;
Gamal El-Din, Mahmoud M.;
Choi, Yunji;
Choi, Jungseung;
Shin, Ji-Sun;
Kang, Shin-Young;
Yoo, Kyung Ho;
Lee, Kyung-Tae;
Baek, Daejin;
Oh, Chang-Hyun

Publication type:

Article

A New Series of Cycloalkane-fused Coumarin Sulfonates: Synthesis and In Vitro Antiproliferative Screening.

Published in:

Bulletin of the Korean Chemical Society, 2016, v. 37, n. 2, p. 184, doi. 10.1002/bkcs.10651

By:

El-Gamal, Mohammed I.;
Baek, Daejin;
Oh, Chang-Hyun

Publication type:

Article

Complexity‐to‐Diversity and Pseudo‐Natural Product Strategies as Powerful Platforms for Deciphering Next‐Generation Therapeutics.

Published in:

ChemMedChem, 2023, v. 18, n. 14, p. 1, doi. 10.1002/cmdc.202300117

By:

Alkubaisi, Bilal O.;
Shahin, Afnan I.;
Zenati, Ruba A.;
Ravi, Anil;
Alchami, Riema;
Alkalla, Mohammad;
Khaled, Rawan;
El‐Gamal, Mohammed I.;
Al‐Tel, Taleb H.

Publication type:

Article

Antiproliferative Diarylpyrazole Derivatives as Dual Inhibitors of the ERK Pathway and COX-2.

Published in:

Chemical Biology & Drug Design, 2013, v. 82, n. 3, p. 336, doi. 10.1111/cbdd.12186

By:

El ‐ Gamal, Mohammed I.;
Choi, Hong Seok;
Yoo, Kyung Ho;
Baek, Daejin;
Oh, Chang ‐ Hyun

Publication type:

Article

Diastereoselective Synthesis of Camptothecin‐like Scaffolds: Construction of a New Class of Pseudo‐natural Products.

Published in:

European Journal of Organic Chemistry, 2023, v. 26, n. 13, p. 1, doi. 10.1002/ejoc.202300080

By:

Srikanth, Gourishetty;
Ravi, Anil;
Sebastian, Anusha;
Joseph, Jobi;
Khanfar, Monther A.;
El‐Gamal, Mohammed I.;
Al‐Qawasmeh, Raed A.;
Shehadi, Ihsan A.;
McN. Sieburth, Scott;
Abu‐Yousef, Imad A.;
Majdalawieh, Amin F.;
Al‐Tel, Taleb H.

Publication type:

Article

Stereodivergent Transformation of Azepino[3,4,5‐cd]indoles En Route to Nature‐Inspired Scaffolds.

Published in:

European Journal of Organic Chemistry, 2023, v. 26, n. 9, p. 1, doi. 10.1002/ejoc.202201354

By:

Srikanth, Gourishetty;
Ravi, Anil;
Sebastian, Anusha;
Joseph, Jobi;
Khanfar, Monther A.;
El‐Gamal, Mohammed I.;
Al‐Qawasmeh, Raed A.;
Abu‐Yousef, Imad A.;
Majdalawieh, Amin F.;
Al‐Tel, Taleb H.

Publication type:

Article

Anti-proliferative activity of RIHMS-Qi-23 against MCF-7 breast cancer cell line is through inhibition of cell proliferation and senescence but not inhibition of targeted kinases.

Published in:

BMC Cancer, 2023, v. 23, n. 1, p. 1, doi. 10.1186/s12885-023-11547-1

By:

El-Gamal, Randa;
Elfarrash, Sara;
EL-Nablaway, Mohammad;
Salem, Asmaa Ahmed;
Zaraei, Seyed-Omar;
Anbar, Hanan S.;
Shoma, Ashraf;
El-Gamal, Mohammed I.

Publication type:

Article

Next generation imidazothiazole and imidazooxazole derivatives as potential drugs against brain-eating amoebae.

Published in:

Parasitology Research, 2024, v. 123, n. 6, p. 1, doi. 10.1007/s00436-024-08255-5

By:

Akbar, Noor;
Siddiqui, Ruqaiyyah;
El-Gamal, Mohammed I.;
Khan, Naveed Ahmed;
Zaraei, Seyed-Omar;
Saeed, Balsam Qubais;
Alharbi, Ahmad M.;
Dash, Nihar Ranjan

Publication type:

Article

The anti-amoebic potential of carboxamide derivatives containing sulfonyl or sulfamoyl moieties against brain-eating Naegleria fowleri.

Published in:

Parasitology Research, 2023, v. 122, n. 11, p. 2539, doi. 10.1007/s00436-023-07953-w

By:

Akbar, Noor;
Siddiqui, Ruqaiyyah;
El-Gamal, Mohammed I.;
Zaraei, Seyed-Omar;
Alawfi, Bader S.;
Khan, Naveed Ahmed

Publication type:

Article

Anti-amoebic activity of a series of benzofuran/benzothiophene derivatives against Acanthamoeba castellanii belonging to the T4 genotype.

Published in:

Journal of Applied Microbiology, 2023, v. 134, n. 1, p. 1, doi. 10.1093/jambio/lxac030

By:

Akbar, Noor;
El-Gamal, Mohammed I;
Zaraei, Seyed-Omar;
Saeed, Balsam Qubais;
Khan, Naveed Ahmed;
Siddiqui, Ruqaiyyah

Publication type:

Article

Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1712, doi. 10.1080/14756366.2020.1819260

By:

Anbar, Hanan S.;
El-Gamal, Mohammed I.;
Tarazi, Hamadeh;
Lee, Bong S.;
Jeon, Hong R.;
Kwon, Dow;
Oh, Chang-Hyun

Publication type:

Article

Design, synthesis, in vitro potent antiproliferative activity, and kinase inhibitory effects of new triarylpyrazole derivatives possessing different heterocycle terminal moieties.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1534, doi. 10.1080/14756366.2019.1653292

By:

Gamal El-Din, Mahmoud M.;
El-Gamal, Mohammed I.;
Abdel-Maksoud, Mohammed S.;
Yoo, Kyung Ho;
Oh, Chang-Hyun

Publication type:

Article

Design, synthesis, in vitro anticancer evaluation, kinase inhibitory effects, and pharmacokinetic profile of new 1,3,4-triarylpyrazole derivatives possessing terminal sulfonamide moiety.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 97, doi. 10.1080/14756366.2018.1530225

By:

Abdel-Maksoud, Mohammed S.;
El-Gamal, Mohammed I.;
Gamal El-Din, Mahmoud M.;
Oh, Chang Hyun

Publication type:

Article

Pyrrolo[3,2-c]pyridine derivatives with potential inhibitory effect against FMS kinase: in vitro biological studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1160, doi. 10.1080/14756366.2018.1491563

By:

El-Gamal, Mohammed I.;
Oh, Chang-Hyun

Publication type:

Article

Tricyclic coumarin sulphonate derivatives with alkaline phosphatase inhibitory effects: in vitro and docking studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 479, doi. 10.1080/14756366.2018.1428193

By:

Iqbal, Jamshed;
El-Gamal, Mohammed I.;
Ejaz, Syeda Abida;
Lecka, Joanna;
Sévigny, Jean;
Oh, Chang-Hyun

Publication type:

Article

Design, synthesis, and in vitro antiproliferative and kinase inhibitory effects of pyrimidinylpyrazole derivatives terminating with arylsulfonamido or cyclic sulfamide substituents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 111, doi. 10.1080/14756366.2016.1190715

By:

Gamal El-Din, Mahmoud M.;
El-Gamal, Mohammed I.;
Abdel-Maksoud, Mohammed S.;
Yoo, Kyung Ho;
Baek, Daejin;
Choi, Jungseung;
Lee, Huiseong;
Oh, Chang-Hyun

Publication type:

Article

Novel Anti-Acanthamoebic Activities of Irosustat and STX140 and Their Nanoformulations.

Published in:

Antibiotics (2079-6382), 2023, v. 12, n. 3, p. 561, doi. 10.3390/antibiotics12030561

By:

Siddiqui, Ruqaiyyah;
Rawas-Qalaji, Mutasem;
El-Gamal, Mohammed I.;
Sajeev, Sreedevi;
Jagal, Jayalakshmi;
Zaraei, Seyed-Omar;
Sbenati, Rawan M.;
Anbar, Hanan S.;
Dohle, Wolfgang;
Potter, Barry V. L.;
Khan, Naveed Ahmed

Publication type:

Article

Imidazothiazole Derivatives Exhibited Potent Effects against Brain-Eating Amoebae.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 11, p. 1515, doi. 10.3390/antibiotics11111515

By:

Siddiqui, Ruqaiyyah;
El-Gamal, Mohammed I.;
Boghossian, Anania;
Saeed, Balsam Qubais;
Oh, Chang-Hyun;
Abdel-Maksoud, Mohammed S.;
Alharbi, Ahmad M.;
Alfahemi, Hasan;
Khan, Naveed Ahmed

Publication type:

Article

Antiamoebic Activity of Imidazothiazole Derivatives against Opportunistic Pathogen Acanthamoeba castellanii.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 9, p. 1183, doi. 10.3390/antibiotics11091183

By:

Akbar, Noor;
El-Gamal, Mohammed I.;
Saeed, Balsam Qubais;
Oh, Chang-Hyun;
Abdel-Maksoud, Mohammed S.;
Khan, Naveed Ahmed;
Alharbi, Ahmad M.;
Alfahemi, Hasan;
Siddiqui, Ruqaiyyah

Publication type:

Article

Steroid sulfatase inhibitors: the current landscape.

Published in:

Expert Opinion on Therapeutic Patents, 2021, v. 31, n. 6, p. 453, doi. 10.1080/13543776.2021.1910237

By:

Anbar, Hanan S.;
Isa, Zahraa;
Elounais, Jana J.;
Jameel, Mariam A.;
Zib, Joudi H.;
Samer, Aya M.;
Jawad, Aya F.;
El-Gamal, Mohammed I.

Publication type:

Article

Recent advances of pyrrolopyridines derivatives: a patent and literature review.

Published in:

Expert Opinion on Therapeutic Patents, 2017, v. 27, n. 5, p. 591, doi. 10.1080/13543776.2017.1280465

By:

El-Gamal, Mohammed I.;
Anbar, Hanan S.

Publication type:

Article

Radiosynthesis and in vitro evaluation of 1-(tetrahydro-5-hydroxy-6-(hydroxymethyl)-2H-pyran-3-yl)-5-[.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2011, v. 54, n. 2, p. 93, doi. 10.1002/jlcr.1819

By:

Jo, Nam Hyun;
Kim, Jung Young;
El-Gamal, Mohammed I.;
Choi, Won-Kyoung;
Park, Jin-Hun;
Kim, Eun Jung;
Cho, Jung-Hyuck;
Ha, Hyun-Joon;
Choi, Tae Hyun;
Oh, Chang-Hyun

Publication type:

Article

FMS Kinase Inhibitors: Current Status and Future Prospects.

Published in:

Medicinal Research Reviews, 2013, v. 33, n. 3, p. 599, doi. 10.1002/med.21258

By:

El-Gamal, Mohammed I.;
Anbar, Hanan S.;
Yoo, Kyung Ho;
Oh, Chang-Hyun

Publication type:

Article

Divergent Strategy for the Synthesis of Indolopyrazines Fused to Benzopyrimidinones and Benzimidazoles: Identification of Antiproliferative Molecules.

Published in:

ChemistrySelect, 2023, v. 8, n. 46, p. 1, doi. 10.1002/slct.202303730

By:

Alkubaisi, Bilal O.;
Sebastian, Anusha;
Bauer, Maximilian;
Sultan, Shaista;
El‐Awady, Raafat;
Wehbe, Ayeh;
Yassin, Mariam;
Vunnam, Srinivasulu;
El‐Gamal, Mohammed I.;
Al‐Tel, Taleb H.

Publication type:

Article

Synthesis and in vitro antibacterial activity of new meropenem analogs.

Published in:

Journal of Antibiotics, 2011, v. 64, n. 10, p. 687, doi. 10.1038/ja.2011.70

By:

El-Gamal, Mohammed I;
Kim, Seong Jong;
Oh, Chang-Hyun

Publication type:

Article