Works by Dolezal, Vladimir

Results: 32

Calcium channels involved in the inhibition of acetylcholine release by presynaptic muscarinic receptors in rat striatum.

Published in:

British Journal of Pharmacology, 1999, v. 127, n. 7, p. 1627, doi. 10.1038/sj.bjp.0702721

By:

Doležal, Vladimír;
Tuček, Stanislav

Publication type:

Article

Agonist-selective activation of individual G-proteins by muscarinic receptors.

Published in:

Scientific Reports, 2024, v. 14, n. 1, p. 1, doi. 10.1038/s41598-024-60259-4

By:

Nelic, Dominik;
Chetverikov, Nikolai;
Hochmalová, Martina;
Diaz, Christina;
Doležal, Vladimír;
Boulos, John;
Jakubík, Jan;
Martemyanov, Kirill;
Janoušková-Randáková, Alena

Publication type:

Article

Towards predictive docking at aminergic G-protein coupled receptors.

Published in:

Journal of Molecular Modeling, 2015, v. 21, n. 11, p. 1, doi. 10.1007/s00894-015-2824-9

By:

Jakubík, Jan;
El-Fakahany, Esam E.;
Doležal, Vladimír

Publication type:

Article

Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors.

Published in:

FEBS Journal, 2009, v. 276, n. 18, p. 5065, doi. 10.1111/j.1742-4658.2009.07203.x

By:

Mordvintsev, Dmitry Yu.;
Polyak, Yakov L.;
Rodionov, Dmitry I.;
Jakubik, Jan;
Dolezal, Vladimir;
Karlsson, Evert;
Tsetlin, Victor I.;
Utkin, Yuri N.

Publication type:

Article

On homology modeling of the M muscarinic acetylcholine receptor subtype.

Published in:

Journal of Computer-Aided Molecular Design, 2013, v. 27, n. 6, p. 525, doi. 10.1007/s10822-013-9660-8

By:

Jakubík, Jan;
Randáková, Alena;
Doležal, Vladimír

Publication type:

Article

Novel M2 -selective, Gi -biased agonists of muscarinic acetylcholine receptors.

Published in:

2020

By:

Randáková, Alena;
Nelic, Dominik;
Ungerová, Dana;
Nwokoye, Peter;
Su, Qiwen;
Doležal, Vladimír;
El‐Fakahany, Esam E.;
Boulos, John;
Jakubík, Jan;
El-Fakahany, Esam E

Publication type:

journal article

Novel long-acting antagonists of muscarinic ACh receptors.

Published in:

2018

By:

Randáková, Alena;
Rudajev, Vladimír;
Doležal, Vladimír;
Boulos, John;
Jakubík, Jan

Publication type:

journal article

The effects of brucine and alcuronium on the inhibition of [3H]acetylcholine release from rat striatum by muscarinic receptor agonists.

Published in:

British Journal of Pharmacology, 1998, v. 124, n. 6, p. 1213, doi. 10.1038/sj.bjp.0701966

By:

Doležal, Vladimír;
Tuček, Stanislav

Publication type:

Article

Changes in Membrane Cholesterol Differentially Influence Preferential and Non-preferential Signaling of the M1 and M3 Muscarinic Acetylcholine Receptors.

Published in:

Neurochemical Research, 2015, v. 40, n. 10, p. 2068, doi. 10.1007/s11064-014-1325-z

By:

Michal, Pavel;
El-Fakahany, Esam;
Doležal, Vladimír

Publication type:

Article

Inhibition of the Synthesis of Acetylcholine in Rat Brain Slices by (−)-Hydroxycitrate and Citrate.

Published in:

Journal of Neurochemistry, 1981, v. 36, n. 4, p. 1331, doi. 10.1111/j.1471-4159.1981.tb00570.x

By:

Tuček, Stanislav;
Doležal, Vladimír;
Sullivan, Ann C

Publication type:

Article

Utilization of Citrate, Acetylcarnitine, Acetate, Pyruvate and Glucose for the Synthesis of Acetylcholine in Rat Brain Slices.

Published in:

Journal of Neurochemistry, 1981, v. 36, n. 4, p. 1323, doi. 10.1111/j.1471-4159.1981.tb00569.x

By:

Doležal, Vladimir;
Tuček, Stanislav

Publication type:

Article

Apolipoprotein E4 reduces evoked hippocampal acetylcholine release in adult mice.

Published in:

Journal of Neurochemistry, 2016, v. 136, n. 3, p. 503, doi. 10.1111/jnc.13417

By:

Dolejší, Eva;
Liraz, Ori;
Rudajev, Vladimír;
Zimčík, Pavel;
Doležal, Vladimír;
Michaelson, Daniel M.

Publication type:

Article

Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators.

Published in:

PLoS ONE, 2019, v. 14, n. 3, p. 1, doi. 10.1371/journal.pone.0214255

By:

Jakubík, Jan;
Randáková, Alena;
El-Fakahany, Esam E.;
Doležal, Vladimír

Publication type:

Article

Stanislav Tuček (1932–2002).

Published in:

Journal of Neurochemistry, 2003, v. 84, n. 1, p. 1, doi. 10.1046/j.1471-4159.2003.01565.x

By:

Doležal, Vladimir;
Dahlström, Annica;
Bachelard, Herman

Publication type:

Article

Presynaptic Nicotinic Receptors Stimulate Increases in Intraterminal Calcium of Chick Sympathetic Neurons in Culture.

Published in:

Journal of Neurochemistry, 1995, v. 65, n. 4, p. 1874, doi. 10.1046/j.1471-4159.1995.65041874.x

By:

Doležal, Vladimír;
Schobert, Angelika;
Hertting, Georg

Publication type:

Article

Positive and Negative Effects of Tacrine (Tetrahydroaminoacridine) and Methoxytacrine on the Metabolism of Acetylcholine in Brain Cortical Prisms Incubated Under 'Resting'Conditions.

Published in:

Journal of Neurochemistry, 1991, v. 56, n. 4, p. 1207, doi. 10.1111/j.1471-4159.1991.tb11412.x

By:

Doležal, Vladimír;
Tuček, Stanislav

Publication type:

Article

Negative Effects of Tacrine (Tetrahydroaminoacridine) and Methoxytacrine on the Metabolism of Acetylcholine in Brain Slices Incubated Under Conditions Stimulating Neurotransmitter Release.

Published in:

Journal of Neurochemistry, 1991, v. 56, n. 4, p. 1216, doi. 10.1111/j.1471-4159.1991.tb11413.x

By:

Tuček, Stanislav;
Doležal, Vladimír

Publication type:

Article

Calcium-Independent Release of Acetylcholine from Electric Organ Synaptosomes and Its Changes by Depolarization and Cholinergic Drugs.

Published in:

Journal of Neurochemistry, 1988, v. 50, n. 2, p. 406, doi. 10.1111/j.1471-4159.1988.tb02927.x

By:

Doležal, Vladimír;
Françoise Diebler, Marie;
Lazereg, Sylvie;
Israël, Maurice;
Tuček, Stanislav

Publication type:

Article

Effect of Lanthanum on the Release of Acetylcholine from the Myenteric Plexus and on Its Activation by Ouabain and Electrical Stimulation.

Published in:

Journal of Neurochemistry, 1987, v. 49, n. 2, p. 503, doi. 10.1111/j.1471-4159.1987.tb02892.x

By:

Doležal, Vladimir;
Somogyi, Gyorgy T.;
Bernath, Sandor;
Tuček, Stanislav;
Vizi, E. Sylvester

Publication type:

Article

Characterization of the Drosophila adenosine receptor: the effect of adenosine analogs on cAMP signaling in Drosophila cells and their utility for in vivo experiments.

Published in:

Journal of Neurochemistry, 2012, v. 121, n. 3/4, p. 383, doi. 10.1111/j.1471-4159.2012.07701.x

By:

Kucerova, Lucie;
Broz, Vaclav;
Fleischmannova, Jana;
Santruckova, Eva;
Sidorov, Roman;
Dolezal, Vladimir;
Zurovec, Michal

Publication type:

Article

A specific multi-nutrient formulation enhances M1 muscarinic acetylcholine receptor responses in vitro.

Published in:

Journal of Neurochemistry, 2012, v. 120, n. 4, p. 631, doi. 10.1111/j.1471-4159.2011.07616.x

By:

Savelkoul, Paul J. M.;
Janickova, Helena;
Kuipers, Almar A. M.;
Hageman, Robert J. J.;
Kamphuis, Patrick J.;
Dolezal, Vladimir;
Broersen, Laus M.

Publication type:

Article

Detection of choline transporter-like 1 protein CTL1 in neuroblastoma × glioma cells and in the CNS, and its role in choline uptake.

Published in:

Journal of Neurochemistry, 2009, v. 110, n. 4, p. 1297, doi. 10.1111/j.1471-4159.2009.06218.x

By:

Machov&3x00E1;, Eva;
O'Regan, Seana;
Newcombe, Jia;
Meunier, François-Marie;
Prentice, Joanna;
Dove, Rosamund;
Lis, Věra;
Doležal, Vladimír

Publication type:

Article

The transcriptional repressor REST is a critical regulator of the neurosecretory phenotype.

Published in:

Journal of Neurochemistry, 2006, v. 98, n. 6, p. 1828, doi. 10.1111/j.1471-4159.2006.04010.x

By:

Bruce, Alexander W.;
Krejčí, Alena;
Ooi, Lezanne;
Deuchars, James;
Wood, Ian C.;
Doležal, Vladimír;
Buckley, Noel J.

Publication type:

Article

Multiple promoters drive tissue-specific expression of the human M2 muscarinic acetylcholine receptor gene.

Published in:

Journal of Neurochemistry, 2004, v. 91, n. 1, p. 88, doi. 10.1111/j.1471-4159.2004.02694.x

By:

Krejci, Alena;
Bruce, Alexander W.;
Dolezal, Vladimir;
Tucek, Stanislav;
Buckley, Noel J.

Publication type:

Article

Determinants of positive cooperativity between strychnine-like allosteric modulators and N-methylscopolamine at muscarinic receptors.

Published in:

Journal of Molecular Neuroscience, 2006, v. 30, n. 1/2, p. 111, doi. 10.1385/JMN:30:1:111

By:

Jakubík, Jan;
Doležal, Vladimír

Publication type:

Article

Docosahexaenoic acid supports cell growth and expression of choline acetyltransferase and muscarinic receptors in NG108-15 cell line.

Published in:

Journal of Molecular Neuroscience, 2006, v. 30, n. 1/2, p. 25, doi. 10.1385/JMN:30:1:25

By:

Machová, Eva;
Nováková, Jana;
Lisá, Věra;
Doležal, Vladimír

Publication type:

Article

The operational model of allosteric modulation of pharmacological agonism.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. N.PAG, doi. 10.1038/s41598-020-71228-y

By:

Jakubík, Jan;
Randáková, Alena;
Chetverikov, Nikolai;
El-Fakahany, Esam E.;
Doležal, Vladimír

Publication type:

Article

Long-Term Activation upon Brief Exposure to Xanomleline Is Unique to M1 and M4 Subtypes of Muscarinic Acetylcholine Receptors.

Published in:

PLoS ONE, 2014, v. 9, n. 2, p. 1, doi. 10.1371/journal.pone.0088910

By:

Šantrůčková, Eva;
Doležal, Vladimír;
El-Fakahany, Esam E.;
Jakubík, Jan

Publication type:

Article

Subtype Differences in Pre-Coupling of Muscarinic Acetylcholine Receptors.

Published in:

PLoS ONE, 2011, v. 6, n. 11, p. 1, doi. 10.1371/journal.pone.0027732

By:

Jakubík, Jan;
Janíčková, Helena;
Randáková, Alena;
El-Fakahany, Esam E.;
Doležal, Vladimír

Publication type:

Article

Pharmacological Evaluation of the Long-Term Effects of Xanomeline on the M1 Muscarinic Acetylcholine Receptor.

Published in:

PLoS ONE, 2010, v. 5, n. 12, p. 1, doi. 10.1371/journal.pone.0015722

By:

Grant, Marianne K. O.;
Noetzel, Meredith J.;
De Lorme, Kayla C.;
Jakubík, Jan;
Doležal, Vladimír;
El-Fakahany, Esam E.

Publication type:

Article

Enhanced muscarinic receptor responses in vitro after multi-nutrient supplementation

Published in:

2011

By:

Savelkoul, Paul;
Merkes, Mandy;
Janiekova, H;
Kuipers, Almar;
Hageman, Robert;
Dolezal, Vladimir;
Broersen, Laus;
Kamphuis, Patrick

Publication type:

Abstract

Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors.

Published in:

Scientific Reports, 2017, p. 40381, doi. 10.1038/srep40381

By:

Jakubík, Jan;
Randáková, Alena;
Zimčík, Pavel;
El-Fakahany, Esam E.;
Doležal, Vladimír

Publication type:

Article

Works by Dolezal, Vladimir

Calcium channels involved in the inhibition of acetylcholine release by presynaptic muscarinic receptors in rat striatum.

Agonist-selective activation of individual G-proteins by muscarinic receptors.

Towards predictive docking at aminergic G-protein coupled receptors.

Weak toxin WTX from Naja kaouthia cobra venom interacts with both nicotinic and muscarinic acetylcholine receptors.

On homology modeling of the M muscarinic acetylcholine receptor subtype.

Novel M<sub>2</sub> -selective, G<sub>i</sub> -biased agonists of muscarinic acetylcholine receptors.

Novel long-acting antagonists of muscarinic ACh receptors.

The effects of brucine and alcuronium on the inhibition of [<sup>3</sup>H]acetylcholine release from rat striatum by muscarinic receptor agonists.

Changes in Membrane Cholesterol Differentially Influence Preferential and Non-preferential Signaling of the M1 and M3 Muscarinic Acetylcholine Receptors.

Inhibition of the Synthesis of Acetylcholine in Rat Brain Slices by (−)-Hydroxycitrate and Citrate.

Utilization of Citrate, Acetylcarnitine, Acetate, Pyruvate and Glucose for the Synthesis of Acetylcholine in Rat Brain Slices.

Apolipoprotein E4 reduces evoked hippocampal acetylcholine release in adult mice.

Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators.

Stanislav Tuček (1932–2002).

Presynaptic Nicotinic Receptors Stimulate Increases in Intraterminal Calcium of Chick Sympathetic Neurons in Culture.

Positive and Negative Effects of Tacrine (Tetrahydroaminoacridine) and Methoxytacrine on the Metabolism of Acetylcholine in Brain Cortical Prisms Incubated Under 'Resting'Conditions.

Negative Effects of Tacrine (Tetrahydroaminoacridine) and Methoxytacrine on the Metabolism of Acetylcholine in Brain Slices Incubated Under Conditions Stimulating Neurotransmitter Release.

Calcium-Independent Release of Acetylcholine from Electric Organ Synaptosomes and Its Changes by Depolarization and Cholinergic Drugs.

Effect of Lanthanum on the Release of Acetylcholine from the Myenteric Plexus and on Its Activation by Ouabain and Electrical Stimulation.

Characterization of the Drosophila adenosine receptor: the effect of adenosine analogs on cAMP signaling in Drosophila cells and their utility for in vivo experiments.

A specific multi-nutrient formulation enhances M1 muscarinic acetylcholine receptor responses in vitro.

Detection of choline transporter-like 1 protein CTL1 in neuroblastoma × glioma cells and in the CNS, and its role in choline uptake.

The transcriptional repressor REST is a critical regulator of the neurosecretory phenotype.

Multiple promoters drive tissue-specific expression of the human M<sub>2</sub> muscarinic acetylcholine receptor gene.

Determinants of positive cooperativity between strychnine-like allosteric modulators and N-methylscopolamine at muscarinic receptors.

Docosahexaenoic acid supports cell growth and expression of choline acetyltransferase and muscarinic receptors in NG108-15 cell line.

The operational model of allosteric modulation of pharmacological agonism.

Long-Term Activation upon Brief Exposure to Xanomleline Is Unique to M<sub>1</sub> and M<sub>4</sub> Subtypes of Muscarinic Acetylcholine Receptors.

Subtype Differences in Pre-Coupling of Muscarinic Acetylcholine Receptors.

Pharmacological Evaluation of the Long-Term Effects of Xanomeline on the M<sub>1</sub> Muscarinic Acetylcholine Receptor.

Enhanced muscarinic receptor responses in vitro after multi-nutrient supplementation

Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors.