Works by Deplano, Alessandro

Results: 8

Design, synthesis and in vitro and in vivo biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 940, doi. 10.1080/14756366.2021.1875459

By:

Deplano, Alessandro;
Karlsson, Jessica;
Moraca, Federica;
Svensson, Mona;
Cristiano, Claudia;
Morgillo, Carmine Marco;
Fowler, Christopher J.;
Russo, Roberto;
Catalanotti, Bruno;
Onnis, Valentina

Publication type:

Article

Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 815, doi. 10.1080/14756366.2020.1743283

By:

Deplano, Alessandro;
Karlsson, Jessica;
Svensson, Mona;
Moraca, Federica;
Catalanotti, Bruno;
Fowler, Christopher J.;
Onnis, Valentina

Publication type:

Article

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 562, doi. 10.1080/14756366.2018.1532418

By:

Deplano, Alessandro;
Cipriano, Mariateresa;
Moraca, Federica;
Novellino, Ettore;
Catalanotti, Bruno;
Fowler, Christopher J.;
Onnis, Valentina

Publication type:

Article

Molecular Basis for Non-Covalent, Non-Competitive FAAH Inhibition.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 24, p. 15502, doi. 10.3390/ijms232415502

By:

Morgillo, Carmine Marco;
Lupia, Antonio;
Deplano, Alessandro;
Pirone, Luciano;
Fiorillo, Bianca;
Pedone, Emilia;
Luque, F. Javier;
Onnis, Valentina;
Moraca, Federica;
Catalanotti, Bruno

Publication type:

Article

Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode.

Published in:

PLoS ONE, 2015, v. 10, n. 10, p. 1, doi. 10.1371/journal.pone.0142711

By:

Karlsson, Jessica;
Morgillo, Carmine M.;
Deplano, Alessandro;
Smaldone, Giovanni;
Pedone, Emilia;
Luque, F. Javier;
Svensson, Mona;
Novellino, Ettore;
Congiu, Cenzo;
Onnis, Valentina;
Catalanotti, Bruno;
Fowler, Christopher J.

Publication type:

Article

Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor.

Published in:

PLoS ONE, 2015, v. 10, n. 9, p. 1, doi. 10.1371/journal.pone.0139212

By:

Gouveia-Figueira, Sandra;
Karlsson, Jessica;
Deplano, Alessandro;
Hashemian, Sanaz;
Svensson, Mona;
Fredriksson Sundbom, Marcus;
Congiu, Cenzo;
Onnis, Valentina;
Fowler, Christopher J.

Publication type:

Article

Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity.

Published in:

Molecules, 2022, v. 27, n. 17, p. 5370, doi. 10.3390/molecules27175370

By:

Moi, Davide;
Deplano, Alessandro;
Angeli, Andrea;
Balboni, Gianfranco;
Supuran, Claudiu T.;
Onnis, Valentina

Publication type:

Article

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones.

Published in:

Molecules, 2016, v. 21, n. 5, p. 579, doi. 10.3390/molecules21050579

By:

Onnis, Valentina;
Demurtas, Monica;
Deplano, Alessandro;
Balboni, Gianfranco;
Baldisserotto, Anna;
StefanoManfredini;
Pacifico, Salvatore;
Liekens, Sandra;
Balzarini, Jan

Publication type:

Article