Works by Delagrange, Philippe

Results: 56

New selective ligands of human cloned melatonin MT1 and MT2 receptors.

Published in:

Naunyn-Schmiedeberg's Archives of Pharmacology, 2003, v. 367, n. 6, p. 553, doi. 10.1007/s00210-003-0751-2

By:

Audinot, Valérie;
Mailliet, François;
Lahaye-Brasseur, Chantal;
Bonnaud, Anne;
Le Gall, Aude;
Amossé, Christophe;
Dromaint, Sandra;
Rodriguez, Marianne;
Nagel, Nadine;
Galizzi, Jean-Pierre;
xEE;t#Malpaux, Beno&;
Guillaumet, Gérald;
Lesieur, Daniel;
Lefoulon, François;
Renard, Pierre;
Delagrange, Philippe;
Boutin, Jean A.

Publication type:

Article

Insights into the redox cycle of human quinone reductase 2.

Published in:

Free Radical Research, 2011, v. 45, n. 10, p. 1184, doi. 10.3109/10715762.2011.605788

By:

Reybier, Karine;
Perio, Pierre;
Ferry, Gilles;
Bouajila, Jalloul;
Delagrange, Philippe;
Boutin, Jean A.;
Nepveu, Françoise

Publication type:

Article

IUPHAR-DB: the IUPHAR database of G protein-coupled receptors and ion channels.

Published in:

Nucleic Acids Research, 2009, v. 37, n. suppl_1, p. D680, doi. 10.1093/nar/gkn728

By:

Harmar, Anthony J.;
Hills, Rebecca A.;
Rosser, Edward M.;
Jones, Martin;
Buneman, O. Peter;
Dunbar, Donald R.;
Greenhill, Stuart D.;
Hale, Valerie A.;
Sharman, Joanna L.;
Bonner, Tom I.;
Catterall, William A.;
Davenport, Anthony P.;
Delagrange, Philippe;
Dollery, Colin T.;
Foord, Steven M.;
Gutman, George A.;
Laudet, Vincent;
Neubig, Richard R.;
Ohlstein, Eliot H.;
Olsen, Richard W.

Publication type:

Article

Molecular organization and dynamics of the melatonin MT1 receptor/RGS20/Gi protein complex reveal asymmetry of receptor dimers for RGS and Gi coupling.

Published in:

EMBO Journal, 2010, v. 29, n. 21, p. 3646, doi. 10.1038/emboj.2010.236

By:

Maurice, Pascal;
Daulat, Avais M;
Turecek, Rostislav;
Ivankova-Susankova, Klara;
Zamponi, Francesco;
Kamal, Maud;
Clement, Nathalie;
Guillaume, Jean-Luc;
Bettler, Bernhard;
Galès, Céline;
Delagrange, Philippe;
Jockers, Ralf

Publication type:

Article

The orphan GPR50 receptor specifically inhibits MT1 melatonin receptor function through heterodimerization.

Published in:

EMBO Journal, 2006, v. 25, n. 13, p. 3012, doi. 10.1038/sj.emboj.7601193

By:

Levoye, Angélique;
Dam, Julie;
Ayoub, Mohammed A.;
Guillaume, Jean-Luc;
Couturier, Cyril;
Delagrange, Philippe;
Jockers, Ralf

Publication type:

Article

Novel Conformationally Constrained Analogues of Agomelatine as New Melatoninergic Ligands.

Published in:

Molecules, 2013, v. 18, n. 1, p. 154, doi. 10.3390/molecules18010154

By:

Rami, Marouan;
Landagaray, Elodie;
Ettaoussi, Mohamed;
Boukhalfa, Koussayla;
Caignard, Daniel-Henri;
Delagrange, Philippe;
Berthelot, Pascal;
Yous, Saïd

Publication type:

Article

New Quinoxaline Derivatives as Potential MT1 and MT2 Receptor Ligands.

Published in:

Molecules, 2012, v. 17, n. 7, p. 7737, doi. 10.3390/molecules17077737

By:

Ancizu, Saioa;
Castrillo, Nerea;
Pérez-Silanes, Silvia;
Aldana, Ignacio;
Monge, Antonio;
Delagrange, Philippe;
Caignard, Daniel-Henry;
Galiano, Silvia

Publication type:

Article

Screening of Ligand Binding on Melatonin Receptor Using Non-Peptide Combinatorial Libraries.

Published in:

Journal of Receptors & Signal Transduction, 2000, v. 20, n. 1, p. 105, doi. 10.3109/10799890009150040

By:

Boutin, Jean A.;
Lahaye, Chantal;
Pegurier, Cecile;
Nicolas, Jean-Paul;
Fauchere, Jean-Luc;
Langlois, Michel;
Renard, Pierre;
Delagrange, Philippe;
Canet, Emmanuel

Publication type:

Article

Are G Protein‐Coupled Receptor Heterodimers of Physiological Relevance?—Focus on Melatonin Receptors.

Published in:

Chronobiology International: The Journal of Biological & Medical Rhythm Research, 2006, v. 23, n. 1/2, p. 419, doi. 10.1080/07420520500521863

By:

Levoye, Angélique;
Jockers, Ralf;
Ayoub, Mohammed A.;
Delagrange, Philippe;
Savaskan, Egemen;
Guillaume, Jean‐Luc

Publication type:

Article

Therapeutic Potential of Melatonin Ligands.

Published in:

Chronobiology International: The Journal of Biological & Medical Rhythm Research, 2006, v. 23, n. 1/2, p. 413, doi. 10.1080/07420520500464387

By:

Delagrange, Philippe;
Boutin, Jean A.

Publication type:

Article

The orphan GPR50 receptor promotes constitutive TGFβ receptor signaling and protects against cancer development.

Published in:

Nature Communications, 2018, v. 9, n. 1, p. 1, doi. 10.1038/s41467-018-03609-x

By:

Wojciech, Stefanie;
Ahmad, Raise;
Belaid-Choucair, Zakia;
Journé, Anne-Sophie;
Gallet, Sarah;
Dam, Julie;
Daulat, Avais;
Ndiaye-Lobry, Delphine;
Lahuna, Olivier;
Karamitri, Angeliki;
Guillaume, Jean-Luc;
Do Cruzeiro, Marcio;
Guillonneau, François;
Saade, Anastasia;
Clément, Nathalie;
Courivaud, Thomas;
Kaabi, Nawel;
Kenjiro Tadagak;
Delagrange, Philippe;
Prévot, Vincent

Publication type:

Article

Prevention of apoptotic and necrotic cell death, caspase‐3 activation, and renal dysfunction by melatonin after ischemia/reperfusion.

Published in:

FASEB Journal, 2003, v. 17, n. 8, p. 1, doi. 10.1096/fj.02-0504fje

By:

Kunduzova, Oxana R.;
Escourrou, Ghislaine;
Seguelas, Marie-Helene;
Delagrange, Philippe;
De La Farge, France;
Cambon, Claudie;
Parini, Angelo

Publication type:

Article

The Role of the Retrochiasmatic Area in the Control of Pineal Metabolism.

Published in:

Neuroendocrinology, 1999, v. 69, n. 2, p. 97, doi. 10.1159/000054407

By:

Cipolla-Neto, José;
Skorupa, Ana Lúcia;
Ribeiro-Barbosa, Érika R.;
Bartol, Ione;
Mota, Sandra Regina;
Castro Afeche, Solange;
Delagrange, Philippe;
Guardiola-Lemaitre, Béatrice;
Canteras, Newton Sabino

Publication type:

Article

Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6‐Dihydroindolo[2,1‐a]isoquinolines and Related Systems.

Published in:

ChemMedChem, 2022, v. 17, n. 12, p. 1, doi. 10.1002/cmdc.202200129

By:

Tsotinis, Andrew;
Afroudakis, Pandelis A.;
Papanastasiou, Ioannis P.;
Sakellaropoulou, Aikaterini;
Boniakou, Marina;
Komiotis, Dimitri;
Garratt, Peter J.;
Delagrange, Philippe;
Bocianowska‐Zbrog, Alina;
Sugden, David

Publication type:

Article

Synthesis and SAR Studies of Isoquinoline and Tetrahydroisoquinoline Derivatives as Melatonin Receptor Ligands.

Published in:

ChemMedChem, 2022, v. 17, n. 3, p. 1, doi. 10.1002/cmdc.202100658

By:

Ettaoussi, Mohamed;
Laversin, Amélie;
Vreulz, Brandon;
Rami, Marouane;
Lebegue, Nicolas;
Delagrange, Philippe;
Caignard, Daniel Henri;
Melnyk, Patricia;
Liberelle, Maxime;
Yous, Saïd

Publication type:

Article

First evidence of neuronal connections between specific parts of the periaqueductal gray (PAG) and the rest of the brain in sheep: placing the sheep PAG in the circuit of emotion.

Published in:

Brain Structure & Function, 2018, v. 223, n. 7, p. 3297, doi. 10.1007/s00429-018-1689-y

By:

Menant, Ophélie;
Prima, Marie-Caroline;
Morisse, Mélody;
Cornilleau, Fabien;
Moussu, Christian;
Gautier, Adeline;
Blanchon, Hélène;
Meurisse, Maryse;
Delagrange, Philippe;
Tillet, Yves;
Chaillou, Elodie

Publication type:

Article

Synthesis and Pharmacological Evaluation of a series of the Agomelatine Analogues as Melatonin MT1/MT2 Agonist and 5-HT2C Antagonist.

Published in:

ChemMedChem, 2013, v. 8, n. 11, p. 1830, doi. 10.1002/cmdc.201300294

By:

Ettaoussi, Mohamed;
Sabaouni, Ahmed;
Pérès, Basile;
Landagaray, Elodie;
Nosjean, Olivier;
Boutin, Jean A.;
Caignard, Daniel‐Henri;
Delagrange, Philippe;
Berthelot, Pascal;
Yous, Saïd

Publication type:

Article

S 23521 Decreases Food Intake and Body Weight Gain in Diet-Induced Obese Rats**.

Published in:

Obesity (19307381), 2004, v. 12, n. 10, p. 1596, doi. 10.1038/oby.2004.199

By:

Claret, Marc;
Corominola, Helena;
Canals, Ignasi;
Nadal, Belén;
Chavanieu, Alain;
Pfeiffer, Bruno;
Renard, Pierre;
Gorostiaga, Carmen;
Delagrange, Philippe;
Grassy, Gérard;
Gomis, Ramon

Publication type:

Article

Impact of treatment with melatonin on cerebral circulation in old rats.

Published in:

British Journal of Pharmacology, 2004, v. 141, n. 3, p. 399, doi. 10.1038/sj.bjp.0705629

By:

Dupuis, François;
Régrigny, Olivier;
Atkinson, Jeffrey;
Limiñana, Patrick;
Delagrange, Philippe;
Scalbert, Elizabeth;
Chillon, Jean-Marc

Publication type:

Article

Melatonin inhibits nitrate tolerance in isolated coronary arteries.

Published in:

2003

By:

O'Rourke, Stephen T.;
Hammad, Hana;
Delagrange, Philippe;
Scalbert, Elizabeth;
Vanhoutte, Paul M.

Publication type:

journal article

Effects of melatonin on rat pial arteriolar diameter in vivo.

Published in:

British Journal of Pharmacology, 1999, v. 127, n. 7, p. 1666, doi. 10.1038/sj.bjp.0702714

By:

Régrigny, Olivier;
Delagrange, Philippe;
Scalbert, Elizabeth;
Lartaud-Idjouadiene, Isabelle;
Atkinson, Jeffrey;
Chillon, Jean-Marc

Publication type:

Article

Differential inhibitory effects of melatonin analogs and three naphthalenic ligands on 2-[125I]iodomelatonin binding to chicken tissues.

Published in:

Journal of Pineal Research, 1997, v. 23, n. 3, p. 148, doi. 10.1111/j.1600-079X.1997.tb00348.x

By:

Pang, Celia S.;
Tang, Pak L;
Song, Yong;
Pang, Shiu F.;
Ng, Kai W.;
Guardiola-Lemaitre, Beatrice;
Delagrange, Philippe;
Brown, Gregory M.

Publication type:

Article

GPR50-Ctail cleavage and nuclear translocation: a new signal transduction mode for G protein-coupled receptors.

Published in:

Cellular & Molecular Life Sciences, 2020, v. 77, n. 24, p. 5189, doi. 10.1007/s00018-019-03440-7

By:

Ahmad, Raise;
Lahuna, Olivier;
Sidibe, Anissa;
Daulat, Avais;
Zhang, Qiang;
Luka, Marine;
Guillaume, Jean-Luc;
Gallet, Sarah;
Guillonneau, François;
Hamroune, Juliette;
Polo, Sophie;
Prévot, Vincent;
Delagrange, Philippe;
Dam, Julie;
Jockers, Ralf

Publication type:

Article

Melatonin receptors limit dopamine reuptake by regulating dopamine transporter cell-surface exposure.

Published in:

Cellular & Molecular Life Sciences, 2018, v. 75, n. 23, p. 4357, doi. 10.1007/s00018-018-2876-y

By:

Benleulmi-Chaachoua, Abla;
Hegron, Alan;
Le Boulch, Marine;
Karamitri, Angeliki;
Wierzbicka, Marta;
Wong, Victoria;
Stagljar, Igor;
Delagrange, Philippe;
Ahmad, Raise;
Jockers, Ralf

Publication type:

Article

Hamster Melatonin Receptors: Cloning and Binding Characterization of MT1 and Attempt to Clone MT2.

Published in:

International Journal of Molecular Sciences, 2018, v. 19, n. 7, p. 1957, doi. 10.3390/ijms19071957

By:

Dufour, Emilie;
Dupré, Clémence;
Lizzo, Giulia;
Caignard, Sarah;
Riest-Fery, Isabelle;
Brasseur, Chantal;
Legros, Céline;
Delagrange, Philippe;
Guenin, Sophie-Pénélope;
Gautier, Célia;
Nosjean, Olivier;
Boutin, Jean A.;
Simonneaux, Valérie

Publication type:

Article

New MT2 Melatonin Receptor-Selective Ligands: Agonists and Partial Agonists.

Published in:

International Journal of Molecular Sciences, 2017, v. 18, n. 7, p. 1347, doi. 10.3390/ijms18071347

By:

Boutin, Jean A.;
Bonnaud, Anne;
Brasseur, Chantal;
Bruno, Olivier;
Lepretre, Nolwenn;
Oosting, Peter;
Coumailleau, Sophie;
Delagrange, Philippe;
Nosjean, Olivier;
Legros, Céline

Publication type:

Article

New Radioligands for Describing the Molecular Pharmacology of MT1 and MT2 Melatonin Receptors.

Published in:

International Journal of Molecular Sciences, 2013, v. 14, n. 5, p. 8948, doi. 10.3390/ijms14058948

By:

Legros, Céline;
Matthey, Ulrich;
Grelak, Teresa;
Pedragona-Moreau, Sandrine;
Hassler, Werner;
Yous, Saïd;
Thomas, Emmanuel;
Suzenet, Franck;
Folleas, Benoît;
Lefoulon, François;
Berthelot, Pascal;
Caignard, Daniel-Henri;
Guillaumet, Gérald;
Delagrange, Philippe;
Brayer, Jean-Louis;
Nosjean, Olivier;
Boutin, Jean A.

Publication type:

Article

Influence of the novel antidepressant and melatonin agonist/serotonin2C receptor antagonist, agomelatine, on the rat sleep–wake cycle architecture.

Published in:

Psychopharmacology, 2009, v. 205, n. 1, p. 93, doi. 10.1007/s00213-009-1519-2

By:

Descamps, Amandine;
Rousset, Colette;
Millan, Mark;
Spedding, Michael;
Delagrange, Philippe;
Cespuglio, Raymond

Publication type:

Article

Influence of the novel antidepressant and melatonin agonist/serotonin2C receptor antagonist, agomelatine, on the rat sleep–wake cycle architecture.

Published in:

2009

By:

Descamps, Amandine;
Rousset, Colette;
Millan, Mark;
Spedding, Michael;
Delagrange, Philippe;
Cespuglio, Raymond

Publication type:

Correction Notice

Quantitative assessment of oligomeric amyloid β peptide binding to α7 nicotinic receptor.

Published in:

2019

By:

Cecon, Erika;
Dam, Julie;
Luka, Marine;
Gautier, Clément;
Chollet, Anne‐Marie;
Delagrange, Philippe;
Danober, Laurence;
Jockers, Ralf;
Chollet, Anne-Marie

Publication type:

journal article

Importance of the second extracellular loop for melatonin MT1 receptor function and absence of melatonin binding in GPR50.

Published in:

2018

By:

Clement, Nathalie;
Renault, Nicolas;
Guillaume, Jean‐Luc;
Cecon, Erika;
Journé, Anne‐Sophie;
Laurent, Xavier;
Tadagaki, Kenjiro;
Cogé, Francis;
Gohier, Arnaud;
Delagrange, Philippe;
Chavatte, Philippe;
Jockers, Ralf;
Guillaume, Jean-Luc;
Journé, Anne-Sophie

Publication type:

journal article

Design and validation of the first cell-impermeant melatonin receptor agonist.

Published in:

2017

By:

Gbahou, Florence;
Cecon, Erika;
Viault, Guillaume;
Gerbier, Romain;
Jean ‐ Alphonse, Frederic;
Karamitri, Angeliki;
Guillaumet, Gérald;
Delagrange, Philippe;
Friedlander, Robert M;
Vilardaga, Jean ‐ Pierre;
Suzenet, Franck;
Jockers, Ralf;
Jean-Alphonse, Frederic;
Guillaumet, Gérald;
Vilardaga, Jean-Pierre

Publication type:

journal article

Update on melatonin receptors: IUPHAR Review 20.

Published in:

2016

By:

Jockers, Ralf;
Delagrange, Philippe;
Dubocovich, Margarita L.;
Markus, Regina P.;
Renault, Nicolas;
Tosini, Gianluca;
Cecon, Erika;
Zlotos, Darius P.

Publication type:

journal article

Melatonin MT₁ and MT₂ receptors display different molecular pharmacologies only in the G-protein coupled state.

Published in:

2014

By:

Legros, Céline;
Devavry, Séverine;
Caignard, Sarah;
Tessier, Clémence;
Delagrange, Philippe;
Ouvry, Christine;
Boutin, Jean A;
Nosjean, Olivier

Publication type:

journal article

Melatonin MT1 and MT2 receptors display different molecular pharmacologies only in the G-protein coupled state.

Published in:

British Journal of Pharmacology, 2014, v. 171, n. 1, p. 186, doi. 10.1111/bph.12457

By:

Legros, Céline;
Devavry, Séverine;
Caignard, Sarah;
Tessier, Clémence;
Delagrange, Philippe;
Ouvry, Christine;
Boutin, Jean A;
Nosjean, Olivier

Publication type:

Article

Negative regulation of melatonin secretion by melatonin receptors in ovine pinealocytes.

Published in:

PLoS ONE, 2021, v. 16, n. 7, p. 1, doi. 10.1371/journal.pone.0255249

By:

Lépinay, Julie;
Taragnat, Catherine;
Dubois, Jean-Philippe;
Chesneau, Didier;
Jockers, Ralf;
Delagrange, Philippe;
Bozon, Véronique

Publication type:

Article

Mathematical modeling of the microtubule detyrosination/tyrosination cycle for cell-based drug screening design.

Published in:

PLoS Computational Biology, 2022, v. 18, n. 6, p. 1, doi. 10.1371/journal.pcbi.1010236

By:

Grignard, Jeremy;
Lamamy, Véronique;
Vermersch, Eva;
Delagrange, Philippe;
Stephan, Jean-Philippe;
Dorval, Thierry;
Fages, François

Publication type:

Article

Melatonin increases pial artery tone and decreases the lower limit of cerebral blood flow autoregulation.

Published in:

Fundamental & Clinical Pharmacology, 2001, v. 15, n. 4, p. 233, doi. 10.1046/j.1472-8206.2001.00037.x

By:

Régrigny, Olivier;
Delagrange, Philippe;
Scalbert, Elizabeth;
Atkinson, Jeffrey;
Chillon, Jean-Marc

Publication type:

Article

Recombinant Human Melatonin Receptor MT1 Isolated in Mixed Detergents Shows Pharmacology Similar to That in Mammalian Cell Membranes.

Published in:

PLoS ONE, 2014, v. 9, n. 6, p. 1, doi. 10.1371/journal.pone.0100616

By:

Logez, Christel;
Berger, Sylvie;
Legros, Céline;
Banères, Jean-Louis;
Cohen, William;
Delagrange, Philippe;
Nosjean, Olivier;
Boutin, Jean A.;
Ferry, Gilles;
Simonin, Frédéric;
Wagner, Renaud

Publication type:

Article

Loss of Quinone Reductase 2 Function Selectively Facilitates Learning Behaviors.

Published in:

Journal of Neuroscience, 2010, v. 30, n. 38, p. 12690, doi. 10.1523/JNEUROSCI.2808-10.2010

By:

Benoit, Charles-Etienne;
Bastianetto, Stephane;
Brouillette, Jonathan;
YiuChung Tse;
Boutin, Jean A.;
Delagrange, Philippe;
TakPan Wong;
Sarret, Philippe;
Quirion, Rémi

Publication type:

Article

Synthesis of 5-Substituted-2,3-dihydro-1,4-benzoxathiins: Biological Evaluation as Melatonin Receptors Ligands.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 2, p. 187, doi. 10.1080/1475636032000096855

By:

Charton, Isabelle;
Suzenet, Franck;
Boutin, Jean A.;
Audinot, Valérie;
Delagrange, Philippe;
Bennejean, Caroline;
Renard, Pierre;
Guillaumet, Gérald

Publication type:

Article

Intrinsic and extrinsic cues regulate the daily profile of mouse lateral habenula neuronal activity.

Published in:

Journal of Physiology, 2014, v. 592, n. 22, p. 5025, doi. 10.1113/jphysiol.2014.280065

By:

Sakhi, Kanwal;
Wegner, Sven;
Belle, Mino D. C.;
Howarth, Michael;
Delagrange, Philippe;
Brown, Timothy M.;
Piggins, Hugh D.

Publication type:

Article

Daily variation in the electrophysiological activity of mouse medial habenula neurones.

Published in:

Journal of Physiology, 2014, v. 592, n. 4, p. 587, doi. 10.1113/jphysiol.2013.263319

By:

Sakhi, Kanwal;
Belle, Mino D. C.;
Gossan, Nicole;
Delagrange, Philippe;
Piggins, Hugh D.

Publication type:

Article

Organs from mice deleted for NRH:quinone oxidoreductase 2 are deprived of the melatonin binding site MT3

Published in:

FEBS Letters, 2004, v. 578, n. 1/2, p. 116, doi. 10.1016/j.febslet.2004.10.083

By:

Mailliet, François;
Ferry, Gilles;
Vella, Fanny;
Thiam, Kader;
Delagrange, Philippe;
Boutin, Jean A.

Publication type:

Article

Tubulin tyrosination regulates synaptic function and is disrupted in Alzheimer's disease.

Published in:

2022

By:

Peris, Leticia;
Parato, Julie;
Qu, Xiaoyi;
Soleilhac, Jean Marc;
Lanté, Fabien;
Kumar, Atul;
Pero, Maria Elena;
Martínez-Hernández, José;
Corrao, Charlotte;
Falivelli, Giulia;
Payet, Floriane;
Gory-Fauré, Sylvie;
Bosc, Christophe;
Ramirez, Marian Blanca;
Sproul, Andrew;
Brocard, Jacques;
Cara, Benjamin Di;
Delagrange, Philippe;
Buisson, Alain;
Goldberg, Yves

Publication type:

journal article

Orphan GPR50 Restrains Neurite Outgrowth and Cell Migration by Activating the G12/13 Protein‐RhoA Pathway in Neural Progenitor Cells and Tanycytes.

Published in:

Journal of Pineal Research, 2025, v. 77, n. 2, p. 1, doi. 10.1111/jpi.70041

By:

Ahmad, Raise;
Luka, Marine;
Journe, Anne‐Sophie;
Gallet, Sarah;
Hegron, Alan;
Do Cruzeiro, Marcio;
Millan, Mark J.;
Delagrange, Philippe;
Masri, Bernard;
Dam, Julie;
Prevot, Vincent;
Jockers, Ralf

Publication type:

Article

Detection of recombinant and endogenous mouse melatonin receptors by monoclonal antibodies targeting the C‐terminal domain.

Published in:

Journal of Pineal Research, 2019, v. 66, n. 2, p. N.PAG, doi. 10.1111/jpi.12540

By:

Cecon, Erika;
Ivanova, Anna;
Luka, Marine;
Gbahou, Florence;
Friederich, Anne;
Guillaume, Jean‐Luc;
Keller, Patrick;
Knoch, Klaus;
Ahmad, Raise;
Delagrange, Philippe;
Solimena, Michele;
Jockers, Ralf

Publication type:

Article

Protein interactome mining defines melatonin MT1 receptors as integral component of presynaptic protein complexes of neurons.

Published in:

Journal of Pineal Research, 2016, v. 60, n. 1, p. 95, doi. 10.1111/jpi.12294

By:

Benleulmi‐Chaachoua, Abla;
Chen, Lina;
Sokolina, Kate;
Wong, Victoria;
Jurisica, Igor;
Emerit, Michel Boris;
Darmon, Michèle;
Espin, Almudena;
Stagljar, Igor;
Tafelmeyer, Petra;
Zamponi, Gerald W.;
Delagrange, Philippe;
Maurice, Pascal;
Jockers, Ralf

Publication type:

Article

Description of the constitutive activity of cloned human melatonin receptors hMT1 and hMT2 and discovery of inverse agonists.

Published in:

Journal of Pineal Research, 2012, v. 53, n. 1, p. 29, doi. 10.1111/j.1600-079X.2011.00968.x

By:

Devavry, Séverine;
Legros, Céline;
Brasseur, Chantal;
Delagrange, Philippe;
Spadoni, Gilberto;
Cohen, William;
Malpaux, Benoît;
Boutin, Jean A.;
Nosjean, Olivier

Publication type:

Article

Molecular and cellular pharmacological properties of 5-methoxycarbonylamino- N-acetyltryptamine (MCA-NAT): a nonspecific MT3 ligand.

Published in:

Journal of Pineal Research, 2010, v. 48, n. 3, p. 222, doi. 10.1111/j.1600-079X.2010.00746.x

By:

Vincent, Ludwig;
Cohen, William;
Delagrange, Philippe;
Boutin, Jean A.;
Nosjean, Olivier

Publication type:

Article