Works matching AU Dal Corso, Alberto

Results: 26

RGD Cyclopeptide Equipped with a Lysine‐Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency.
Published in:
Chemistry - A European Journal, 2023, v. 29, n. 19, p. 1, doi. 10.1002/chem.202203768
By:
- Sacco, Giovanni;
- Arosio, Daniela;
- Paolillo, Mayra;
- Gloger, Andreas;
- Scheuermann, Jörg;
- Pignataro, Luca;
- Belvisi, Laura;
- Dal Corso, Alberto;
- Gennari, Cesare
Publication type:
Article
Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.
Published in:
Angewandte Chemie, 2020, v. 132, n. 10, p. 4205, doi. 10.1002/ange.201916394
By:
- Dal Corso, Alberto;
- Borlandelli, Valentina;
- Corno, Cristina;
- Perego, Paola;
- Belvisi, Laura;
- Pignataro, Luca;
- Gennari, Cesare
Publication type:
Article
Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.
Published in:
Angewandte Chemie, 2018, v. 130, n. 52, p. 17424, doi. 10.1002/ange.201811650
By:
- Dal Corso, Alberto;
- Catalano, Marco;
- Schmid, Anja;
- Scheuermann, Jörg;
- Neri, Dario
Publication type:
Article
Amine‐Carbamate Self‐Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads.
Published in:
ChemBioChem, 2024, v. 25, n. 8, p. 1, doi. 10.1002/cbic.202400174
By:
- Mason, Mattia;
- Bisbal Lopez, Lydia;
- Bashiri, Fazel;
- Herrero, Aurélie;
- Baron, Aurélien;
- Bucci, Raffaella;
- Pignataro, Luca;
- Gennari, Cesare;
- Dal Corso, Alberto
Publication type:
Article
A Tight Contact: The Expanding Application of Salicylaldehydes in Lysine‐Targeting Covalent Drugs.
Published in:
ChemBioChem, 2024, v. 25, n. 7, p. 1, doi. 10.1002/cbic.202300743
By:
- Mason, Mattia;
- Belvisi, Laura;
- Pignataro, Luca;
- Dal Corso, Alberto
Publication type:
Article
Targeted Small‐Molecule Conjugates: The Future is Now.
Published in:
ChemBioChem, 2020, v. 21, n. 23, p. 3321, doi. 10.1002/cbic.202000507
By:
- Dal Corso, Alberto
Publication type:
Article
Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors.
Published in:
ChemistryOpen, 2015, v. 4, n. 5, p. 633, doi. 10.1002/open.201500062
By:
- Zanella, Simone;
- Mingozzi, Michele;
- Dal Corso, Alberto;
- Fanelli, Roberto;
- Arosio, Daniela;
- Cosentino, Marco;
- Schembri, Laura;
- Marino, Franca;
- De Zotti, Marta;
- Formaggio, Fernando;
- Pignataro, Luca;
- Belvisi, Laura;
- Piarulli, Umberto;
- Gennari, Cesare
Publication type:
Article
Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker.
Published in:
Frontiers in Pharmacology, 2023, p. 1, doi. 10.3389/fphar.2023.1320524
By:
- Lopez, Lydia Bisbal;
- Ravazza, Domenico;
- Bocci, Matilde;
- Zana, Aureliano;
- Principi, Lucrezia;
- Plaza, Sheila Dakhel;
- Galbiati, Andrea;
- Gilardoni, Ettore;
- Scheuermann, Jörg;
- Neri, Dario;
- Pignataro, Luca;
- Gennari, Cesare;
- Cazzamalli, Samuele;
- Dal Corso, Alberto
Publication type:
Article
Synthesis of Noncoded Amino Acids Bearing a Salicylaldehyde Tag for the Design of Reversible‐Covalent Peptides.
Published in:
European Journal of Organic Chemistry, 2024, v. 27, n. 22, p. 1, doi. 10.1002/ejoc.202400229
By:
- Mason, Mattia;
- Nava, Beatrice;
- Belvisi, Laura;
- Pignataro, Luca;
- Dal Corso, Alberto
Publication type:
Article
Metallaphotoredox C−O and C−N Cross‐Coupling Using Donor‐Acceptor Cyanoarene Photocatalysts.
Published in:
ChemCatChem, 2022, v. 14, n. 23, p. 1, doi. 10.1002/cctc.202200990
By:
- Gandini, Tommaso;
- Dolcini, Luigi;
- Di Leo, Lorenzo;
- Fornara, Matthieu;
- Bossi, Alberto;
- Penconi, Marta;
- Dal Corso, Alberto;
- Gennari, Cesare;
- Pignataro, Luca
Publication type:
Article
Functionalized 2‐Hydroxybenzaldehyde‐PEG Modules as Portable Tags for the Engagement of Protein Lysine ϵ‐Amino Groups.
Published in:
European Journal of Organic Chemistry, 2021, v. 2021, n. 11, p. 1763, doi. 10.1002/ejoc.202100160
By:
- Sacco, Giovanni;
- Stammwitz, Simon;
- Belvisi, Laura;
- Pignataro, Luca;
- Dal Corso, Alberto;
- Gennari, Cesare
Publication type:
Article
Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and αVβ3‐Integrin Ligands for Tumor Targeting.
Published in:
European Journal of Organic Chemistry, 2018, v. 2018, n. 23, p. 2902, doi. 10.1002/ejoc.201800447
By:
- López Rivas, Paula;
- Ranđelović, Ivan;
- Raposo Moreira Dias, André;
- Pina, Arianna;
- Arosio, Daniela;
- Tóvári, József;
- Mező, Gábor;
- Dal Corso, Alberto;
- Pignataro, Luca;
- Gennari, Cesare
Publication type:
Article
Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.
Published in:
Angewandte Chemie International Edition, 2020, v. 59, n. 10, p. 4176, doi. 10.1002/anie.201916394
By:
- Dal Corso, Alberto;
- Borlandelli, Valentina;
- Corno, Cristina;
- Perego, Paola;
- Belvisi, Laura;
- Pignataro, Luca;
- Gennari, Cesare
Publication type:
Article
Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.
Published in:
Angewandte Chemie International Edition, 2018, v. 57, n. 52, p. 17178, doi. 10.1002/anie.201811650
By:
- Dal Corso, Alberto;
- Catalano, Marco;
- Schmid, Anja;
- Scheuermann, Jörg;
- Neri, Dario
Publication type:
Article
Advanced Pyrrolidine‐Carbamate Self‐Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release.
Published in:
ChemMedChem, 2022, v. 17, n. 15, p. 1, doi. 10.1002/cmdc.202200279
By:
- Dal Corso, Alberto;
- Frigoli, Margaux;
- Prevosti, Martina;
- Mason, Mattia;
- Bucci, Raffaella;
- Belvisi, Laura;
- Pignataro, Luca;
- Gennari, Cesare
Publication type:
Article
Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin αVβ3.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 938, doi. 10.1002/cmdc.201900049
By:
- Raposo Moreira Dias, André;
- Bodero, Lizeth;
- Martins, Ana;
- Arosio, Daniela;
- Gazzola, Silvia;
- Belvisi, Laura;
- Pignataro, Luca;
- Steinkühler, Christian;
- Dal Corso, Alberto;
- Gennari, Cesare;
- Piarulli, Umberto
Publication type:
Article
Impact of a Central Scaffold on the Binding Affinity of Fragment Pairs Isolated from DNA-Encoded Self-Assembling Chemical Libraries.
Published in:
ChemMedChem, 2017, v. 12, n. 21, p. 1748, doi. 10.1002/cmdc.201700569
By:
- Bigatti, Martina;
- Dal Corso, Alberto;
- Vanetti, Sara;
- Cazzamalli, Samuele;
- Rieder, Ulrike;
- Scheuermann, Jörg;
- Neri, Dario;
- Sladojevich, Filippo
Publication type:
Article
Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake.
Published in:
Chemistry - A European Journal, 2020, v. 26, n. 33, p. 7492, doi. 10.1002/chem.202001115
By:
- Pina, Arianna;
- Kadri, Malika;
- Arosio, Daniela;
- Dal Corso, Alberto;
- Coll, Jean‐Luc;
- Gennari, Cesare;
- Boturyn, Didier
Publication type:
Article
Frontispiece: Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.
Published in:
Chemistry - A European Journal, 2019, v. 25, n. 65, p. N.PAG, doi. 10.1002/chem.201986561
By:
- Dal Corso, Alberto;
- Pignataro, Luca;
- Belvisi, Laura;
- Gennari, Cesare
Publication type:
Article
Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.
Published in:
Chemistry - A European Journal, 2019, v. 25, n. 65, p. 14740, doi. 10.1002/chem.201903127
By:
- Dal Corso, Alberto;
- Pignataro, Luca;
- Belvisi, Laura;
- Gennari, Cesare
Publication type:
Article
Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin‐Targeted Conjugate.
Published in:
Chemistry - A European Journal, 2019, v. 25, n. 7, p. 1696, doi. 10.1002/chem.201805447
By:
- Raposo Moreira Dias, André;
- Pina, Arianna;
- Dean, Amelia;
- Lerchen, Hans‐Georg;
- Caruso, Michele;
- Gasparri, Fabio;
- Fraietta, Ivan;
- Troiani, Sonia;
- Arosio, Daniela;
- Belvisi, Laura;
- Pignataro, Luca;
- Dal Corso, Alberto;
- Gennari, Cesare
Publication type:
Article
Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αVβ3.
Published in:
Chemistry - A European Journal, 2017, v. 23, n. 58, p. n/a, doi. 10.1002/chem.201703093
By:
- Raposo Moreira Dias, André;
- Pina, Arianna;
- Dal Corso, Alberto;
- Arosio, Daniela;
- Belvisi, Laura;
- Pignataro, Luca;
- Caruso, Michele;
- Gennari, Cesare
Publication type:
Article
Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αVβ3.
Published in:
Chemistry - A European Journal, 2017, v. 23, n. 58, p. 14410, doi. 10.1002/chem.201703093
By:
- Raposo Moreira Dias, André;
- Pina, Arianna;
- Dal Corso, Alberto;
- Arosio, Daniela;
- Belvisi, Laura;
- Pignataro, Luca;
- Caruso, Michele;
- Gennari, Cesare
Publication type:
Article
Synthesis and Biological Evaluation of RGD Peptidomimetic-Paclitaxel Conjugates Bearing Lysosomally Cleavable Linkers.
Published in:
Chemistry - A European Journal, 2015, v. 21, n. 18, p. 6921, doi. 10.1002/chem.201500158
By:
- Dal Corso, Alberto;
- Caruso, Michele;
- Belvisi, Laura;
- Arosio, Daniela;
- Piarulli, Umberto;
- Albanese, Clara;
- Gasparri, Fabio;
- Marsiglio, Aurelio;
- Sola, Francesco;
- Troiani, Sonia;
- Valsasina, Barbara;
- Pignataro, Luca;
- Donati, Daniele;
- Gennari, Cesare
Publication type:
Article
Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists.
Published in:
Chemistry - A European Journal, 2015, v. 21, n. 16, p. 6265, doi. 10.1002/chem.201406567
By:
- Panzeri, Silvia;
- Zanella, Simone;
- Arosio, Daniela;
- Vahdati, Leila;
- Dal Corso, Alberto;
- Pignataro, Luca;
- Paolillo, Mayra;
- Schinelli, Sergio;
- Belvisi, Laura;
- Gennari, Cesare;
- Piarulli, Umberto
Publication type:
Article
Cyclic isoDGR Peptidomimetics as Low-Nanomolar αvβ3 Integrin Ligands.
Published in:
Chemistry - A European Journal, 2013, v. 19, n. 11, p. 3563, doi. 10.1002/chem.201204639
By:
- Mingozzi, Michele;
- Dal Corso, Alberto;
- Marchini, Mattia;
- Guzzetti, Ileana;
- Civera, Monica;
- Piarulli, Umberto;
- Arosio, Daniela;
- Belvisi, Laura;
- Potenza, Donatella;
- Pignataro, Luca;
- Gennari, Cesare
Publication type:
Article

Works matching AU Dal Corso, Alberto

RGD Cyclopeptide Equipped with a Lysine‐Engaging Salicylaldehyde Showing Enhanced Integrin Affinity and Cell Detachment Potency.

Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.

Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.

Amine‐Carbamate Self‐Immolative Spacers Counterintuitively Release 3° Alcohol at Much Faster Rates than 1° Alcohol Payloads.

A Tight Contact: The Expanding Application of Salicylaldehydes in Lysine‐Targeting Covalent Drugs.

Targeted Small‐Molecule Conjugates: The Future is Now.

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting α<sub>v</sub>β<sub>3</sub> Integrin and VEGF Receptors.

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker.

Synthesis of Noncoded Amino Acids Bearing a Salicylaldehyde Tag for the Design of Reversible‐Covalent Peptides.

Metallaphotoredox C−O and C−N Cross‐Coupling Using Donor‐Acceptor Cyanoarene Photocatalysts.

Functionalized 2‐Hydroxybenzaldehyde‐PEG Modules as Portable Tags for the Engagement of Protein Lysine ϵ‐Amino Groups.

Synthesis and Biological Evaluation of Paclitaxel Conjugates Involving Linkers Cleavable by Lysosomal Enzymes and α<sub>V</sub>β<sub>3</sub>‐Integrin Ligands for Tumor Targeting.

Fast Cyclization of a Proline‐Derived Self‐Immolative Spacer Improves the Efficacy of Carbamate Prodrugs.

Affinity Enhancement of Protein Ligands by Reversible Covalent Modification of Neighboring Lysine Residues.

Advanced Pyrrolidine‐Carbamate Self‐Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release.

Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin α<sub>V</sub>β<sub>3</sub>.

Impact of a Central Scaffold on the Binding Affinity of Fragment Pairs Isolated from DNA-Encoded Self-Assembling Chemical Libraries.

Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake.

Frontispiece: Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.

Innovative Linker Strategies for Tumor‐Targeted Drug Conjugates.

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin‐Targeted Conjugate.

Frontispiece: Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α<sub>V</sub>β<sub>3</sub>.

Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α<sub>V</sub>β<sub>3</sub>.

Synthesis and Biological Evaluation of RGD Peptidomimetic-Paclitaxel Conjugates Bearing Lysosomally Cleavable Linkers.

Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists.

Cyclic isoDGR Peptidomimetics as Low-Nanomolar α<sub>v</sub>β<sub>3</sub> Integrin Ligands.