Works by Da Settimo, Federico

Results: 56

New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects.

Published in:

Archiv der Pharmazie, 2022, v. 355, n. 11, p. 1, doi. 10.1002/ardp.202200295

By:

Robello, Marco;
Salerno, Silvia;
Barresi, Elisabetta;
Orlandi, Paola;
Vaglini, Francesca;
Banchi, Marta;
Simorini, Francesca;
Baglini, Emma;
Poggetti, Valeria;
Taliani, Sabrina;
Da Settimo, Federico;
Bocci, Guido

Publication type:

Article

Anti-ischaemic activity of an antioxidant aldose reductase inhibitor on diabetic and non-diabetic rat hearts.

Published in:

Journal of Pharmacy & Pharmacology, 2010, v. 62, n. 1, p. 107, doi. 10.1211/jpp.62.01.0012

By:

Calderone, Vincenzo;
Testai, Lara;
Martelli, Alma;
Motta, Concettina La;
Sartini, Stefania;
Settimo, Federico Da;
Breschi, Maria C.

Publication type:

Article

Genetic analysis of dTSPO, an outer mitochondrial membrane protein, reveals its functions in apoptosis, longevity, and Aβ42-induced neurodegeneration.

Published in:

Aging Cell, 2014, v. 13, n. 3, p. 507, doi. 10.1111/acel.12200

By:

Lin, Ran;
Angelin, Alessia;
Da Settimo, Federico;
Martini, Claudia;
Taliani, Sabrina;
Zhu, Shigong;
Wallace, Douglas C.

Publication type:

Article

Synthesis and in vitro antiproliferative activity of new substituted benzo[3′,2′:5,6]thiopyrano[4,3- d]pyrimidines.

Published in:

Journal of Heterocyclic Chemistry, 2008, v. 45, n. 3, p. 745, doi. 10.1002/jhet.5570450318

By:

Marini, Anna Maria;
Da Settimo, Federico;
Salerno, Silvia;
La Motta, Concettina;
Simorini, Francesca;
Taliani, Sabrina;
Bertini, Daniele;
Gia, Ornella;
Dalla Via, Lisa

Publication type:

Article

Synthesis of New Heterocyclic Ring Systems via [1,3,5]Triazino[1,2- a]benzimidazole Derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2005, v. 42, n. 7, p. 1417, doi. 10.1002/jhet.5570420725

By:

Primofiore, Giampaolo;
Da Settimo, Federico;
Pardi, Gianluca;
Simorini, Francesca;
La Motta, Concettina;
Salemo, Silvia;
Taliani, Sabrina;
Marini, Anna Maria

Publication type:

Article

Synthesis of novel 1,4-dihydropyrido[3′,2′:5,6]thiopyrano[4,3- c]-pyrazoles and 5 H-pyrido[3′,2′:5,6]thiopyrano[4,3- d]pyrimidines as potential antiproliferative agents.

Published in:

Journal of Heterocyclic Chemistry, 2003, v. 40, n. 5, p. 783, doi. 10.1002/jhet.5570400506

By:

Primofiore, Giampaolo;
Marini, Anna Maria;
Da Settimo, Federico;
Salerno, Silvia;
Bertini, Daniele;
Dalla Via, Lisa;
Magno, Sebastiano Marciani

Publication type:

Article

An approach to novel fused triazole or tetrazole derivatives starting from benzimidazo[1,2- a]quinazoline-5(7 H)-one and 5,7-dihydro-5-oxopyrido[3′,2′:5,6]pyrimido[1,2- a]benzimidazole.

Published in:

Journal of Heterocyclic Chemistry, 2002, v. 39, n. 5, p. 1007, doi. 10.1002/jhet.5570390523

By:

Da Settimo, Antonio;
Primofiore, Giampaolo;
Da Settimo, Federico;
Pardi, Gianluca;
Simorini, Francesca;
Marini, Anna Maria

Publication type:

Article

Synthesis of novel pyrido[3′,2′:5,6]thiopyrano[3,2- b]indol-5(6 H)-ones and 6 H-pyrido[3′,2′:5,6]thiopyrano[4,3- b]quinolines, two new heterocyclic ring systems.

Published in:

Journal of Heterocyclic Chemistry, 2002, v. 39, n. 5, p. 1001, doi. 10.1002/jhet.5570390522

By:

Da Settimo, Antonio;
Marini, Anna María;
Primofiore, Giampaolo;
Da Settimo, Federico;
Salerno, Silvia;
Simorini, Francesca;
Pardi, Gianluca;
La Motta, Concettina;
Bertini, Daniele

Publication type:

Article

Facile synthesis of 3-substituted [1,2,4]triazino[3,4- f]purine-4,6,8-trione derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2001, v. 38, n. 3, p. 607, doi. 10.1002/jhet.5570380309

By:

Settimo, Federico Da;
Marini, Anna Maria;
Pardi, Gianluca;
Primofiore, Giampaolo;
Salerno, Silvia;
Simorini, Francesca

Publication type:

Article

Synthesis of novel 5 H, 11 H-pyrido[2′,3′:2,3]thiopyrano[4,3- b]-indoles by fischer-indole cyclization.

Published in:

Journal of Heterocyclic Chemistry, 2000, v. 37, n. 2, p. 379, doi. 10.1002/jhet.5570370224

By:

Da Settimo, Antonio;
Marini, Anna Maria;
Primofiore, Giampaolo;
Da Settimo, Federico;
Salerno, Silvia;
La Motta, Concettina;
Pardi, Gianluca;
Ferrarini, Pier Luigi;
Mori, Claudio

Publication type:

Article

Synthesis of a novel purine-containing heterocyclic ring system: 8,10-Dimethylindolo[2′,3′:5,6][1,2,4]triazino[4,3- f]purine-9,11(8 H, 10 H, 13 H)-dione.

Published in:

Journal of Heterocyclic Chemistry, 2000, v. 37, n. 2, p. 373, doi. 10.1002/jhet.5570370223

By:

Da Settimo, Antonio;
Primofiore, Giampaolo;
Da Settimo, Federico;
Simorini, Francesca;
Marini, Anna Maria;
La Motta, Concettina;
Taliani, Sabrina

Publication type:

Article

Synthesis of purinobenzodiazepine and purinobenzotriazocine derivatives, two new heterocyclic ring systems.

Published in:

Journal of Heterocyclic Chemistry, 1999, v. 36, n. 3, p. 639, doi. 10.1002/jhet.5570360311

By:

Settimo, Antonio Da;
Primofiore, Giampaolo;
Marini, Anna Maria;
Settimo, Federico Da;
La Motta, Concettina;
Salerno, Silvia

Publication type:

Article

Synthesis of purinobenzothiazine and pyridothiazinopurine derivatives. Two new heterocyclic ring systems.

Published in:

Journal of Heterocyclic Chemistry, 1998, v. 35, n. 1, p. 57, doi. 10.1002/jhet.5570350111

By:

Settimo, Antonio Da;
Marini, Anna Maria;
Primofiore, Giampaolo;
Settimo, Federico Da;
Bertini, Daniele

Publication type:

Article

Synthesis of fused purinoquinazolines. Three new heterocyclic ring systems.

Published in:

Journal of Heterocyclic Chemistry, 1995, v. 32, n. 3, p. 941, doi. 10.1002/jhet.5570320345

By:

Da Settimo, Antonio;
Primofiore, Giampaolo;
Cristina, Bertacchi Maria;
Da Settimo, Federico;
Marini, Anna Maria

Publication type:

Article

Synthesis of novel 1-aryl[1]benzoxepino[5,4- c]pyrazole and [1]benzoxepino[5,4- d]pyrimidine derivatives.

Published in:

Journal of Heterocyclic Chemistry, 1993, v. 30, n. 6, p. 1653, doi. 10.1002/jhet.5570300632

By:

Chetoni, Fabio;
Da Settimo, Federico;
La Motta, Concettina;
Primofiore, Giampaolo

Publication type:

Article

Synthesis of some 5 H,12 H-[1]benzoxepino[4,3- b]indol-6-ones. A new heterocyclic ring system.

Published in:

Journal of Heterocyclic Chemistry, 1993, v. 30, n. 6, p. 1481, doi. 10.1002/jhet.5570300603

By:

Chetoni, Fabio;
Da Settimo, Federico;
Marini, Anna Maria;
Primofiore, Giampaolo

Publication type:

Article

Synthesis and Biological Evaluation of 2′-Oxo-2,3-dihydro-3′ H- spiro[chromene-4,5′-[1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors.

Published in:

Archiv der Pharmazie, 2011, v. 344, n. 6, p. 372, doi. 10.1002/ardp.201000302

By:

Rapposelli, Simona;
Da Settimo, Federico;
Digiacomo, Maria;
La Motta, Concettina;
Lapucci, Annalina;
Sartini, Stefania;
Vanni, Michael

Publication type:

Article

Synthesis and Benzodiazepine Receptor Affinity of Derivatives of the New Tricyclic Heteroaromatic System Pyrido[3′,2′:5,6]thiopyrano[4,3-c]pyridazin-3(2H,5H)-one.

Published in:

Archiv der Pharmazie, 2005, v. 338, n. 2/3, p. 126, doi. 10.1002/ardp.200400948

By:

Giampaolo Primofiore;
Federico Da Settimo;
Anna Maria Marini;
Francesca Simorini;
Concettina La Motta;
Sabrina Taliani;
Sonia Laneri;
Letizia Trincavelli;
Claudia Martini

Publication type:

Article

Geometrically Constrained Analogues of N-Benzylindolylglyoxylylamides: [1, 2, 4]Triazino[4, 3-a]benzimidazol-4(10H)-one Derivatives as Potential New Ligands at the Benzodiazepine Receptor.

Published in:

Archiv der Pharmazie, 2003, v. 336, n. 9, p. 413, doi. 10.1002/ardp.200300788

By:

Giampaolo Primofiore;
Federico Da Settimo;
Sabrina Taliani;
Anna Maria Marini;
Francesca Simorini;
Ettore Novellino;
Giovanni Greco;
Letizia Trincavelli;
Claudia Martini

Publication type:

Article

Target-Based Anticancer Indole Derivatives for the Development of Anti-Glioblastoma Agents.

Published in:

Molecules, 2023, v. 28, n. 6, p. 2587, doi. 10.3390/molecules28062587

By:

Salerno, Silvia;
Barresi, Elisabetta;
Baglini, Emma;
Poggetti, Valeria;
Da Settimo, Federico;
Taliani, Sabrina

Publication type:

Article

Carbonic Anhydrase Activators for Neurodegeneration: An Overview.

Published in:

Molecules, 2022, v. 27, n. 8, p. N.PAG, doi. 10.3390/molecules27082544

By:

Poggetti, Valeria;
Salerno, Silvia;
Baglini, Emma;
Barresi, Elisabetta;
Da Settimo, Federico;
Taliani, Sabrina

Publication type:

Article

Enriching the Arsenal of Pharmacological Tools against MICAL2.

Published in:

Molecules, 2021, v. 26, n. 24, p. 7519, doi. 10.3390/molecules26247519

By:

Barravecchia, Ivana;
Barresi, Elisabetta;
Russo, Camilla;
Scebba, Francesca;
De Cesari, Chiara;
Mignucci, Valerio;
De Luca, Davide;
Salerno, Silvia;
La Pietra, Valeria;
Giustiniano, Mariateresa;
Pelliccia, Sveva;
Brancaccio, Diego;
Donati, Greta;
Da Settimo, Federico;
Taliani, Sabrina;
Angeloni, Debora;
Marinelli, Luciana

Publication type:

Article

Exploiting the Indole Scaffold to Design Compounds Binding to Different Pharmacological Targets †.

Published in:

Molecules, 2020, v. 25, n. 10, p. 2331, doi. 10.3390/molecules25102331

By:

Taliani, Sabrina;
Da Settimo, Federico;
Martini, Claudia;
Laneri, Sonia;
Novellino, Ettore;
Greco, Giovanni;
Catto, Marco;
Altomare, Cosimo Damiano

Publication type:

Article

PIGA ( N, N-Di- n-butyl-5-chloro-2-(4-chlorophenyl)indol-3-ylglyoxylamide), a New Mitochondrial Benzodiazepine-Receptor Ligand, Induces Apoptosis in C6 glioma Cells.

Published in:

ChemBioChem, 2005, v. 6, n. 6, p. 1082, doi. 10.1002/cbic.200400350

By:

Chelli, Beatrice;
Rossi, Leonardo;
Da Pozzo, Eleonora;
Costa, Barbara;
Spinetti, Francesca;
Rechichi, Mariarosa;
Salvetti, Alessandra;
Lena, Annalisa;
Simorini, Francesca;
Vanacore, Renato;
Scatena, Fabrizio;
Da Settimo, Federico;
Gremigni, Vittorio;
Martini, Claudia

Publication type:

Article

Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N, N-Dialkyl-2-arylindol-3-ylglyoxylamides.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1275, doi. 10.1002/cmdc.201700220

By:

Costa, Barbara;
Taliani, Sabrina;
Da Pozzo, Eleonora;
Barresi, Elisabetta;
Robello, Marco;
Cavallini, Chiara;
Cosconati, Sandro;
Da Settimo, Federico;
Novellino, Ettore;
Martini, Claudia

Publication type:

Article

4-amino-6-alkyloxy-2-alkylthiopyrimidine derivatives as novel non-nucleoside agonists for the adenosine A1 receptor.

Published in:

Chemical Biology & Drug Design, 2016, v. 88, n. 5, p. 724, doi. 10.1111/cbdd.12801

By:

Cosimelli, Barbara;
Greco, Giovanni;
Laneri, Sonia;
Novellino, Ettore;
Sacchi, Antonia;
Trincavelli, Maria Letizia;
Giacomelli, Chiara;
Taliani, Sabrina;
Da Settimo, Federico;
Martini, Claudia

Publication type:

Article

Structure-Activity Relationships on Purine and 2,3-Dihydropurine Derivatives as Antitubercular Agents: a Data Mining Approach.

Published in:

Chemical Biology & Drug Design, 2011, v. 78, n. 4, p. 718, doi. 10.1111/j.1747-0285.2011.01181.x

By:

Pietra, Daniele;
Imbriani, Marcello;
Borghini, Alice;
Giorgi, Irene;
Settimo, Federico Da;
Breschi, Maria Cristina;
Campa, Mario;
Batoni, Giovanna;
Brancatisano, Franca Lisa;
Bianucci, Anna Maria

Publication type:

Article

Apoptosis Therapy in Cancer: The First Single-molecule Co-activating p53 and the Translocator Protein in Glioblastoma.

Published in:

Scientific Reports, 2014, p. 1, doi. 10.1038/srep04749

By:

Daniele, Simona;
Taliani, Sabrina;
Da Pozzo, Eleonora;
Giacomelli, Chiara;
Costa, Barbara;
Trincavelli, Maria Letizia;
Rossi, Leonardo;
Pietra, Valeria La;
Barresi, Elisabetta;
Carotenuto, Alfonso;
Limatola, Antonio;
Lamberti, Anna;
Marinelli, Luciana;
Novellino, Ettore;
Da Settimo, Federico;
Martini, Claudia

Publication type:

Article

Derivatives of Benzimidazol-2-ylquinoline and Benzimidazol-2-ylisoquinoline as Selective A1 Adenosine Receptor Antagonists with Stimulant Activity on Human Colon Motility.

Published in:

ChemMedChem, 2011, v. 6, n. 10, p. 1909, doi. 10.1002/cmdc.201100284

By:

Cosimelli, Barbara;
Taliani, Sabrina;
Greco, Giovanni;
Novellino, Ettore;
Sala, Annalisa;
Severi, Elda;
Da Settimo, Federico;
La Motta, Concettina;
Pugliesi, Isabella;
Antonioli, Luca;
Fornai, Matteo;
Colucci, Rocchina;
Blandizzi, Corrado;
Daniele, Simona;
Trincavelli, Maria Letizia;
Martini, Claudia

Publication type:

Article

A Virtual Screening Study of the 18 kDa Translocator Protein using Pharmacophore Models Combined with 3D-QSAR Studies.

Published in:

ChemMedChem, 2009, v. 4, n. 10, p. 1686, doi. 10.1002/cmdc.200900254

By:

Tuccinardi, Tiziano;
Taliani, Sabrina;
Bellandi, Marusca;
Da Settimo, Federico;
Da Pozzo, Eleonora;
Martini, Claudia;
Martinelli, Adriano

Publication type:

Article

Highlighting the New Advances in Drug Discovery and Development.

Published in:

ChemMedChem, 2008, v. 3, n. 1, p. 181, doi. 10.1002/cmdc.200700268

By:

Taliani, Sabrina;
Da Settimo, Federico

Publication type:

Article

Targeting the 18-kDa translocator protein: recent perspectives for neuroprotection.

Published in:

Biochemical Society Transactions, 2015, v. 43, n. 4, p. 559, doi. 10.1042/BST20150028

By:

Da Pozzo, Eleonora;
Giacomelli, Chiara;
Barresi, Elisabetta;
Costa, Barbara;
Taliani, Sabrina;
Da Settimo Passetti, Federico;
Martini, Claudia

Publication type:

Article

Allosterism vs. Orthosterism: Recent Findings and Future Perspectives on A2B AR Physio-Pathological Implications.

Published in:

Frontiers in Pharmacology, 2021, v. 11, p. N.PAG, doi. 10.3389/fphar.2021.652121

By:

Barresi, Elisabetta;
Martini, Claudia;
Da Settimo, Federico;
Greco, Giovanni;
Taliani, Sabrina;
Giacomelli, Chiara;
Trincavelli, Maria Letizia

Publication type:

Article

11C-ER176, a Radioligand for 18-kDa Translocator Protein, Has Adequate Sensitivity to Robustly Image All Three Affinity Genotypes in Human Brain.

Published in:

Journal of Nuclear Medicine, 2017, v. 58, n. 2, p. 320, doi. 10.2967/jnumed.116.178996

By:

Ikawa, Masamichi;
Lohith, Talakad G.;
Shrestha, Stal;
Telu, Sanjay;
Zoghbi, Sami S.;
Castellano, Sabrina;
Taliani, Sabrina;
Da Settimo, Federico;
Fujita, Masahiro;
Pike, Victor W.;
Innis, Robert B.

Publication type:

Article

A1 adenosine receptor antagonists, 3-aryl[1,2,4]triazino[4,3- a]benzimidazol-4-(10 H)-ones (ATBIs) and N-alkyl and N-acyl-(7-substituted-2-phenylimidazo[1,2- a][1,3,5]triazin-4-yl)amines (ITAs): Different recognition of bovine and human binding sites

Published in:

Drug Development Research, 2004, v. 63, n. 1, p. 1, doi. 10.1002/ddr.10366

By:

Da Settimo, Federico;
Primofiore, Giampaolo;
Taliani, Sabrina;
La Motta, Concettina;
Novellino, Ettore;
Greco, Giovanni;
Lavecchia, Antonio;
Cosimelli, Barbara;
Iadanza, Manuela;
Klotz, Karl-Norbert;
Tuscano, Daniela;
Trincavelli, Maria Letizia;
Martini, Claudia

Publication type:

Article

Anti-Proliferative Properties of the Novel Hybrid Drug Met-ITC, Composed of the Native Drug Metformin with the Addition of an Isothiocyanate H 2 S Donor Moiety, in Different Cancer Cell Lines.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 22, p. 16131, doi. 10.3390/ijms242216131

By:

Citi, Valentina;
Barresi, Elisabetta;
Piragine, Eugenia;
Spezzini, Jacopo;
Testai, Lara;
Da Settimo, Federico;
Martelli, Alma;
Taliani, Sabrina;
Calderone, Vincenzo

Publication type:

Article

Microglial Pro-Inflammatory and Anti-Inflammatory Phenotypes Are Modulated by Translocator Protein Activation.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 18, p. 4467, doi. 10.3390/ijms20184467

By:

Da Pozzo, Eleonora;
Tremolanti, Chiara;
Costa, Barbara;
Giacomelli, Chiara;
Milenkovic, Vladimir M.;
Bader, Stefanie;
Wetzel, Christian H.;
Rupprecht, Rainer;
Taliani, Sabrina;
Da Settimo, Federico;
Martini, Claudia

Publication type:

Article

TSPO PIGA Ligands Promote Neurosteroidogenesis and Human Astrocyte Well-Being.

Published in:

International Journal of Molecular Sciences, 2016, v. 17, n. 7, p. 1028, doi. 10.3390/ijms17071028

By:

Da Pozzo, Eleonora;
Giacomelli, Chiara;
Costa, Barbara;
Cavallini, Chiara;
Taliani, Sabrina;
Barresi, Elisabetta;
Da Settimo, Federico;
Martini, Claudia

Publication type:

Article

Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A3 Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy.

Published in:

Chirality, 2016, v. 28, n. 5, p. 434, doi. 10.1002/chir.22599

By:

Rossi, Daniela;
Nasti, Rita;
Marra, Annamaria;
Meneghini, Silvia;
Mazzeo, Giuseppe;
Longhi, Giovanna;
Memo, Maurizio;
Cosimelli, Barbara;
Greco, Giovanni;
Novellino, Ettore;
Da Settimo, Federico;
Martini, Claudia;
Taliani, Sabrina;
Abbate, Sergio;
Collina, Simona

Publication type:

Article

Tyrosine kinase inhibitors (TKIs) for ovarian cancer treatment: from organic to inorganic chemotherapeutics towards selectivity—a perspective overview.

Published in:

BioMetals, 2024, v. 37, n. 2, p. 275, doi. 10.1007/s10534-023-00547-0

By:

Baglini, Emma;
Chiaverini, Lorenzo;
Tolbatov, Iogann;
Taliani, Sabrina;
Da Settimo, Federico;
La Mendola, Diego;
Barresi, Elisabetta;
Marzo, Tiziano

Publication type:

Article

A complex bearing TSPO PIGA ligand coordinated to the [Au(PEt3)]+ pharmacophore is highly cytotoxic against ovarian cancer cells.

Published in:

BioMetals, 2023, v. 36, n. 5, p. 961, doi. 10.1007/s10534-023-00496-8

By:

Chiaverini, Lorenzo;
Baglini, Emma;
Mannelli, Michele;
Poggetti, Valeria;
Da Settimo, Federico;
Taliani, Sabrina;
Gamberi, Tania;
Barresi, Elisabetta;
La Mendola, Diego;
Marzo, Tiziano

Publication type:

Article

TSPO ligand residence time: a new parameter to predict compound neurosteroidogenic efficacy.

Published in:

Scientific Reports, 2016, p. 18164, doi. 10.1038/srep18164

By:

Costa, Barbara;
Da Pozzo, Eleonora;
Giacomelli, Chiara;
Barresi, Elisabetta;
Taliani, Sabrina;
Da Settimo, Federico;
Martini, Claudia

Publication type:

Article

Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 7, p. 997, doi. 10.3390/ph16070997

By:

Barresi, Elisabetta;
Robello, Marco;
Baglini, Emma;
Poggetti, Valeria;
Viviano, Monica;
Salerno, Silvia;
Da Settimo, Federico;
Taliani, Sabrina

Publication type:

Article

A New Approach to Control the Enigmatic Activity of Aldose Reductase.

Published in:

PLoS ONE, 2013, v. 8, n. 9, p. 1, doi. 10.1371/journal.pone.0074076

By:

Del-Corso, Antonella;
Balestri, Francesco;
Di Bugno, Elisa;
Moschini, Roberta;
Cappiello, Mario;
Sartini, Stefania;
La-Motta, Concettina;
Da-Settimo, Federico;
Mura, Umberto

Publication type:

Article

18 kDa TSPO targeting drives polarized human microglia towards a protective and restorative neurosteroidome profile.

Published in:

Cellular & Molecular Life Sciences, 2025, v. 82, n. 1, p. 1, doi. 10.1007/s00018-024-05544-1

By:

Germelli, Lorenzo;
Angeloni, Elisa;
Da Pozzo, Eleonora;
Tremolanti, Chiara;
De Felice, Martina;
Giacomelli, Chiara;
Marchetti, Laura;
Muscatello, Beatrice;
Barresi, Elisabetta;
Taliani, Sabrina;
Da Settimo Passetti, Federico;
Trincavelli, Maria Letizia;
Martini, Claudia;
Costa, Barbara

Publication type:

Article

Carbonic anhydrase activation profile of indole-based derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1783, doi. 10.1080/14756366.2021.1959573

By:

Barresi, Elisabetta;
Ravichandran, Rahul;
Germelli, Lorenzo;
Angeli, Andrea;
Baglini, Emma;
Salerno, Silvia;
Marini, Anna Maria;
Costa, Barbara;
Da Pozzo, Eleonora;
Martini, Claudia;
Da Settimo, Federico;
Supuran, Claudiu;
Cosconati, Sandro;
Taliani, Sabrina

Publication type:

Article

Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1874, doi. 10.1080/14756366.2021.1956913

By:

Baglini, Emma;
Ravichandran, Rahul;
Berrino, Emanuela;
Salerno, Silvia;
Barresi, Elisabetta;
Marini, Anna Maria;
Viviano, Monica;
Castellano, Sabrina;
Da Settimo, Federico;
Supuran, Claudiu T.;
Cosconati, Sandro;
Taliani, Sabrina

Publication type:

Article

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 287, doi. 10.1080/14756366.2020.1862103

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Barresi, Elisabetta;
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Greco, Giovanni;
Da Settimo, Federico;
Martini, Claudia;
Trincavelli, Maria Letizia;
Taliani, Sabrina

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1697, doi. 10.1080/14756366.2019.1666836

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Milite, Ciro;
Amendola, Giorgio;
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Feoli, Alessandra;
Novellino, Ettore;
Da Settimo, Federico;
Supuran, Claudiu T.;
Castellano, Sabrina;
Cosconati, Sandro;
Taliani, Sabrina

Publication type:

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Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 350, doi. 10.1080/14756366.2018.1553166

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Sorce, Carlo;
Cappiello, Mario;
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Moschini, Roberta;
Pineschi, Carlotta;
Braca, Alessandra;
La Motta, Concettina;
Da Settimo, Federico;
Del-Corso, Antonella;
Mura, Umberto

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Article