Works matching AU Da Settimo, Federico


Results: 55
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    Enantiomeric 4-Acylamino-6-alkyloxy-2 Alkylthiopyrimidines As Potential A<sub>3</sub> Adenosine Receptor Antagonists: HPLC Chiral Resolution and Absolute Configuration Assignment by a Full Set of Chiroptical Spectroscopy.

    Published in:
    Chirality, 2016, v. 28, n. 5, p. 434, doi. 10.1002/chir.22599
    By:
    • Rossi, Daniela;
    • Nasti, Rita;
    • Marra, Annamaria;
    • Meneghini, Silvia;
    • Mazzeo, Giuseppe;
    • Longhi, Giovanna;
    • Memo, Maurizio;
    • Cosimelli, Barbara;
    • Greco, Giovanni;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Martini, Claudia;
    • Taliani, Sabrina;
    • Abbate, Sergio;
    • Collina, Simona
    Publication type:
    Article
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    18 kDa TSPO targeting drives polarized human microglia towards a protective and restorative neurosteroidome profile.

    Published in:
    Cellular & Molecular Life Sciences, 2025, v. 82, n. 1, p. 1, doi. 10.1007/s00018-024-05544-1
    By:
    • Germelli, Lorenzo;
    • Angeloni, Elisa;
    • Da Pozzo, Eleonora;
    • Tremolanti, Chiara;
    • De Felice, Martina;
    • Giacomelli, Chiara;
    • Marchetti, Laura;
    • Muscatello, Beatrice;
    • Barresi, Elisabetta;
    • Taliani, Sabrina;
    • Da Settimo Passetti, Federico;
    • Trincavelli, Maria Letizia;
    • Martini, Claudia;
    • Costa, Barbara
    Publication type:
    Article
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    A<sub>1</sub> adenosine receptor antagonists, 3-aryl[1,2,4]triazino[4,3- a]benzimidazol-4-(10 H)-ones (ATBIs) and N-alkyl and N-acyl-(7-substituted-2-phenylimidazo[1,2- a][1,3,5]triazin-4-yl)amines (ITAs): Different recognition of bovine and human binding sites

    Published in:
    Drug Development Research, 2004, v. 63, n. 1, p. 1, doi. 10.1002/ddr.10366
    By:
    • Da Settimo, Federico;
    • Primofiore, Giampaolo;
    • Taliani, Sabrina;
    • La Motta, Concettina;
    • Novellino, Ettore;
    • Greco, Giovanni;
    • Lavecchia, Antonio;
    • Cosimelli, Barbara;
    • Iadanza, Manuela;
    • Klotz, Karl-Norbert;
    • Tuscano, Daniela;
    • Trincavelli, Maria Letizia;
    • Martini, Claudia
    Publication type:
    Article
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    Carbonic anhydrase activation profile of indole-based derivatives.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1783, doi. 10.1080/14756366.2021.1959573
    By:
    • Barresi, Elisabetta;
    • Ravichandran, Rahul;
    • Germelli, Lorenzo;
    • Angeli, Andrea;
    • Baglini, Emma;
    • Salerno, Silvia;
    • Marini, Anna Maria;
    • Costa, Barbara;
    • Da Pozzo, Eleonora;
    • Martini, Claudia;
    • Da Settimo, Federico;
    • Supuran, Claudiu;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1874, doi. 10.1080/14756366.2021.1956913
    By:
    • Baglini, Emma;
    • Ravichandran, Rahul;
    • Berrino, Emanuela;
    • Salerno, Silvia;
    • Barresi, Elisabetta;
    • Marini, Anna Maria;
    • Viviano, Monica;
    • Castellano, Sabrina;
    • Da Settimo, Federico;
    • Supuran, Claudiu T.;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1697, doi. 10.1080/14756366.2019.1666836
    By:
    • Milite, Ciro;
    • Amendola, Giorgio;
    • Nocentini, Alessio;
    • Bua, Silvia;
    • Cipriano, Alessandra;
    • Barresi, Elisabetta;
    • Feoli, Alessandra;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Supuran, Claudiu T.;
    • Castellano, Sabrina;
    • Cosconati, Sandro;
    • Taliani, Sabrina
    Publication type:
    Article
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    Soyasaponins from Zolfino bean as aldose reductase differential inhibitors.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 350, doi. 10.1080/14756366.2018.1553166
    By:
    • Balestri, Francesco;
    • De Leo, Marinella;
    • Sorce, Carlo;
    • Cappiello, Mario;
    • Quattrini, Luca;
    • Moschini, Roberta;
    • Pineschi, Carlotta;
    • Braca, Alessandra;
    • La Motta, Concettina;
    • Da Settimo, Federico;
    • Del-Corso, Antonella;
    • Mura, Umberto
    Publication type:
    Article
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    PIGA ( N, N-Di- n-butyl-5-chloro-2-(4-chlorophenyl)indol-3-ylglyoxylamide), a New Mitochondrial Benzodiazepine-Receptor Ligand, Induces Apoptosis in C6 glioma Cells.

    Published in:
    ChemBioChem, 2005, v. 6, n. 6, p. 1082, doi. 10.1002/cbic.200400350
    By:
    • Chelli, Beatrice;
    • Rossi, Leonardo;
    • Da Pozzo, Eleonora;
    • Costa, Barbara;
    • Spinetti, Francesca;
    • Rechichi, Mariarosa;
    • Salvetti, Alessandra;
    • Lena, Annalisa;
    • Simorini, Francesca;
    • Vanacore, Renato;
    • Scatena, Fabrizio;
    • Da Settimo, Federico;
    • Gremigni, Vittorio;
    • Martini, Claudia
    Publication type:
    Article
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    TSPO Radioligands for Neuroinflammation: An Overview.

    Published in:
    Molecules, 2024, v. 29, n. 17, p. 4212, doi. 10.3390/molecules29174212
    By:
    • Salerno, Silvia;
    • Viviano, Monica;
    • Baglini, Emma;
    • Poggetti, Valeria;
    • Giorgini, Doralice;
    • Castagnoli, Jacopo;
    • Barresi, Elisabetta;
    • Castellano, Sabrina;
    • Da Settimo, Federico;
    • Taliani, Sabrina
    Publication type:
    Article
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    Enriching the Arsenal of Pharmacological Tools against MICAL2.

    Published in:
    Molecules, 2021, v. 26, n. 24, p. 7519, doi. 10.3390/molecules26247519
    By:
    • Barravecchia, Ivana;
    • Barresi, Elisabetta;
    • Russo, Camilla;
    • Scebba, Francesca;
    • De Cesari, Chiara;
    • Mignucci, Valerio;
    • De Luca, Davide;
    • Salerno, Silvia;
    • La Pietra, Valeria;
    • Giustiniano, Mariateresa;
    • Pelliccia, Sveva;
    • Brancaccio, Diego;
    • Donati, Greta;
    • Da Settimo, Federico;
    • Taliani, Sabrina;
    • Angeloni, Debora;
    • Marinelli, Luciana
    Publication type:
    Article
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    CLM3, a Multitarget Tyrosine Kinase Inhibitor With Antiangiogenic Properties, Is Active Against Primary Anaplastic Thyroid Cancer In Vitro and In Vivo.

    Published in:
    2014
    By:
    • Antonelli, Alessandro;
    • Bocci, Guido;
    • Fallahi, Poupak;
    • La Motta, Concettina;
    • Ferrari, Silvia Martina;
    • Mancusi, Caterina;
    • Fioravanti, Anna;
    • Di Desidero, Teresa;
    • Sartini, Stefania;
    • Corti, Alessandro;
    • Piaggi, Simona;
    • Materazzi, Gabriele;
    • Spinelli, Claudio;
    • Fontanini, Gabriella;
    • Danesi, Romano;
    • Da Settimo, Federico;
    • Miccoli, Paolo
    Publication type:
    Journal Article
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    Novel Pyrazolopyrimidine Derivatives as Tyrosine Kinase Inhibitors with Antitumoral Activity in Vitro and in Vivo in Papillary Dedifferentiated Thyroid Cancer.

    Published in:
    Journal of Clinical Endocrinology & Metabolism, 2011, v. 96, n. 2, p. E288, doi. 10.1210/jc.2010-1905
    By:
    • Antonelli, Alessandro;
    • Bocci, Guido;
    • La Motta, Concettina;
    • Ferrari, Silvia Martina;
    • Fallahi, Poupak;
    • Fioravanti, Anna;
    • Sartini, Stefania;
    • Minuto, Michele;
    • Piaggi, Simona;
    • Corti, Alessandro;
    • Alì, Greta;
    • Berti, Piero;
    • Fontanini, Gabriella;
    • Danesi, Romano;
    • Da Settimo, Federico;
    • Miccoli, Paolo
    Publication type:
    Article
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    Apoptosis Therapy in Cancer: The First Single-molecule Co-activating p53 and the Translocator Protein in Glioblastoma.

    Published in:
    Scientific Reports, 2014, p. 1, doi. 10.1038/srep04749
    By:
    • Daniele, Simona;
    • Taliani, Sabrina;
    • Da Pozzo, Eleonora;
    • Giacomelli, Chiara;
    • Costa, Barbara;
    • Trincavelli, Maria Letizia;
    • Rossi, Leonardo;
    • Pietra, Valeria La;
    • Barresi, Elisabetta;
    • Carotenuto, Alfonso;
    • Limatola, Antonio;
    • Lamberti, Anna;
    • Marinelli, Luciana;
    • Novellino, Ettore;
    • Da Settimo, Federico;
    • Martini, Claudia
    Publication type:
    Article
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