Works by Džubák, Petr

Results: 34

Secondary metabolite profiles and anti‐SARS‐CoV‐2 activity of ethanolic extracts from nine genotypes of Cannabis sativa L.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400607

By:

Schadich, Ermin;
Kaczorová, Dominika;
Béres, Tibor;
Džubák, Petr;
Hajdúch, Marián;
Tarkowski, Petr;
Ćavar Zeljković, Sanja

Publication type:

Article

New Imidazo[1,2- c]pyrimidin-5(6 H)-Ones Derived from Cytosine: Synthesis, Structure, and Cytotoxic Activity.

Published in:

Journal of Heterocyclic Chemistry, 2015, v. 52, n. 5, p. 1382, doi. 10.1002/jhet.2243

By:

Jansa, Josef;
Lyčka, Antonín;
Padělková, Zdeňka;
Grepl, Martin;
Konečný, Petr;
Hajdúch, Marián;
Džubák, Petr

Publication type:

Article

A unique case of AH-dominant type nodular pulmonary amyloidosis presenting as a spontaneous pneumothorax: a case report and review of the literature.

Published in:

Pathology & Oncology Research, 2023, p. 1, doi. 10.3389/pore.2023.1611390

By:

Skopelidou, Valeria;
Hurník, Pavel;
Tulinský, Lubomír;
Židlík, Vladimir;
Lenz, Jiří;
Delongová, Patricie;
Hornychová, Helena;
Flodr, Patrik;
Jelínek, Tomáš;
Muroňová, Ludmila;
Holub, Dušan;
Džubák, Petr;
Hajdúch, Marián

Publication type:

Article

Synthesis, Leishmanicidal, Trypanocidal, Antiproliferative Assay and Apoptotic Induction of (2-Phenoxypyridin-3-yl)naphthalene-1(2 H)-one Derivatives.

Published in:

Molecules, 2022, v. 27, n. 17, p. 5626, doi. 10.3390/molecules27175626

By:

Blanco, Zuleima;
Fernandez-Moreira, Esteban;
Mijares, Michael R.;
Celis, Carmen;
Martínez, Gricelis;
De Sanctis, Juan B.;
Gurská, Soňa;
Džubák, Petr;
Hajdůch, Marián;
Mijoba, Ali;
García, Yael;
Serrano, Xenón;
Herrera, Nahum;
Correa-Abril, Jhonny;
Parra, Yonathan;
Ángel, Jorge;
Ramírez, Hegira;
Charris, Jaime E.

Publication type:

Article

Betulinic Acid Decorated with Polar Groups and Blue Emitting BODIPY Dye: Synthesis, Cytotoxicity, Cell-Cycle Analysis and Anti-HIV Profiling.

Published in:

Biomedicines, 2021, v. 9, n. 9, p. 1104, doi. 10.3390/biomedicines9091104

By:

Kodr, David;
Stanková, Jarmila;
Rumlová, Michaela;
Džubák, Petr;
Řehulka, Jiří;
Zimmermann, Tomáš;
Křížová, Ivana;
Gurská, Soňa;
Hajdúch, Marián;
Drašar, Pavel B.;
Jurášek, Michal

Publication type:

Article

Isomeric Naphtho‐Fused 7‐Deazapurine Nucleosides and Nucleotides: Synthesis, Biological Activity, Photophysical Properties and Enzymatic Incorporation to Nucleic Acids.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 37, p. 5092, doi. 10.1002/ejoc.201800165

By:

Ghosh, Ketaki;
Perlíková, Pavla;
Havlíček, Vojtěch;
Yang, Chao;
Pohl, Radek;
Tloušťová, Eva;
Hodek, Jan;
Gurská, Soňa;
Džubák, Petr;
Hajdúch, Marián;
Hocek, Michal

Publication type:

Article

Improved syntheses of P2X7 ligands based on substituted benzyl amide of pyroglutamic acid motif labelled with iodine-123 or iodine-125.

Published in:

Journal of Radioanalytical & Nuclear Chemistry, 2023, v. 332, n. 10, p. 4191, doi. 10.1007/s10967-023-09081-2

By:

Marešová, Anna;
Jurášek, Michal;
Zimmermann, Tomáš;
Drašar, Pavel;
Petřík, Miloš;
Džubák, Petr;
Lindegren, Sture;
Cumming, Paul;
Pichler, Robert;
Popkov, Alexander

Publication type:

Article

Steroid Glycosides Hyrcanoside and Deglucohyrcanoside: On Isolation, Structural Identification, and Anticancer Activity.

Published in:

Foods, 2021, v. 10, n. 1, p. 136, doi. 10.3390/foods10010136

By:

Rimpelová, Silvie;
Zimmermann, Tomáš;
Drašar, Pavel B.;
Dolenský, Bohumil;
Bejček, Jiří;
Kmoníčková, Eva;
Cihlářová, Petra;
Gurská, Soňa;
Kuklíková, Lucie;
Hajdůch, Marián;
Ruml, Tomáš;
Opletal, Lubomír;
Džubák, Petr;
Jurášek, Michal

Publication type:

Article

Effects of Ginger Phenylpropanoids and Quercetin on Nrf2-ARE Pathway in Human BJ Fibroblasts and HaCaT Keratinocytes.

Published in:

BioMed Research International, 2016, v. 2016, p. 1, doi. 10.1155/2016/2173275

By:

Schadich, Ermin;
Hlaváč, Jan;
Volná, Tereza;
Varanasi, Lakshman;
Hajdúch, Marián;
Džubák, Petr

Publication type:

Article

Differential Regulation of Methylation-Regulating Enzymes by Senescent Stromal Cells Drives Colorectal Cancer Cell Response to DNA-Demethylating Epi-Drugs.

Published in:

Stem Cells International, 2018, p. 1, doi. 10.1155/2018/6013728

By:

Agrawal, Khushboo;
Das, Viswanath;
Táborská, Natálie;
Gurský, Ján;
Džubák, Petr;
Hajdúch, Marián

Publication type:

Article

Synthesis and Biological Evaluation of Oxindole Sulfonamide Derivatives as Bruton's Tyrosine Kinase Inhibitors.

Published in:

ChemMedChem, 2024, v. 19, n. 1, p. 1, doi. 10.1002/cmdc.202300511

By:

Koraboina, Chandra Prakash;
Maddipati, Venkatanarayana Chowdary;
Annadurai, Narendran;
Gurská, Soňa;
Džubák, Petr;
Hajdúch, Marián;
Das, Viswanath;
Gundla, Rambabu

Publication type:

Article

<italic>N</italic>‐Benzyl Substitution of Polyhydroxypyrrolidines: The Way to Selective Inhibitors of Golgi α‐Mannosidase II.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 373, doi. 10.1002/cmdc.201700607

By:

Šesták, Sergej;
Bella, Maroš;
Klunda, Tomáš;
Gurská, Soňa;
Džubák, Petr;
Wöls, Florian;
Wilson, Iain B. H.;
Sladek, Vladimir;
Hajdúch, Marián;
Poláková, Monika;
Kóňa, Juraj

Publication type:

Article

Antiviral Activity of Selected Lamiaceae Essential Oils and Their Monoterpenes Against SARS-Cov-2.

Published in:

Frontiers in Pharmacology, 2022, v. 13, p. 1, doi. 10.3389/fphar.2022.893634

By:

Ćavar Zeljković, Sanja;
Schadich, Ermin;
Džubák, Petr;
Hajdúch, Marián;
Tarkowski, Petr

Publication type:

Article

Synthesis and Biological Activity of 2,6‐Disubstituted 7‐Deazapurine Ribonucleosides.

Published in:

European Journal of Organic Chemistry, 2025, v. 28, n. 5, p. 1, doi. 10.1002/ejoc.202401187

By:

Šinkevičiūtė, Ugnė;
Dvořáková, Marcela;
Tichý, Michal;
Gurská, Soňa;
Ječmeňová, Kateřina;
Poštová Slavětínská, Lenka;
Džubák, Petr;
Hajdúch, Marián;
Hocek, Michal

Publication type:

Article

Synthesis and Biological Profiling of Benzofuro‐Fused 7‐Deazapurine Nucleosides.

Published in:

European Journal of Organic Chemistry, 2023, v. 26, n. 44, p. 1, doi. 10.1002/ejoc.202300723

By:

Yang, Chao;
Tichý, Michal;
Poštová Slavětínská, Lenka;
Vaiedelich, Enzo;
Gurská, Soňa;
Džubák, Petr;
Hajdúch, Marián;
Hocek, Michal

Publication type:

Article

C‐5 Aryl Substituted Azaspirooxindolinones Derivatives: Synthesis and Biological Evaluation as Potential Inhibitors of Tec Family Kinases.

Published in:

European Journal of Organic Chemistry, 2021, v. 2021, n. 33, p. 4630, doi. 10.1002/ejoc.202100699

By:

Mudasani, Gopal;
Paidikondala, Kalyani;
Gurská, Soňa;
Maddirala, Shambabu Joseph;
Džubák, Petr;
Das, Viswanath;
Gundla, Rambabu

Publication type:

Article

2-Substituted 6-(Het)aryl-7-deazapurine Ribonucleosides: Synthesis, Inhibition of Adenosine Kinases, and Antimycobacterial Activity.

Published in:

ChemMedChem, 2015, v. 10, n. 6, p. 1079, doi. 10.1002/cmdc.201500081

By:

Malnuit, Vincent;
Slavětínská, Lenka Poštová;
Nauš, Petr;
Džubák, Petr;
Hajdúch, Marián;
Stolaříková, Jiřina;
Snášel, Jan;
Pichová, Iva;
Hocek, Michal

Publication type:

Article

Covidové prsty.

Published in:

Pediatrie pro Praxi, 2021, v. 22, n. 3, p. 233, doi. 10.36290/ped.2021.047

By:

Kopřiva, František;
Džubák, Petr

Publication type:

Article

Microtubule affinity-regulating kinases are potential druggable targets for Alzheimer's disease.

Published in:

Cellular & Molecular Life Sciences, 2017, v. 74, n. 22, p. 4159, doi. 10.1007/s00018-017-2574-1

By:

Annadurai, Narendran;
Agrawal, Khushboo;
Džubák, Petr;
Hajdúch, Marián;
Das, Viswanath

Publication type:

Article

Thienopyrrolo[2, 3‐d]pyrimidines, New Tricyclic Nucleobase Analogues: Synthesis and Biological Activities.

Published in:

ChemistrySelect, 2018, v. 3, n. 31, p. 9144, doi. 10.1002/slct.201802190

By:

Tichý, Michal;
Smoleń, Sabina;
Deingruber, Tomáš;
Džubák, Petr;
Pohl, Radek;
Slavětínská, Lenka Poštová;
Hajdúch, Marián;
Hocek, Michal

Publication type:

Article

Proteome Mapping of Cervical Mucus and Its Potential as a Source of Biomarkers in Female Tract Disorders.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 2, p. 1038, doi. 10.3390/ijms24021038

By:

Oždian, Tomáš;
Vodička, Jan;
Dostál, Jiří;
Holub, Dušan;
Václavková, Jana;
Ješeta, Michal;
Hamerníková, Barbora;
Kouřilová, Pavla;
Malchar, Ondřej;
Dvořák, Vladimír;
Hejtmánek, Pavel;
Sobková, Kateřina;
Ventruba, Pavel;
Pilka, Radovan;
Džubák, Petr;
Hajdúch, Marián

Publication type:

Article

Mixture Effects of Tryptophan Intestinal Microbial Metabolites on Aryl Hydrocarbon Receptor Activity.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 18, p. N.PAG, doi. 10.3390/ijms231810825

By:

Vrzalová, Aneta;
Pečinková, Petra;
Illés, Peter;
Gurská, Soňa;
Džubák, Petr;
Szotkowski, Martin;
Hajdúch, Marián;
Mani, Sridhar;
Dvořák, Zdeněk

Publication type:

Article

Current Adenosinergic Therapies: What Do Cancer Cells Stand to Gain and Lose?

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 22, p. 12569, doi. 10.3390/ijms222212569

By:

Kotulová, Jana;
Hajdúch, Marián;
Džubák, Petr

Publication type:

Article

Cell-based DNA demethylation detection system for screening of epigenetic drugs in 2D, 3D, and xenograft models.

Published in:

Cytometry. Part A, 2017, v. 91, n. 2, p. 133, doi. 10.1002/cyto.a.23004

By:

Agrawal, Khushboo;
Das, Viswanath;
Otmar, Miroslav;
Krečmerová, Marcela;
Džubák, Petr;
Hajdúch, Marián

Publication type:

Article

Functional p53 in cells contributes to the anticancer effect of the cyclin-dependent kinase inhibitor roscovitine.

Published in:

Journal of Cellular Biochemistry, 2009, v. 107, n. 3, p. 428, doi. 10.1002/jcb.22139

By:

Paprskářová, Martina;
Kryštof, Vladimír;
Jorda, Radek;
Džubák, Petr;
Hajdúch, Marián;
Węsierska-Gądek, Józefa;
Strnad, Miroslav

Publication type:

Article

Síntesis y actividad antiproliferativa de una mezcla de derivados de (+ / -) 7-cloro-(4-tioalquilquinolina). Inducción de apoptosis y daño sobre el ADN/ARN.

Published in:

Revista Colombiana de Química, 2023, v. 52, n. 1, p. 10, doi. 10.15446/rev.colomb.quim.v52n1.110787

By:

Gutiérrez, Joyce E.;
Fernández-Moreira, Esteban;
De Sanctis, Juan B.;
Gurská, Soňa;
Džubák, Petr;
Hajdůch, Marián;
Ramírez, Hegira;
Charris, Jaime E.

Publication type:

Article

Synthesis, Antimalarial, Antileishmanial, and Cytotoxicity Activities and Preliminary In Silico ADMET Studies of 2-(7-Chloroquinolin-4-ylamino)ethyl Benzoate Derivatives.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 12, p. 1709, doi. 10.3390/ph16121709

By:

Gutiérrez, Joyce E.;
Ramírez, Hegira;
Fernandez-Moreira, Esteban;
Acosta, María E.;
Mijares, Michael R.;
De Sanctis, Juan Bautista;
Gurská, Soňa;
Džubák, Petr;
Hajdúch, Marián;
Labrador-Fagúndez, Liesangerli;
Stella, Bruno G.;
Díaz-Pérez, Luis José;
Benaim, Gustavo;
Charris, Jaime E.

Publication type:

Article

Novel 7-Chloro-(4-thioalkylquinoline) Derivatives: Synthesis and Antiproliferative Activity through Inducing Apoptosis and DNA/RNA Damage.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 10, p. 1234, doi. 10.3390/ph15101234

By:

Gutiérrez, Joyce E.;
Fernandez-Moreira, Esteban;
Rodríguez, Miguel A.;
Mijares, Michael R.;
De Sanctis, Juan Bautista;
Gurská, Soňa;
Džubák, Petr;
Hajdůch, Marián;
Bruno-Colmenarez, Julia;
Rojas, Luis;
Deffieux, Denis;
Pouységu, Laurent;
Quideau, Stéphane;
Charris, Jaime;
Ramírez, Hegira

Publication type:

Article

Synthesis and Cytotoxic and Antiviral Activity Profiling of All‐Four Isomeric Series of Pyrido‐Fused 7‐Deazapurine Ribonucleosides.

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 57, p. 13002, doi. 10.1002/chem.202001124

By:

Veselovská, Lucia;
Kudlová, Natálie;
Gurská, Soňa;
Lišková, Barbora;
Medvedíková, Martina;
Hodek, Ondřej;
Tloušťová, Eva;
Milisavljevic, Nemanja;
Tichý, Michal;
Perlíková, Pavla;
Mertlíková‐Kaiserová, Helena;
Trylčová, Jana;
Pohl, Radek;
Klepetářová, Blanka;
Džubák, Petr;
Hajdúch, Marián;
Hocek, Michal

Publication type:

Article

Click estradiol dimers with novel aromatic bridging units: synthesis and anticancer evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2367139

By:

Řehulka, Jiří;
Jurášek, Michal;
Dráber, Pavel;
Ivanová, Aleksandra;
Gurská, Soňa;
Ječmeňová, Kateřina;
Mokshyna, Olena;
Hajdúch, Marián;
Polishchuk, Pavel;
Drašar, Pavel B.;
Džubák, Petr

Publication type:

Article

Toll-Like Receptor 7/8 Ligand, S28463, Suppresses Ascaris suum-induced Allergic Asthma in Nonhuman Primates.

Published in:

American Journal of Respiratory Cell & Molecular Biology, 2018, v. 58, n. 1, p. 55, doi. 10.1165/rcmb.2017-0184OC

By:

Camateros, Pierre;
Kanagaratham, Cynthia;
Najdekr, Lukáš;
Holub, Dušan;
Vrbkova, Jana;
Coté, Lucie;
Fournier, Jocelyn;
Gourdon, Jim;
Creery, David;
Olivenstein, Ron;
Kopriva, Frantisek;
Adam, Tomáš;
Friedecký, David;
Džubák, Petr;
Hajdúh, Marian;
Radzioch, Danuta

Publication type:

Article

Cytotoxicity of Amino‐BODIPY Modulated via Conjugation with 2‐Phenyl‐3‐Hydroxy‐4(1H)‐Quinolinones.

Published in:

ChemistryOpen, 2021, v. 10, n. 11, p. 1104, doi. 10.1002/open.202100025

By:

Porubský, Martin;
Vychodilová, Kristýna;
Milićević, David;
Buděšinský, Miloš;
Stanková, Jarmila;
Džubák, Petr;
Hajdúch, Marián;
Hlaváč, Jan

Publication type:

Article

Synthesis and evaluation of the anticancer activity of some semisynthetic derivatives of rutaecarpine and evodiamine.

Published in:

Synthetic Communications, 2021, v. 51, n. 21, p. 3237, doi. 10.1080/00397911.2021.1919712

By:

Patrykei, Serhii;
Korobko, Yulia;
Ogorodniichuk, Oleksandr;
Garazd, Myroslav;
Polishchuk, Pavel;
Džubák, Petr;
Gurská, Soňa;
Hajdúch, Marián;
Lesyk, Roman

Publication type:

Article

Synthesis and antitumour activity of varitriol and its analogues.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2012, p. 365

By:

Caletková, Oľga;
Lásiková, Angelika;
Hajdúch, Marián;
Džubák, Petr;
Graczaa, Tibor

Publication type:

Article

Works by Džubák, Petr

Secondary metabolite profiles and anti‐SARS‐CoV‐2 activity of ethanolic extracts from nine genotypes of Cannabis sativa L.

New Imidazo[1,2- c]pyrimidin-5(6 H)-Ones Derived from Cytosine: Synthesis, Structure, and Cytotoxic Activity.

A unique case of AH-dominant type nodular pulmonary amyloidosis presenting as a spontaneous pneumothorax: a case report and review of the literature.

Synthesis, Leishmanicidal, Trypanocidal, Antiproliferative Assay and Apoptotic Induction of (2-Phenoxypyridin-3-yl)naphthalene-1(2 H)-one Derivatives.

Betulinic Acid Decorated with Polar Groups and Blue Emitting BODIPY Dye: Synthesis, Cytotoxicity, Cell-Cycle Analysis and Anti-HIV Profiling.

Isomeric Naphtho‐Fused 7‐Deazapurine Nucleosides and Nucleotides: Synthesis, Biological Activity, Photophysical Properties and Enzymatic Incorporation to Nucleic Acids.

Improved syntheses of P2X<sub>7</sub> ligands based on substituted benzyl amide of pyroglutamic acid motif labelled with iodine-123 or iodine-125.

Steroid Glycosides Hyrcanoside and Deglucohyrcanoside: On Isolation, Structural Identification, and Anticancer Activity.

Effects of Ginger Phenylpropanoids and Quercetin on Nrf2-ARE Pathway in Human BJ Fibroblasts and HaCaT Keratinocytes.

Differential Regulation of Methylation-Regulating Enzymes by Senescent Stromal Cells Drives Colorectal Cancer Cell Response to DNA-Demethylating Epi-Drugs.

Synthesis and Biological Evaluation of Oxindole Sulfonamide Derivatives as Bruton's Tyrosine Kinase Inhibitors.

<italic>N</italic>‐Benzyl Substitution of Polyhydroxypyrrolidines: The Way to Selective Inhibitors of Golgi α‐Mannosidase II.

Antiviral Activity of Selected Lamiaceae Essential Oils and Their Monoterpenes Against SARS-Cov-2.

Synthesis and Biological Activity of 2,6‐Disubstituted 7‐Deazapurine Ribonucleosides.

Synthesis and Biological Profiling of Benzofuro‐Fused 7‐Deazapurine Nucleosides.

C‐5 Aryl Substituted Azaspirooxindolinones Derivatives: Synthesis and Biological Evaluation as Potential Inhibitors of Tec Family Kinases.

2-Substituted 6-(Het)aryl-7-deazapurine Ribonucleosides: Synthesis, Inhibition of Adenosine Kinases, and Antimycobacterial Activity.

Covidové prsty.

Microtubule affinity-regulating kinases are potential druggable targets for Alzheimer's disease.

Thienopyrrolo[2, 3‐d]pyrimidines, New Tricyclic Nucleobase Analogues: Synthesis and Biological Activities.

Proteome Mapping of Cervical Mucus and Its Potential as a Source of Biomarkers in Female Tract Disorders.

Mixture Effects of Tryptophan Intestinal Microbial Metabolites on Aryl Hydrocarbon Receptor Activity.

Current Adenosinergic Therapies: What Do Cancer Cells Stand to Gain and Lose?

Cell-based DNA demethylation detection system for screening of epigenetic drugs in 2D, 3D, and xenograft models.

Functional p53 in cells contributes to the anticancer effect of the cyclin-dependent kinase inhibitor roscovitine.

Síntesis y actividad antiproliferativa de una mezcla de derivados de (<sup>+</sup> / <sub>-</sub>) 7-cloro-(4-tioalquilquinolina). Inducción de apoptosis y daño sobre el ADN/ARN.

Synthesis, Antimalarial, Antileishmanial, and Cytotoxicity Activities and Preliminary In Silico ADMET Studies of 2-(7-Chloroquinolin-4-ylamino)ethyl Benzoate Derivatives.

Novel 7-Chloro-(4-thioalkylquinoline) Derivatives: Synthesis and Antiproliferative Activity through Inducing Apoptosis and DNA/RNA Damage.

Synthesis and Cytotoxic and Antiviral Activity Profiling of All‐Four Isomeric Series of Pyrido‐Fused 7‐Deazapurine Ribonucleosides.

Click estradiol dimers with novel aromatic bridging units: synthesis and anticancer evaluation.

Toll-Like Receptor 7/8 Ligand, S28463, Suppresses Ascaris suum-induced Allergic Asthma in Nonhuman Primates.

Cytotoxicity of Amino‐BODIPY Modulated via Conjugation with 2‐Phenyl‐3‐Hydroxy‐4(1H)‐Quinolinones.

Synthesis and evaluation of the anticancer activity of some semisynthetic derivatives of rutaecarpine and evodiamine.

Synthesis and antitumour activity of varitriol and its analogues.