An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains.
- Published in:
- Angewandte Chemie, 2019, v. 131, n. 4, p. 1019, doi. 10.1002/ange.201807825
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- Publication type:
- Article
Works by D'Ascenzio, Melissa
Results: 11
1
2
4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 597, doi. 10.1080/14756366.2019.1571272
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- Publication type:
- Article
3
Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 51, doi. 10.1080/14756366.2016.1235040
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- Publication type:
- Article
4
(Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 908, doi. 10.3109/14756366.2014.987138
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- Publication type:
- Article
5
An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains.
- Published in:
- Angewandte Chemie International Edition, 2019, v. 58, n. 4, p. 1007, doi. 10.1002/anie.201807825
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- Publication type:
- Article
6
Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines.
- Published in:
- Journal of Heterocyclic Chemistry, 2014, v. 51, n. 6, p. 1856, doi. 10.1002/jhet.1856
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- Publication type:
- Article
7
Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and Their In Vitro Inhibition of Human Cyclooxygenase.
- Published in:
- Journal of Heterocyclic Chemistry, 2012, v. 49, n. 5, p. 1187, doi. 10.1002/jhet.1058
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- Publication type:
- Article
8
Synthesis and anti- Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives.
- Published in:
- Journal of Heterocyclic Chemistry, 2010, v. 47, n. 6, p. 1269, doi. 10.1002/jhet.464
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- Publication type:
- Article
9
A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases.
- Published in:
- Chemistry - A European Journal, 2016, v. 22, n. 1, p. 97, doi. 10.1002/chem.201503748
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- Publication type:
- Article
10
Selective MAO-B inhibitors: a lesson from natural products.
- Published in:
- Molecular Diversity, 2014, v. 18, n. 1, p. 219, doi. 10.1007/s11030-013-9490-6
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- Publication type:
- Article
11
Synthesis and Selective Human Monoamine Oxidase B Inhibition of Heterocyclic Hybrids Based on Hydrazine and Thiazole Scaffolds.
- Published in:
- Archiv der Pharmazie, 2013, v. 346, n. 1, p. 17, doi. 10.1002/ardp.201200318
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- Publication type:
- Article