Works by D'Agostino, Ilaria

Results: 23

Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400776

By:

Paciotti, Roberto;
Carradori, Simone;
Angeli, Andrea;
D'Agostino, Ilaria;
Ferraroni, Marta;
Coletti, Cecilia;
Supuran, Claudiu T.

Publication type:

Article

Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2024, v. 357, n. 11, p. 1, doi. 10.1002/ardp.202400548

By:

Gumus, Arzu;
D'Agostino, Ilaria;
Puca, Valentina;
Crocetta, Valentina;
Carradori, Simone;
Cutarella, Luigi;
Mori, Mattia;
Carta, Fabrizio;
Angeli, Andrea;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

A New Vista of Aldehyde Dehydrogenase 1A3 (ALDH1A3): New Specific Inhibitors and Activity-Based Probes Targeting ALDH1A3 Dependent Pathways in Glioblastoma, Mesothelioma and Other Cancers.

Published in:

Cancers, 2024, v. 16, n. 13, p. 2397, doi. 10.3390/cancers16132397

By:

Magrassi, Lorenzo;
Pinton, Giulia;
Luzzi, Sabino;
Comincini, Sergio;
Scravaglieri, Andrea;
Gigliotti, Valentina;
Bernardoni, Bianca Laura;
D'Agostino, Ilaria;
Juretich, Francesca;
La Motta, Concettina;
Garavaglia, Silvia

Publication type:

Article

Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment.

Published in:

Drug Development Research, 2024, v. 85, n. 1, p. 1, doi. 10.1002/ddr.22158

By:

Vagaggini, Chiara;
Petroni, Debora;
D'Agostino, Ilaria;
Poggialini, Federica;
Cavallini, Chiara;
Cianciusi, Annarita;
Salis, Annalisa;
D'Antona, Lucia;
Francesconi, Valeria;
Manetti, Fabrizio;
Damonte, Gianluca;
Musumeci, Francesca;
Menichetti, Luca;
Dreassi, Elena;
Carbone, Anna;
Schenone, Silvia

Publication type:

Article

Negative Modulation of the Angiogenic Cascade Induced by Allosteric Kinesin Eg5 Inhibitors in a Gastric Adenocarcinoma In Vitro Model.

Published in:

Molecules, 2022, v. 27, n. 3, p. 957, doi. 10.3390/molecules27030957

By:

Ricci, Alessia;
Gallorini, Marialucia;
Del Bufalo, Donatella;
Cataldi, Amelia;
D'Agostino, Ilaria;
Carradori, Simone;
Zara, Susi

Publication type:

Article

Synthetic Heterocyclic Derivatives as Kinase Inhibitors Tested for the Treatment of Neuroblastoma †.

Published in:

Molecules, 2021, v. 26, n. 23, p. 7069, doi. 10.3390/molecules26237069

By:

Musumeci, Francesca;
Cianciusi, Annarita;
D'Agostino, Ilaria;
Grossi, Giancarlo;
Carbone, Anna;
Schenone, Silvia

Publication type:

Article

The antiplatelet agent revacept prevents the increase of systemic thromboxane A2 biosynthesis and neointima hyperplasia.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-77934-x

By:

Alberti, Sara;
Zhang, Qianqian;
D'Agostino, Ilaria;
Bruno, Annalisa;
Tacconelli, Stefania;
Contursi, Annalisa;
Guarnieri, Simone;
Dovizio, Melania;
Falcone, Lorenza;
Ballerini, Patrizia;
Münch, Götz;
Yu, Ying;
Patrignani, Paola

Publication type:

Article

Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400601

By:

Kilbile, Jaydeo T.;
Sapkal, Suryakant B.;
Renzi, Gioele;
D'Agostino, Ilaria;
Boudjelal, Mohamed;
Tamboli, Yasinalli;
Cutarella, Luigi;
Mori, Mattia;
Sgambellone, Silvia;
Villano, Serafina;
Marri, Silvia;
Lucarini, Laura;
Carradori, Simone;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Antimalarial Agents Targeting Plasmodium falciparum Carbonic Anhydrase: Towards Artesunate Hybrid Compounds with Dual Mechanism of Action.

Published in:

ChemMedChem, 2023, v. 18, n. 21, p. 1, doi. 10.1002/cmdc.202300267

By:

D'Agostino, Ilaria;
Zara, Susi;
Carradori, Simone;
De Luca, Viviana;
Capasso, Clemente;
Kocken, Clemens H. M.;
Zeeman, Anne‐Marie;
Angeli, Andrea;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Nature as a source and inspiration for human monoamine oxidase B (hMAO-B) inhibition: A review of the recent advances in chemical modification of natural compounds.

Published in:

Expert Opinion on Drug Discovery, 2023, v. 18, n. 8, p. 851, doi. 10.1080/17460441.2023.2226860

By:

Melfi, Francesco;
Carradori, Simone;
Angeli, Andrea;
D'Agostino, Ilaria

Publication type:

Article

A Journey Around Boronic Acids: Sulfonyl Hydrazone‐Containing Derivatives as Carbonic Anhydrase Inhibitors.

Published in:

Chemical Biology & Drug Design, 2025, v. 105, n. 4, p. 1, doi. 10.1111/cbdd.70108

By:

Anakök, Deniz A.;
Angeli, Andrea;
D'Agostino, Ilaria;
Renzi, Gioele;
Massardi, Maria Luisa;
Tavani, Camilla;
Çete, Servet;
Carradori, Simone;
Ronca, Roberto;
Capasso, Clemente;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas.

Published in:

Molecular Diversity, 2023, v. 27, n. 3, p. 1489, doi. 10.1007/s11030-022-10505-6

By:

Ardino, Claudia;
Sannio, Filomena;
Pasero, Carolina;
Botta, Lorenzo;
Dreassi, Elena;
Docquier, Jean-Denis;
D'Agostino, Ilaria

Publication type:

Article

Focused library of phenyl-fused macrocyclic amidinoureas as antifungal agents.

Published in:

Molecular Diversity, 2022, v. 26, n. 6, p. 3399, doi. 10.1007/s11030-022-10388-7

By:

Balestri, Lorenzo J. I.;
D'Agostino, Ilaria;
Rango, Enrico;
Vagaggini, Chiara;
Marchitiello, Rosalba;
Mariotti, Melinda;
Casian, Alexandru;
Deodato, Davide;
Truglio, Giuseppina I.;
Orofino, Francesco;
Sanguinetti, Maurizio;
Bugli, Francesca;
Botta, Lorenzo;
Dreassi, Elena

Publication type:

Article

Assessment of The Green Corrosion Inhibition Performances of Thymus Algeriensis Microwave-Assisted Extracts on Mild Steel in Acid Solution.

Published in:

Analytical & Bioanalytical Electrochemistry, 2023, v. 15, n. 11, p. 938, doi. 10.22034/abec.2023.709095

By:

Boutaoui, Nassima;
Acila, Meryem;
Boulahbel, Hani;
Achouri, Billel;
Zaiter, Lahcene;
Benayache, Fadila;
Benayache, Samir;
D'Agostino, Ilaria;
Campestre, Cristina;
Locatelli, Marcello

Publication type:

Article

Reduced Variability to Aspirin Antiplatelet Effect by the Coadministration of Statins in High‐Risk Patients for Cardiovascular Disease.

Published in:

Clinical Pharmacology & Therapeutics, 2018, v. 104, n. 1, p. 111, doi. 10.1002/cpt.1075

By:

Tacconelli, Stefania;
Dovizio, Melania;
Di Francesco, Luigia;
D'Agostino, Ilaria;
Bruno, Annalisa;
Patrignani, Paola;
Capone, Marta L.;
Grossi, Linda;
Ballerini, Patrizia;
Meneguzzi, Alessandra;
Fava, Cristiano;
Minuz, Pietro;
Evangelista, Virgilio;
Manarini, Stefano;
Porreca, Ettore;
Di Febbo, Concetta;
Levantesi, Giacomo

Publication type:

Article

Antimicrobial and Antibiofilm Activities of Carvacrol, Amoxicillin and Salicylhydroxamic Acid Alone and in Combination vs. Helicobacter pylori: Towards a New Multi-Targeted Therapy.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 5, p. 4455, doi. 10.3390/ijms24054455

By:

Puca, Valentina;
Turacchio, Gabriele;
Marinacci, Beatrice;
Supuran, Claudiu T.;
Capasso, Clemente;
Di Giovanni, Pamela;
D'Agostino, Ilaria;
Carradori, Simone;
Grande, Rossella

Publication type:

Article

Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies.

Published in:

Pharmaceuticals (14248247), 2024, v. 17, n. 8, p. 1027, doi. 10.3390/ph17081027

By:

Giampietro, Letizia;
Marinacci, Beatrice;
Della Valle, Alice;
D'Agostino, Ilaria;
Lauro, Aldo;
Mori, Mattia;
Carradori, Simone;
Ammazzalorso, Alessandra;
De Filippis, Barbara;
Maccallini, Cristina;
Angeli, Andrea;
Capasso, Clemente;
Francati, Santolo;
Mollica, Adriano;
Grande, Rossella;
Supuran, Claudiu T.

Publication type:

Article

Nature-Inspired Compounds: Synthesis and Antibacterial Susceptibility Testing of Eugenol Derivatives against H. pylori Strains.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 9, p. 1317, doi. 10.3390/ph16091317

By:

Carradori, Simone;
Ammazzalorso, Alessandra;
Niccolai, Sofia;
Tanini, Damiano;
D'Agostino, Ilaria;
Melfi, Francesco;
Capperucci, Antonella;
Grande, Rossella;
Sisto, Francesca

Publication type:

Article

Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201402

By:

Fantacuzzi, Marialuigia;
D'Agostino, Ilaria;
Carradori, Simone;
Liguori, Francesco;
Carta, Fabrizio;
Agamennone, Mariangela;
Angeli, Andrea;
Sannio, Filomena;
Docquier, Jean-Denis;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 986, doi. 10.1080/14756366.2022.2055009

By:

D'Agostino, Ilaria;
Mathew, Githa Elizabeth;
Angelini, Paola;
Venanzoni, Roberto;
Flores, Giancarlo Angeles;
Angeli, Andrea;
Carradori, Simone;
Marinacci, Beatrice;
Menghini, Luigi;
Abdelgawad, Mohamed A.;
Ghoneim, Mohammed M.;
Mathew, Bijo;
Supuran, Claudiu T.

Publication type:

Article

The challenging inhibition of Aldose Reductase for the treatment of diabetic complications: a 2019–2023 update of the patent literature.

Published in:

Expert Opinion on Therapeutic Patents, 2024, v. 34, n. 11, p. 1085, doi. 10.1080/13543776.2024.2412573

By:

Bernardoni, Bianca Laura;
D'Agostino, Ilaria;
Scianò, Fabio;
La Motta, Concettina

Publication type:

Article

An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans, the pivotal pathogens in the oral cavity.

Published in:

Expert Opinion on Therapeutic Patents, 2024, v. 34, n. 6, p. 433, doi. 10.1080/13543776.2024.2349739

By:

Bernardoni, Bianca Laura;
D'Agostino, Ilaria;
La Motta, Concettina;
Angeli, Andrea

Publication type:

Article

Emerging compounds and therapeutic strategies to treat infections from Trypanosoma brucei: an overhaul of the last 5-years patents.

Published in:

Expert Opinion on Therapeutic Patents, 2023, v. 33, n. 3, p. 247, doi. 10.1080/13543776.2023.2193328

By:

Melfi, Francesco;
Carradori, Simone;
Campestre, Cristina;
Haloci, Entela;
Ammazzalorso, Alessandra;
Grande, Rossella;
D'Agostino, Ilaria

Publication type:

Article