Works by Courageux, Charlotte

Results: 8

Chemoselective Hydrogenation of 6‐Alkynyl‐3‐fluoro‐2‐pyridinaldoximes: Access to First‐in‐Class 6‐Alkyl‐3‐Fluoro‐2‐pyridinaldoxime Scaffolds as New Reactivators of Sarin‐Inhibited Human Acetylcholinesterase with Increased Blood–Brain Barrier Permeability

Published in:

Chemistry - A European Journal, 2020, v. 26, n. 65, p. 15035, doi. 10.1002/chem.202002012

By:

Yerri, Jagadeesh;
Dias, José;
Nimmakayala, Mallikajurna Reddy;
Razafindrainibe, Franck;
Courageux, Charlotte;
Gastellier, Anne‐Julie;
Jegoux, Johanne;
Coisne, Caroline;
Landry, Christophe;
Gosselet, Fabien;
Hachani, Johan;
Goossens, Jean‐François;
Dehouck, Marie‐Pierre;
Nachon, Florian;
Baati, Rachid

Publication type:

Article

Discovery of drug‐like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database.

Published in:

Chemical Biology & Drug Design, 2021, v. 97, n. 5, p. 1048, doi. 10.1111/cbdd.13825

By:

Miles, Jared A.;
Ng, Jia Hui;
Sreenivas, B. Yogi;
Courageux, Charlotte;
Igert, Alexandre;
Dias, José;
McGeary, Ross P.;
Brazzolotto, Xavier;
Ross, Benjamin P.

Publication type:

Article

Cover Image.

Published in:

Chemical Biology & Drug Design, 2021, v. 97, n. 5, p. i, doi. 10.1111/cbdd.13717

By:

Miles, Jared A.;
Ng, Jia Hui;
Sreenivas, B. Yogi;
Courageux, Charlotte;
Igert, Alexandre;
Dias, José;
McGeary, Ross P.;
Brazzolotto, Xavier;
Ross, Benjamin P.

Publication type:

Article

Development of versatile and potent monoquaternary reactivators of acetylcholinesterase.

Published in:

Archives of Toxicology, 2021, v. 95, n. 3, p. 985, doi. 10.1007/s00204-021-02981-w

By:

Gorecki, Lukas;
Hepnarova, Vendula;
Karasova, Jana Zdarova;
Hrabinova, Martina;
Courageux, Charlotte;
Dias, José;
Kucera, Tomas;
Kobrlova, Tereza;
Muckova, Lubica;
Prchal, Lukas;
Malinak, David;
Jun, Daniel;
Musilek, Kamil;
Worek, Franz;
Nachon, Florian;
Soukup, Ondrej;
Korabecny, Jan

Publication type:

Article

Efficacy Assessment of an Uncharged Reactivator of NOP-Inhibited Acetylcholinesterase Based on Tetrahydroacridine Pyridine-Aldoxime Hybrid in Mouse Compared to Pralidoxime.

Published in:

Biomolecules (2218-273X), 2020, v. 10, n. 6, p. 858, doi. 10.3390/biom10060858

By:

Calas, André-Guilhem;
Hanak, Anne-Sophie;
Jaffré, Nina;
Nervo, Aurélie;
Dias, José;
Rousseau, Catherine;
Courageux, Charlotte;
Brazzolotto, Xavier;
Villa, Pascal;
Obrecht, Adeline;
Goossens, Jean-François;
Landry, Christophe;
Hachani, Johan;
Gosselet, Fabien;
Dehouck, Marie-Pierre;
Yerri, Jagadeesh;
Kliachyna, Maria;
Baati, Rachid;
Nachon, Florian

Publication type:

Article

Genes coding for transcription factors involved in stem cell maintenance are repressed by TGF-β and downstream of Slug/Snail2 in COPD bronchial epithelial progenitors.

Published in:

Molecular Biology Reports, 2021, v. 48, n. 10, p. 6729, doi. 10.1007/s11033-021-06664-8

By:

de la Grange, Pierre;
Jolly, Ariane;
Courageux, Charlotte;
Ben Brahim, Chamseddine;
Leroy, Pascale

Publication type:

Article

Grid‐Type Quaternary Metallosupramolecular Compounds Inhibit Human Cholinesterases through Dynamic Multivalent Interactions.

Published in:

ChemBioChem, 2022, v. 23, n. 23, p. 1, doi. 10.1002/cbic.202200456

By:

Nachon, Florian;
Brazzolotto, Xavier;
Dias, José;
Courageux, Charlotte;
Drożdż, Wojciech;
Cao, Xiao‐Yu;
Stefankiewicz, Artur R.;
Lehn, Jean‐Marie

Publication type:

Article

DESIGN, SYNTHESIS AND IN VITRO EVALUATION OF A PROMISING NEW CLASS OF BIFUNCTIONAL UNCHARGED HYBRID REACTIVATORS FOR NERVE AGENT-INHIBITED HUMAN ACETYLCHOLINESTERASE.

Published in:

Military Medical Science Letters / Vojenské zdravotnické Listy, 2018, v. 87, p. 100

By:

Dias, José;
De Sousa, Julien;
Jagadeesh, Yerri;
Courageux, Charlotte;
Gastellier, Anne-Julie;
Timperley, Christopher;
Brown, Richard;
Santoni, Gianluca;
Weik, Martin;
Baati, Rachid;
Nachon, Florian

Publication type:

Article