Works by Corona, Angela


Results: 59
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    Targeting SARS-CoV-2 nsp13 Helicase and Assessment of Druggability Pockets: Identification of Two Potent Inhibitors by a Multi-Site In Silico Drug Repurposing Approach.

    Published in:
    Molecules, 2022, v. 27, n. 21, p. 7522, doi. 10.3390/molecules27217522
    By:
    • Romeo, Isabella;
    • Ambrosio, Francesca Alessandra;
    • Costa, Giosuè;
    • Corona, Angela;
    • Alkhatib, Mohammad;
    • Salpini, Romina;
    • Lemme, Saverio;
    • Vergni, Davide;
    • Svicher, Valentina;
    • Santoro, Maria Mercedes;
    • Tramontano, Enzo;
    • Ceccherini-Silberstein, Francesca;
    • Artese, Anna;
    • Alcaro, Stefano
    Publication type:
    Article
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    Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding.

    Published in:
    ChemBioChem, 2017, v. 18, n. 4, p. 374, doi. 10.1002/cbic.201600592
    By:
    • Martini, Riccardo;
    • Esposito, Francesca;
    • Corona, Angela;
    • Ferrarese, Roberto;
    • Ceresola, Elisa Rita;
    • Visconti, Laura;
    • Tintori, Cristina;
    • Barbieri, Alessandro;
    • Calcaterra, Andrea;
    • Iovine, Valentina;
    • Canducci, Filippo;
    • Tramontano, Enzo;
    • Botta, Maurizio
    Publication type:
    Article
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    Cytopathic SARS-CoV-2 screening on VERO-E6 cells in a large-scale repurposing effort.

    Published in:
    Scientific Data, 2022, v. 9, n. 1, p. 1, doi. 10.1038/s41597-022-01532-x
    By:
    • Zaliani, Andrea;
    • Vangeel, Laura;
    • Reinshagen, Jeanette;
    • Iaconis, Daniela;
    • Kuzikov, Maria;
    • Keminer, Oliver;
    • Wolf, Markus;
    • Ellinger, Bernhard;
    • Esposito, Francesca;
    • Corona, Angela;
    • Tramontano, Enzo;
    • Manelfi, Candida;
    • Herzog, Katja;
    • Jochmans, Dirk;
    • De Jonghe, Steven;
    • Chiu, Winston;
    • Francken, Thibault;
    • Schepers, Joost;
    • Collard, Caroline;
    • Abbasi, Kayvan
    Publication type:
    Article
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    Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).

    Published in:
    ChemMedChem, 2016, v. 11, n. 16, p. 1669, doi. 10.1002/cmdc.201600392
    By:
    • Corona, Angela;
    • Desantis, Jenny;
    • Massari, Serena;
    • Distinto, Simona;
    • Masaoka, Takashi;
    • Sabatini, Stefano;
    • Esposito, Francesca;
    • Manfroni, Giuseppe;
    • Maccioni, Elias;
    • Cecchetti, Violetta;
    • Pannecouque, Christophe;
    • Le Grice, Stuart F. J.;
    • Tramontano, Enzo;
    • Tabarrini, Oriana
    Publication type:
    Article
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    Design, Synthesis, and Biological Evaluation of 1,3-Diarylpropenones as Dual Inhibitors of HIV-1 Reverse Transcriptase.

    Published in:
    ChemMedChem, 2014, v. 9, n. 8, p. 1869, doi. 10.1002/cmdc.201402015
    By:
    • Meleddu, Rita;
    • Cannas, Valeria;
    • Distinto, Simona;
    • Sarais, Giorgia;
    • Del Vecchio, Claudia;
    • Esposito, Francesca;
    • Bianco, Giulia;
    • Corona, Angela;
    • Cottiglia, Filippo;
    • Alcaro, Stefano;
    • Parolin, Cristina;
    • Artese, Anna;
    • Scalise, Daniela;
    • Fresta, Massimo;
    • Arridu, Antonella;
    • Ortuso, Francesco;
    • Maccioni, Elias;
    • Tramontano, Enzo
    Publication type:
    Article
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    Biological Activities of Aerial Parts Extracts of Euphorbia characias.

    Published in:
    BioMed Research International, 2016, v. 2016, p. 1, doi. 10.1155/2016/1538703
    By:
    • Pisano, Maria Barbara;
    • Cosentino, Sofia;
    • Viale, Silvia;
    • Spanò, Delia;
    • Corona, Angela;
    • Esposito, Francesca;
    • Tramontano, Enzo;
    • Montoro, Paola;
    • Tuberoso, Carlo Ignazio Giovanni;
    • Medda, Rosaria;
    • Pintus, Francesca
    Publication type:
    Article
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    New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors.

    Published in:
    Pharmaceuticals (14248247), 2024, v. 17, n. 5, p. 650, doi. 10.3390/ph17050650
    By:
    • Messore, Antonella;
    • Malune, Paolo;
    • Patacchini, Elisa;
    • Madia, Valentina Noemi;
    • Ialongo, Davide;
    • Arpacioglu, Merve;
    • Albano, Aurora;
    • Ruggieri, Giuseppe;
    • Saccoliti, Francesco;
    • Scipione, Luigi;
    • Tramontano, Enzo;
    • Canton, Serena;
    • Corona, Angela;
    • Scognamiglio, Sante;
    • Paulis, Annalaura;
    • Suleiman, Mustapha;
    • Al-Maqtari, Helmi Mohammed;
    • Abid, Fatma Mohamed A.;
    • Kawsar, Sarkar M. A.;
    • Sankaranarayanan, Murugesan
    Publication type:
    Article
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    DHFR Inhibitors Display a Pleiotropic Anti-Viral Activity against SARS-CoV-2: Insights into the Mechanisms of Action.

    Published in:
    Viruses (1999-4915), 2023, v. 15, n. 5, p. 1128, doi. 10.3390/v15051128
    By:
    • Iaconis, Daniela;
    • Caccuri, Francesca;
    • Manelfi, Candida;
    • Talarico, Carmine;
    • Bugatti, Antonella;
    • Filippini, Federica;
    • Zani, Alberto;
    • Novelli, Rubina;
    • Kuzikov, Maria;
    • Ellinger, Bernhard;
    • Gribbon, Philip;
    • Riecken, Kristoffer;
    • Esposito, Francesca;
    • Corona, Angela;
    • Tramontano, Enzo;
    • Beccari, Andrea Rosario;
    • Caruso, Arnaldo;
    • Allegretti, Marcello
    Publication type:
    Article
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    Alizarine derivatives as new dual inhibitors of the HIV-1 reverse transcriptase-associated DNA polymerase and RNase H activities effective also on the RNase H activity of non-nucleoside resistant reverse transcriptases.

    Published in:
    FEBS Journal, 2011, v. 278, n. 9, p. 1444, doi. 10.1111/j.1742-4658.2011.08057.x
    By:
    • Esposito, Francesca;
    • Kharlamova, Tatyana;
    • Distinto, Simona;
    • Zinzula, Luca;
    • Cheng, Yung-Chi;
    • Dutschman, Ginger;
    • Floris, Giovanni;
    • Markt, Patrick;
    • Corona, Angela;
    • Tramontano, Enzo
    Publication type:
    Article
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    Scaffold hopping and optimisation of 3',4'-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1953, doi. 10.1080/14756366.2020.1835884
    By:
    • Tocco, Graziella;
    • Esposito, Francesca;
    • Caboni, Pierluigi;
    • Laus, Antonio;
    • Beutler, John A.;
    • Wilson, Jennifer A.;
    • Corona, Angela;
    • Le Grice, Stuart F. J.;
    • Tramontano, Enzo
    Publication type:
    Article