Works by Colabufo, Nicola Antonio
Results: 29
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 974, doi. 10.1080/14756366.2020.1747449
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- Article
Distribution of sigma receptors in EMT-6 cells: preliminary biological evaluation of PB167 and potential for in-vivo PET.
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- Journal of Pharmacy & Pharmacology, 2005, v. 57, n. 11, p. 1453
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- Article
A conformational rearrangement of the SARS-CoV-2 host protein sigma-1 is required for antiviral activity: insights from a combined in-silico/in-vitro approach.
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- Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-39662-w
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- Article
Herbal Medicines in Brazil: Pharmacokinetic Profile and Potential Herb-Drug Interactions.
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- Frontiers in Pharmacology, 2014, v. 5, p. 1, doi. 10.3389/fphar.2014.00162
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- Article
ABC transporters in CSCs membranes as a novel target for treating tumour relapse.
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- Frontiers in Pharmacology, 2014, v. 5, p. 1, doi. 10.3389/fphar.2014.00163
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- Article
Antiproliferative and cytotoxic effects of some σ<sub>2</sub> agonists and σ<sub>1</sub> antagonists in tumour cell lines.
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- Naunyn-Schmiedeberg's Archives of Pharmacology, 2004, v. 370, n. 2, p. 106
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- Article
Inhibition of hERG potassium channel by the antiarrhythmic agent mexiletine and its metabolite m-hydroxymexiletine.
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- Pharmacology Research & Perspectives, 2015, v. 3, n. 5, p. 1, doi. 10.1002/prp2.160
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- Article
Guinea-pig ileum as ex vivo model useful to characterize ligands displaying Imidazoline I<sub>2</sub> and Adrenergic alpha<sub>2</sub> mixed activity: a preliminary study.
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- Drugs & Therapy Studies, 2013, v. 3, n. 1, p. 1, doi. 10.4081/dts.2013.e1
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- Article
Design, synthesis, biological evaluation, NMR and DFT studies of structurally simplified trimethoxy benzamides as selective P-glycoprotein inhibitors: the role of molecular flatness.
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- Chemical Biology & Drug Design, 2016, v. 88, n. 6, p. 820, doi. 10.1111/cbdd.12811
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- Article
PB28, the Sigma-1 and Sigma-2 Receptors Modulator With Potent Anti–SARS-CoV-2 Activity: A Review About Its Pharmacological Properties and Structure Affinity Relationships.
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- Frontiers in Pharmacology, 2020, v. 11, p. N.PAG, doi. 10.3389/fphar.2020.589810
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- Article
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4‐Substituted Quinazoline Derivatives.
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- ChemMedChem, 2022, v. 17, n. 12, p. 1, doi. 10.1002/cmdc.202200027
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- Article
Corrigendum: Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels.
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- ChemMedChem, 2022, v. 17, n. 7, p. 1, doi. 10.1002/cmdc.202200131
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- Article
Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels.
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- ChemMedChem, 2021, v. 16, n. 23, p. 3588, doi. 10.1002/cmdc.202100496
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- Article
Structure-Activity Relationship Studies on 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Multidrug Resistance Reversers.
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- ChemMedChem, 2017, v. 12, n. 16, p. 1369, doi. 10.1002/cmdc.201700239
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- Article
A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression.
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- ChemMedChem, 2016, v. 11, n. 4, p. 374, doi. 10.1002/cmdc.201500538
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- Article
<sup>11</sup>C- and <sup>18</sup>F-Labeled Radioligands for P-Glycoprotein Imaging by Positron Emission Tomography.
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- ChemMedChem, 2016, v. 11, n. 1, p. 108, doi. 10.1002/cmdc.201500420
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- Article
Arylamino Esters As P-Glycoprotein Modulators: SAR Studies to Establish Requirements for Potency and Selectivity.
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- ChemMedChem, 2015, v. 10, n. 8, p. 1339, doi. 10.1002/cmdc.201500143
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- Article
PET Radiotracers for Imaging P-glycoprotein: The Challenge for Early Diagnosis in AD.
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- ChemMedChem, 2014, v. 9, n. 1, p. 38, doi. 10.1002/cmdc.201300362
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- Article
Inside Cover: Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity (ChemMedChem 12/2013).
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- ChemMedChem, 2013, v. 8, n. 12, p. 1898, doi. 10.1002/cmdc.201390051
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- Article
Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity.
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- ChemMedChem, 2013, v. 8, n. 12, p. 2026, doi. 10.1002/cmdc.201300291
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- Article
A Benzopyrane Derivative as a P-Glycoprotein Stimulator: A Potential Agent to Decrease β-Amyloid Accumulation in Alzheimer's Disease.
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- ChemMedChem, 2012, v. 7, n. 3, p. 391, doi. 10.1002/cmdc.201100469
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- Article
Inside Cover: 1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity (ChemMedChem 1/2011).
- Published in:
- ChemMedChem, 2011, v. 6, n. 1, p. 2, doi. 10.1002/cmdc.201090062
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- Article
1-Cyclohexyl-4-(4-arylcyclohexyl)piperazines: Mixed σ and Human Δ<sub>8</sub>-Δ<sub>7</sub> Sterol Isomerase Ligands with Antiproliferative and P-Glycoprotein Inhibitory Activity.
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- ChemMedChem, 2011, v. 6, n. 1, p. 73, doi. 10.1002/cmdc.201000371
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- Article
Chiral Aryloxyalkylamines: Selective 5-HT<sub>1B/1D</sub> Activation and Analgesic Activity.
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- ChemMedChem, 2010, v. 5, n. 5, p. 696, doi. 10.1002/cmdc.200900530
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- Article
Gut-Derived Uremic Toxins in CKD: An Improved Approach for the Evaluation of Serum Indoxyl Sulfate in Clinical Practice.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 6, p. 5142, doi. 10.3390/ijms24065142
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- Article
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold †.
- Published in:
- Molecules, 2024, v. 29, n. 14, p. 3290, doi. 10.3390/molecules29143290
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- Article
miRNAs for the Detection of MultiDrug Resistance: Overview and Perspectives.
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- Molecules, 2014, v. 19, n. 5, p. 5611, doi. 10.3390/molecules19055611
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- Article
Small and innovative molecules as new strategy to revert MDR.
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- Frontiers in Oncology, 2014, v. 3, p. 1, doi. 10.3389/fonc.2014.00002
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- Article
The interaction of celecoxib with MDR transporters enhances the activity of mitomycin C in a bladder cancer cell line.
- Published in:
- Molecular Cancer, 2013, v. 12, n. 1, p. 1, doi. 10.1186/1476-4598-12-47
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- Article