Works matching AU Colabufo, Nicola A.


Results: 65
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    A conformational rearrangement of the SARS-CoV-2 host protein sigma-1 is required for antiviral activity: insights from a combined in-silico/in-vitro approach.

    Published in:
    Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-39662-w
    By:
    • Abatematteo, Francesca Serena;
    • Delre, Pietro;
    • Mercurio, Ivan;
    • Rezelj, Veronica V.;
    • Siliqi, Dritan;
    • Beaucourt, Stephanie;
    • Lattanzi, Gianluca;
    • Colabufo, Nicola Antonio;
    • Leopoldo, Marcello;
    • Saviano, Michele;
    • Vignuzzi, Marco;
    • Mangiatordi, Giuseppe Felice;
    • Abate, Carmen
    Publication type:
    Article
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    6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 974, doi. 10.1080/14756366.2020.1747449
    By:
    • Braconi, Laura;
    • Bartolucci, Gianluca;
    • Contino, Marialessandra;
    • Chiaramonte, Niccolò;
    • Giampietro, Roberta;
    • Manetti, Dina;
    • Perrone, Maria Grazia;
    • Romanelli, Maria Novella;
    • Colabufo, Nicola Antonio;
    • Riganti, Chiara;
    • Dei, Silvia;
    • Teodori, Elisabetta
    Publication type:
    Article
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    Sugar-based bactericides targeting phosphatidylethanolamine-enriched membranes.

    Published in:
    Nature Communications, 2018, v. 9, n. 1, p. 1, doi. 10.1038/s41467-018-06488-4
    By:
    • Dias, Catarina;
    • Pais, João P.;
    • Nunes, Rafael;
    • Blázquez-Sánchez, Maria-Teresa;
    • Marquês, Joaquim T.;
    • Almeida, Andreia F.;
    • Serra, Patrícia;
    • Xavier, Nuno M.;
    • Vila-Viçosa, Diogo;
    • Machuqueiro, Miguel;
    • Viana, Ana S.;
    • Martins, Alice;
    • Santos, Maria S.;
    • Pelerito, Ana;
    • Dias, Ricardo;
    • Tenreiro, Rogério;
    • Oliveira, Maria C.;
    • Contino, Marialessandra;
    • Colabufo, Nicola A.;
    • de Almeida, Rodrigo F. M.
    Publication type:
    Article
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    Head-to-head comparison of (R)-[<sup>11</sup>C]verapamil and [<sup>18</sup>F]MC225 in non-human primates, tracers for measuring P-glycoprotein function.

    Published in:
    European Journal of Nuclear Medicine & Molecular Imaging, 2021, v. 48, n. 13, p. 4307, doi. 10.1007/s00259-021-05411-2
    By:
    • García-Varela, Lara;
    • Vállez García, David;
    • Aguiar, Pablo;
    • Kakiuchi, Takeharu;
    • Ohba, Hiroyuki;
    • Harada, Norihiro;
    • Nishiyama, Shingo;
    • Tago, Tetsuro;
    • Elsinga, Philip H.;
    • Tsukada, Hideo;
    • Colabufo, Nicola A.;
    • Dierckx, Rudi A. J. O.;
    • van Waarde, Aren;
    • Toyohara, Jun;
    • Boellaard, Ronald;
    • Luurtsema, Gert
    Publication type:
    Article
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    Evaluation of P-glycoprotein function at the blood–brain barrier using [<sup>18</sup>F]MC225-PET.

    Published in:
    European Journal of Nuclear Medicine & Molecular Imaging, 2021, v. 48, n. 12, p. 4105, doi. 10.1007/s00259-021-05419-8
    By:
    • Mossel, Pascalle;
    • Garcia Varela, Lara;
    • Arif, Wejdan M.;
    • van der Weijden, Chris W. J.;
    • Boersma, Hendrikus H.;
    • Willemsen, Antoon T. M.;
    • Boellaard, Ronald;
    • Elsinga, Philip H.;
    • Borra, Ronald J. H.;
    • Colabufo, Nicola A.;
    • Toyohara, Jun;
    • de Deyn, Peter Paul;
    • Dierckx, Rudi A. J. O.;
    • Lammertsma, Adriaan A.;
    • Bartels, Anna L.;
    • Luurtsema, Gert
    Publication type:
    Article
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    Nature-Inspired 1-Phenylpyrrolo[2,1- a ]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance.

    Published in:
    Pharmaceuticals (14248247), 2024, v. 17, n. 4, p. 539, doi. 10.3390/ph17040539
    By:
    • Nevskaya, Alisa A.;
    • Purgatorio, Rosa;
    • Borisova, Tatiana N.;
    • Varlamov, Alexey V.;
    • Anikina, Lada V.;
    • Obydennik, Arina Yu.;
    • Nevskaya, Elena Yu.;
    • Niso, Mauro;
    • Colabufo, Nicola A.;
    • Carrieri, Antonio;
    • Catto, Marco;
    • de Candia, Modesto;
    • Voskressensky, Leonid G.;
    • Altomare, Cosimo D.
    Publication type:
    Article
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    Exploring Mannosylpurines as Copper Chelators and Cholinesterase Inhibitors with Potential for Alzheimer's Disease.

    Published in:
    Pharmaceuticals (14248247), 2023, v. 16, n. 1, p. 54, doi. 10.3390/ph16010054
    By:
    • Schino, Ignazio;
    • Cantore, Mariangela;
    • de Candia, Modesto;
    • Altomare, Cosimo D.;
    • Maria, Catarina;
    • Barros, João;
    • Cachatra, Vasco;
    • Calado, Patrícia;
    • Shimizu, Karina;
    • Freitas, Adilson A.;
    • Oliveira, Maria C.;
    • Ferreira, Maria J.;
    • Lopes, José N. C.;
    • Colabufo, Nicola A.;
    • Rauter, Amélia P.
    Publication type:
    Article
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    Design and Synthesis of CNS-targeted Flavones and Analogues with Neuroprotective Potential Against H2O2- and Aβ1-42-Induced Toxicity in SH-SY5Y Human Neuroblastoma Cells.

    Published in:
    Pharmaceuticals (14248247), 2019, v. 12, n. 2, p. 98, doi. 10.3390/ph12020098
    By:
    • de Matos, Ana M.;
    • Martins, Alice;
    • Man, Teresa;
    • Evans, David;
    • Walter, Magnus;
    • Oliveira, Maria Conceição;
    • López, Óscar;
    • Fernandez-Bolaños, José G.;
    • Dätwyler, Philipp;
    • Ernst, Beat;
    • Macedo, M. Paula;
    • Contino, Marialessandra;
    • Colabufo, Nicola A.;
    • Rauter, Amélia P.
    Publication type:
    Article
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    Radiosynthesis and in vivo Evaluation of Carbon-11 (2 S)-3-(1 H-Indol-3-yl)-2-{[(4-methoxyphenyl)carbamoyl]amino}- N-{[1-(5-methoxypyridin-2-yl)cyclohexyl]methyl}propanamide: An Attempt to Visualize Brain Formyl Peptide Receptors in Mouse Models of Neuroinflammation

    Published in:
    Chemistry & Biodiversity, 2016, v. 13, n. 7, p. 875, doi. 10.1002/cbdv.201500281
    By:
    • Lacivita, Enza;
    • Stama, Madia Letizia;
    • Maeda, Jun;
    • Fujinaga, Masayuki;
    • Hatori, Akiko;
    • Zhang, Ming‐Rong;
    • Colabufo, Nicola A.;
    • Perrone, Roberto;
    • Higuchi, Makoto;
    • Suhara, Tetsuya;
    • Leopoldo, Marcello
    Publication type:
    Article
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    Corrigendum: Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels.

    Published in:
    ChemMedChem, 2022, v. 17, n. 7, p. 1, doi. 10.1002/cmdc.202200131
    By:
    • Milani, Gualtiero;
    • Cavalluzzi, Maria Maddalena;
    • Altamura, Concetta;
    • Santoro, Antonella;
    • Perrone, Mariagrazia;
    • Muraglia, Marilena;
    • Colabufo, Nicola Antonio;
    • Corbo, Filomena;
    • Casalino, Elisabetta;
    • Franchini, Carlo;
    • Pisano, Isabella;
    • Desaphy, Jean‐François;
    • Carrieri, Antonio;
    • Carocci, Alessia;
    • Lentini, Giovanni
    Publication type:
    Article
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    Bioisosteric Modification of To042: Synthesis and Evaluation of Promising Use‐Dependent Inhibitors of Voltage‐Gated Sodium Channels.

    Published in:
    ChemMedChem, 2021, v. 16, n. 23, p. 3588, doi. 10.1002/cmdc.202100496
    By:
    • Milani, Gualtiero;
    • Cavalluzzi, Maria Maddalena;
    • Altamura, Concetta;
    • Santoro, Antonella;
    • Perrone, Mariagrazia;
    • Muraglia, Marilena;
    • Colabufo, Nicola Antonio;
    • Corbo, Filomena;
    • Casalino, Elisabetta;
    • Franchini, Carlo;
    • Pisano, Isabella;
    • Desaphy, Jean‐François;
    • Carrieri, Antonio;
    • Carocci, Alessia;
    • Lentini, Giovanni
    Publication type:
    Article