Works matching AU Cilibrizzi, Agostino

Results: 29

Drug Susceptibility, Siderophore Production, and Genome Analysis of Staphylococcus aureus Clinical Isolates from a University Hospital in Chiang Mai, Thailand.

Published in:

Antibiotics (2079-6382), 2025, v. 14, n. 5, p. 521, doi. 10.3390/antibiotics14050521

By:

Prommachote, Warinda;
Deeudom, Manu;
Koonyosying, Pimpisid;
Srichomphoo, Phronpawee;
Somnabut, Ratchanee;
Khamnoi, Phadungkiat;
Cilibrizzi, Agostino;
Ravikumar, Yuvaraj;
Srichairatanakool, Somdet

Publication type:

Article

The synthesis and properties of mitochondrial targeted iron chelators.

Published in:

BioMetals, 2023, v. 36, n. 2, p. 321, doi. 10.1007/s10534-022-00383-8

By:

Cilibrizzi, Agostino;
Pourzand, Charareh;
Abbate, Vincenzo;
Reelfs, Olivier;
Versari, Laura;
Floresta, Giuseppe;
Hider, Robert

Publication type:

Article

Glutathione and the intracellular labile heme pool.

Published in:

BioMetals, 2021, v. 34, n. 2, p. 221, doi. 10.1007/s10534-020-00274-w

By:

O'Keeffe, Rosemary;
Latunde-Dada, Gladys Oluyemisi;
Chen, Yu-Lin;
Kong, Xiaole L.;
Cilibrizzi, Agostino;
Hider, Robert C.

Publication type:

Article

Synthesis, HPLC Enantioresolution, and X-ray Analysis of a New Series of C5-methyl Pyridazines as N-Formyl Peptide Receptor (FPR) Agonists.

Published in:

Chirality, 2013, v. 25, n. 7, p. 400, doi. 10.1002/chir.22162

By:

Cilibrizzi, Agostino;
Crocetti, Letizia;
Paola Giovannoni, Maria;
Graziano, Alessia;
Vergelli, Claudia;
Bartolucci, Gianluca;
Soldani, Giacomo;
Quinn, Mark T.;
Schepetkin, Igor A.;
Faggi, Cristina

Publication type:

Article

Synthesis, biological evaluation, molecular modeling, and structural analysis of new pyrazole and pyrazolone derivatives as N‐formyl peptide receptors agonists.

Published in:

Chemical Biology & Drug Design, 2021, v. 98, n. 4, p. 582, doi. 10.1111/cbdd.13913

By:

Vergelli, Claudia;
Khlebnikov, Andrei I.;
Crocetti, Letizia;
Guerrini, Gabriella;
Cantini, Niccolò;
Kirpotina, Liliya N.;
Schepetkin, Igor A.;
Cilibrizzi, Agostino;
Quinn, Mark T.;
Rossi, Patrizia;
Paoli, Paola;
Giovannoni, Maria Paola

Publication type:

Article

'Main Mechanical Forces‐Chemical Interactions' Interplay as a Tool to Elucidate Folding Mechanisms.

Published in:

Peptide Science, 2024, v. 116, n. 5, p. 1, doi. 10.1002/pep2.24365

By:

Larocca, Michele;
Floresta, Giuseppe;
Verderese, Daniele;
Cilibrizzi, Agostino

Publication type:

Article

Repurposing strategies on pyridazinone-based series by pharmacophore- and structure-driven screening.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1137, doi. 10.1080/14756366.2020.1760261

By:

Floresta, Giuseppe;
Crocetti, Letizia;
Giovannoni, Maria Paola;
Biagini, Pierfrancesco;
Cilibrizzi, Agostino

Publication type:

Article

iVS analysis to evaluate the impact of scaffold diversity in the binding to cellular targets relevant in cancer.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 44, doi. 10.1080/14756366.2018.1518960

By:

Cilibrizzi, Agostino;
Floresta, Giuseppe;
Abbate, Vincenzo;
Giovannoni, Maria Paola

Publication type:

Article

Cinnoline derivatives as human neutrophil elastase inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 4, p. 628, doi. 10.3109/14756366.2015.1057718

By:

Giovannoni, Maria Paola;
Schepetkin, Igor A.;
Crocetti, Letizia;
Ciciani, Giovanna;
Cilibrizzi, Agostino;
Guerrini, Gabriella;
Khlebnikov, Andrei I.;
Quinn, Mark T.;
Vergelli, Claudia

Publication type:

Article

Correspondence: Compound 17b and formyl peptide receptor biased agonism in relation to cardioprotective effects in ischaemia-reperfusion injury.

Published in:

Nature Communications, 2018, v. 9, n. 1, p. 1, doi. 10.1038/s41467-017-02654-2

By:

Cilibrizzi, Agostino

Publication type:

Article

The role of mitochondrial labile iron in Friedreich's ataxia skin fibroblasts sensitivity to ultraviolet A.

Published in:

Metallomics, 2019, v. 11, n. 3, p. 656, doi. 10.1039/c8mt00257f

By:

Reelfs, Olivier;
Abbate, Vincenzo;
Cilibrizzi, Agostino;
Pook, Mark A.;
Hider, Robert C.;
Pourzand, Charareh

Publication type:

Article

Synthesis of Five- and Six-Membered N-Phenylacetamido Substituted Heterocycles as Formyl Peptide Receptor Agonists.

Published in:

Drug Development Research, 2017, v. 78, n. 1, p. 49, doi. 10.1002/ddr.21370

By:

Vergelli, Claudia;
Schepetkin, Igor A.;
Ciciani, Giovanna;
Cilibrizzi, Agostino;
Crocetti, Letizia;
Giovannoni, Maria Paola;
Guerrini, Gabriella;
Iacovone, Antonella;
Kirpotina, Liliya N.;
Ye, Richard D.;
Quinn, Mark T.

Publication type:

Article

Synthesis and Pharmacological Evaluation of New Pyridazin-Based Thioderivatives as Formyl Peptide Receptor ( FPR) Agonists.

Published in:

Drug Development Research, 2013, v. 74, n. 4, p. 259, doi. 10.1002/ddr.21076

By:

Crocetti, Letizia;
Vergelli, Claudia;
Cilibrizzi, Agostino;
Graziano, Alessia;
Khlebnikov, Andrei I.;
Kirpotina, Liliya N.;
Schepetkin, Igor A.;
Quinn, Mark T.;
Giovannoni, Maria Paola

Publication type:

Article

Synthesis and Evaluation as Antitubercular Agents of 5-Arylethenyl and 5-(Hetero)aryl-3-Isoxazolecarboxylate.

Published in:

Drug Development Research, 2013, v. 74, n. 3, p. 162, doi. 10.1002/ddr.21057

By:

Vergelli, Claudia;
Cilibrizzi, Agostino;
Crocetti, Letizia;
Graziano, Alessia;
Dal Piaz, Vittorio;
Wan, Baojie;
Wang, Yuehong;
Franzblau, Scott;
Giovannoni, Maria Paola

Publication type:

Article

Synthesis and evaluation as PDE4 inhibitors of pyrimidine-2,4-dione derivatives.

Published in:

Drug Development Research, 2011, v. 72, n. 3, p. 274, doi. 10.1002/ddr.20395

By:

Giovannoni, Maria P.;
Graziano, Alessia;
Matucci, Rosanna;
Nesi, Marta;
Cesari, Nicoletta;
Vergelli, Claudia;
Biancalani, Claudio;
Crocetti, Letizia;
Cilibrizzi, Agostino;
Dal Piaz, Vittorio

Publication type:

Article

Optimization of 4‐amino‐pyridazin‐3(2H)‐one as a valid core scaffold for FABP4 inhibitors.

Published in:

Archiv der Pharmazie, 2023, v. 356, n. 10, p. 1, doi. 10.1002/ardp.202300314

By:

Floresta, Giuseppe;
Crocetti, Letizia;
Silva, Renan Rodrigues de Oliveira;
Patamia, Vincenzo;
Mazzacuva, Francesca;
Chen, Yu Chee Sonia;
Vergelli, Claudia;
Cilibrizzi, Agostino

Publication type:

Article

Optical Imaging Opportunities to Inspect the Nature of Cytosolic Iron Pools.

Published in:

Molecules, 2023, v. 28, n. 18, p. 6467, doi. 10.3390/molecules28186467

By:

Hider, Robert Charles;
Pourzand, Charareh;
Ma, Yongmin;
Cilibrizzi, Agostino

Publication type:

Article

Steered Molecular Dynamics Simulations Study on FABP4 Inhibitors.

Published in:

Molecules, 2023, v. 28, n. 6, p. 2731, doi. 10.3390/molecules28062731

By:

Tomarchio, Rosario;
Patamia, Vincenzo;
Zagni, Chiara;
Crocetti, Letizia;
Cilibrizzi, Agostino;
Floresta, Giuseppe;
Rescifina, Antonio

Publication type:

Article

An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022.

Published in:

Molecules, 2022, v. 27, n. 15, p. 4964, doi. 10.3390/molecules27154964

By:

Crocetti, Letizia;
Floresta, Giuseppe;
Cilibrizzi, Agostino;
Giovannoni, Maria Paola

Publication type:

Article

Synthesis and analytical characterization of new thiazol-2-( 3H)-ones as human neutrophil elastase (HNE) inhibitors.

Published in:

Chemistry Central Journal, 2017, v. 11, n. 1, p. 1, doi. 10.1186/s13065-017-0358-1

By:

Crocetti, Letizia;
Bartolucci, Gianluca;
Cilibrizzi, Agostino;
Giovannoni, Maria;
Guerrini, Gabriella;
Iacovone, Antonella;
Menicatti, Marta;
Schepetkin, Igor;
Khlebnikov, Andrei;
Quinn, Mark;
Vergelli, Claudia

Publication type:

Article

Ligand Growing Experiments Suggested 4-amino and 4-ureido pyridazin-3(2 H)-one as Novel Scaffold for FABP4 Inhibition.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 11, p. 1335, doi. 10.3390/ph15111335

By:

Crocetti, Letizia;
Floresta, Giuseppe;
Zagni, Chiara;
Merugu, Divya;
Mazzacuva, Francesca;
de Oliveira Silva, Renan Rodrigues;
Vergelli, Claudia;
Giovannoni, Maria Paola;
Cilibrizzi, Agostino

Publication type:

Article

Pharmacokinetics of Mephedrone Enantiomers in Whole Blood after a Controlled Intranasal Administration to Healthy Human Volunteers.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 1, p. 5, doi. 10.3390/ph14010005

By:

Czerwinska, Joanna;
Parkin, Mark C.;
Cilibrizzi, Agostino;
George, Claire;
Kicman, Andrew T.;
Dargan, Paul I.;
Abbate, Vincenzo

Publication type:

Article

Dominant Chemical Interactions Governing the Folding Mechanism of Oligopeptides.

Published in:

International Journal of Molecular Sciences, 2024, v. 25, n. 17, p. 9586, doi. 10.3390/ijms25179586

By:

Larocca, Michele;
Floresta, Giuseppe;
Verderese, Daniele;
Cilibrizzi, Agostino

Publication type:

Article

PDE4 Inhibitors: Profiling Hits through the Multitude of Structural Classes.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 14, p. 11518, doi. 10.3390/ijms241411518

By:

Jin, Jian;
Mazzacuva, Francesca;
Crocetti, Letizia;
Giovannoni, Maria Paola;
Cilibrizzi, Agostino

Publication type:

Article

The Colorimetric Detection of the Hydroxyl Radical.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 4162, doi. 10.3390/ijms24044162

By:

Ran, Yandong;
Moursy, Mohammed;
Hider, Robert C.;
Cilibrizzi, Agostino

Publication type:

Article

Solid-Phase Synthesis and In-Silico Analysis of Iron-Binding Catecholato Chelators.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 20, p. 7498, doi. 10.3390/ijms21207498

By:

Gacesa, Ranko;
Tripodi, Andrea A. P.;
Cilibrizzi, Agostino;
Leggio, Antonella;
Hider, Robert;
Abbate, Vincenzo

Publication type:

Article

New Pyrazolo[1',5':1,6]pyrimido[4,5-d]pyridazin-4 (3H)-ones Fluoroderivatives as Human A<sub>1</sub> Adenosine Receptor Ligands.

Published in:

Acta Chimica Slovenica, 2012, v. 59, n. 3, p. 648

By:

Graziano, Alessia;
Giovannoni, Maria Paola;
Cilibrizzi, Agostino;
Crocetti, Letizia;
Piaz, Vittorio Dal;
Vergelli, Claudia;
Trincavelli, Maria Letizia;
Martini, Claudia;
Giacomelli, Chiara

Publication type:

Article

Synthesis and Evaluation of Novel Pyrrolo[2,3-d] and Thieno[2,3-d]Pyridazinones as in Vitro Antiproliferative Agents.

Published in:

Acta Chimica Slovenica, 2009, v. 56, n. 3, p. 571

By:

Dal Piaz, Vittorio;
Vergelli, Claudia;
Giovannoni, Maria Paola;
Biancalani, Claudio;
Cilibrizzi, Agostino;
Graziano, Alessia;
Cesari, Nicoletta

Publication type:

Article

Analytical characterization of three cathinone derivatives, 4-MPD, 4F-PHP and bk-EPDP, purchased as bulk powder from online vendors.

Published in:

Drug Testing & Analysis, 2018, v. 10, n. 2, p. 372, doi. 10.1002/dta.2218

By:

Apirakkan, Orapan;
Frinculescu, Anca;
Shine, Trevor;
Parkin, Mark C.;
Cilibrizzi, Agostino;
Frascione, Nunzianda;
Abbate, Vincenzo

Publication type:

Article