Works by Christodoulou, Michael S.

Results: 36

Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus.

Published in:

Frontiers in Pharmacology, 2025, p. 1, doi. 10.3389/fphar.2025.1549288

By:

Molina Panadero, Irene;
Falcón Torres, Javier;
Hmadcha, Abdelkrim;
Princiotto, Salvatore;
Cutarella, Luigi;
Mori, Mattia;
Dallavalle, Sabrina;
Christodoulou, Michael S.;
Smani, Younes

Publication type:

Article

Antioxidant-mediated suppression of ferroptosis in Pyricularia oryzae : a novel approach to rice blast management for sustainable rice production.

Published in:

2025

By:

Santoni, Mattia;
Molina-Hernandez, Junior Bernardo;
Kunova, Andrea;
Cortesi, Paolo;
Brunetti, Barbara;
Rocculi, Pietro;
Christodoulou, Michael S.;
Danesi, Francesca

Publication type:

Literature Review

Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-45851-6

By:

Pinzi, Luca;
Conze, Christian;
Bisi, Nicolo;
Torre, Gabriele Dalla;
Soliman, Ahmed;
Monteiro-Abreu, Nanci;
Trushina, Nataliya I.;
Krusenbaum, Andrea;
Dolouei, Maryam Khodaei;
Hellwig, Andrea;
Christodoulou, Michael S.;
Passarella, Daniele;
Bakota, Lidia;
Rastelli, Giulio;
Brandt, Roland

Publication type:

Article

Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-45851-6

By:

Pinzi, Luca;
Conze, Christian;
Bisi, Nicolo;
Torre, Gabriele Dalla;
Soliman, Ahmed;
Monteiro-Abreu, Nanci;
Trushina, Nataliya I.;
Krusenbaum, Andrea;
Dolouei, Maryam Khodaei;
Hellwig, Andrea;
Christodoulou, Michael S.;
Passarella, Daniele;
Bakota, Lidia;
Rastelli, Giulio;
Brandt, Roland

Publication type:

Article

Antiproliferative effects of chalcones on T cell acute lymphoblastic leukemia‐derived cells: Role of PKCβ.

Published in:

Archiv der Pharmazie, 2020, v. 353, n. 7, p. 1, doi. 10.1002/ardp.202000062

By:

Corsini, Emanuela;
Facchetti, Giorgio;
Esposito, Sara;
Maddalon, Ambra;
Rimoldi, Isabella;
Christodoulou, Michael S.

Publication type:

Article

Biological Properties of New Chiral 2-Methyl-5,6,7,8-tetrahydroquinolin-8-amine-based Compounds.

Published in:

Molecules, 2020, v. 25, n. 23, p. 5561, doi. 10.3390/molecules25235561

By:

Facchetti, Giorgio;
Christodoulou, Michael S.;
Mendoza, Lina Barragán;
Cusinato, Federico;
Dalla Via, Lisa;
Rimoldi, Isabella;
Jampilek, Josef;
Musioł, Robert

Publication type:

Article

Vancomycin-Iridium (III) Interaction: An Unexplored Route for Enantioselective Imine Reduction.

Published in:

Molecules, 2019, v. 24, n. 15, p. 2771, doi. 10.3390/molecules24152771

By:

Facchetti, Giorgio;
Pellegrino, Sara;
Bucci, Raffaella;
Nava, Donatella;
Gandolfi, Raffaella;
Christodoulou, Michael S.;
Rimoldi, Isabella

Publication type:

Article

Chiral Flavanones from Amygdalus lycioides Spach: Structural Elucidation and Identification of TNFalpha Inhibitors by Bioactivity-guided Fractionation.

Published in:

Molecules, 2012, v. 17, n. 2, p. 1665, doi. 10.3390/molecules17021665

By:

Gaggeri, Raffaella;
Rossi, Daniela;
Christodoulou, Michael S.;
Passarella, Daniele;
Leoni, Flavio;
Azzolina, Ornella;
Collina, Simona

Publication type:

Article

A small library of chalcones induce liver cancer cell death through Akt phosphorylation inhibition.

Published in:

Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-68775-9

By:

Sahin, Irem Durmaz;
Christodoulou, Michael S.;
Guzelcan, Ece Akhan;
Koyas, Altay;
Karaca, Cigdem;
Passarella, Daniele;
Cetin-Atalay, Rengul

Publication type:

Article

Engineered Ferritin Nanoparticles for the Bioluminescence Tracking of Nanodrug Delivery in Cancer.

Published in:

Small, 2020, v. 16, n. 39, p. 1, doi. 10.1002/smll.202001450

By:

Bellini, Michela;
Riva, Benedetta;
Tinelli, Veronica;
Rizzuto, Maria Antonietta;
Salvioni, Lucia;
Colombo, Miriam;
Mingozzi, Francesca;
Visioli, Alberto;
Marongiu, Laura;
Frascotti, Gianni;
Christodoulou, Michael S.;
Passarella, Daniele;
Prosperi, Davide;
Fiandra, Luisa

Publication type:

Article

Divergent Palladium‐ and Platinum‐Catalyzed Intramolecular Hydroamination/Hydroarylation of O‐Propargyl‐2‐aminophenols.

Published in:

European Journal of Organic Chemistry, 2018, v. 2018, n. 44, p. 6176, doi. 10.1002/ejoc.201801103

By:

Christodoulou, Michael S.;
Giofrè, Sabrina;
Broggini, Gianluigi;
Mazza, Alberto;
Sala, Roberto;
Beccalli, Egle M.

Publication type:

Article

Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders.

Published in:

European Journal of Organic Chemistry, 2016, v. 2016, n. 11, p. 2029, doi. 10.1002/ejoc.201600130

By:

Marucci, Cristina;
Christodoulou, Michael S.;
Pieraccini, Stefano;
Sironi, Maurizio;
Dapiaggi, Federico;
Cartelli, Daniele;
Calogero, Alessandra M.;
Cappelletti, Graziella;
Vilanova, Concepción;
Gazzola, Silvia;
Broggini, Gianluigi;
Passarella, Daniele

Publication type:

Article

Cover Feature: 2‐Phenyloxazole‐4‐carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B (ChemMedChem 18/2019).

Published in:

ChemMedChem, 2019, v. 14, n. 18, p. 1619, doi. 10.1002/cmdc.201900504

By:

Di Paolo, Maria L.;
Christodoulou, Michael S.;
Calogero, Alessandra M.;
Pinzi, Luca;
Rastelli, Giulio;
Passarella, Daniele;
Cappelletti, Graziella;
Dalla Via, Lisa

Publication type:

Article

2‐Phenyloxazole‐4‐carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B.

Published in:

ChemMedChem, 2019, v. 14, n. 18, p. 1641, doi. 10.1002/cmdc.201900261

By:

Di Paolo, Maria L.;
Christodoulou, Michael S.;
Calogero, Alessandra M.;
Pinzi, Luca;
Rastelli, Giulio;
Passarella, Daniele;
Cappelletti, Graziella;
Dalla Via, Lisa

Publication type:

Article

Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR.

Published in:

ChemMedChem, 2018, v. 13, n. 24, p. 2627, doi. 10.1002/cmdc.201800687

By:

Carlino, Luca;
Christodoulou, Michael S.;
Restelli, Valentina;
Caporuscio, Fabiana;
Foschi, Francesca;
Semrau, Marta S.;
Costanzi, Elisa;
Tinivella, Annachiara;
Pinzi, Luca;
Lo Presti, Leonardo;
Battistutta, Roberto;
Storici, Paola;
Broggini, Massimo;
Passarella, Daniele;
Rastelli, Giulio

Publication type:

Article

Correlation between Perturbation of Redox Homeostasis and Antibiofilm Capacity of Phytochemicals at Non-Lethal Concentrations.

Published in:

Antioxidants, 2022, v. 11, n. 12, p. 2451, doi. 10.3390/antiox11122451

By:

Christodoulou, Michael S.;
Villa, Federica;
Pinto, Andrea;
Cappitelli, Francesca

Publication type:

Article

Cascade Reaction by Chemo‐ and Biocatalytic Approaches to Obtain Chiral Hydroxy Ketones and anti 1,3‐Diols.

Published in:

ChemistryOpen, 2018, v. 7, n. 5, p. 393, doi. 10.1002/open.201800056

By:

Gandolfi, Raffaella;
Facchetti, Giorgio;
Christodoulou, Michael S.;
Fusè, Marco;
Meneghetti, Fiorella;
Rimoldi, Isabella

Publication type:

Article

Ruthenium‐Catalyzed Decarboxylative Rearrangement of 4‐Alkenyl‐isoxazol‐5‐ones to Pyrrole Derivatives.

Published in:

European Journal of Organic Chemistry, 2022, v. 2022, n. 25, p. 1, doi. 10.1002/ejoc.202200496

By:

Molteni, Letizia;
Loro, Camilla;
Christodoulou, Michael S.;
Papis, Marta;
Foschi, Francesca;
Beccalli, Egle M.;
Broggini, Gianluigi

Publication type:

Article

Probing an Allosteric Pocket of CDK2 with Small Molecules.

Published in:

ChemMedChem, 2017, v. 12, n. 1, p. 33, doi. 10.1002/cmdc.201600474

By:

Christodoulou, Michael S.;
Caporuscio, Fabiana;
Restelli, Valentina;
Carlino, Luca;
Cannazza, Giuseppe;
Costanzi, Elisa;
Citti, Cinzia;
Lo Presti, Leonardo;
Pisani, Pasquale;
Battistutta, Roberto;
Broggini, Massimo;
Passarella, Daniele;
Rastelli, Giulio

Publication type:

Article

Inside Cover: Probing an Allosteric Pocket of CDK2 with Small Molecules (ChemMedChem 1/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 1, p. 2, doi. 10.1002/cmdc.201600623

By:

Christodoulou, Michael S.;
Caporuscio, Fabiana;
Restelli, Valentina;
Carlino, Luca;
Cannazza, Giuseppe;
Costanzi, Elisa;
Citti, Cinzia;
Lo Presti, Leonardo;
Pisani, Pasquale;
Battistutta, Roberto;
Broggini, Massimo;
Passarella, Daniele;
Rastelli, Giulio

Publication type:

Article

Camptothecin-7-yl-methanthiole: Semisynthesis and Biological Evaluation.

Published in:

ChemMedChem, 2012, v. 7, n. 12, p. 2134, doi. 10.1002/cmdc.201200322

By:

Christodoulou, Michael S.;
Zunino, Franco;
Zuco, Valentina;
Borrelli, Stella;
Comi, Daniela;
Fontana, Gabriele;
Martinelli, Marisa;
Lorens, James B.;
Evensen, Lasse;
Sironi, Maurizio;
Pieraccini, Stefano;
Dalla Via, Lisa;
Gia, Ornella Maria;
Passarella, Daniele

Publication type:

Article

Exploration of Novel Scaffolds Targeting Cytochrome b of Pyricularia oryzae.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 3, p. 2705, doi. 10.3390/ijms24032705

By:

Pinna, Cecilia;
Laurenzi, Tommaso;
Forlani, Fabio;
Palazzolo, Luca;
Nolan, Claire Beatrice;
Christodoulou, Michael S.;
Cortesi, Paolo;
Pinto, Andrea;
Eberini, Ivano;
Kunova, Andrea;
Dallavalle, Sabrina

Publication type:

Article

Enzymatic Kinetic Resolution of 2-Piperidineethanol for the Enantioselective Targeted and Diversity Oriented Synthesis.

Published in:

International Journal of Molecular Sciences, 2016, v. 17, n. 1, p. 17, doi. 10.3390/ijms17010017

By:

Perdicchia, Dario;
Christodoulou, Michael S.;
Fumagalli, Gaia;
Calogero, Francesco;
Marucci, Cristina;
Passarella, Daniele

Publication type:

Article

Nanolipid-Trehalose Conjugates and Nano-Assemblies as Putative Autophagy Inducers.

Published in:

Pharmaceutics, 2019, v. 11, n. 8, p. 422, doi. 10.3390/pharmaceutics11080422

By:

Colombo, Eleonora;
Biocotino, Michele;
Frapporti, Giulia;
Randazzo, Pietro;
Christodoulou, Michael S.;
Piccoli, Giovanni;
Polito, Laura;
Seneci, Pierfausto;
Passarella, Daniele

Publication type:

Article

Targeting Ovarian Cancer with Chalcone Derivatives: Cytotoxicity and Apoptosis Induction in HGSOC Cells.

Published in:

Molecules, 2023, v. 28, n. 23, p. 7777, doi. 10.3390/molecules28237777

By:

Merve Aydin, Elif;
Canıtez, İdil Su;
Colombo, Eleonora;
Princiotto, Salvatore;
Passarella, Daniele;
Dallavalle, Sabrina;
Christodoulou, Michael S.;
Durmaz Şahin, Irem

Publication type:

Article

Design and Synthesis of Hsp90 Inhibitors with B‐Raf and PDHK1 Multi‐Target Activity.

Published in:

ChemistryOpen, 2021, v. 10, n. 12, p. 1177, doi. 10.1002/open.202100131

By:

Pinzi, Luca;
Foschi, Francesca;
Christodoulou, Michael S.;
Passarella, Daniele;
Rastelli, Giulio

Publication type:

Article

Asymmetric Hydrogenation of 1-aryl substituted-3,4-Dihydroisoquinolines with Iridium Catalysts Bearing Different Phosphorus-Based Ligands.

Published in:

Catalysts (2073-4344), 2020, v. 10, n. 8, p. 914, doi. 10.3390/catal10080914

By:

Facchetti, Giorgio;
Christodoulou, Michael S.;
Binda, Eleonora;
Fusè, Marco;
Rimoldi, Isabella

Publication type:

Article

Palladium-Catalyzed Benzodiazepines Synthesis.

Published in:

Catalysts (2073-4344), 2020, v. 10, n. 6, p. 634, doi. 10.3390/catal10060634

By:

Christodoulou, Michael S.;
Beccalli, Egle M.;
Giofrè, Sabrina

Publication type:

Article

Synthesis of Thicolchicine‐Based Conjugates: Investigation towards Bivalent Tubulin/Microtubules Binders.

Published in:

ChemPlusChem, 2019, v. 84, n. 1, p. 98, doi. 10.1002/cplu.201800497

By:

Bonandi, Elisa;
Foschi, Francesca;
Marucci, Cristina;
Dapiaggi, Federico;
Sironi, Maurizio;
Pieraccini, Stefano;
Christodoulou, Michael S.;
de Asís Balaguer, Francisco;
Díaz, J. Fernando;
Zidar, Nace;
Passarella, Daniele

Publication type:

Article

Cyclopamine-Paclitaxel-Containing Nanoparticles: Internalization in Cells Detected by Confocal and Super-Resolution Microscopy.

Published in:

ChemPlusChem, 2015, v. 80, n. 9, p. 1380, doi. 10.1002/cplu.201500156

By:

Fumagalli, Gaia;
Mazza, Davide;
Christodoulou, Michael S.;
Damia, Giovanna;
Ricci, Francesca;
Perdicchia, Dario;
Stella, Barbara;
Dosio, Franco;
Sotiropoulou, Panagiota A.;
Passarella, Daniele

Publication type:

Article

Click Reaction as a Tool to Combine Pharmacophores: The Case of Vismodegib.

Published in:

ChemPlusChem, 2015, v. 80, n. 6, p. 938, doi. 10.1002/cplu.201402435

By:

Christodoulou, Michael S.;
Mori, Mattia;
Pantano, Rebecca;
Alfonsi, Romina;
Infante, Paola;
Botta, Maurizio;
Damia, Giovanna;
Ricci, Francesca;
Sotiropoulou, Panagiota A.;
Liekens, Sandra;
Botta, Bruno;
Passarella, Daniele

Publication type:

Article

Self-Assembled Squalene-based Fluorescent Heteronanoparticles.

Published in:

ChemPlusChem, 2015, v. 80, n. 1, p. 47, doi. 10.1002/cplu.201402239

By:

Borrelli, Stella;
Cartelli, Daniele;
Secundo, Francesco;
Fumagalli, Gaia;
Christodoulou, Michael S.;
Borroni, Ambra;
Perdicchia, Dario;
Dosio, Franco;
Milla, Paola;
Cappelletti, Graziella;
Passarella, Daniele

Publication type:

Article

9-Fluorenone-2-Carboxylic Acid as a Scaffold for Tubulin Interacting Compounds.

Published in:

ChemPlusChem, 2013, v. 78, n. 7, p. 663, doi. 10.1002/cplu.201300036

By:

Calogero, Francesco;
Borrelli, Stella;
Speciale, Gaetano;
Christodoulou, Michael S.;
Cartelli, Daniele;
Ballinari, Dario;
Sola, Francesco;
Albanese, Clara;
Ciavolella, Antonella;
Passarella, Daniele;
Cappelletti, Graziella;
Pieraccini, Stefano;
Sironi, Maurizio

Publication type:

Article

Preparation of Fluorescent Tubulin Binders.

Published in:

ChemPlusChem, 2013, v. 78, n. 3, p. 222, doi. 10.1002/cplu.201200260

By:

Riva, Elena;
Mattarella, Martin;
Borrelli, Stella;
Christodoulou, Michael S.;
Cartelli, Daniele;
Main, Marcus;
Faulkner, Stephen;
Sykes, Daniel;
Cappelletti, Graziella;
Snaith, John S.;
Passarella, Daniele

Publication type:

Article

Preparation of Fluorescent Tubulin Binders.

Published in:

2013

By:

Riva, Elena;
Mattarella, Martin;
Borrelli, Stella;
Christodoulou, Michael S.;
Cartelli, Daniele;
Main, Marcus;
Faulkner, Stephen;
Sykes, Daniel;
Cappelletti, Graziella;
Snaith, John S.;
Passarella, Daniele

Publication type:

Other

Cover Picture: Preparation of Fluorescent Tubulin Binders (ChemPlusChem 3/2013).

Published in:

ChemPlusChem, 2013, v. 78, n. 3, p. 201, doi. 10.1002/cplu.201390010

By:

Riva, Elena;
Mattarella, Martin;
Borrelli, Stella;
Christodoulou, Michael S.;
Cartelli, Daniele;
Main, Marcus;
Faulkner, Stephen;
Sykes, Daniel;
Cappelletti, Graziella;
Snaith, John S.;
Passarella, Daniele

Publication type:

Article