Works by Ceruso, Mariangela

Results: 14

Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity.

Published in:

ChemBioChem, 2017, v. 18, n. 2, p. 213, doi. 10.1002/cbic.201600513

By:

Bhatt, Avni;
Mahon, Brian P.;
Cruzeiro, Vinicius Wilian D.;
Cornelio, Benedetta;
Laronze‐Cochard, Marie;
Ceruso, Mariangela;
Sapi, Janos;
Rance, Graham A.;
Khlobystov, Andrei N.;
Fontana, Antonella;
Roitberg, Adrian;
Supuran, Claudiu T.;
McKenna, Robert

Publication type:

Article

Real-world Treatment Sequencing and Outcomes With Cabozantinib After First-line Immune Checkpoint Inhibitor-based Combination Therapy For Patients With Advanced Renal Cell Carcinoma: CARINA Study Results.

Published in:

Clinical Genitourinary Cancer, 2024, v. 22, n. 5, p. N.PAG, doi. 10.1016/j.clgc.2024.102141

By:

Nathan, Paul;
Venugopal, Balaji;
Ali, Jamshed;
Allison, Jennifer;
Ceruso, Mariangela;
Charnley, Natalie;
Griffiths, Richard;
Michael, Agnieszka;
Moore, Kathryn;
Perrot, Valérie;
Prendergast, Áine;
Sharma, Anand;
Szabados, Bernadett;
Larkin, James

Publication type:

Article

Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 7, p. 2621, doi. 10.3390/ijms21072621

By:

Hargunani, Priya;
Tadge, Nikhil;
Ceruso, Mariangela;
Leitans, Janis;
Kazaks, Andris;
Tars, Kaspars;
Gratteri, Paola;
Supuran, Claudiu T.;
Nocentini, Alessio;
Toraskar, Mrunmayee P.

Publication type:

Article

Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 255, doi. 10.1080/14756366.2017.1413097

By:

Monti, Simona Maria;
Meccariello, Angela;
Ceruso, Mariangela;
Szafrański, Krzysztof;
Sławiński, Jarosław;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 798, doi. 10.1080/14756366.2017.1327522

By:

De Vita, Daniela;
Angeli, Andrea;
Pandolfi, Fabiana;
Bortolami, Martina;
Costi, Roberta;
Di Santo, Roberto;
Suffredini, Elisabetta;
Ceruso, Mariangela;
Del Prete, Sonia;
Capasso, Clemente;
Scipione, Luigi;
Supuran, Claudiu T.

Publication type:

Article

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 51, doi. 10.1080/14756366.2016.1235040

By:

D'Ascenzio, Melissa;
Guglielmi, Paolo;
Carradori, Simone;
Secci, Daniela;
Florio, Rosalba;
Mollica, Adriano;
Ceruso, Mariangela;
Akdemir, Atilla;
Sobolev, Anatoly P.;
Supuran, Claudiu T.

Publication type:

Article

Overexpression of the transmembrane carbonic anhydrase isoforms IX and XII in the inflamed synovium.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 60, doi. 10.1080/14756366.2016.1217857

By:

Margheri, Francesca;
Ceruso, Mariangela;
Carta, Fabrizio;
Laurenzana, Anna;
Maggi, Laura;
Lazzeri, Simone;
Simonini, Gabriele;
Annunziato, Francesco;
Del Rosso, Mario;
Supuran, Claudiu T.;
Cimaz, Rolando

Publication type:

Article

7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1226, doi. 10.3109/14756366.2015.1115401

By:

Nocentini, Alessio;
Ceruso, Mariangela;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and inhibition potency of novel ureido benzenesulfonamides incorporating GABA as tumor-associated carbonic anhydrase IX and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 2, p. 205, doi. 10.3109/14756366.2015.1014477

By:

Ceruso, Mariangela;
Antel, Sabrina;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 6, p. 901, doi. 10.3109/14756366.2014.986118

By:

Singasane, Namrata;
Kharkar, Prashant S.;
Ceruso, Mariangela;
Supuran, Claudiu T.;
Toraskar, Mrunmayee P.

Publication type:

Article

Inhibition studies of quinazoline-sulfonamide derivatives against the γ-CA (PgiCA) from the pathogenic bacterium, Porphyromonas gingivalis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 592, doi. 10.3109/14756366.2014.957202

By:

Alafeefy, Ahmed M.;
Ceruso, Mariangela;
Al-Tamimi, Abdul-Malek S.;
Prete, Sonia Del;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

A new class of quinazoline-sulfonamides acting as efficient inhibitors against the α-carbonic anhydrase from Trypanosoma cruzi.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 4, p. 581, doi. 10.3109/14756366.2014.956309

By:

Alafeefy, Ahmed M.;
Ceruso, Mariangela;
Al-Jaber, Nabila A.;
Parkkila, Seppo;
Vermelho, Alane Beatriz;
Supuran, Claudiu T.

Publication type:

Article

New series of sulfonamides containing amino acid moiety act as effective and selective inhibitors of tumor-associated carbonic anhydrase XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 3, p. 430, doi. 10.3109/14756366.2014.942659

By:

Ceruso, Mariangela;
Bragagni, Marco;
AlOthman, Zeid;
Osman, Sameh M.;
Supuran, Claudiu T.

Publication type:

Article

Sulfonamides incorporating fluorine and 1,3,5-triazine moieties are effective inhibitors of three β-class carbonic anhydrases from Mycobacterium tuberculosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 5, p. 686, doi. 10.3109/14756366.2013.842233

By:

Ceruso, Mariangela;
Vullo, Daniela;
Scozzafava, Andrea;
Supuran, Claudiu T.

Publication type:

Article