Works by Cerecetto, Hugo


Results: 63
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    Novel and Selective Rhipicephalus microplus Triosephosphate Isomerase Inhibitors with Acaricidal Activity.

    Published in:
    Veterinary Sciences, 2018, v. 5, n. 3, p. 1, doi. 10.3390/vetsci5030074
    By:
    • Saramago, Luiz;
    • Gomes, Helga;
    • Aguilera, Elena;
    • Cerecetto, Hugo;
    • González, Mercedes;
    • Cabrera, Mauricio;
    • Alzugaray, Maria Fernanda;
    • da Silva Vaz Junior, Itabajara;
    • da Fonseca, Rodrigo Nunes;
    • Aguirre-López, Beatriz;
    • Cabrera, Nallely;
    • Pérez-Montfort, Ruy;
    • Merlino, Alicia;
    • Moraes, Jorge;
    • Álvarez, Guzmán
    Publication type:
    Article
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    Sunitinib-Containing Carborane Pharmacophore with the Ability to Inhibit Tyrosine Kinases Receptors FLT3, KIT and PDGFR-β, Exhibits Powerful In Vivo Anti-Glioblastoma Activity.

    Published in:
    Cancers, 2020, v. 12, n. 11, p. 3423, doi. 10.3390/cancers12113423
    By:
    • Alamón, Catalina;
    • Dávila, Belén;
    • García, María Fernanda;
    • Sánchez, Carina;
    • Kovacs, Mariángeles;
    • Trias, Emiliano;
    • Barbeito, Luis;
    • Gabay, Martín;
    • Zeineh, Nidal;
    • Gavish, Moshe;
    • Teixidor, Francesc;
    • Viñas, Clara;
    • Couto, Marcos;
    • Cerecetto, Hugo
    Publication type:
    Article
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    Potent and Selective Inhibitors of Trypanosoma cruzi Triosephosphate Isomerase with Concomitant Inhibition of Cruzipain: Inhibition of Parasite Growth through Multitarget Activity.

    Published in:
    ChemMedChem, 2016, v. 11, n. 12, p. 1328, doi. 10.1002/cmdc.201500385
    By:
    • Aguilera, Elena;
    • Varela, Javier;
    • Birriel, Estefanía;
    • Serna, Elva;
    • Torres, Susana;
    • Yaluff, Gloria;
    • de Bilbao, Ninfa Vera;
    • Aguirre‐López, Beatriz;
    • Cabrera, Nallely;
    • Díaz Mazariegos, Selma;
    • de Gómez‐Puyou, Marieta Tuena;
    • Gómez‐Puyou, Armando;
    • Pérez‐Montfort, Ruy;
    • Minini, Lucia;
    • Merlino, Alicia;
    • Cerecetto, Hugo;
    • González, Mercedes;
    • Alvarez, Guzmán
    Publication type:
    Article
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    Back Cover: Potent and Selective Inhibitors of Trypanosoma cruzi Triosephosphate Isomerase with Concomitant Inhibition of Cruzipain: Inhibition of Parasite Growth through Multitarget Activity (ChemMedChem 12/2016).

    Published in:
    ChemMedChem, 2016, v. 11, n. 12, p. 1395, doi. 10.1002/cmdc.201600287
    By:
    • Aguilera, Elena;
    • Varela, Javier;
    • Birriel, Estefanía;
    • Serna, Elva;
    • Torres, Susana;
    • Yaluff, Gloria;
    • de Bilbao, Ninfa Vera;
    • Aguirre‐López, Beatriz;
    • Cabrera, Nallely;
    • Díaz Mazariegos, Selma;
    • de Gómez‐Puyou, Marieta Tuena;
    • Gómez‐Puyou, Armando;
    • Pérez‐Montfort, Ruy;
    • Minini, Lucia;
    • Merlino, Alicia;
    • Cerecetto, Hugo;
    • González, Mercedes;
    • Alvarez, Guzmán
    Publication type:
    Article
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    Morphological evidence of the protective effects of a synthetic chalcone against the striatal myelin damage induced by glutaric acid.

    Published in:
    International Journal of Developmental Neuroscience, 2023, v. 83, n. 3, p. 274, doi. 10.1002/jdn.10256
    By:
    • Casanova, Gabriela;
    • Rosillo, Juan Carlos;
    • Jiménez, Marcie;
    • Fernández, Anabel;
    • Rodao, Magela;
    • Martínez, Gaby;
    • Isasi, Eugenia;
    • Presa Gau, Nadia;
    • Otero, Gabriel;
    • Cabrera, Mauricio;
    • Díaz‐Amarilla, Pablo;
    • Cerecetto, Hugo;
    • González, Mercedes;
    • Olivera‐Bravo, Silvia
    Publication type:
    Article
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    Novel coumarins active against Trypanosoma cruzi and toxicity assessment using the animal model Caenorhabditis elegans.

    Published in:
    BMC Pharmacology & Toxicology, 2019, v. 20, p. 1, doi. 10.1186/s40360-019-0357-z
    By:
    • Soares, Fabiana Gomes Nascimento;
    • Göethel, Gabriela;
    • Kagami, Luciano Porto;
    • das Neves, Gustavo Machado;
    • Sauer, Elisa;
    • Birriel, Estefania;
    • Varela, Javier;
    • Gonçalves, Itamar Luís;
    • Von Poser, Gilsane;
    • González, Mercedes;
    • Kawano, Daniel Fábio;
    • Paula, Fávero Reisdorfer;
    • de Melo, Eduardo Borges;
    • Garcia, Solange Cristina;
    • Cerecetto, Hugo;
    • Eifler-Lima, Vera Lucia
    Publication type:
    Article
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    Potent in vitro anti- Trypanosoma cruzi activity of pyridine-2-thiol N-oxide metal complexes having an inhibitory effect on parasite-specific fumarate reductase.

    Published in:
    Journal of Biological Inorganic Chemistry (JBIC), 2008, v. 13, n. 5, p. 723, doi. 10.1007/s00775-008-0358-7
    By:
    • Vieites, Marisol;
    • Smircich, Pablo;
    • Parajón-Costa, Beatriz;
    • Rodríguez, Jorge;
    • Galaz, Verónica;
    • Olea-Azar, Claudio;
    • Otero, Lucía;
    • Aguirre, Gabriela;
    • Cerecetto, Hugo;
    • González, Mercedes;
    • Gómez-Barrio, Alicia;
    • Garat, Beatriz;
    • Gambino, Dinorah
    Publication type:
    Article
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    Preclinical Studies and Drug Combination of Low-Cost Molecules for Chagas Disease.

    Published in:
    Pharmaceuticals (14248247), 2023, v. 16, n. 1, p. 20, doi. 10.3390/ph16010020
    By:
    • Aguilera, Elena;
    • Sánchez, Carina;
    • Cruces, María Eugenia;
    • Dávila, Belén;
    • Minini, Lucía;
    • Mosquillo, Florencia;
    • Pérez-Díaz, Leticia;
    • Serna, Elva;
    • Torres, Susana;
    • Schini, Alicia;
    • Sanabria, Luis;
    • Vera de Bilbao, Ninfa I.;
    • Yaluff, Gloria;
    • Zolessi, Flavio R.;
    • Ceilas, Luis Fabian;
    • Cerecetto, Hugo;
    • Alvarez, Guzmán
    Publication type:
    Article
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    Cover Feature: Discovery of Potent EGFR Inhibitors through the Incorporation of a 3D‐Aromatic‐Boron‐Rich‐Cluster into the 4‐Anilinoquinazoline Scaffold: Potential Drugs for Glioma Treatment (Chem. Eur. J. 13/2018).

    Published in:
    Chemistry - A European Journal, 2018, v. 24, n. 13, p. 3071, doi. 10.1002/chem.201706010
    By:
    • Alamón, Catalina;
    • Couto, Marcos;
    • Cerecetto, Hugo;
    • Teixidor, Francesc;
    • Viñas, Clara;
    • García, María Fernanda;
    • Cabral, Pablo;
    • Cabrera, Mauricio;
    • Merlino, Alicia
    Publication type:
    Article
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