Works by Cadelis, Melissa M.

Results: 23

Structure–Activity Relationship Studies of Indolglyoxyl-Polyamine Conjugates as Antimicrobials and Antibiotic Potentiators.

Published in:

Pharmaceuticals (14248247), 2023, v. 16, n. 6, p. 823, doi. 10.3390/ph16060823

By:

Cadelis, Melissa M.;
Liu, Tim;
Sue, Kenneth;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Synthesis and Antibacterial Activity of Alkylamine-Linked Pleuromutilin Derivatives.

Published in:

Antibiotics (2079-6382), 2024, v. 13, n. 11, p. 1018, doi. 10.3390/antibiotics13111018

By:

Hainsworth, Kerrin;
Cadelis, Melissa M.;
Rouvier, Florent;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Investigation of Naphthyl–Polyamine Conjugates as Antimicrobials and Antibiotic Enhancers.

Published in:

Antibiotics (2079-6382), 2023, v. 12, n. 6, p. 1014, doi. 10.3390/antibiotics12061014

By:

Cadelis, Melissa M.;
Edmeades, Liam R.;
Chen, Dan;
Gill, Evangelene S.;
Fraser, Kyle;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Investigation of α,ω-Disubstituted Polyamine-Cholic Acid Conjugates Identifies Hyodeoxycholic and Chenodeoxycholic Scaffolds as Non-Toxic, Potent Antimicrobials.

Published in:

Antibiotics (2079-6382), 2023, v. 12, n. 2, p. 404, doi. 10.3390/antibiotics12020404

By:

Sue, Kenneth;
Cadelis, Melissa M.;
Troia, Thomas;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Discovery and Preliminary Structure-Activity Investigation of 3-Substituted-1 H -imidazol-5-yl-1 H -indoles with In Vitro Activity towards Methicillin-Resistant Staphylococcus aureus.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 10, p. N.PAG, doi. 10.3390/antibiotics11101450

By:

Li, Steven A.;
Zheng, Rebecca J.;
Sue, Kenneth;
Bourguet-Kondracki, Marie-Lise;
Troudi, Azza;
Brunel, Jean Michel;
Copp, Brent R.;
Cadelis, Melissa M.

Publication type:

Article

A Review of Fungal Protoilludane Sesquiterpenoid Natural Products.

Published in:

Antibiotics (2079-6382), 2020, v. 9, n. 12, p. 928, doi. 10.3390/antibiotics9120928

By:

Cadelis, Melissa M.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

Screening of Fungi for Antimycobacterial Activity Using a Medium-Throughput Bioluminescence-Based Assay.

Published in:

Frontiers in Microbiology, 2021, v. 12, p. 1, doi. 10.3389/fmicb.2021.739995

By:

Grey, Alexander B. J.;
Cadelis, Melissa M.;
Diao, Yiwei;
Park, Duckchul;
Lumley, Thomas;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

α,ω-Diacyl-Substituted Analogues of Natural and Unnatural Polyamines: Identification of Potent Bactericides That Selectively Target Bacterial Membranes.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 6, p. 5882, doi. 10.3390/ijms24065882

By:

Chen, Dan;
Cadelis, Melissa M.;
Rouvier, Florent;
Troia, Thomas;
Edmeades, Liam R.;
Fraser, Kyle;
Gill, Evangelene S.;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Antimicrobial Indole-3-Carboxamido-Polyamine Conjugates Target Bacterial Membranes and Are Antibiotic Potentiators.

Published in:

Biomolecules (2218-273X), 2024, v. 14, n. 3, p. 261, doi. 10.3390/biom14030261

By:

Sue, Kenneth;
Cadelis, Melissa M.;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Indole-3-Acetamido-Polyamines as Antimicrobial Agents and Antibiotic Adjuvants.

Published in:

Biomolecules (2218-273X), 2023, v. 13, n. 8, p. 1226, doi. 10.3390/biom13081226

By:

Sue, Kenneth;
Cadelis, Melissa M.;
Gill, Evangelene S.;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Exploration of Bis-Cinnamido-Polyamines as Intrinsic Antimicrobial Agents and Antibiotic Enhancers.

Published in:

Biomolecules (2218-273X), 2023, v. 13, n. 7, p. 1087, doi. 10.3390/biom13071087

By:

Cadelis, Melissa M.;
Kim, Jisoo;
Rouvier, Florent;
Gill, Evangelene S.;
Fraser, Kyle;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Preliminary SAR of Novel Pleuromutilin–Polyamine Conjugates.

Published in:

Microorganisms, 2023, v. 11, n. 11, p. 2791, doi. 10.3390/microorganisms11112791

By:

Sue, Kenneth;
Cadelis, Melissa M.;
Hainsworth, Kerrin;
Rouvier, Florent;
Bourguet-Kondracki, Marie-Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Spermine Derivatives of Indole‐3‐carboxylic Acid, Indole‐3‐acetic Acid and Indole‐3‐acrylic Acid as Gram‐Negative Antibiotic Adjuvants.

Published in:

ChemMedChem, 2021, v. 16, n. 3, p. 513, doi. 10.1002/cmdc.202000359

By:

Cadelis, Melissa M.;
Li, Steven A.;
Bourguet‐Kondracki, Marie‐Lise;
Blanchet, Marine;
Douafer, Hana;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Exploration of the Electrophilic Reactivity of the Cytotoxic Marine Alkaloid Discorhabdin C and Subsequent Discovery of a New Dimeric C-1/N-13-Linked Discorhabdin Natural Product.

Published in:

Marine Drugs, 2020, v. 18, n. 8, p. 404, doi. 10.3390/md18080404

By:

Lam, Cary F. C.;
Cadelis, Melissa M.;
Copp, Brent R.

Publication type:

Article

Preclinical Evaluation of Discorhabdins in Antiangiogenic and Antitumor Models.

Published in:

Marine Drugs, 2018, v. 16, n. 7, p. 241, doi. 10.3390/md16070241

By:

Harris, Emily M.;
Strope, Jonathan D.;
Beedie, Shaunna L.;
Huang, Phoebe A.;
Goey, Andrew K. L.;
Cook, Kristina M.;
Schofield, Christopher J.;
Chau, Cindy H.;
Cadelis, Melissa M.;
Copp, Brent R.;
Gustafson, Kirk R.;
Figg, William D.

Publication type:

Article

Antimicrobial Natural Products from Plant Pathogenic Fungi.

Published in:

Molecules, 2023, v. 28, n. 3, p. 1142, doi. 10.3390/molecules28031142

By:

Cadelis, Melissa M.;
Li, Steven A.;
van de Pas, Shara J.;
Grey, Alex;
Mulholland, Daniel;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

Total Synthesis of the Four Stereoisomers of Cyclo(l-Trp-l-Arg) Raises Uncertainty of the Structures of the Natural Products and Invalidates Their Promising Antimicrobial Activities.

Published in:

Molecules, 2022, v. 27, n. 18, p. 5913, doi. 10.3390/molecules27185913

By:

Chen, Dan;
Park, Daniel J.;
Cadelis, Melissa M.;
Douafer, Hana;
Bourguet-Kondracki, Marie Lise;
Brunel, Jean Michel;
Copp, Brent R.

Publication type:

Article

Antimicrobial Polyketide Metabolites from Penicillium bissettii and P. glabrum.

Published in:

Molecules, 2022, v. 27, n. 1, p. 240, doi. 10.3390/molecules27010240

By:

Cadelis, Melissa M.;
Nipper, Natasha S. L.;
Grey, Alex;
Geese, Soeren;
van de Pas, Shara J.;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

Isolation of a Novel Polyketide from Neodidymelliopsis sp.

Published in:

Molecules, 2021, v. 26, n. 11, p. 3235, doi. 10.3390/molecules26113235

By:

Cadelis, Melissa M.;
Gordon, Hugo;
Grey, Alex;
Geese, Soeren;
Mulholland, Daniel R.;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

Antimicrobial Metabolites against Methicillin-Resistant Staphylococcus aureus from the Endophytic Fungus Neofusicoccum australe.

Published in:

Molecules, 2021, v. 26, n. 4, p. 1094, doi. 10.3390/molecules26041094

By:

Cadelis, Melissa M.;
Geese, Soeren;
Uy, Benedict B.;
Mulholland, Daniel R.;
van de Pas, Shara J.;
Grey, Alex;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie;
Brycki, Bogumil E.;
Borges, Fernanda;
Gaspar, Alexandra;
Fagin, Fernando Cagide

Publication type:

Article

Epipyrone A, a Broad-Spectrum Antifungal Compound Produced by Epicoccum nigrum ICMP 19927.

Published in:

Molecules, 2020, v. 25, n. 24, p. 5997, doi. 10.3390/molecules25245997

By:

Lee, Alex J.;
Cadelis, Melissa M.;
Kim, Sang H.;
Swift, Simon;
Copp, Brent R.;
Villas-Boas, Silas G.;
Patron, Rosa Durán

Publication type:

Article

A Revised Structure and Assigned Absolute Configuration of Theissenolactone A.

Published in:

Molecules, 2020, v. 25, n. 20, p. 4823, doi. 10.3390/molecules25204823

By:

Cadelis, Melissa M.;
Geese, Soeren;
Gris, Lauren;
Weir, Bevan S.;
Copp, Brent R.;
Wiles, Siouxsie

Publication type:

Article

Synthesis and Antibacterial Analysis of Analogues of the Marine Alkaloid Pseudoceratidine.

Published in:

Molecules, 2020, v. 25, n. 11, p. 2713, doi. 10.3390/molecules25112713

By:

Barker, David;
Lee, Stephanie;
Varnava, Kyriakos G.;
Sparrow, Kevin;
van Rensburg, Michelle;
Deed, Rebecca C.;
Cadelis, Melissa M.;
Li, Steven A.;
Copp, Brent R.;
Sarojini, Vijayalekshmi;
Pilkington, Lisa I.;
Schmidt, Thomas J.

Publication type:

Article