Works by Burns, H. Donald

Results: 46

The synthesis of tritium labelled neurokinin-1 receptor ligands.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2004, v. 47, n. 2, p. 99

By:

Terence G. Hamill;
H. Donald Burns

Publication type:

Article

Radioiodinated α1-adrenergic receptor ligands.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2001, v. 44, n. 1, p. 61, doi. 10.1002/jlcr.433

By:

Hamill, Terence G.;
Burns, H. Donald;
Gibson, Raymond E.

Publication type:

Article

Radiosynthesis of a potent endothelin receptor antagonist: [11C] L-753,037.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2000, v. 43, n. 12, p. 1205, doi. 10.1002/1099-1344(20001030)43:12<1205::AID-JLCR407>3.0.CO;2-1

By:

Ravert, Hayden T.;
Mathews, William B.;
Hamill, Terence G.;
Donald Burns, H.;
Dannals, Robert F.

Publication type:

Article

Non-peptide fibrinogen receptor antagonists. 31. The synthesis of [3H]L-767,685 and [3H]L-767,679.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1998, v. 41, n. 7, p. 677, doi. 10.1002/(SICI)1099-1344(199807)41:7<677::AID-JLCR118>3.0.CO;2-L

By:

Hamill, Terence G.;
Hutchinson, John H.;
Hartman, George D.;
Burns, H. Donald

Publication type:

Article

Non-peptide fibrinogen receptor antagonists. 21. The synthesis of [3H]L-738,167.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1998, v. 41, n. 4, p. 273, doi. 10.1002/(SICI)1099-1344(199804)41:4<273::AID-JLCR76>3.0.CO;2-1

By:

Hamill, Terence G.;
Askew, Ben C.;
Hartman, George D.;
Claremon, David A.;
McIntyre, Charles J.;
Burns, H. Donald

Publication type:

Article

The synthesis of several tritiated non-nucleoside, HIV-1 reverse transcriptase inhibitors.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1998, v. 41, n. 4, p. 319, doi. 10.1002/(SICI)1099-1344(199804)41:4<319::AID-JLCR84>3.0.CO;2-S

By:

Hamill, Terence G.;
Brenner, Nancy J.;
Eng, Wai-si;
Burns, H. Donald

Publication type:

Article

Carbon-11 labeling of a potent, nonpeptide, at1-selective angiotensin-II receptor antagonist: MK-996.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1995, v. 36, n. 8, p. 729, doi. 10.1002/jlcr.2580360804

By:

Mathews, William B.;
Burns, H. Donald;
Dannals, Robert F.;
Ravert, Hayden T.;
Naylor, Elizabeth M.

Publication type:

Article

Radiosynthesis of [11C]nifedipine and [11C]nicardipine.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1989, v. 27, n. 5, p. 589, doi. 10.1002/jlcr.2580270513

By:

Wilson, Alan A.;
Dannals, Robert F.;
Ravert, Hayden T.;
Donald Burns, H.;
Lever, Susan Z.;
Wagner, Henry N.

Publication type:

Article

I-125 and I-123 labelled iodobenzyl bromide, a useful alkylating agent for radiolabelling biologically important molecules.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1986, v. 23, n. 1, p. 83, doi. 10.1002/jlcr.2580230111

By:

Wilson, Alan A.;
Dannals, Robert F.;
Ravert, Hayden T.;
Burns, H. Donald;
Wagner, Henry N.

Publication type:

Article

The plasma-occupancy relationship of the novel GABAA receptor benzodiazepine site ligand, alpha5IA, is similar in rats and primates.

Published in:

2009

By:

Atack, John R.;
Wai-si Eng;
Gibson, Ray E.;
Ryan, Christine;
Francis, Barbara;
Sohal, Bindi;
Dawson, Gerard R.;
Hargreaves, Richard J.;
Burns, H. Donald;
Eng, Wai-Si

Publication type:

journal article

11C-MK-8278 PET as a Tool for Pharmacodynamic Brain Occupancy of Histamine 3 Receptor Inverse Agonists.

Published in:

Journal of Nuclear Medicine, 2014, v. 55, n. 1, p. 65, doi. 10.2967/jnumed.113.122515

By:

Van Laere, Koenraad J.;
Sanabria-Bohórquez, Sandra M.;
Mozley, David P.;
Burns, Donald H.;
Hamill, Terence G.;
Van Hecken, Anne;
De Lepeleire, Inge;
Koole, Michel;
Bormans, Guy;
de Hoon, Jan;
Depré, Marleen;
Cerchio, Kristine;
Plalcza, John;
Lingling Han;
Renger, John;
Hargreaves, Richard J.;
Iannone, Robert

Publication type:

Article

Whole-Body Biodistribution and Radiation Dosimetry of the Human Cannabinoid Type-1 Receptor Ligand 18F-MK-9470 in Healthy Subjects.

Published in:

Journal of Nuclear Medicine, 2008, v. 49, n. 3, p. 439, doi. 10.2967/jnumed.107.047290

By:

Van Laere, Koen;
Koole, Michel;
Bohorquez, Sandra M. Sanabria;
Goffin, Karolien;
Guenther, Ilonka;
Belanger, Marie J.;
Cote, Josee;
Rothenberg, Paul;
De Lepeleire, Inge;
Grachev, Igor D.;
Hargreaves, Richard J.;
Bormans, Guy;
Burns, H. Donald

Publication type:

Article

Human Biodistribution and Radiation Dosimetry of the Tachykinin NK1 Antagonist Radioligand [18F]SPA-RQ: Comparison of Thin-Slice, Bisected, and 2-Dimensional Planar Image Analysis.

Published in:

Journal of Nuclear Medicine, 2007, v. 48, n. 1, p. 100

By:

Sprague, David R.;
Chin, Frederick T.;
Jeih-San Liow;
Fujita, Masahiro;
Burns, H. Donald;
Hargreaves, Richard;
Stubbs, James B.;
Pike, Victor W.;
Innis, Robert B.;
Mozley, P. David

Publication type:

Article

In Vivo Labeling of Endothelin Receptors with [11C]L-753,037: Studies in Mice and a Dog.

Published in:

Journal of Nuclear Medicine, 2001, v. 42, n. 8, p. 1274

By:

Aleksic, Sasa;
Szabo, Zsolt;
Scheffel, Ursula;
Ravert, Hayden T.;
Mathews, William B.;
Kerenyi, Levente;
Rauseo, Paige A.;
Gibson, Raymond E.;
Burns, H. Donald;
Dannals, Robert F.

Publication type:

Article

The synthesis and preclinical evaluation in rhesus monkey of [.

Published in:

Synapse, 2011, v. 65, n. 4, p. 261, doi. 10.1002/syn.20842

By:

HAMILL, TERENCE G.;
WAISI ENG;
JENNINGS, ANDREW;
LEWIS, RICHARD;
THOMAS, STEVEN;
WOOD, SUZANNE;
STREET, LESLIE;
WISNOSKI, DAVID;
WOLKENBERG, SCOTT;
LINDSLEY, CRAIG;
SANABRIA-BOHÓRQUEZ, SANDRA M.;
PATEL, SHIL;
RIFFEL, KERRY;
RYAN, CHRISTINE;
COOK, JACQUELYNN;
SUR, CYRILLE;
BURNS, H. DONALD;
HARGREAVES, RICHARD

Publication type:

Article

Synthesis, characterization, and monkey PET studies of [18F]MK-1312, a PET tracer for quantification of mGluR1 receptor occupancy by MK-5435.

Published in:

Synapse, 2011, v. 65, n. 2, p. 125, doi. 10.1002/syn.20826

By:

Hostetler, Eric D.;
Eng, Waisi;
Joshi, Aniket D.;
Sanabria-Bohórquez, Sandra;
Kawamoto, Hiroshi;
Ito, Satoru;
O'Malley, Stacey;
Krause, Stephen;
Ryan, Christine;
Patel, Shil;
Williams, Mangay;
Riffel, Kerry;
Suzuki, Gentaroh;
Ozaki, Satoshi;
Ohta, Hisashi;
Cook, Jacquelynn;
Burns, H. Donald;
Hargreaves, Richard

Publication type:

Article

Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18.

Published in:

Synapse, 2009, v. 63, n. 12, p. 1122, doi. 10.1002/syn.20689

By:

Hamill, Terence G.;
Sato, Nagaaki;
Jitsuoka, Makoto;
Tokita, Shigeru;
Sanabria, Sandra;
Eng, Waisi;
Ryan, Christine;
Krause, Stephen;
Takenaga, Norihiro;
Patel, Shil;
Zeng, Zhizhen;
Williams, David;
Sur, Cyrille;
Hargreaves, Richard;
Burns, H. Donald

Publication type:

Article

Synthesis, characterization, and first successful monkey imaging studies of metabotropic glutamate receptor subtype 5 (mGluR5) PET radiotracers.

Published in:

Synapse, 2005, v. 56, n. 4, p. 205, doi. 10.1002/syn.20147

By:

Hamill, Terence G.;
Krause, Stephen;
Ryan, Christine;
Bonnefous, Celine;
Govek, Steve;
Seiders, T. Jon;
Cosford, Nicholas D.P.;
Roppe, Jeffrey;
Kamenecka, Ted;
Patel, Shil;
Gibson, Raymond E.;
Sanabria, Sandra;
Riffel, Kerry;
Eng, Waisi;
King, Christopher;
Yang, Xiaoqing;
Green, Mitchell D.;
O'malley, Stacey S.;
Hargreaves, Richard;
Burns, H. Donald

Publication type:

Article

Radiosynthesis of the HIV integrase inhibitor [18F]MK-0518 (Isentress).

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2010, v. 53, n. 7, p. 517, doi. 10.1002/jlcr.1778

By:

Li, Wenping;
Thompson, Wayne;
Fisher, Thorsten;
Wai, John S.;
Hazuda, Daria;
Burns, H. Donald;
Hamill, Terence G.

Publication type:

Article

An improved synthesis of substituted [11C]toluenes via Suzuki coupling with [11C]methyl iodide.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2005, v. 48, n. 9, p. 629, doi. 10.1002/jlcr.953

By:

Hostetler, Eric D.;
Terry, Garth E.;
Donald Burns, H.

Publication type:

Article

The synthesis of a benzamidine-containing NR2B-selective NMDA receptor ligand labelled with tritium or fluorine-18.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2005, v. 48, n. 1, p. 1, doi. 10.1002/jlcr.871

By:

Hamill, Terence G.;
McCauley, John A.;
Burns, H. Donald

Publication type:

Article

PET imaging studies in rhesus monkey with the cannabinoid-1 (CB1) receptor ligand [11C]CB-119.

Published in:

2009

By:

Hamill, Terence G;
Lin, Linus S;
Hagmann, William;
Liu, Ping;
Jewell, James;
Sanabria, Sandra;
Eng, WaiSi;
Ryan, Christine;
Fong, Tung M;
Connolly, Brett;
Vanko, Amy;
Hargreaves, Richard;
Goulet, Mark T;
Burns, H Donald

Publication type:

journal article

Screening cascade and development of potential Positron Emission Tomography radiotracers for mGluR5: in vitro and in vivo characterization.

Published in:

2005

By:

Patel, Shil;
Ndubizu, Obinna;
Hamill, Terence;
Chaudhary, A;
Burns, H Donald;
Hargreaves, R;
Gibson, Raymond E

Publication type:

journal article

Synthesis and characterization of a potent, selective, radiolabeled substance-P antagonist for NK1 receptor quantitation: ([18F]SPA-RQ)

Published in:

2004

By:

Solin, Olof;
Eskola, Olli;
Hamill, Terence G.;
Bergman, Jörgen;
Lehikoinen, Pertti;
Grönroos, Tove;
Forsback, Sarita;
Haaparanta, Merja;
Viljanen, Tapio;
Ryan, Christine;
Gibson, Raymond;
Kieczykowski, Gerard;
Hietala, Jarmo;
Hargreaves, Richard;
Burns, H. Donald;
Bergman, Jörgen;
Grönroos, Tove

Publication type:

journal article

[Re symposium: "Approaches to optimize the discovery of CNS receptor imaging probes for use in drug discovery and development"].

Published in:

2003

By:

Waterhouse, Rikki N;
McCarthy, Timothy J;
Collier, T Lee;
Burns, H Donald

Publication type:

journal article

Invited commentary

Published in:

Molecular Imaging & Biology, 2003, v. 5, n. 6, p. 347, doi. 10.1016/j.mibio.2003.10.002

By:

Waterhouse, Rikki N.;
McCarthy, Timothy J.;
Collier, T. Lee;
Burns, H. Donald

Publication type:

Article

Image-derived input function for [11C]flumazenil kinetic analysis in human brain.

Published in:

2003

By:

Sanabria-Bohórquez, Sandra M;
Maes, Alex;
Dupont, Patrick;
Bormans, Guy;
de Groot, Tjibbe;
Coimbra, Alexandre;
Eng, WaiSi;
Laethem, Tine;
De Lepeleire, Inge;
Gambale, Jay;
Vega, Jose M;
Burns, H Donald

Publication type:

journal article

Image-Derived Input Function for [11C]Flumazenil Kinetic Analysis in Human Brain

Published in:

Molecular Imaging & Biology, 2003, v. 5, n. 2, p. 72, doi. 10.1016/S1536-1632(03)00046-5

By:

Sanabria-Bohórquez, Sandra M.;
Maes, Alex;
Dupont, Patrick;
Bormans, Guy;
Groot, Tjibbe de;
Coimbra, Alexandre;
Eng, WaiSi;
Laethem, Tine;
Lepeleire, Inge De;
Gambale, Jay;
Vega, Jose M.;
Burns, H. Donald

Publication type:

Article

An In Vitro Assay for Predicting Successful Imaging Radiotracers

Published in:

2003

By:

Patel, Shil;
Hamill, Terence;
Hostetler, Eric;
Burns, H. Donald;
Gibson, Raymond E.

Publication type:

journal article

Society of Noninvasive Imaging in Drug Development Joins the Academy of Molecular Imaging

Published in:

2002

By:

Burns, H. Donald;
Eckelman, William C.

Publication type:

Editorial

Assessment of dopamine receptor densities in the human brain with carbon-11-labeled N-methylspiperone.

Published in:

Annals of Neurology, 1984, v. 15, n. S1, p. 79, doi. 10.1002/ana.410150715

By:

Wagner, Henry N.;
Burns, H. Donald;
Dannals, Robert F.;
Wong, Dean F.;
Langström, Bengt;
Duelfer, Timothy;
Frost, J. James;
Ravert, Hayden T.;
Links, Jonathan M.;
Rosenbloom, Shelley B.;
Lukas, Scott E.;
Kramer, Alfred V.;
Kuhar, Michael J.

Publication type:

Article

In vivo studies of opiate receptors.

Published in:

Annals of Neurology, 1984, v. 15, n. S1, p. 85, doi. 10.1002/ana.410150716

By:

Frost, J. James;
Dannals, Robert F.;
Duelfer, Timothy;
Burns, H. Donald;
Ravert, Hayden T.;
Langströ, Bengt;
Balasubramanian, V.;
Wagner, Henry N.

Publication type:

Article

Kinetic analysis of the cannabinoid-1 receptor PET tracer [18F]MK-9470 in human brain.

Published in:

European Journal of Nuclear Medicine & Molecular Imaging, 2010, v. 37, n. 5, p. 920, doi. 10.1007/s00259-009-1340-5

By:

Sanabria-Bohórquez, Sandra Marina;
Hamill, Terence G.;
Goffin, Karolien;
de Lepeleire, Inge;
Bormans, Guy;
Burns, H. Donald;
van Laere, Koen

Publication type:

Article

PREPARATION OF 1-ARYL-3-(TETRA-0-ACETYL-2-DEOXY-D-GLUCOS-2-YL)UREAS.

Published in:

Organic Preparations & Procedures International, 1975, v. 7, n. 6, p. 291, doi. 10.1080/00304947509355164

By:

Heindel, Ned D.;
Burns, H. Donald;
Honda, Takashi;
Risch, Victor R.;
Brady, Luther W.

Publication type:

Article

A SIMPLE, TWO STEP SYNTHESIS OF 1-(2-CHLOROETHYL)-1-NITROSO-3-(D-GLUCOS-2-YL) UREA.

Published in:

Organic Preparations & Procedures International, 1974, v. 6, n. 6, p. 259, doi. 10.1080/00304947409355117

By:

Burns, H. Donald;
Heindel, Ned D.

Publication type:

Article

Symposium abstracts.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1977, v. 13, n. 2, p. 235, doi. 10.1002/jlcr.2580130202

By:

Burns, H. Donald;
Worley, Paul;
Wagner, Henry N.

Publication type:

Article

Symposium abstracts.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 1977, v. 13, n. 2, p. 235, doi. 10.1002/jlcr.2580130202

By:

Burns, H. Donald;
Worley, Paul;
Wagner, Henry N.

Publication type:

Article

The 1,3,4-oxadiazole moiety, a protective synthon for indirect radioiodination.

Published in:

Journal of Heterocyclic Chemistry, 1985, v. 22, n. 1, p. 209, doi. 10.1002/jhet.5570220149

By:

Heindel, Ned D.;
Van Dort, Marcian;
Cahn, Maurice;
Schneider, Richard;
Burns, H. Donald

Publication type:

Article

Imaging and its Applications to Drug Delivery.

Published in:

Drug Development & Industrial Pharmacy, 1990, v. 16, n. 18, p. 2655, doi. 10.3109/03639049009058553

By:

Solomon, Howard F.;
Burns, H. Donald;
Gibson, Raymond E.

Publication type:

Article

Investigation of Angiotensin II/AT1 Receptors with Carbon-11-L-1 59,884: A Selective AT1 Antagonist.

Published in:

Journal of Nuclear Medicine, 1998, v. 39, n. 7, p. 1209

By:

Szabo, Zsolt;
Pan Fu Kao;
Burns, H. Donald;
Gibson, Raymond E.;
Hamill, Terence G.;
Ravert, Hayden T.;
Sang Eun Kim;
Mathews, William B.;
Musachio, John L.;
Scheffel, Ursula;
Dannals, Robert F.

Publication type:

Article

In Vivo Labeling of Angiotensin II Receptors with a Carbon- 11-Labeled Selective Nonpeptide Antagonist.

Published in:

Journal of Nuclear Medicine, 1996, v. 37, n. 2, p. 307

By:

Sang Eun Kim;
Scheffel, Ursula;
Szabo, Zsolt;
Burns, H. Donald;
Gibson, Raymond E.;
Ravert, Hayden T.;
Mathews, William B.;
Hamill, Terence G.;
Dannals, Robert F.

Publication type:

Article

Comparison of Technetium-99m Aminoalkyl Diaminodithiol (DADT) Analogs as Potential Brain Blood Flow Imaging Agents.

Published in:

Journal of Nuclear Medicine, 1988, v. 29, n. 1, p. 73

By:

Scheffel, Ursula;
Goldfarb, Howard W.;
Lever, Susan Z.;
Gungon, Ramon L.;
Burns, H. Donald;
Wagner Jr., Henry N.

Publication type:

Article

Design, Preparation, and Biodistribution of a Technetium-99m Triaminedithiol Complex to Assess Regional Cerebral Blood Flow.

Published in:

Journal of Nuclear Medicine, 1985, v. 26, n. 11, p. 1287

By:

Lever, S. Zemyan;
Burns, H. Donald;
Kervitsky, Therese M.;
Goldfarb, Howard W.;
Woo, David V.;
Wong, Dean F.;
Epps, Leon A.;
Kramer, Alfred V.;
Wagner Jr., Henry N.

Publication type:

Article

(3-N-[11C]Methyl)Spiperone, A Ligand Binding to Dopamine Receptors: Radiochemical Synthesis and Biodistribution Studies in Mice.

Published in:

Journal of Nuclear Medicine, 1984, v. 25, n. 11, p. 1222

By:

Burns, H. Donald;
Dannals, Robert F.;
Langström, Bengt;
Ravert, Hayden T.;
Zemyan, Susan E.;
Dueller, Timothy;
Wong, Dean F.;
Frost, J. James;
Kuhar, Michael J.;
Wagner, Henry N.

Publication type:

Article

4-[125l] lodophenyltrimethylammonium Ion, an lodinated Acetylcholinesterase Inhibitor with Potential as a Myocardial Imaging Agent.

Published in:

Journal of Nuclear Medicine, 1980, v. 21, n. 9, p. 875

By:

Burns, H. Donald;
Marzilli, Luigi G.;
Dannals, Robert F.;
Dannals, Thomas E.;
Trageser, Timothy C.;
Conti, Peter;
Wagner Jr., Henry N.

Publication type:

Article

A New Electrophoretic Method for Determining Ligand: Technetium Stoichiometry in Carrier Free 99mTc-Radiopharmaceuticals.

Published in:

Journal of Nuclear Medicine, 1979, v. 20, n. 8, p. 871

By:

Marzilli, Luigi G.;
Worley, Paul;
Burns, H. Donald

Publication type:

Article