Works matching AU Brogi, Simone


Results: 65
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    Design, synthesis, and biological investigation of oxadiazolyl, thiadiazolyl, and pyrimidinyl linked antipyrine derivatives as potential non-acidic anti-inflammatory agents.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2022.2162511
    By:
    • Al-Sanea, Mohammad M.;
    • Hamdi, Abdelrahman;
    • Brogi, Simone;
    • S. Tawfik, Samar;
    • Othman, Dina I. A.;
    • Elshal, Mahmoud;
    • Ur Rahman, Hidayat;
    • Parambi, Della G. T.;
    • M. Elbargisy, Rehab;
    • Selim, Samy;
    • Mostafa, Ehab M.;
    • Mohamed, Ahmed A. B.
    Publication type:
    Article
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    The Citrus Flavonoid Naringenin Protects the Myocardium from Ageing-Dependent Dysfunction: Potential Role of SIRT1.

    Published in:
    Oxidative Medicine & Cellular Longevity, 2020, p. 1, doi. 10.1155/2020/4650207
    By:
    • Testai, Lara;
    • Piragine, Eugenia;
    • Piano, Ilaria;
    • Flori, Lorenzo;
    • Da Pozzo, Eleonora;
    • Miragliotta, Vincenzo;
    • Pirone, Andrea;
    • Citi, Valentina;
    • Di Cesare Mannelli, Lorenzo;
    • Brogi, Simone;
    • Carpi, Sara;
    • Martelli, Alma;
    • Nieri, Paola;
    • Martini, Claudia;
    • Ghelardini, Carla;
    • Gargini, Claudia;
    • Calderone, Vincenzo
    Publication type:
    Article
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    Resveratrol-like Compounds as SIRT1 Activators.

    Published in:
    International Journal of Molecular Sciences, 2022, v. 23, n. 23, p. 15105, doi. 10.3390/ijms232315105
    By:
    • Ciccone, Lidia;
    • Piragine, Eugenia;
    • Brogi, Simone;
    • Camodeca, Caterina;
    • Fucci, Raffaele;
    • Calderone, Vincenzo;
    • Nencetti, Susanna;
    • Martelli, Alma;
    • Orlandini, Elisabetta
    Publication type:
    Article
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    Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain.

    Published in:
    ChemMedChem, 2018, v. 13, n. 19, p. 2090, doi. 10.1002/cmdc.201800397
    By:
    • Brindisi, Margherita;
    • Borrelli, Giuseppe;
    • Brogi, Simone;
    • Grillo, Alessandro;
    • Maramai, Samuele;
    • Paolino, Marco;
    • Benedusi, Mascia;
    • Pecorelli, Alessandra;
    • Valacchi, Giuseppe;
    • Di Cesare Mannelli, Lorenzo;
    • Ghelardini, Carla;
    • Allarà, Marco;
    • Ligresti, Alessia;
    • Minetti, Patrizia;
    • Campiani, Giuseppe;
    • di Marzo, Vincenzo;
    • Butini, Stefania;
    • Gemma, Sandra
    Publication type:
    Article
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    New Visions on Natural Products and Cancer Therapy: Autophagy and Related Regulatory Pathways.

    Published in:
    Cancers, 2022, v. 14, n. 23, p. 5839, doi. 10.3390/cancers14235839
    By:
    • Martelli, Alma;
    • Omrani, Marzieh;
    • Zarghooni, Maryam;
    • Citi, Valentina;
    • Brogi, Simone;
    • Calderone, Vincenzo;
    • Sureda, Antoni;
    • Lorzadeh, Shahrokh;
    • da Silva Rosa, Simone C.;
    • Grabarek, Beniamin Oscar;
    • Staszkiewicz, Rafał;
    • Los, Marek J.;
    • Nabavi, Seyed Fazel;
    • Nabavi, Seyed Mohammad;
    • Mehrbod, Parvaneh;
    • Klionsky, Daniel J.;
    • Ghavami, Saeid
    Publication type:
    Article
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    Synthesis and biological investigation of peptidomimetic SARS‐CoV‐2 main protease inhibitors bearing quinoline‐based heterocycles at P<sub>3</sub>.

    Published in:
    Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400812
    By:
    • Rossi, Sara;
    • Deidda, Graziano;
    • Fiaschi, Lia;
    • Ibba, Roberta;
    • Pieroni, Mariachiara;
    • Dichiara, Maria;
    • Carullo, Gabriele;
    • Butini, Stefania;
    • Ramunno, Anna;
    • Brogi, Simone;
    • Lolicato, Marco;
    • Arrigoni, Cristina;
    • Cabella, Noemi;
    • Bavagnoli, Laura;
    • Maga, Giovanni;
    • Varasi, Ilenia;
    • Biba, Camilla;
    • Vicenti, Ilaria;
    • Gemma, Sandra;
    • Crespan, Emmanuele
    Publication type:
    Article
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    Myxobacterial depsipeptide chondramides interrupt SARS-CoV-2 entry by targeting its broad, cell tropic spike protein.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2022, v. 40, n. 22, p. 12209, doi. 10.1080/07391102.2021.1969281
    By:
    • Fernandez, Rey Arturo;
    • Quimque, Mark Tristan;
    • Notarte, Kin Israel;
    • Manzano, Joe Anthony;
    • Pilapil IV, Delfin Yñigo;
    • de Leon, Von Novi;
    • San Jose, John Jeric;
    • Villalobos, Omar;
    • Muralidharan, Nisha Harur;
    • Gromiha, M. Michael;
    • Brogi, Simone;
    • Macabeo, Allan Patrick G.
    Publication type:
    Article
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    Front Cover: Synthesis of Unsymmetrical Squaramides as Allosteric GSK‐3β Inhibitors Promoting β‐Catenin‐Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial Cells (ChemMedChem 24/2022).

    Published in:
    ChemMedChem, 2022, v. 17, n. 24, p. 1, doi. 10.1002/cmdc.202200663
    By:
    • Carullo, Gabriele;
    • Bottoni, Laura;
    • Pasquini, Silvia;
    • Papa, Alessandro;
    • Contri, Chiara;
    • Brogi, Simone;
    • Calderone, Vincenzo;
    • Orlandini, Maurizio;
    • Gemma, Sandra;
    • Varani, Katia;
    • Butini, Stefania;
    • Galvagni, Federico;
    • Vincenzi, Fabrizio;
    • Campiani, Giuseppe
    Publication type:
    Article
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    Synthesis of Unsymmetrical Squaramides as Allosteric GSK‐3β Inhibitors Promoting β‐Catenin‐Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial Cells.

    Published in:
    ChemMedChem, 2022, v. 17, n. 24, p. 1, doi. 10.1002/cmdc.202200456
    By:
    • Carullo, Gabriele;
    • Bottoni, Laura;
    • Pasquini, Silvia;
    • Papa, Alessandro;
    • Contri, Chiara;
    • Brogi, Simone;
    • Calderone, Vincenzo;
    • Orlandini, Maurizio;
    • Gemma, Sandra;
    • Varani, Katia;
    • Butini, Stefania;
    • Galvagni, Federico;
    • Vincenzi, Fabrizio;
    • Campiani, Giuseppe
    Publication type:
    Article
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    Design and Synthesis of Oligopeptidic Parvulin Inhibitors.

    Published in:
    ChemMedChem, 2022, v. 17, n. 11, p. 1, doi. 10.1002/cmdc.202200050
    By:
    • Relitti, Nicola;
    • Prasanth Saraswati, A.;
    • Carullo, Gabriele;
    • Papa, Alessandro;
    • Monti, Alessandra;
    • Benedetti, Rosaria;
    • Passaro, Eugenia;
    • Brogi, Simone;
    • Calderone, Vincenzo;
    • Butini, Stefania;
    • Gemma, Sandra;
    • Altucci, Lucia;
    • Campiani, Giuseppe;
    • Doti, Nunzianna
    Publication type:
    Article
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