Works matching AU Bojarski, Andrzej J.

Results: 83

Electrospray mass spectrometric studies of noncovalent complexes of buspirone hydrochloride and other serotonin 5-HT1A receptor ligands containing arylpiperazine moieties.

Published in:

Rapid Communications in Mass Spectrometry: RCM, 2003, v. 17, n. 18, p. 2139, doi. 10.1002/rcm.1166

By:

Kowalski, Piotr;
Suder, Piotr;
Kowalska, Teresa;
Silberring, Jerzy;
Duszyńska, Beata;
Bojarski, Andrzej J.

Publication type:

Article

Conformational analysis of 4-(2′-furyl)-2-(methylamino)pyrimidine.

Published in:

Journal of Heterocyclic Chemistry, 1996, v. 33, n. 4, p. 1207, doi. 10.1002/jhet.5570330434

By:

Mokrosz, Jerzy L.;
Bojarski, Andrzej J.;
Harden, Donald B.;
Strekowski, Lucjan

Publication type:

Article

Novel 1,4-Benzoxazin-3( 4H)-one, 1,2-Benzoxazolin-3-one and 1,3-Benzoxazolin-2,4-dione Arylpiperazine Derivatives with Different 5-HT1A and Antagonistic 5-HT2A Activities.

Published in:

Archiv der Pharmazie, 1999, v. 332, n. 11, p. 373, doi. 10.1002/(SICI)1521-4184(199911)332:11<373::AID-ARDP373>3.0.CO;2-L

By:

Mokrosz, Maria J.;
Kowalski, Piotr;
Kowalska, Teresa;
Majka, Zbigniew;
Duszynska, Beata;
Bojarski, Andrzej J.;
Fruzinski, Andrzej;
Karolak-Wojciechowska, Janina;
Wesolowska, Anna;
Klodzinska, Aleksandra;
Tatarczynska, Ewa;
Chojnacka-Wojcik, Ewa

Publication type:

Article

Crystal and Molecular Structure of 4-[ω-(Benzotriazolyl)alkyl]-1-(2-methoxyphenyl)piperazines with a Different Pharmacological Activity.

Published in:

Archiv der Pharmazie, 1998, v. 331, n. 10, p. 299, doi. 10.1002/(sici)1521-4184(199810)331:10<299::aid-ardp299>3.3.co;2-v

By:

Karolak-Wojciechowska, Janina;
Fruziński, Andrzej;
Bojarski, Andrzej J.;
Paluchowska, Maria H.;
Mokrosz, Maria J.

Publication type:

Article

Structure-Activity Relationship Studies of CNS Agents, Part 25: 4,6-Di(heteroaryl)-2-( N-methylpiperazino)pyrimidines as New, Potent 5-HT2A Receptor Ligands: A Verification of the Topographic Model.

Published in:

Archiv der Pharmazie, 1995, v. 328, n. 9, p. 659, doi. 10.1002/ardp.19953280906

By:

Mokrosz, Maria J.;
Strekowski, Lucjan;
Kozak, Wei Xing;
Duszyńska, Beata;
Bojarski, Andrzej J.;
Kłodzinska, Aleksandra;
Czarny, Agnieszka;
Cegła, Marek T.;
Dereń-Wesołek, Anna;
Chojnacka-Wójcik, Ewa;
Dove, Stefan;
Mokrosz, Jerzy L.

Publication type:

Article

Structure-Activity Relationship Studies of CNS Agents, Part 23[1]): N-(3-Phenylpropyl)- and N-[3( E)-Cinnamyl]-1,2,3,4-tetrahydroisoquinoline Mimic 1-Phenylpiperazine at 5-HT1A Receptors.

Published in:

Archiv der Pharmazie, 1995, v. 328, n. 7/8, p. 604, doi. 10.1002/ardp.19953280707

By:

Mokrosz, Jerzy L.;
Bojarski, Andrzej J.;
Charakchieva-Minol, Sijka;
Duszynska, Beata;
Mokrosz, Maria J.;
Paluchowska, Maria H.

Publication type:

Article

Structure-Activity Relationship Studies of CNS Agents, XXI: Two Derivatives of 1-( o-Methoxyphenyl)piperazine with an Opposite Function at 5-HT1A Receptors Struktur-Wirkung-Beziehungen ZNS-aktiver Substanzen, 21. Mitt.1): Zwei Derivate von 1-( o-Methoxyphenyl)piperazin mit entgegengesetzter Wirkung auf 5-HT1A Rezeptoren

Published in:

Archiv der Pharmazie, 1995, v. 328, n. 4, p. 381, doi. 10.1002/ardp.19953280417

By:

Mokrosz, Jerzy L.;
Klodzinska, Aleksandra;
Boksa, Jan;
Bojarski, Andrzej J.;
Duszynska, Beata;
Chojnacka-Wójcik, Ewa

Publication type:

Article

Structure-Activity Relationship Studies of CNS Agents, XIX: Quantitative Analysis of the Alkyl Chain Effects on the 5-HT1A and 5-HT2 Receptor Affinities of 4-Alkyl-1-arylpiperazines and Their Analogs.

Published in:

Archiv der Pharmazie, 1995, v. 328, n. 2, p. 143, doi. 10.1002/ardp.19953280210

By:

Mokrosz, Jerzy L.;
Mokrosz, Maria J.;
Charakchieva-Minol, Sijka;
Paluchowska, Maria H.;
Bojarski, Andrzej J.;
Duszyńska, Beata

Publication type:

Article

Robust optimization of SVM hyperparameters in the classification of bioactive compounds.

Published in:

Journal of Cheminformatics, 2015, v. 7, n. 1, p. 1, doi. 10.1186/s13321-015-0088-0

By:

Czarnecki, Wojciech M.;
Podlewska, Sabina;
Bojarski, Andrzej J.

Publication type:

Article

Multiple conformational states in retrospective virtual screening - homology models vs. crystal structures: beta-2 adrenergic receptor case study.

Published in:

Journal of Cheminformatics, 2015, v. 7, n. 1, p. 1, doi. 10.1186/s13321-015-0062-x

By:

Mordalski, Stefan;
Witek, Jagna;
Smusz, Sabina;
Rataj, Krzysztof;
Bojarski, Andrzej J.

Publication type:

Article

The influence of negative training set size on machine learning-based virtual screening.

Published in:

Journal of Cheminformatics, 2014, v. 6, n. 1, p. 1, doi. 10.1186/1758-2946-6-32

By:

Kurczab, Rafał;
Smusz, Sabina;
Bojarski, Andrzej J.

Publication type:

Article

The influence of the inactives subset generation on the performance of machine learning methods.

Published in:

Journal of Cheminformatics, 2013, v. 5, n. 1, p. 1, doi. 10.1186/1758-2946-5-17

By:

Smusz, Sabina;
Kurczab, Rafał;
Bojarski, Andrzej J.

Publication type:

Article

The influence of training actives/inactives ratio on machine learning performance.

Published in:

2013

By:

Kurczab, Rafał;
Smusz, Sabina;
Bojarski, Andrzej J.

Publication type:

Conference Paper/Materials

Application of Structural Interaction Fingerpints (SIFts) into post-docking analysis - insight into activity and selectivity.

Published in:

2013

By:

Witek, Jagna;
Krzysztof Rataj,, Krzysztof;
Mordalski, Stefan;
Smusz, Sabina;
Kosciolek, Tomasz;
Bojarski, Andrzej J.

Publication type:

Conference Paper/Materials

The influence of hashed fingerprints density on the machine learning methods performance.

Published in:

2013

By:

Smusz, Sabina;
Kurczab, Rafał;
Bojarski, Andrzej J.

Publication type:

Conference Paper/Materials

The importance of template choice in homology modeling. A 5-HT6R case study.

Published in:

Journal of Cheminformatics, 2013, v. 5, n. S1, p. 1, doi. 10.1186/1758-2946-5-S1-P8

By:

Rataj, Krzysztof;
Witek, Jagna;
Mordalski, Stefan;
Kościółek, Tomasz;
Bojarski, Andrzej J.

Publication type:

Article

Asymmetric Clustering Index in a Case Study of 5-HT1A Receptor Ligands.

Published in:

PLoS ONE, 2014, v. 9, n. 7, p. 1, doi. 10.1371/journal.pone.0102069

By:

Śmieja, Marek;
Warszycki, Dawid;
Tabor, Jacek;
Bojarski, Andrzej J.

Publication type:

Article

A Linear Combination of Pharmacophore Hypotheses as a New Tool in Search of New Active Compounds – An Application for 5-HT1A Receptor Ligands.

Published in:

PLoS ONE, 2013, v. 8, n. 12, p. 1, doi. 10.1371/journal.pone.0084510

By:

Warszycki, Dawid;
Mordalski, Stefan;
Kristiansen, Kurt;
Kafel, Rafał;
Sylte, Ingebrigt;
Chilmonczyk, Zdzisław;
Bojarski, Andrzej J.

Publication type:

Article

In the search for a lead structure among series of potent and selective hydantoin 5- HT7R agents: The drug-likeness in vitro study.

Published in:

Chemical Biology & Drug Design, 2017, v. 90, n. 6, p. 1295, doi. 10.1111/cbdd.13106

By:

Latacz, Gniewomir;
Lubelska, Annamaria;
Jastrzębska‐Więsek, Magdalena;
Partyka, Anna;
Sobiło, Andrzej;
Olejarz, Agnieszka;
Kucwaj‐Brysz, Katarzyna;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Wesołowska, Anna;
Kieć‐Kononowicz, Katarzyna;
Handzlik, Jadwiga

Publication type:

Article

Solid-Supported Synthesis and 5- HT7/5- HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1 H)-one.

Published in:

Chemical Biology & Drug Design, 2015, v. 86, n. 4, p. 697, doi. 10.1111/cbdd.12539

By:

Grychowska, Katarzyna;
Masurier, Nicolas;
Verdié, Pascal;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Martinez, Jean;
Pawłowski, Maciej;
Subra, Gilles;
Zajdel, Paweł

Publication type:

Article

Synthesis, Antidepressant Evaluation and Docking Studies of Long-Chain Alkylnitroquipazines as Serotonin Transporter Inhibitors.

Published in:

Chemical Biology & Drug Design, 2013, v. 81, n. 6, p. 695, doi. 10.1111/cbdd.12116

By:

Gabrielsen, Mari;
Wołosewicz, Karol;
Zawadzka, Anna;
Kossakowski, Jerzy;
Nowak, Gabriel;
Wolak, Małgorzata;
Stachowicz, Katarzyna;
Siwek, Agata;
Ravna, Aina W.;
Kufareva, Irina;
Kozerski, Lech;
Bednarek, Elżbieta;
Sitkowski, Jerzy;
Bocian, Wojciech;
Abagyan, Ruben;
Bojarski, Andrzej J.;
Sylte, Ingebrigt;
Chilmonczyk, Zdzisław

Publication type:

Article

Functional characterization of a novel opioid, PZM21, and its effects on the behavioural responses to morphine.

Published in:

2019

By:

Kudla, Lucja;
Bugno, Ryszard;
Skupio, Urszula;
Wiktorowska, Lucja;
Solecki, Wojciech;
Wojtas, Adam;
Golembiowska, Krystyna;
Zádor, Ferenc;
Benyhe, Sándor;
Buda, Szymon;
Makuch, Wioletta;
Przewlocka, Barbara;
Bojarski, Andrzej J.;
Przewlocki, Ryszard

Publication type:

journal article

Structural determinants influencing halogen bonding: a case study on azinesulfonamide analogs of aripiprazole as 5-HT1A, 5-HT7, and D2 receptor ligands.

Published in:

Chemistry Central Journal, 2018, v. 12, n. 1, p. 1, doi. 10.1186/s13065-018-0422-5

By:

Marciniec, Krzysztof;
Kurczab, Rafał;
Książek, Maria;
Bębenek, Ewa;
Chrobak, Elwira;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Kusz, Joachim;
Zajdel, Paweł

Publication type:

Article

5-HT1A receptor ligands and their therapeutic applications: review of new patents.

Published in:

Expert Opinion on Therapeutic Patents, 2018, v. 28, n. 9, p. 679, doi. 10.1080/13543776.2018.1514011

By:

Staroń, Jakub;
Bugno, Ryszard;
Hogendorf, Adam S.;
Bojarski, Andrzej J.

Publication type:

Article

Amisulpride as a potential disease‐modifying drug in the treatment of tauopathies.

Published in:

Alzheimer's & Dementia: The Journal of the Alzheimer's Association, 2023, v. 19, n. 12, p. 5482, doi. 10.1002/alz.13090

By:

Jahreis, Kathrin;
Brüge, Alina;
Borsdorf, Saskia;
Müller, Franziska E.;
Sun, Weilun;
Jia, Shaobo;
Kang, Dong Min;
Boesen, Nicolette;
Shin, Seulgi;
Lim, Sungsu;
Koroleva, Anastasia;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Rakuša, Elena;
Fink, Anne;
Doblhammer‐Reiter, Gabriele;
Kim, Yun Kyung;
Dityatev, Alexander;
Ponimaskin, Evgeni;
Labus, Josephine

Publication type:

Article

Radiolabeling and in vivo evaluation of [11C]AGH-44: a potential lead structure to develop a positron emission tomography radioligand for the 5-HT7 receptor.

Published in:

Journal of Radioanalytical & Nuclear Chemistry, 2019, v. 322, n. 2, p. 847, doi. 10.1007/s10967-019-06687-3

By:

L'Estrade, Elina T.;
Petersen, Ida N.;
Xiong, Mengfei;
Hogendorf, Adam S.;
Hogendorf, Agata;
Kristensen, Jesper L.;
Kjær, Andreas;
Bojarski, Andrzej J.;
Erlandsson, Maria;
Ohlsson, Tomas;
Knudsen, Gitte M.;
Herth, Matthias M.

Publication type:

Article

Erratum: Synthesis of Some Aminophosphonates Bearing N-(Fluorophenyl)-piperazynyl Moiety and Their Activity toward Serotonin Receptors.

Published in:

Heteroatom Chemistry, 2016, v. 27, n. 2, p. 135, doi. 10.1002/hc.21312

By:

Lewkowski, Jarosław;
Jóźwiak, Andrzej;
Tokarz, Paweł;
Zagórski, Piotr M.;
Hamera, Róża;
Cal, Dariusz;
Satała, Grzegorz;
Bojarski, Andrzej J.

Publication type:

Article

Synthesis of Some Aminophosphonates Bearing N-(Fluorophenyl)-piperazynyl Moiety and Their Activity toward Serotonin Receptors.

Published in:

Heteroatom Chemistry, 2015, v. 26, n. 4, p. 290, doi. 10.1002/hc.21259

By:

Lewkowski, Jarosław;
Jóźwiak, Andrzej;
Tokarz, Paweł;
Zagórski, Piotr M.;
Hamera, Róża;
Cal, Dariusz;
Satała, Grzegorz;
Bojarski, Andrzej J.

Publication type:

Article

New 1,2,4-oxadiazole derivatives with positive mGlu4 receptor modulation activity and antipsychotic-like properties.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 211, doi. 10.1080/14756366.2021.1998022

By:

Stankiewicz, Anna;
Kaczorowska, Katarzyna;
Bugno, Ryszard;
Kozioł, Aneta;
Paluchowska, Maria H.;
Burnat, Grzegorz;
Chruścicka, Barbara;
Chorobik, Paulina;
Brański, Piotr;
Wierońska, Joanna M.;
Duszyńska, Beata;
Pilc, Andrzej;
Bojarski, Andrzej J.

Publication type:

Article

Arylpiperazinylalkyl derivatives of 8-amino-1,3-dimethylpurine-2,6-dione as novel multitarget 5-HT/D receptor agents with potential antipsychotic activity.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1048, doi. 10.3109/14756366.2015.1088844

By:

Chłoń-Rzepa, Grażyna;
Bucki, Adam;
Kołaczkowski, Marcin;
Partyka, Anna;
Jastrzębska-Więsek, Magdalena;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Kalinowska-Tłuścik, Justyna;
Kazek, Grzegorz;
Mordyl, Barbara;
Głuch-Lutwin, Monika;
Wesołowska, Anna

Publication type:

Article

Variation, Natural Selection, and Information Content - A Simulation.

Published in:

Chemistry & Biodiversity, 2007, v. 4, n. 10, p. 2458, doi. 10.1002/cbdv.200790200

By:

Testa, Bernard;
Bojarski, Andrzej J.

Publication type:

Article

Conformational Fluctuations versus Constraints in Amino Acid Side Chains: The Evolution of Information Content from Free Amino Acids to Proteins.

Published in:

Chemistry & Biodiversity, 2006, v. 3, n. 3, p. 245, doi. 10.1002/cbdv.200690029

By:

Bojarski, Andrzej J.;
Nowak, Mateusz;
Testa, Bernard

Publication type:

Article

The influence of the negative-positive ratio and screening database size on the performance of machine learning-based virtual screening.

Published in:

PLoS ONE, 2017, v. 12, n. 4, p. 1, doi. 10.1371/journal.pone.0175410

By:

Kurczab, Rafał;
Bojarski, Andrzej J.

Publication type:

Article

Ligand-guided homology modelling of the GABAB2 subunit of the GABAB receptor.

Published in:

PLoS ONE, 2017, v. 12, n. 3, p. 1, doi. 10.1371/journal.pone.0173889

By:

Freyd, Thibaud;
Warszycki, Dawid;
Mordalski, Stefan;
Bojarski, Andrzej J.;
Sylte, Ingebrigt;
Gabrielsen, Mari

Publication type:

Article

1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT 6 R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity.

Published in:

Biomolecules (2218-273X), 2023, v. 13, n. 1, p. 12, doi. 10.3390/biom13010012

By:

Canale, Vittorio;
Trybała, Wojciech;
Chaumont-Dubel, Séverine;
Koczurkiewicz-Adamczyk, Paulina;
Satała, Grzegorz;
Bento, Ophélie;
Blicharz-Futera, Klaudia;
Bantreil, Xavier;
Pękala, Elżbieta;
Bojarski, Andrzej J.;
Lamaty, Frédéric;
Marin, Philippe;
Zajdel, Paweł

Publication type:

Article

Data-Driven Analysis of Fluorination of Ligands of Aminergic G Protein Coupled Receptors.

Published in:

Biomolecules (2218-273X), 2021, v. 11, n. 11, p. 1647, doi. 10.3390/biom11111647

By:

Pietruś, Wojciech;
Kurczab, Rafał;
Stumpfe, Dagmar;
Bojarski, Andrzej J.;
Bajorath, Jürgen

Publication type:

Article

Exploring protein hotspots by optimized fragment pharmacophores.

Published in:

Nature Communications, 2021, v. 12, n. 1, p. 1, doi. 10.1038/s41467-021-23443-y

By:

Bajusz, Dávid;
Wade, Warren S.;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Ilaš, Janez;
Ebner, Jessica;
Grebien, Florian;
Papp, Henrietta;
Jakab, Ferenc;
Douangamath, Alice;
Fearon, Daren;
von Delft, Frank;
Schuller, Marion;
Ahel, Ivan;
Wakefield, Amanda;
Vajda, Sándor;
Gerencsér, János;
Pallai, Péter;
Keserű, György M.

Publication type:

Article

ONIOM and FMO‐EDA study of metabotropic glutamate receptor 1: Quantum insights into the allosteric binding site.

Published in:

International Journal of Quantum Chemistry, 2018, v. 118, n. 15, p. 1, doi. 10.1002/qua.25617

By:

Śliwa, Paweł;
Kurczab, Rafał;
Bojarski, Andrzej J.

Publication type:

Article

Allosteric Inhibition of Serotonin 5-HT7 Receptors by Zinc Ions.

Published in:

Molecular Neurobiology, 2018, v. 55, n. 4, p. 2897, doi. 10.1007/s12035-017-0536-0

By:

Satała, Grzegorz;
Duszyńska, Beata;
Lenda, Tomasz;
Nowak, Gabriel;
Bojarski, Andrzej J.

Publication type:

Article

Structure-5-HT/D2 Receptor Affinity Relationship in a New Group of 1-Arylpiperazynylalkyl Derivatives of 8-Dialkylamino-3,7-dimethyl-1 H-purine-2,6(3 H,7 H)-dione.

Published in:

Archiv der Pharmazie, 2016, v. 349, n. 10, p. 774, doi. 10.1002/ardp.201600162

By:

Żmudzki, Paweł;
Satała, Grzegorz;
Chłoń ‐ Rzepa, Grażyna;
Bojarski, Andrzej J.;
Kazek, Grzegorz;
Siwek, Agata;
Gryboś, Anna;
Głuch ‐ Lutwin, Monika;
Wesołowska, Anna;
Pawłowski, Maciej

Publication type:

Article

New Arylpiperazinylalkyl Derivatives of 8-Alkoxy-purine-2,6-dione and Dihydro[1,3]oxazolo[2,3- f]purinedione Targeting the Serotonin 5-HT1A/5-HT2A/5-HT7 and Dopamine D2 Receptors.

Published in:

Archiv der Pharmazie, 2015, v. 348, n. 4, p. 242, doi. 10.1002/ardp.201500015

By:

Chłoń ‐ Rzepa, Grażyna;
Zagórska, Agnieszka;
Bucki, Adam;
Kołaczkowski, Marcin;
Pawłowski, Maciej;
Satała, Grzegorz;
Bojarski, Andrzej J.;
Partyka, Anna;
Wesołowska, Anna;
Pękala, Elżbieta;
Słoczyńska, Karolina

Publication type:

Article

Structure-5-HT Receptor Affinity Relationship in a New Group of 7-Arylpiperazynylalkyl and 7-Tetrahydroisoquinolinylalkyl Derivatives of 8-Amino-1,3-dimethyl-1 H-purine-2,6(3 H,7 H)-dione.

Published in:

Archiv der Pharmazie, 2015, v. 348, n. 4, p. 229, doi. 10.1002/ardp.201400392

By:

Żmudzki, Paweł;
Chłoń ‐ Rzepa, Grażyna;
Bojarski, Andrzej J.;
Zygmunt, Małgorzata;
Kazek, Grzegorz;
Mordyl, Barbara;
Pawłowski, Maciej

Publication type:

Article

New Arylpiperazines with Flexible versus Partly Constrained Linker as Serotonin 5-HT1A/5-HT7 Receptor Ligands.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 5, p. 339, doi. 10.1002/ardp.201300011

By:

Kowalski, Piotr;
Mitka, Katarzyna;
Jaśkowska, Jolanta;
Duszyńska, Beata;
Bojarski, Andrzej J.

Publication type:

Article

Quinolinesulfonamides of Aryloxy-/Arylthio-ethyl Piperidines: Influence of an Arylether Fragment on 5-HT1A/5-HT7 Receptor Selectivity.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 3, p. 180, doi. 10.1002/ardp.201200322

By:

Grychowska, Katarzyna;
Marciniec, Krzysztof;
Canale, Vittorio;
Szymiec, Michał;
Glanowski, Grzegorz;
Satała, Grzegorz;
Maślankiewicz, Andrzej;
Pawłowski, Maciej;
Bojarski, Andrzej J.;
Zajdel, Paweł

Publication type:

Article

Novel Mannich Bases, 5-Arylimidazolidine-2,4-dione Derivatives with Dual 5-HT1A Receptor and Serotonin Transporter Affinity.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 2, p. 98, doi. 10.1002/ardp.201200378

By:

Czopek, Anna;
Kołaczkowski, Marcin;
Bucki, Adam;
Byrtus, Hanna;
Pawłowski, Maciej;
Siwek, Agata;
Bojarski, Andrzej J.;
Bednarski, Marek;
Wróbel, Dagmara;
Wesołowska, Anna

Publication type:

Article

Conformational Restriction in Novel NAN-190 and MP3022 Analogs and Their 5-HT1A Receptor Activity.

Published in:

Archiv der Pharmazie, 2006, v. 339, n. 9, p. 498

By:

Ryszard Bugno;
Sijka Charakchieva-Minol;
Andrzej J. Bojarski;
Ewa Tatarczyńska;
Ewa Chojnacka-Wójcik

Publication type:

Article

Modification of the Structure of 4, 6-Disubstituted 2-(4-Alkyl-1-piperazinyl)pyridines: Synthesis and Their 5-HT2A Receptor Activity.

Published in:

Archiv der Pharmazie, 2003, v. 336, n. 2, p. 104, doi. 10.1002/ardp.200390006

By:

Maria H. Paluchowska;
Andrzej J. Bojarski;
Ryszard Bugno;
Sijka Charakchieva-Minol;
Anna Wesołowska

Publication type:

Article

Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT 6 and D 3 R Affinity in the 1 H -Pyrrolo[3,2- c ]quinoline Series.

Published in:

Molecules, 2023, v. 28, n. 3, p. 1096, doi. 10.3390/molecules28031096

By:

Grychowska, Katarzyna;
Pietruś, Wojciech;
Kulawik, Ludmiła;
Bento, Ophélie;
Satała, Grzegorz;
Bantreil, Xavier;
Lamaty, Frédéric;
Bojarski, Andrzej J.;
Gołębiowska, Joanna;
Nikiforuk, Agnieszka;
Marin, Philippe;
Chaumont-Dubel, Séverine;
Kurczab, Rafał;
Zajdel, Paweł

Publication type:

Article

Isomeric Activity Cliffs—A Case Study for Fluorine Substitution of Aminergic G Protein-Coupled Receptor Ligands.

Published in:

Molecules, 2023, v. 28, n. 2, p. 490, doi. 10.3390/molecules28020490

By:

Pietruś, Wojciech;
Kurczab, Rafał;
Warszycki, Dawid;
Bojarski, Andrzej J.;
Bajorath, Jürgen

Publication type:

Article

Hydrogen Bonds with Fluorine in Ligand–Protein Complexes-the PDB Analysis and Energy Calculations.

Published in:

Molecules, 2022, v. 27, n. 3, p. 1005, doi. 10.3390/molecules27031005

By:

Pietruś, Wojciech;
Kafel, Rafał;
Bojarski, Andrzej J.;
Kurczab, Rafał

Publication type:

Article