Works by Bergare, Jonas

Results: 12

Synthesis of C‐14 labeled Rac‐(3R,2S)‐glycopyrronium bromide.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2020, v. 63, n. 10, p. 456, doi. 10.1002/jlcr.3864

By:

Bergare, Jonas;
Nixon, Neil;
Newsome, Jeffery;
Thunberg, Linda;
Elmore, Charles S.

Publication type:

Article

The synthesis of one H‐2 labeled and two H‐3 labeled leukotriene C4 synthase inhibitors.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2020, v. 63, n. 10, p. 434, doi. 10.1002/jlcr.3862

By:

Bergare, Jonas;
Kingston, Lee;
Guly, Dominic J.;
Dolan, James;
Lewis, Richard J.;
Elmore, Charles S.

Publication type:

Article

Synthesis, 3H‐labelling and in vitro evaluation of a substituted dipiperidine alcohol as a potential ligand for chemokine receptor 2.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2019, v. 62, n. 6, p. 265, doi. 10.1002/jlcr.3731

By:

Artelsmair, Markus;
Miranda‐Azpiazu, Patricia;
Kingston, Lee;
Bergare, Jonas;
Schou, Magnus;
Varrone, Andrea;
Elmore, Charles S.

Publication type:

Article

Synthesis of 2 C-14 labeled cathepsin C inhibitors: The use of a cyanide to displace a Benzotriazole.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2017, v. 60, n. 6, p. 294, doi. 10.1002/jlcr.3502

By:

Kingston, Lee;
Bergare, Jonas;
Lönn, Hans;
Ericsson, Cecilia;
Grönberg, Gunnar;
Chen, Song;
Elmore, Charles S.

Publication type:

Article

Synthesis of 1β-hydroxydeoxycholic acid in H-2 and unlabeled forms.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2017, v. 60, n. 4, p. 221, doi. 10.1002/jlcr.3495

By:

Hayes, Martin A.;
Roberts, Ieuan;
Grönberg, Gunnar;
Lv, Kexin;
Lin, Baorui;
Bergare, Jonas;
Elmore, Charles S.

Publication type:

Article

Selective Deuteration and Tritiation of Pharmaceutically Relevant Sulfoximines.

Published in:

Angewandte Chemie International Edition, 2025, v. 64, n. 5, p. 1, doi. 10.1002/anie.202417179

By:

Smith, Blair I. P.;
Knight, Nathan M. L.;
Knox, Gary J.;
Lindsay, David M.;
Paterson, Laura C.;
Bergare, Jonas;
Elmore, Charles S.;
Bragg, Ryan A.;
Kerr, William J.

Publication type:

Article

Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone.

Published in:

Journal of Labelled Compounds & Radiopharmaceuticals, 2024, v. 67, n. 4, p. 145, doi. 10.1002/jlcr.4089

By:

Bergare, Jonas;
Bailey, Christopher;
Sörensen, Henrik;
Grönberg, Gunnar;
Broberg, Karl;
Berglund, Monica;
Grecu, Tudor;
Sanchez, Carolina;
Emtenäs, Hans;
Bragg, Ryan A.;
Elmore, Charles S.

Publication type:

Article

Selective Deuteration and Tritiation of Pharmaceutically Relevant Sulfoximines.

Published in:

Angewandte Chemie, 2025, v. 137, n. 5, p. 1, doi. 10.1002/ange.202417179

By:

Smith, Blair I. P.;
Knight, Nathan M. L.;
Knox, Gary J.;
Lindsay, David M.;
Paterson, Laura C.;
Bergare, Jonas;
Elmore, Charles S.;
Bragg, Ryan A.;
Kerr, William J.

Publication type:

Article

Pharmacokinetic Evaluation of New Drugs Using a Multi-Labelling Approach and PET Imaging: Application to a Drug Candidate with Potential Application in Neuromuscular Disorders.

Published in:

Biomedicines, 2023, v. 11, n. 2, p. 253, doi. 10.3390/biomedicines11020253

By:

Passannante, Rossana;
Gómez-Vallejo, Vanessa;
Sagartzazu-Aizpurua, Maialen;
Vignau Arsuaga, Laura;
Marco-Moreno, Pablo;
Aldanondo, Garazi;
Vallejo-Illarramendi, Ainara;
Aguiar, Pablo;
Cossío, Unai;
Martín, Abraham;
Bergare, Jonas;
Kingston, Lee;
Elmore, Charles S.;
Morcillo, Miguel Angel;
Ferrón, Pablo;
Aizpurua, Jesus M.;
Llop, Jordi

Publication type:

Article

Rapid and Efficient Synthesis of 11C‐Labeled Benzimidazolones Using [11C]Carbon Dioxide.

Published in:

ChemistrySelect, 2019, v. 4, n. 6, p. 1846, doi. 10.1002/slct.201803561

By:

Horkka, Kaisa;
Dahl, Kenneth;
Bergare, Jonas;
Elmore, Charles S.;
Halldin, Christer;
Schou, Magnus

Publication type:

Article

Efficient palladium-catalyzed electrocarboxylation enables late-stage carbon isotope labelling.

Published in:

Nature Communications, 2024, v. 15, n. 1, p. 1, doi. 10.1038/s41467-024-46820-9

By:

Batista, Gabriel M. F.;
Ebenbauer, Ruth;
Day, Craig;
Bergare, Jonas;
Neumann, Karoline T.;
Hopmann, Kathrin H.;
Elmore, Charles S.;
Rosas-Hernández, Alonso;
Skrydstrup, Troels

Publication type:

Article

Synthesis and preclinical evaluation of [11C]EAI045 as a PET tracer for imaging tumors expressing mutated epidermal growth factor receptor.

Published in:

EJNMMI Research, 2024, v. 14, p. 1, doi. 10.1186/s13550-024-01078-6

By:

Högnäsbacka, Antonia A.;
Poot, Alex J.;
Plisson, Christophe;
Bergare, Jonas;
Bonsall, David R.;
McCluskey, Stuart P.;
Wells, Lisa A.;
Kooijman, Esther;
Schuit, Robert C.;
Verlaan, Mariska;
Beaino, Wissam;
van Dongen, Guus A. M. S.;
Vugts, Danielle J.;
Elmore, Charles S.;
Passchier, Jan;
Windhorst, Albert D.

Publication type:

Article

Works by Bergare, Jonas

Synthesis of C‐14 labeled Rac‐(3R,2S)‐glycopyrronium bromide.

The synthesis of one H‐2 labeled and two H‐3 labeled leukotriene C4 synthase inhibitors.

Synthesis, <sup>3</sup>H‐labelling and in vitro evaluation of a substituted dipiperidine alcohol as a potential ligand for chemokine receptor 2.

Synthesis of 2 C-14 labeled cathepsin C inhibitors: The use of a cyanide to displace a Benzotriazole.

Synthesis of 1β-hydroxydeoxycholic acid in H-2 and unlabeled forms.

Selective Deuteration and Tritiation of Pharmaceutically Relevant Sulfoximines.

Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone.

Selective Deuteration and Tritiation of Pharmaceutically Relevant Sulfoximines.

Pharmacokinetic Evaluation of New Drugs Using a Multi-Labelling Approach and PET Imaging: Application to a Drug Candidate with Potential Application in Neuromuscular Disorders.

Rapid and Efficient Synthesis of <sup>11</sup>C‐Labeled Benzimidazolones Using [<sup>11</sup>C]Carbon Dioxide.

Efficient palladium-catalyzed electrocarboxylation enables late-stage carbon isotope labelling.

Synthesis and preclinical evaluation of [<sup>11</sup>C]EAI045 as a PET tracer for imaging tumors expressing mutated epidermal growth factor receptor.