Works matching AU Bach, Stéphane


Results: 50
    1

    New Insights into the Anticancer Effects and Toxicogenomic Safety of Two β-Lapachone Derivatives.

    Published in:
    Pharmaceuticals (14248247), 2025, v. 18, n. 6, p. 837, doi. 10.3390/ph18060837
    By:
    • De Lima, José Rivaldo;
    • Da Silva Góes, Alexandre José;
    • De Oliveira Borba, Elizabeth Fernanda;
    • da Silva, Meykson Alexandre;
    • Caiana, Rodrigo Ribeiro Alves;
    • Rodrigues, Maria do Desterro;
    • De Lima Silva, Mariza Severina;
    • Chagas, Cristiano Aparecido;
    • Baratte, Blandine;
    • Robert, Thomas;
    • Bach, Stéphane;
    • Ourliac-Garnier, Isabelle;
    • Marchand, Pascal;
    • Da Silva, Teresinha Gonçalves
    Publication type:
    Article
    2

    Development of a novel family of antifungal agents based on a quinone methide oxime framework.

    Published in:
    Scientific Reports, 2025, v. 15, n. 1, p. 1, doi. 10.1038/s41598-025-98609-5
    By:
    • Janeczko, Monika;
    • Masłyk, Maciej;
    • Demchuk, Oleg M.;
    • Kurowska-Okoń, Antonina;
    • Kwaśnik, Mateusz;
    • Górka, Kamila;
    • Martyna, Aleksandra;
    • Foll-Josselin, Béatrice;
    • Ruchaud, Sandrine;
    • Bach, Stéphane;
    • Woliński, Przemysław;
    • Jasiński, Radomir;
    • Mirosław, Barbara;
    • Sadczuk, Małgorzata;
    • Kubiński, Konrad
    Publication type:
    Article
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    Biological Evaluation of Arylsemicarbazone Derivatives as Potential Anticancer Agents.

    Published in:
    Pharmaceuticals (14248247), 2019, v. 12, n. 4, p. 169, doi. 10.3390/ph12040169
    By:
    • Nascimento da Cruz, Anne Cecília;
    • Brondani, Dalci José;
    • I´talo de Santana, Temístocles;
    • Oliveira da Silva, Lucas;
    • da Oliveira Borba, Elizabeth Fernanda;
    • de Faria, Antônio Rodolfo;
    • Ferreira Cavalcanti de Albuquerque, Julianna;
    • Piessard, Sylvie;
    • Matos Ximenes, Rafael;
    • Baratte, Blandine;
    • Bach, Stéphane;
    • Ruchaud, Sandrine;
    • Bezerra Mendonça Junior, Francisco Jaime;
    • Bazin, Marc-Antoine;
    • Montenegro Rabello, Marcelo;
    • Zaldini Hernandes, Marcelo;
    • Marchand, Pascal;
    • Gonçalves da Silva, Teresinha
    Publication type:
    Article
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    Design of new disubstituted imidazo[1,2-b]pyridazine derivatives as selective Haspin inhibitors. Synthesis, binding mode and anticancer biological evaluation.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1840, doi. 10.1080/14756366.2020.1825408
    By:
    • Elie, Jonathan;
    • Feizbakhsh, Omid;
    • Desban, Nathalie;
    • Josselin, Béatrice;
    • Baratte, Blandine;
    • Bescond, Amandine;
    • Duez, Julien;
    • Fant, Xavier;
    • Bach, Stéphane;
    • Marie, Dominique;
    • Place, Matthieu;
    • Ben Salah, Sami;
    • Chartier, Agnes;
    • Berteina-Raboin, Sabine;
    • Chaikuad, Apirat;
    • Knapp, Stefan;
    • Carles, Fabrice;
    • Bonnet, Pascal;
    • Buron, Frédéric;
    • Routier, Sylvain
    Publication type:
    Article
    9

    An Optimized Workflow for the Discovery of New Antimicrobial Compounds Targeting Bacterial RNA Polymerase Complex Formation.

    Published in:
    Antibiotics (2079-6382), 2022, v. 11, n. 10, p. N.PAG, doi. 10.3390/antibiotics11101449
    By:
    • Caputo, Alessia;
    • Sartini, Sara;
    • Levati, Elisabetta;
    • Minato, Ilaria;
    • Elisi, Gian Marco;
    • Di Stasi, Adriana;
    • Guillou, Catherine;
    • Goekjian, Peter G.;
    • Garcia, Pierre;
    • Gueyrard, David;
    • Bach, Stéphane;
    • Comte, Arnaud;
    • Ottonello, Simone;
    • Rivara, Silvia;
    • Montanini, Barbara
    Publication type:
    Article
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    Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N-Arylation Reactions and Biological Properties.

    Published in:
    European Journal of Organic Chemistry, 2017, v. 2017, n. 39, p. 5903, doi. 10.1002/ejoc.201701004
    By:
    • Hedidi, Madani;
    • Maillard, Julien;
    • Erb, William;
    • Lassagne, Frédéric;
    • Halauko, Yury S.;
    • Ivashkevich, Oleg A.;
    • Matulis, Vadim E.;
    • Roisnel, Thierry;
    • Dorcet, Vincent;
    • Hamzé, Monzer;
    • Fajloun, Ziad;
    • Baratte, Blandine;
    • Ruchaud, Sandrine;
    • Bach, Stéphane;
    • Bentabed‐Ababsa, Ghenia;
    • Mongin, Florence
    Publication type:
    Article
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    Le criblage à Roscoff.

    Published in:
    Médecine Sciences, 2015, v. 31, n. 5, p. 538, doi. 10.1051/medsci/20153105016
    By:
    • Baratte, Blandine;
    • Serive, Benoît;
    • Bach, Stéphane
    Publication type:
    Article
    20

    Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases.

    Published in:
    Molecules, 2015, v. 20, n. 7, p. 12412, doi. 10.3390/molecules200712412
    By:
    • Dago, Camille Déliko;
    • Ambeu, Christelle N´ta;
    • Coulibaly, Wacothon-Karime;
    • Békro, Yves-Alain;
    • Mamyrbékova, Janat;
    • Defontaine, Audrey;
    • Baratte, Blandine;
    • Bach, Stéphane;
    • Ruchaud, Sandrine;
    • Le Guével, Rémy;
    • Ravache, Myriam;
    • Corlu, Anne;
    • Bazureau, Jean-Pierre
    Publication type:
    Article
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    Protein Folding Activity of Ribosomal RNA Is a Selective Target of Two Unrelated Antiprion Drugs.

    Published in:
    PLoS ONE, 2008, v. 3, n. 5, p. 1, doi. 10.1371/journal.pone.0002174
    By:
    • Tribouillard-Tanvier, Déborah;
    • Reis, Suzana Dos;
    • Gug, Fabienne;
    • Voisset, Cécile;
    • Béringue, Vincent;
    • Sabate, Raimon;
    • Kikovska, Ema;
    • Talarek, Nicolas;
    • Bach, Stéphane;
    • Huang, Chenhui;
    • Desban, Nathalie;
    • Saupe, Sven J.;
    • Supattapone, Surachai;
    • Thuret, Jean-Yves;
    • Chédin, Stéphane;
    • Vilette, Didier;
    • Galons, Hervé;
    • Sanyal, Suparna;
    • Blondel, Marc
    Publication type:
    Article
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    Using budding yeast to screen for anti-prion drugs.

    Published in:
    Biotechnology Journal, 2006, v. 1, n. 1, p. 58, doi. 10.1002/biot.200500001
    By:
    • Tribouillard, Déborah;
    • Bach, Stéphane;
    • Gug, Fabienne;
    • Desban, Nathalie;
    • Beringue, Vincent;
    • Andrieu, Thibault;
    • Dormont, Dominique;
    • Galons, Hervé;
    • Laude, Hubert;
    • Vilette, Didier;
    • Blondel, Marc
    Publication type:
    Article
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    Nigratine as dual inhibitor of necroptosis and ferroptosis regulated cell death.

    Published in:
    Scientific Reports, 2022, v. 12, n. 1, p. 1, doi. 10.1038/s41598-022-09019-w
    By:
    • Delehouzé, Claire;
    • Comte, Arnaud;
    • Leon-Icaza, Stephen Adonai;
    • Cougoule, Céline;
    • Hauteville, Marcelle;
    • Goekjian, Peter;
    • Bulinski, Jeannette Chloë;
    • Dimanche-Boitrel, Marie-Thérèse;
    • Meunier, Etienne;
    • Rousselot, Morgane;
    • Bach, Stéphane
    Publication type:
    Article
    32

    Investigating the C2 Modulation of the Imidazo[1,2‐a]pyrazine‐Based Hit Compound CTN1122: Synthesis, in vitro Antileishmanial Activity, Cytotoxicity and Casein Kinase 1 Inhibition.

    Published in:
    ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400862
    By:
    • Tisseur, Lhana;
    • Cojean, Sandrine;
    • Gassama, Khadidiatou;
    • Logé, Cédric;
    • Pagniez, Fabrice;
    • Cavé, Christian;
    • Bernadat, Guillaume;
    • Loiseau, Philippe M.;
    • Bach, Stéphane;
    • Thiéfaine, Jérôme;
    • Picot, Carine;
    • Tomasoni, Christophe;
    • Leclercq, Olivier;
    • Baratte, Blandine;
    • Robert, Thomas;
    • Le Pape, Patrice;
    • Rachidi, Najma;
    • Bazin, Marc‐Antoine;
    • Marchand, Pascal
    Publication type:
    Article
    33

    New Fusarochromanone Derivatives from the Marine Fungus Fusarium equiseti UBOCC-A-117302.

    Published in:
    Marine Drugs, 2024, v. 22, n. 10, p. 444, doi. 10.3390/md22100444
    By:
    • Pham, Giang Nam;
    • Josselin, Béatrice;
    • Cousseau, Arnaud;
    • Baratte, Blandine;
    • Dayras, Marie;
    • Le Meur, Christophe;
    • Debaets, Stella;
    • Weill, Amélie;
    • Robert, Thomas;
    • Burgaud, Gaëtan;
    • Probert, Ian;
    • Abdoul-Latif, Fatouma Mohamed;
    • Boyer, Laurent;
    • Bach, Stéphane;
    • Mehiri, Mohamed
    Publication type:
    Article
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    Bioprospecting Marine Plankton.

    Published in:
    Marine Drugs, 2013, v. 11, n. 11, p. 4594, doi. 10.3390/md11114594
    By:
    • Abida, Heni;
    • Ruchaud, Sandrine;
    • Rios, Laurent;
    • Humeau, Anne;
    • Probert, Ian;
    • De Vargas, Colomban;
    • Bach, Stéphane;
    • Bowler, Chris
    Publication type:
    Article
    39

    Structure Activity Relationship Studies around DB18 , a Potent and Selective Inhibitor of CLK Kinases.

    Published in:
    Molecules, 2022, v. 27, n. 19, p. 6149, doi. 10.3390/molecules27196149
    By:
    • Brahmaiah, Dabbugoddu;
    • Bhavani, Anagani Kanaka Durga;
    • Aparna, Pasula;
    • Kumar, Nangunoori Sampath;
    • Solhi, Hélène;
    • Le Guevel, Rémy;
    • Baratte, Blandine;
    • Robert, Thomas;
    • Ruchaud, Sandrine;
    • Bach, Stéphane;
    • Jadav, Surender Singh;
    • Reddy, Chada Raji;
    • Mosset, Paul;
    • Gouault, Nicolas;
    • Levoin, Nicolas;
    • Grée, René
    Publication type:
    Article
    40

    Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases.

    Published in:
    Molecules, 2021, v. 26, n. 21, p. 6572, doi. 10.3390/molecules26216572
    By:
    • Dao, Viet Hung;
    • Ourliac-Garnier, Isabelle;
    • Logé, Cédric;
    • McCarthy, Florence O.;
    • Bach, Stéphane;
    • da Silva, Teresinha Gonçalves;
    • Denevault-Sabourin, Caroline;
    • Thiéfaine, Jérôme;
    • Baratte, Blandine;
    • Robert, Thomas;
    • Gouilleux, Fabrice;
    • Brachet-Botineau, Marie;
    • Bazin, Marc-Antoine;
    • Marchand, Pascal
    Publication type:
    Article
    41

    Betulin, a Newly Characterized Compound in Acacia auriculiformis Bark, Is a Multi-Target Protein Kinase Inhibitor.

    Published in:
    Molecules, 2021, v. 26, n. 15, p. 4599, doi. 10.3390/molecules26154599
    By:
    • Ahmadu, Augustine A.;
    • Delehouzé, Claire;
    • Haruna, Anas;
    • Mustapha, Lukman;
    • Lawal, Bilqis A.;
    • Udobre, Aniefiok;
    • Baratte, Blandine;
    • Triscornia, Camilla;
    • Autret, Axelle;
    • Robert, Thomas;
    • Bulinski, Jeannette Chloë;
    • Rousselot, Morgane;
    • Simoes Eugénio, Mélanie;
    • Dimanche-Boitrel, Marie-Thérèse;
    • Petzer, Jacobus P.;
    • Legoabe, Lesetja J.;
    • Bach, Stéphane
    Publication type:
    Article
    42

    New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation.

    Published in:
    Molecules, 2021, v. 26, n. 4, p. 867, doi. 10.3390/molecules26040867
    By:
    • Oyallon, Bruno;
    • Brachet-Botineau, Marie;
    • Logé, Cédric;
    • Robert, Thomas;
    • Bach, Stéphane;
    • Ibrahim, Sajida;
    • Raoul, William;
    • Croix, Cécile;
    • Berthelot, Pascal;
    • Guillon, Jean;
    • Pinaud, Noël;
    • Gouilleux, Fabrice;
    • Viaud-Massuard, Marie-Claude;
    • Denevault-Sabourin, Caroline;
    • Denny, William A.;
    • Chiara, Brullo
    Publication type:
    Article
    43

    The Anti-Candida albicans Agent 4-AN Inhibits Multiple Protein Kinases.

    Published in:
    Molecules, 2019, v. 24, n. 1, p. 153, doi. 10.3390/molecules24010153
    By:
    • Masłyk, Maciej;
    • Janeczko, Monika;
    • Martyna, Aleksandra;
    • Czernik, Sławomir;
    • Tokarska-Rodak, Małgorzata;
    • Chwedczuk, Marta;
    • Foll-Josselin, Béatrice;
    • Ruchaud, Sandrine;
    • Bach, Stéphane;
    • Demchuk, Oleg M.;
    • Kubiński, Konrad
    Publication type:
    Article
    44

    From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines.

    Published in:
    Molecules, 2018, v. 23, n. 11, p. 2961, doi. 10.3390/molecules23112961
    By:
    • Lassagne, Frédéric;
    • Langlais, Timothy;
    • Caytan, Elsa;
    • Limanton, Emmanuelle;
    • Paquin, Ludovic;
    • Boullard, Manon;
    • Courtel, Coline;
    • Curbet, Idriss;
    • Gédéon, Clément;
    • Lebreton, Julien;
    • Picot, Laurent;
    • Thiéry, Valérie;
    • Souab, Mohamed;
    • Baratte, Blandine;
    • Ruchaud, Sandrine;
    • Bach, Stéphane;
    • Roisnel, Thierry;
    • Mongin, Florence;
    • Bunce, Richard A.
    Publication type:
    Article
    45

    Design and Synthesis of Functionalized 2,4-Diamino-1,3,5-Triazines, Potential Inhibitors Involved in Immune and Inflammatory Response.

    Published in:
    International Journal of Pharmaceutical Research & Allied Sciences, 2024, v. 13, n. 4, p. 1, doi. 10.51847/hsT2C61XWx
    By:
    • Diakité, Amelanh Sica;
    • Ambeu-Loko, Christelle N'ta Mélissa;
    • Yapi, Ange Désiré;
    • Logé, Cédric;
    • Kacou, Alain;
    • Kra, Stéphanie;
    • Baratte, Blandine;
    • Bach, Stéphane;
    • Ruchaud, Sandrine;
    • Sissouma, Drissa;
    • Ouattara, Mahama;
    • Robert, Jean-michel
    Publication type:
    Article
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    Correction to: Phenytoin inhibits necroptosis.

    Published in:
    2018
    By:
    • von Mässenhausen, Anne;
    • Tonnus, Wulf;
    • Himmerkus, Nina;
    • Parmentier, Simon;
    • Saleh, Danish;
    • Rodriguez, Diego;
    • Ousingsawat, Jiraporn;
    • Ang, Rosalind L.;
    • Weinberg, Joel M.;
    • Sanz, Ana B.;
    • Ortiz, Alberto;
    • Zierleyn, Adrian;
    • Becker, Jan Ulrich;
    • Baratte, Blandine;
    • Desban, Nathalie;
    • Bach, Stéphane;
    • Schiessl, Ina Maria;
    • Nogusa, Shoko;
    • Balachandran, Siddharth;
    • Anders, Hans Joachim
    Publication type:
    Correction Notice
    48

    Phenytoin inhibits necroptosis.

    Published in:
    Cell Death & Disease, 2018, v. 9, n. 3, p. 1, doi. 10.1038/s41419-018-0394-3
    By:
    • von Mässenhausen, Anne;
    • Tonnus, Wulf;
    • Himmerkus, Nina;
    • Parmentier, Simon;
    • Saleh, Danish;
    • Rodriguez, Diego;
    • Ousingsawat, Jiraporn;
    • Ang, Rosalind L.;
    • Weinberg, Joel M.;
    • Sanz, Ana B.;
    • Ortiz, Alberto;
    • Zierleyn, Adrian;
    • Becker, Jan Ulrich;
    • Baratte, Blandine;
    • Desban, Nathalie;
    • Bach, Stéphane;
    • Schiessl, Ina Maria;
    • Nogusa, Shoko;
    • Balachandran, Siddharth;
    • Anders, Hans Joachim
    Publication type:
    Article
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    Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis.

    Published in:
    FEBS Journal, 2017, v. 284, n. 18, p. 3050, doi. 10.1111/febs.14176
    By:
    • Le Cann, Fabienne;
    • Delehouzé, Claire;
    • Leverrier ‐ Penna, Sabrina;
    • Filliol, Aveline;
    • Comte, Arnaud;
    • Delalande, Olivier;
    • Desban, Nathalie;
    • Baratte, Blandine;
    • Gallais, Isabelle;
    • Piquet ‐ Pellorce, Claire;
    • Faurez, Florence;
    • Bonnet, Marion;
    • Mettey, Yvette;
    • Goekjian, Peter;
    • Samson, Michel;
    • Vandenabeele, Peter;
    • Bach, Stéphane;
    • Dimanche ‐ Boitrel, Marie ‐ Thérèse
    Publication type:
    Article