Works by Awad, Samir M.

Results: 15

Synthesis and evaluation of antipyrine derivatives bearing a thiazole moiety as antibacterial and antifungal agents.

Published in:

Synthetic Communications, 2023, v. 53, n. 21, p. 1812, doi. 10.1080/00397911.2023.2248306

By:

Abbas, Samir Y.;
Abd El-Aziz, Maha M.;
Awad, Samir M.;
Mohamed, Mosaad S.

Publication type:

Article

Structural hybrids of sulfonamide and thiazole moieties: Synthesis and evaluation of antimicrobial activity.

Published in:

Synthetic Communications, 2023, v. 53, n. 1, p. 68, doi. 10.1080/00397911.2022.2150086

By:

Abbas, Samir Y.;
Abd El-Aziz, Maha M.;
Awad, Samir M.;
Mohamed, Mosaad S.

Publication type:

Article

Design, synthesis, molecular modelling and biological evaluation of novel 6-amino-5-cyano-2-thiopyrimidine derivatives as potent anticancer agents against leukemia and apoptotic inducers.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2024, v. 39, n. 1, p. 1, doi. 10.1080/14756366.2024.2304625

By:

Ahmed, Naglaa M.;
Mohamed, Mosaad S.;
Awad, Samir M.;
El-tawab, Neama A. Abd;
Gaballah, Mohamed S.;
Said, Ahmed M.

Publication type:

Article

Novel benzo chromene derivatives: design, synthesis, molecular docking, cell cycle arrest, and apoptosis induction in human acute myeloid leukemia HL-60 cells.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 405, doi. 10.1080/14756366.2022.2151592

By:

Abd El-Hameed, Rania H.;
Mohamed, Mosaad S.;
Awad, Samir M.;
Hassan, Bardes B.;
Khodair, Marwa Abd El-Fattah;
Mansour, Yara E.

Publication type:

Article

Antineoplastic Effect of New Synthesized Compounds of 2-Thiouracil Sulfonamide Derivatives against Ovarian and Breast Carcinoma Cells "In Vitro Study".

Published in:

Systematic Reviews in Pharmacy, 2020, v. 11, n. 4, p. 229, doi. 10.31838/srp.2020.4.33

By:

Ahjel, Salam W.;
Hassan, Saif M.;
Hussein, Sinan F.;
Hadi, Najah R.;
Awad, Samir M.

Publication type:

Article

Synthesis of Novel 2-Thiouracil-5-Sulfonamide Derivatives as Potent Inducers of Cell Cycle Arrest and CDK2A Inhibition Supported by Molecular Docking.

Published in:

International Journal of Molecular Sciences, 2021, v. 22, n. 21, p. 11957, doi. 10.3390/ijms222111957

By:

Fatahala, Samar S.;
Sayed, Amira I.;
Mahgoub, Shahenda;
Taha, Heba;
El-Sayed, Mohamed-I kotb;
El-Shehry, Mohamed F.;
Awad, Samir M.;
Abd El-Hameed, Rania H.

Publication type:

Article

Effect of new synthesized compounds of 2-Thiouracil Sulfonamide Derivatives against colon and liver carcinoma cells "In Vitro Study".

Published in:

International Journal of Pharmaceutical Research (09752366), 2020, v. 12, n. 4, p. 2012, doi. 10.31838/ijpr/2020.12.04.286

By:

HASSAN, SAIF M.;
AL-JAF, ASHWAQ NAJEMALDEEN ABBAS;
HUSSIEN, YASMEEN ALI;
AWAD, SAMIR M.;
ABDULKHALEQ, MAYSAA ALI;
HADI, NAJAH R.

Publication type:

Article

Development of nifedipine isosteres: an integrated approach to the design, synthesis, and biological assessment of calcium channel blockers.

Published in:

Frontiers in Chemistry, 2025, p. 1, doi. 10.3389/fchem.2025.1581037

By:

Zohny, Yasser M.;
Awad, Samir M.;
Alsaidan, Omar;
Rabie, Maha A.

Publication type:

Article

Studies on the Reactivity of Amino-1-(6-phenyl-pyridazin-3-yl)-1 H-pyrazole-4-carboxylic Acid Hydrazide Towards Some Reagents for Biological Evaluation.

Published in:

Journal of Heterocyclic Chemistry, 2014, v. 51, n. 4, p. 899, doi. 10.1002/jhet.1724

By:

Shamroukh, Ahmed H.;
Rashad, Aymn E.;
Ali, Hatem S.;
Awad, Samir M.

Publication type:

Article

Synthesis of Certain Pyrimidine Derivatives as Antimicrobial Agents and Anti-Inflammatory Agents.

Published in:

Molecules, 2010, v. 15, n. 3, p. 1882, doi. 10.3390/molecules15031882

By:

Mohamed, Mosaad S.;
Awad, Samir M.;
Sayed, Amira Ibrahim

Publication type:

Article

Synthesis, Anti-Cancer Activity, Cell Cycle Arrest, Apoptosis Induction, and Docking Study of Fused Benzo[ h ]chromeno[2,3- d ]pyrimidine on Human Breast Cancer Cell Line MCF-7.

Published in:

Molecules, 2024, v. 29, n. 19, p. 4697, doi. 10.3390/molecules29194697

By:

Khoder, Zainab M.;
Mohamed, Mosaad S.;
Awad, Samir M.;
Gharib, Amal F.;
Aly, Omnia;
Khodair, Marwa Abd El-Fattah;
Fatahala, Samar S.;
El-Hameed, Rania H. Abd

Publication type:

Article

Design, Synthesis, Molecular Modeling, and Biological Evaluation of Novel Pyrimidine Derivatives as Potential Calcium Channel Blockers.

Published in:

Molecules, 2023, v. 28, n. 12, p. 4869, doi. 10.3390/molecules28124869

By:

Zohny, Yasser M.;
Awad, Samir M.;
Rabie, Maha A.;
Alsaidan, Omar Awad

Publication type:

Article

Novel 2-Thiouracil-5-Sulfonamide Derivatives: Design, Synthesis, Molecular Docking, and Biological Evaluation as Antioxidants with 15-LOX Inhibition.

Published in:

Molecules, 2023, v. 28, n. 4, p. 1925, doi. 10.3390/molecules28041925

By:

Ahmed, Naglaa M.;
Lotfallah, Ahmed H.;
Gaballah, Mohamed S.;
Awad, Samir M.;
Soltan, Moustafa K.

Publication type:

Article

Synthesis of Dihydropyrimidines: Isosteres of Nifedipine and Evaluation of Their Calcium Channel Blocking Efficiency.

Published in:

Molecules, 2023, v. 28, n. 2, p. 784, doi. 10.3390/molecules28020784

By:

Zohny, Yasser M.;
Awad, Samir M.;
Rabie, Maha A.;
Al-Saidan, Omar A.

Publication type:

Article

Design, Synthesis, Molecular Modeling, and Biological Evaluation of Novel Thiouracil Derivatives as Potential Antithyroid Agents.

Published in:

Molecules, 2018, v. 23, n. 11, p. 2913, doi. 10.3390/molecules23112913

By:

Awad, Samir M.;
Zohny, Yasser M.;
Ali, Sahar A.;
Mahgoub, Shahenda;
Said, Ahmed M.

Publication type:

Article