Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond.
- Published in:
- Archiv der Pharmazie, 2025, v. 358, n. 1, p. 1, doi. 10.1002/ardp.202400776
- By:
- Publication type:
- Article
Works matching AU Angeli, Andrea
Results: 181
1
2
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors.
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- Archiv der Pharmazie, 2024, v. 357, n. 11, p. 1, doi. 10.1002/ardp.202400548
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- Publication type:
- Article
3
Sulfonamide‐incorporated bis(α‐aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X‐ray crystallographic studies.
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- Archiv der Pharmazie, 2024, v. 357, n. 7, p. 1, doi. 10.1002/ardp.202400038
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- Publication type:
- Article
4
Design, synthesis, and biological evaluation of 3‐benzenesulfonamide‐linked 3‐hydrazinoisatin derivatives as carbonic anhydrase inhibitors.
- Published in:
- Archiv der Pharmazie, 2024, v. 357, n. 6, p. 1, doi. 10.1002/ardp.202300718
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- Publication type:
- Article
5
Identification of 3‐(5‐cyano‐6‐oxo‐pyridin‐2‐yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity.
- Published in:
- Archiv der Pharmazie, 2024, v. 357, n. 1, p. 1, doi. 10.1002/ardp.202300449
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- Publication type:
- Article
6
Design, synthesis, and structure–activity studies of new rhodanine derivatives as carbonic anhydrase II, IX inhibitors.
- Published in:
- Archiv der Pharmazie, 2023, v. 356, n. 9, p. 1, doi. 10.1002/ardp.202300205
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- Publication type:
- Article
7
Tail approach synthesis of triazolylthiazolotriazole bearing benzenesulfonamides as carbonic anhydrase inhibitors capable of inducing apoptosis.
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- Archiv der Pharmazie, 2023, v. 356, n. 2, p. 1, doi. 10.1002/ardp.202200439
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- Publication type:
- Article
8
Benzenesulfonamides with trisubstituted triazole motif as selective carbonic anhydrase I, II, IV, and IX inhibitors.
- Published in:
- Archiv der Pharmazie, 2023, v. 356, n. 1, p. 1, doi. 10.1002/ardp.202200391
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- Publication type:
- Article
9
Structure‐guided identification of a selective sulfonamide‐based inhibitor targeting the human carbonic anhydrase VA isoform.
- Published in:
- Archiv der Pharmazie, 2023, v. 356, n. 1, p. 1, doi. 10.1002/ardp.202200383
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- Publication type:
- Article
10
Synthesis and biological evaluation of coumarin‐thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors.
- Published in:
- Archiv der Pharmazie, 2022, v. 355, n. 12, p. 1, doi. 10.1002/ardp.202200232
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- Publication type:
- Article
11
Synthesis and biological evaluation of sulfonamide‐based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae.
- Published in:
- Archiv der Pharmazie, 2022, v. 355, n. 10, p. 1, doi. 10.1002/ardp.202200070
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- Publication type:
- Article
12
Design, synthesis, SAR, and biological evaluation of saccharin‐based hybrids as carbonic anhydrase inhibitors.
- Published in:
- Archiv der Pharmazie, 2022, v. 355, n. 8, p. 1, doi. 10.1002/ardp.202200019
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- Publication type:
- Article
13
Design and development of novel series of indole‐3‐sulfonamide ureido derivatives as selective carbonic anhydrase II inhibitors.
- Published in:
- Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100333
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- Publication type:
- Article
14
Novel benzenesulfonamide‐bearing pyrazoles and 1,2,4‐thiadiazoles as selective carbonic anhydrase inhibitors.
- Published in:
- Archiv der Pharmazie, 2022, v. 355, n. 1, p. 1, doi. 10.1002/ardp.202100241
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- Publication type:
- Article
15
Synthesis of new 7‐amino‐3,4‐dihydroquinolin‐2(1H)‐one‐peptide derivatives and their carbonic anhydrase enzyme inhibition, antioxidant, and cytotoxic activities.
- Published in:
- Archiv der Pharmazie, 2021, v. 354, n. 11, p. 1, doi. 10.1002/ardp.202100122
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- Publication type:
- Article
16
Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐b][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors.
- Published in:
- Archiv der Pharmazie, 2021, v. 354, n. 7, p. 1, doi. 10.1002/ardp.202100028
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- Publication type:
- Article
17
Multiplexed cellular profiling identifies an organoselenium compound as an inhibitor of CRM1‐mediated nuclear export.
- Published in:
- Traffic, 2022, v. 23, n. 12, p. 587, doi. 10.1111/tra.12872
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- Publication type:
- Article
18
Vagar e ocupar: dez anos de narrativas no TOCCA - saberes e práticas transdisciplinares entre as artes e a saúde.
- Published in:
- Interface - Comunicação, Saúde, Educação, 2021, v. 25, p. 1, doi. 10.1590/interface.210218
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- Publication type:
- Article
19
O cotidiano, o lúdico e as redes relacionais: a artesania do cuidar em terapia ocupacional no hospital.
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- Interface - Comunicação, Saúde, Educação, 2012, v. 16, n. 40, p. 261, doi. 10.1590/S1414-32832012005000016
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- Publication type:
- Article
20
Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors.
- Published in:
- Molecules, 2023, v. 28, n. 7, p. 3220, doi. 10.3390/molecules28073220
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- Publication type:
- Article
21
New Insights into Conformationally Restricted Carbonic Anhydrase Inhibitors.
- Published in:
- Molecules, 2023, v. 28, n. 2, p. 890, doi. 10.3390/molecules28020890
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- Publication type:
- Article
22
Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors.
- Published in:
- Molecules, 2023, v. 28, n. 1, p. 91, doi. 10.3390/molecules28010091
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- Publication type:
- Article
23
Design, Synthesis and Biological Assessment of Rhodanine-Linked Benzenesulfonamide Derivatives as Selective and Potent Human Carbonic Anhydrase Inhibitors.
- Published in:
- Molecules, 2022, v. 27, n. 22, p. 8028, doi. 10.3390/molecules27228028
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- Publication type:
- Article
24
Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies.
- Published in:
- Molecules, 2022, v. 27, n. 22, p. 7884, doi. 10.3390/molecules27227884
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- Publication type:
- Article
25
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?
- Published in:
- Molecules, 2022, v. 27, n. 22, p. 7816, doi. 10.3390/molecules27227816
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- Publication type:
- Article
26
Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity.
- Published in:
- Molecules, 2022, v. 27, n. 17, p. 5370, doi. 10.3390/molecules27175370
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- Publication type:
- Article
27
Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII.
- Published in:
- Molecules, 2022, v. 27, n. 14, p. N.PAG, doi. 10.3390/molecules27144610
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- Publication type:
- Article
28
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators.
- Published in:
- Molecules, 2022, v. 27, n. 2, p. 545, doi. 10.3390/molecules27020545
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- Publication type:
- Article
29
Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators.
- Published in:
- Molecules, 2021, v. 26, n. 23, p. 7331, doi. 10.3390/molecules26237331
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- Publication type:
- Article
30
Carbonic Anhydrase Inhibition with Sulfonamides Incorporating Pyrazole- and Pyridazinecarboxamide Moieties Provides Examples of Isoform-Selective Inhibitors.
- Published in:
- Molecules, 2021, v. 26, n. 22, p. 7023, doi. 10.3390/molecules26227023
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- Publication type:
- Article
31
Targeting the RdRp of Emerging RNA Viruses: The Structure-Based Drug Design Challenge.
- Published in:
- Molecules, 2020, v. 25, n. 23, p. 5695, doi. 10.3390/molecules25235695
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- Publication type:
- Article
32
Chagas Disease: Perspectives on the Past and Present and Challenges in Drug Discovery.
- Published in:
- Molecules, 2020, v. 25, n. 22, p. 5483, doi. 10.3390/molecules25225483
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- Publication type:
- Article
33
Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation.
- Published in:
- Molecules, 2020, v. 25, n. 10, p. 2347, doi. 10.3390/molecules25102347
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- Publication type:
- Article
34
Crystal Structure of a Tetrameric Type II β-Carbonic Anhydrase from the Pathogenic Bacterium Burkholderia pseudomallei.
- Published in:
- Molecules, 2020, v. 25, n. 10, p. 2269, doi. 10.3390/molecules25102269
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- Publication type:
- Article
35
Five- and Six-Membered Nitrogen-Containing Compounds as Selective Carbonic Anhydrase Activators.
- Published in:
- Molecules, 2017, v. 22, n. 12, p. 2178, doi. 10.3390/molecules22122178
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- Publication type:
- Article
36
Crystal structure and chemical inhibition of essential schistosome host-interactive virulence factor carbonic anhydrase SmCA.
- Published in:
- Communications Biology, 2019, v. 2, n. 1, p. N.PAG, doi. 10.1038/s42003-019-0578-0
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- Publication type:
- Article
37
Um corpo: cartografando trajetórias de vida de sujeitos com sequelas de acidente vascular cerebral.
- Published in:
- Brazilian Journal of Occupational Therapy / Cadernos Brasileiros de Terapia Ocupacional, 2019, v. 27, n. 1, p. 149, doi. 10.4322/2526-8910.ctoAO1697
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- Publication type:
- Article
38
Towards a standard measure of sea anemone size: assessing the accuracy and precision of morphological measures for cantilever-like animals.
- Published in:
- Marine Ecology, 2016, v. 37, n. 5, p. 1019, doi. 10.1111/maec.12315
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- Publication type:
- Article
39
Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase.
- Published in:
- Natural Product Research, 2022, v. 36, n. 6, p. 1558, doi. 10.1080/14786419.2021.1880406
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- Publication type:
- Article
40
The production and biochemical characterization of α-carbonic anhydrase from Lactobacillus rhamnosus GG.
- Published in:
- Applied Microbiology & Biotechnology, 2022, v. 106, n. 11, p. 4065, doi. 10.1007/s00253-022-11990-3
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- Publication type:
- Article
41
Discovery of a new potent oxindole multi-kinase inhibitor among a series of designed 3-alkenyl-oxindoles with ancillary carbonic anhydrase inhibitory activity as antiproliferative agents.
- Published in:
- BMC Chemistry, 2023, v. 17, n. 1, p. 1, doi. 10.1186/s13065-023-00994-3
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- Publication type:
- Article
42
Thia‐ and Seleno‐Michael Reactions for the Synthesis of Carbonic Anhydrases Inhibitors.
- Published in:
- ChemMedChem, 2024, v. 19, n. 20, p. 1, doi. 10.1002/cmdc.202400345
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- Publication type:
- Article
43
Phthalazine Sulfonamide Derivatives as Carbonic Anhydrase Inhibitors. Synthesis, Biological and in silico Evaluation.
- Published in:
- ChemMedChem, 2024, v. 19, n. 15, p. 1, doi. 10.1002/cmdc.202400147
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- Publication type:
- Article
44
Antimalarial Agents Targeting Plasmodium falciparum Carbonic Anhydrase: Towards Artesunate Hybrid Compounds with Dual Mechanism of Action.
- Published in:
- ChemMedChem, 2023, v. 18, n. 21, p. 1, doi. 10.1002/cmdc.202300267
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- Publication type:
- Article
45
Screening Campaign and Docking Investigations in Identifying New Hit Compounds as Inhibitors of Human Carbonic Anhydrases Expressed In Tumour Cells.
- Published in:
- ChemMedChem, 2023, v. 18, n. 20, p. 1, doi. 10.1002/cmdc.202300330
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- Publication type:
- Article
46
Small Molecule Alkoxy Oriented Selectiveness on Human Carbonic Anhydrase II and IX Inhibition.
- Published in:
- ChemMedChem, 2022, v. 17, n. 11, p. 1, doi. 10.1002/cmdc.202200148
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- Publication type:
- Article
47
Selenocarbamates As a Prodrug‐Based Approach to Carbonic Anhydrase Inhibition.
- Published in:
- ChemMedChem, 2022, v. 17, n. 11, p. 1, doi. 10.1002/cmdc.202200085
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- Publication type:
- Article
48
Ureidosulfocoumarin Derivatives As Selective and Potent Carbonic Anhydrase IX and XII Inhibitors.
- Published in:
- ChemMedChem, 2022, v. 17, n. 5, p. 1, doi. 10.1002/cmdc.202100725
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- Publication type:
- Article
49
4‐Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae.
- Published in:
- ChemMedChem, 2021, v. 16, n. 24, p. 3787, doi. 10.1002/cmdc.202100510
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- Publication type:
- Article
50
Coumarin‐Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action.
- Published in:
- ChemMedChem, 2021, v. 16, n. 8, p. 1252, doi. 10.1002/cmdc.202000915
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- Publication type:
- Article