Works matching AU Amoroso, Rosa
Results: 53
New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1631, doi. 10.1080/14756366.2021.1954918
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- Article
Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1400, doi. 10.1080/14756366.2019.1651315
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- Article
Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1051, doi. 10.1080/14756366.2019.1611801
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- Article
Candida rugosa lipase-catalysed kinetic resolution of 2-substituted-aryloxyacetic esters with dimethylsulfoxide and isopropanol as additives.
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- Chirality, 2008, v. 20, n. 2, p. 115, doi. 10.1002/chir.20505
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- Article
A sulfonimide derivative of bezafibrate as a dual inhibitor of cyclooxygenase-2 and PPARα.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1488722
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- Article
QSAR, QSPR and QSRR in Terms of 3-D-MoRSE Descriptors for In Silico Screening of Clofibric Acid Analogues.
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- Molecular Informatics, 2012, v. 31, n. 6/7, p. 453, doi. 10.1002/minf.201200001
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- Article
Titanium-Promoted Acylation of Sulfonamides to N -Acylsulfonamide PPAR α Antagonists.
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- Synthetic Communications, 2015, v. 45, n. 22, p. 2546, doi. 10.1080/00397911.2015.1092552
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- Article
Stilbene derivatives as new perspective in antifungal medicinal chemistry.
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- Drug Development Research, 2019, v. 80, n. 3, p. 285, doi. 10.1002/ddr.21525
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- Article
Geometric Isomerism of an Acetamidino Derivative Determined by NMR Investigations.
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- ChemistrySelect, 2017, v. 2, n. 30, p. 9706, doi. 10.1002/slct.201701646
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- Article
PPAR Ligands Induce Antiviral Effects Targeting Perturbed Lipid Metabolism during SARS-CoV-2, HCV, and HCMV Infection.
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- Biology (2079-7737), 2022, v. 11, n. 1, p. 114, doi. 10.3390/biology11010114
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- Article
N-acylsulfonamides: Synthetic routes and biological potential in medicinal chemistry.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 6, p. 1094, doi. 10.1111/cbdd.13043
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- Article
Cytotoxic effect of a family of peroxisome proliferator-activated receptor antagonists in colorectal and pancreatic cancer cell lines.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 5, p. 1029, doi. 10.1111/cbdd.13026
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- Article
Synthesis of Naphthyl-, Quinolin- and Anthracenyl Analogues of Clofibric Acid as PPAR α Agonists.
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- Chemical Biology & Drug Design, 2016, v. 87, n. 3, p. 467, doi. 10.1111/cbdd.12677
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- Article
Synthesis of diastereomerically enriched 2-bromoesters and their reaction with nucleophiles.
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- Chirality, 2001, v. 13, n. 2, p. 102, doi. 10.1002/1520-636X(2001)13:2<102::AID-CHIR1005>3.0.CO;2-E
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- Article
Different behavior toward racemization in basic media from chiral analogs of clofibric acid, the active metabolite of the antilipidemic drug clofibrate.
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- Chirality, 2000, v. 12, n. 10, p. 697, doi. 10.1002/1520-636X(2000)12:10<697::AID-CHIR1>3.0.CO;2-L
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- Article
Synthesis of 2-aryloxy acids analogues of clofibrate via dynamic kinetic resolution.
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- Chirality, 1999, v. 11, n. 5/6, p. 483, doi. 10.1002/(SICI)1520-636X(1999)11:5/6<483::AID-CHIR21>3.0.CO;2-I
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- Article
A Novel Prodrug of a nNOS Inhibitor with Improved Pharmacokinetic Potential.
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- ChemMedChem, 2020, v. 15, n. 22, p. 2157, doi. 10.1002/cmdc.202000349
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- Article
Targeting iNOS As a Valuable Strategy for the Therapy of Glioma.
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- ChemMedChem, 2020, v. 15, n. 4, p. 339, doi. 10.1002/cmdc.201900580
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- Article
Development of Fibrates as Important Scaffolds in Medicinal Chemistry.
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- ChemMedChem, 2019, v. 14, n. 11, p. 1051, doi. 10.1002/cmdc.201900128
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- Article
The Anticancer Potential of Peroxisome Proliferator‐Activated Receptor Antagonists.
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- ChemMedChem, 2018, v. 13, n. 3, p. 209, doi. 10.1002/cmdc.201700703
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- Article
Anticancer Activity of Stilbene-Based Derivatives.
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- ChemMedChem, 2017, v. 12, n. 8, p. 558, doi. 10.1002/cmdc.201700045
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- Article
Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.
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- ChemMedChem, 2016, v. 11, n. 16, p. 1695, doi. 10.1002/cmdc.201600204
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- Article
Blocking the Peroxisome Proliferator-Activated Receptor (PPAR): An Overview.
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- ChemMedChem, 2013, v. 8, n. 10, p. 1609, doi. 10.1002/cmdc.201300250
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- Article
Selective Inhibition of iNOS by Benzyl- and Dibenzyl Derivatives of N-(3-Aminobenzyl)acetamidine.
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- ChemMedChem, 2011, v. 6, n. 7, p. 1203, doi. 10.1002/cmdc.201100125
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- Article
Advancements in the Research of New Modulators of Nitric Oxide Synthases Activity.
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- International Journal of Molecular Sciences, 2024, v. 25, n. 15, p. 8486, doi. 10.3390/ijms25158486
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- Article
Emerging Effects of Resveratrol Derivatives in Cells Involved in Oral Wound Healing: A Preliminary Study.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 4, p. 3276, doi. 10.3390/ijms24043276
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- Article
Resveratrol Derivative Exhibits Marked Antiproliferative Actions, Affecting Stemness in Pancreatic Cancer Cells.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 3, p. 1977, doi. 10.3390/ijms24031977
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- Article
Phenylsulfonimide PPARα Antagonists Enhance Nrf2 Activation and Promote Oxidative Stress-Induced Apoptosis/Pyroptosis in MCF7 Breast Cancer Cells.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 2, p. 1316, doi. 10.3390/ijms24021316
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- Article
The Inhibition of the Inducible Nitric Oxide Synthase Enhances the DPSC Mineralization under LPS-Induced Inflammation.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 23, p. 14560, doi. 10.3390/ijms232314560
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- Article
The Selective Acetamidine-Based iNOS Inhibitor CM544 Reduces Glioma Cell Proliferation by Enhancing PARP-1 Cleavage In Vitro.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 3, p. 495, doi. 10.3390/ijms20030495
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- Article
Seeking for Non-Zinc-Binding MMP-2 Inhibitors: Synthesis, Biological Evaluation and Molecular Modelling Studies.
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- International Journal of Molecular Sciences, 2016, v. 17, n. 10, p. 1768, doi. 10.3390/ijms17101768
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- Article
Reversed-phase high-performance liquid chromatography method with fluorescence detection to screen nitric oxide synthases inhibitors.
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- Journal of Separation Science, 2014, v. 37, n. 12, p. 1380, doi. 10.1002/jssc.201400059
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- Article
Azobenzene as Multi-Targeted Scaffold in Medicinal Chemistry.
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- Molecules, 2024, v. 29, n. 24, p. 5872, doi. 10.3390/molecules29245872
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- Article
Neuronal Nitric Oxide Synthase and Post-Translational Modifications in the Development of Central Nervous System Diseases: Implications and Regulation.
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- Molecules, 2023, v. 28, n. 18, p. 6691, doi. 10.3390/molecules28186691
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- Article
Preface to Nitric Oxide Modulators in Health and Disease I.
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- Molecules, 2022, v. 27, n. 20, p. 6820, doi. 10.3390/molecules27206820
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- Article
Choline Chloride-Based DES as Solvents/Catalysts/Chemical Donors in Pharmaceutical Synthesis.
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- Molecules, 2021, v. 26, n. 20, p. 6286, doi. 10.3390/molecules26206286
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- Article
Selective Inhibitors of the Inducible Nitric Oxide Synthase as Modulators of Cell Responses in LPS-Stimulated Human Monocytes.
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- Molecules, 2021, v. 26, n. 15, p. 4419, doi. 10.3390/molecules26154419
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- Article
Redox and Antioxidant Modulation of Circadian Rhythms: Effects of Nitroxyl, N-Acetylcysteine and Glutathione.
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- Molecules, 2021, v. 26, n. 9, p. 2514, doi. 10.3390/molecules26092514
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- Article
The Role of Single-Nucleotide Variants of NOS1 , NOS2, and NOS3 Genes in the Comorbidity of Arterial Hypertension and Tension-Type Headache.
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- Molecules, 2021, v. 26, n. 6, p. 1556, doi. 10.3390/molecules26061556
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- Article
In Vivo Targeted Metabolomic Profiling of Prostanit, a Novel Anti-PAD NO-Donating Alprostadil-Based Drug.
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- Molecules, 2020, v. 25, n. 24, p. 5896, doi. 10.3390/molecules25245896
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- Article
Synthesis and Biological Evaluation of Halogenated E -Stilbenols as Promising Antiaging Agents.
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- Molecules, 2020, v. 25, n. 23, p. 5770, doi. 10.3390/molecules25235770
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- Article
Acetamidine-Based iNOS Inhibitors as Molecular Tools to Counteract Inflammation in BV2 Microglial Cells.
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- Molecules, 2020, v. 25, n. 11, p. 2646, doi. 10.3390/molecules25112646
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- Article
Development of a Rapid Mass Spectrometric Determination of AMP and Cyclic AMP for PDE3 Activity Study: Application and Computational Analysis for Evaluating the Effect of a Novel 2-oxo-1,2-dihydropyridine-3-carbonitrile Derivative as PDE-3 Inhibitor.
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- Molecules, 2020, v. 25, n. 8, p. 1817, doi. 10.3390/molecules25081817
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- Article
Activators of Nrf2 to Counteract Neurodegenerative Diseases.
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- Antioxidants, 2023, v. 12, n. 3, p. 778, doi. 10.3390/antiox12030778
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- Article
The Positive Regulation of eNOS Signaling by PPAR Agonists in Cardiovascular Diseases.
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- American Journal of Cardiovascular Drugs, 2017, v. 17, n. 4, p. 273, doi. 10.1007/s40256-017-0220-9
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- Article
Anti-Inflammatory, Antioxidant, and WAT/BAT-Conversion Stimulation Induced by Novel PPAR Ligands: Results from Ex Vivo and In Vitro Studies.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 3, p. 346, doi. 10.3390/ph16030346
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- Article
Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure–Activity Relationship Studies and Target Prediction Analysis.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 8, p. 937, doi. 10.3390/ph15080937
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- Article
HDAC Inhibitors for the Therapy of Triple Negative Breast Cancer.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 6, p. 667, doi. 10.3390/ph15060667
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- Article
Design, Synthesis and Biological Evaluation of Aromatase Inhibitors Based on Sulfonates and Sulfonamides of Resveratrol.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 10, p. 984, doi. 10.3390/ph14100984
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- Article
PPARα Antagonist AA452 Triggers Metabolic Reprogramming and Increases Sensitivity to Radiation Therapy in Human Glioblastoma Primary Cells.
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- Journal of Cellular Physiology, 2017, v. 232, n. 6, p. 1458, doi. 10.1002/jcp.25648
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- Article