Works matching AU Ammazzalorso, Alessandra
Results: 48
New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1631, doi. 10.1080/14756366.2021.1954918
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- Article
Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.
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- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1051, doi. 10.1080/14756366.2019.1611801
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- Article
Candida rugosa lipase-catalysed kinetic resolution of 2-substituted-aryloxyacetic esters with dimethylsulfoxide and isopropanol as additives.
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- Chirality, 2008, v. 20, n. 2, p. 115, doi. 10.1002/chir.20505
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- Article
A sulfonimide derivative of bezafibrate as a dual inhibitor of cyclooxygenase-2 and PPARα.
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- Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1488722
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- Article
QSAR, QSPR and QSRR in Terms of 3-D-MoRSE Descriptors for In Silico Screening of Clofibric Acid Analogues.
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- Molecular Informatics, 2012, v. 31, n. 6/7, p. 453, doi. 10.1002/minf.201200001
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- Article
Titanium-Promoted Acylation of Sulfonamides to N -Acylsulfonamide PPAR α Antagonists.
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- Synthetic Communications, 2015, v. 45, n. 22, p. 2546, doi. 10.1080/00397911.2015.1092552
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- Article
Stilbene derivatives as new perspective in antifungal medicinal chemistry.
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- Drug Development Research, 2019, v. 80, n. 3, p. 285, doi. 10.1002/ddr.21525
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- Article
Geometric Isomerism of an Acetamidino Derivative Determined by NMR Investigations.
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- ChemistrySelect, 2017, v. 2, n. 30, p. 9706, doi. 10.1002/slct.201701646
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- Article
PPAR Ligands Induce Antiviral Effects Targeting Perturbed Lipid Metabolism during SARS-CoV-2, HCV, and HCMV Infection.
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- Biology (2079-7737), 2022, v. 11, n. 1, p. 114, doi. 10.3390/biology11010114
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- Article
N-acylsulfonamides: Synthetic routes and biological potential in medicinal chemistry.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 6, p. 1094, doi. 10.1111/cbdd.13043
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- Article
Cytotoxic effect of a family of peroxisome proliferator-activated receptor antagonists in colorectal and pancreatic cancer cell lines.
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- Chemical Biology & Drug Design, 2017, v. 90, n. 5, p. 1029, doi. 10.1111/cbdd.13026
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- Article
Synthesis of Naphthyl-, Quinolin- and Anthracenyl Analogues of Clofibric Acid as PPAR α Agonists.
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- Chemical Biology & Drug Design, 2016, v. 87, n. 3, p. 467, doi. 10.1111/cbdd.12677
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- Article
Synthesis of diastereomerically enriched 2-bromoesters and their reaction with nucleophiles.
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- Chirality, 2001, v. 13, n. 2, p. 102, doi. 10.1002/1520-636X(2001)13:2<102::AID-CHIR1005>3.0.CO;2-E
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- Article
Effects of PPARα inhibition in head and neck paraganglioma cells.
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- PLoS ONE, 2017, v. 12, n. 6, p. 1, doi. 10.1371/journal.pone.0178995
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- Article
Development of Fibrates as Important Scaffolds in Medicinal Chemistry.
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- ChemMedChem, 2019, v. 14, n. 11, p. 1051, doi. 10.1002/cmdc.201900128
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- Article
The Anticancer Potential of Peroxisome Proliferator‐Activated Receptor Antagonists.
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- ChemMedChem, 2018, v. 13, n. 3, p. 209, doi. 10.1002/cmdc.201700703
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- Article
Anticancer Activity of Stilbene-Based Derivatives.
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- ChemMedChem, 2017, v. 12, n. 8, p. 558, doi. 10.1002/cmdc.201700045
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- Article
Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.
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- ChemMedChem, 2016, v. 11, n. 16, p. 1695, doi. 10.1002/cmdc.201600204
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- Article
Blocking the Peroxisome Proliferator-Activated Receptor (PPAR): An Overview.
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- ChemMedChem, 2013, v. 8, n. 10, p. 1609, doi. 10.1002/cmdc.201300250
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- Article
Selective Inhibition of iNOS by Benzyl- and Dibenzyl Derivatives of N-(3-Aminobenzyl)acetamidine.
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- ChemMedChem, 2011, v. 6, n. 7, p. 1203, doi. 10.1002/cmdc.201100125
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- Article
Anticancer Activity of Natural Products and Related Compounds.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 22, p. 16507, doi. 10.3390/ijms242216507
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- Article
Phenylsulfonimide PPARα Antagonists Enhance Nrf2 Activation and Promote Oxidative Stress-Induced Apoptosis/Pyroptosis in MCF7 Breast Cancer Cells.
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- International Journal of Molecular Sciences, 2023, v. 24, n. 2, p. 1316, doi. 10.3390/ijms24021316
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- Article
The Selective Acetamidine-Based iNOS Inhibitor CM544 Reduces Glioma Cell Proliferation by Enhancing PARP-1 Cleavage In Vitro.
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- International Journal of Molecular Sciences, 2019, v. 20, n. 3, p. 495, doi. 10.3390/ijms20030495
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- Article
Seeking for Non-Zinc-Binding MMP-2 Inhibitors: Synthesis, Biological Evaluation and Molecular Modelling Studies.
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- International Journal of Molecular Sciences, 2016, v. 17, n. 10, p. 1768, doi. 10.3390/ijms17101768
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- Article
Reversed-phase high-performance liquid chromatography method with fluorescence detection to screen nitric oxide synthases inhibitors.
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- Journal of Separation Science, 2014, v. 37, n. 12, p. 1380, doi. 10.1002/jssc.201400059
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- Article
Azobenzene as Multi-Targeted Scaffold in Medicinal Chemistry.
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- Molecules, 2024, v. 29, n. 24, p. 5872, doi. 10.3390/molecules29245872
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- Article
Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?
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- Molecules, 2022, v. 27, n. 22, p. 7816, doi. 10.3390/molecules27227816
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- Article
Anticancer Inhibitors.
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- Molecules, 2022, v. 27, n. 14, p. N.PAG, doi. 10.3390/molecules27144650
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- Article
Development of CDK4/6 Inhibitors: A Five Years Update.
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- Molecules, 2021, v. 26, n. 5, p. 1488, doi. 10.3390/molecules26051488
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- Article
Targeting Toxins toward Tumors.
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- Molecules, 2021, v. 26, n. 5, p. 1292, doi. 10.3390/molecules26051292
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- Article
Tacrine-Coumarin Derivatives as Topoisomerase Inhibitors with Antitumor Effects on A549 Human Lung Carcinoma Cancer Cell Lines.
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- Molecules, 2021, v. 26, n. 4, p. 1133, doi. 10.3390/molecules26041133
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- Article
Saponins Extracted from Tea (Camellia Sinensis) Flowers Induces Autophagy in Ovarian Cancer Cells.
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- Molecules, 2020, v. 25, n. 22, p. 5254, doi. 10.3390/molecules25225254
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- Article
Engineering Stem Cell Factor Ligands with Different c-Kit Agonistic Potencies.
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- Molecules, 2020, v. 25, n. 20, p. 4850, doi. 10.3390/molecules25204850
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- Article
The Potential Role of Cathepsin K in Non-Small Cell Lung Cancer.
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- Molecules, 2020, v. 25, n. 18, p. 4136, doi. 10.3390/molecules25184136
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- Article
Structural Basis of Beneficial Design for Effective Nicotinamide Phosphoribosyltransferase Inhibitors.
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- Molecules, 2020, v. 25, n. 16, p. 3633, doi. 10.3390/molecules25163633
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- Article
Standardized Saponin Extract from Baiye No.1 Tea (Camellia sinensis) Flowers Induced S Phase Cell Cycle Arrest and Apoptosis via AKT-MDM2-p53 Signaling Pathway in Ovarian Cancer Cells.
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- Molecules, 2020, v. 25, n. 15, p. 3515, doi. 10.3390/molecules25153515
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- Article
Tamoxifen and the PI3K Inhibitor: LY294002 Synergistically Induce Apoptosis and Cell Cycle Arrest in Breast Cancer MCF-7 Cells.
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- Molecules, 2020, v. 25, n. 15, p. 3355, doi. 10.3390/molecules25153355
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- Article
Development of a Rapid Mass Spectrometric Determination of AMP and Cyclic AMP for PDE3 Activity Study: Application and Computational Analysis for Evaluating the Effect of a Novel 2-oxo-1,2-dihydropyridine-3-carbonitrile Derivative as PDE-3 Inhibitor.
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- Molecules, 2020, v. 25, n. 8, p. 1817, doi. 10.3390/molecules25081817
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- Article
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies.
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- Pharmaceuticals (14248247), 2024, v. 17, n. 8, p. 1027, doi. 10.3390/ph17081027
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- Article
Nature-Inspired Compounds: Synthesis and Antibacterial Susceptibility Testing of Eugenol Derivatives against H. pylori Strains.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 9, p. 1317, doi. 10.3390/ph16091317
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- Article
Anti-Inflammatory, Antioxidant, and WAT/BAT-Conversion Stimulation Induced by Novel PPAR Ligands: Results from Ex Vivo and In Vitro Studies.
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- Pharmaceuticals (14248247), 2023, v. 16, n. 3, p. 346, doi. 10.3390/ph16030346
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- Article
Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure–Activity Relationship Studies and Target Prediction Analysis.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 8, p. 937, doi. 10.3390/ph15080937
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- Article
HDAC Inhibitors for the Therapy of Triple Negative Breast Cancer.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 6, p. 667, doi. 10.3390/ph15060667
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- Article
Design, Synthesis and Biological Evaluation of Aromatase Inhibitors Based on Sulfonates and Sulfonamides of Resveratrol.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 10, p. 984, doi. 10.3390/ph14100984
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- Article
CAPE derivatives: Multifaceted agents for chronic wound healing.
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- Archiv der Pharmazie, 2024, v. 357, n. 10, p. 1, doi. 10.1002/ardp.202400165
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- Article
Synthesis and in vitro cytotoxicity of benzoxazole‐based PPARα/γ antagonists in colorectal cancer cell lines.
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- Archiv der Pharmazie, 2024, v. 357, n. 9, p. 1, doi. 10.1002/ardp.202400086
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- Article
PPARα Antagonist AA452 Triggers Metabolic Reprogramming and Increases Sensitivity to Radiation Therapy in Human Glioblastoma Primary Cells.
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- Journal of Cellular Physiology, 2017, v. 232, n. 6, p. 1458, doi. 10.1002/jcp.25648
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- Article
Azole-Based Compounds That Are Active against Candida Biofilm: In Vitro , In Vivo and In Silico Studies.
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- Antibiotics (2079-6382), 2022, v. 11, n. 10, p. N.PAG, doi. 10.3390/antibiotics11101375
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- Article