Works by Al-Rashood, Sara T.


Results: 40
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    Design and statistical optimisation of emulsomal nanoparticles for improved anti-SARS-CoV-2 activity of N-(5-nitrothiazol-2-yl)-carboxamido candidates: in vitro and in silico studies.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2202357
    By:
    • Al-Karmalawy, Ahmed A.;
    • El-Gamil, Dalia S.;
    • El-Shesheny, Rabeh;
    • Sharaky, Marwa;
    • Alnajjar, Radwan;
    • Kutkat, Omnia;
    • Moatasim, Yassmin;
    • Elagawany, Mohamed;
    • Al-Rashood, Sara T.;
    • Binjubair, Faizah A.;
    • Eldehna, Wagdy M.;
    • Noreddin, Ayman M.;
    • Zakaria, Mohamed Y.
    Publication type:
    Article
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    Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201407
    By:
    • Badawi, Waleed A.;
    • Rashed, Mahmoud;
    • Nocentini, Alessio;
    • Bonardi, Alessandro;
    • Abd-Alhaseeb, Mohammad M.;
    • Al-Rashood, Sara T.;
    • Veerakanellore, Giri Babu;
    • Majrashi, Taghreed A.;
    • Elkaeed, Eslam B.;
    • Elgendy, Bahaa;
    • Gratteri, Paola;
    • Supuran, Claudiu T.;
    • Eldehna, Wagdy M.;
    • Elagawany, Mohamed
    Publication type:
    Article
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    Metabolomic profile, anti-trypanosomal potential and molecular docking studies of Thunbergia grandifolia.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2199950
    By:
    • El-Nashar, Heba A. S.;
    • Sayed, Ahmed M.;
    • El-Sherief, Hany A. M.;
    • Rateb, Mostafa E.;
    • Akil, Lina;
    • Khadra, Ibrahim;
    • Majrashi, Taghreed A.;
    • Al-Rashood, Sara T.;
    • Binjubair, Faizah A.;
    • El Hassab, Mahmoud A.;
    • Eldehna, Wagdy M.;
    • Abdelmohsen, Usama Ramadan;
    • Mostafa, Nada M.
    Publication type:
    Article
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    Cancer stem cells CD133 inhibition and cytotoxicity of certain 3-phenylthiazolo[3,2- a ]benzimidazoles: design, direct synthesis, crystal study and in vitro biological evaluation.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 986, doi. 10.1080/14756366.2017.1347166
    By:
    • Al-Ansary, Ghada H.;
    • Eldehna, Wagdy M.;
    • Ghabbour, Hazem A.;
    • Al-Rashood, Sara T. A.;
    • Al-Rashood, Khalid A.;
    • Eladwy, Radwa A.;
    • Al-Dhfyan, Abdullah;
    • Kabil, Maha M.;
    • Abdel-Aziz, Hatem A.
    Publication type:
    Article
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    Anticoagulants as Potential SARS-CoV-2 M pro Inhibitors for COVID-19 Patients: In Vitro, Molecular Docking, Molecular Dynamics, DFT, and SAR Studies.

    Published in:
    International Journal of Molecular Sciences, 2022, v. 23, n. 20, p. 12235, doi. 10.3390/ijms232012235
    By:
    • Abo Elmaaty, Ayman;
    • Eldehna, Wagdy M.;
    • Khattab, Muhammad;
    • Kutkat, Omnia;
    • Alnajjar, Radwan;
    • El-Taweel, Ahmed N.;
    • Al-Rashood, Sara T.;
    • Abourehab, Mohammed A. S.;
    • Binjubair, Faizah A.;
    • Saleh, Mohamed A.;
    • Belal, Amany;
    • Al-Karmalawy, Ahmed A.
    Publication type:
    Article
    18

    Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.

    Published in:
    International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484
    By:
    • Abdelrahman, Mohamed A.;
    • Eldehna, Wagdy M.;
    • Nocentini, Alessio;
    • Bua, Silvia;
    • Al-Rashood, Sara T.;
    • Hassan, Ghada S.;
    • Bonardi, Alessandro;
    • Almehizia, Abdulrahman A.;
    • Alkahtani, Hamad M.;
    • Alharbi, Amal;
    • Gratteri, Paola;
    • Supuran, Claudiu T.
    Publication type:
    Article
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    Molecular docking, DFT and antiproliferative properties of 4‐(3,4‐dimethoxyphenyl)−3‐(4‐methoxyphenyl)−1‐phenyl‐1H‐pyrazolo[3,4‐b]pyridine as potent anticancer agent with CDK2 and PIM1 inhibition potency

    Published in:
    Drug Development Research, 2024, v. 85, n. 7, p. 1, doi. 10.1002/ddr.70009
    By:
    • Binjubair, Faizah A.;
    • Almansour, Basma S.;
    • Ziedan, Noha I.;
    • Abdel‐Aziz, Alaa A.‐M.;
    • Al‐Rashood, Sara T.;
    • Elgohary, Mohamed K.;
    • Elkotamy, Mahmoud S.;
    • Abdel‐Aziz, Hatem A.
    Publication type:
    Article
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    Investigating the promising SARS-CoV-2 main protease inhibitory activity of secoiridoids isolated from Jasminum humile; in silico and in Vitro assessments with structure-activity relationship.

    Published in:
    Journal of Biomolecular Structure & Dynamics, 2024, v. 42, n. 13, p. 6941, doi. 10.1080/07391102.2023.2240419
    By:
    • Al-Karmalawy, Ahmed A.;
    • Alnajjar, Radwan;
    • Elmaaty, Ayman Abo;
    • Binjubair, Faizah A.;
    • Al-Rashood, Sara T.;
    • Mansour, Basma S.;
    • Elkamhawy, Ahmed;
    • Eldehna, Wagdy M.;
    • Mansour, Khaled Ahmed
    Publication type:
    Article
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