Works by Al-Masoudi, Najim A.

Results: 50

Synthesis and In Vitro Anti-HIV Activity of Some New Schiff Base Ligands Derived from 5-Amino-4-phenyl-4H-1,2,4-triazole-3-thiol and Their Metal Complexes.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2009, v. 184, n. 11, p. 2891, doi. 10.1080/10426500802591630

By:

Al-Masoudi, Najim A.;
Aziz, Nazik M.;
Mohammed, Abdulalah T.

Publication type:

Article

Synthesis and Anti-HIV Activity of New 6-Thioarylpyrimidines and Related Compounds.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2008, v. 183, n. 7, p. 1571, doi. 10.1080/10426500701693453

By:

Al-Masoudi, Iman A.;
Al-Soud, Yaseen A.;
Al-Masoudi, Najim A.;
Noori, Saman H.;
Schuppler, Thilo

Publication type:

Article

Synthesis, Anti–HIV, and Antifungal Activity of New Benzensulfonamides Bearing the 2,5-Disubstituted-1,3,4-Oxadiazole Moiety.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2007, v. 182, n. 2, p. 281, doi. 10.1080/10426500600919074

By:

Zareef, Muhammad;
Iqbal, Rashid;
Al-Masoudi, Najim A.;
Zaidi, Javid H.;
Arfan, Muhammad;
Shahzad, Sohail A.

Publication type:

Article

Synthesis and Reactions of New 3′-Deoxy-5′-thioalkyl-β- D - erythro -pentofuranosylthymines and Related Analogues.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2003, v. 178, n. 12, p. 2551, doi. 10.1080/718990492

By:

Al-Masoudi, Najim A.;
Al-Soud, Yaseen A.

Publication type:

Article

Some 2′-Modified 4′-Thionucleosides via Sulfur Participation and Synthesis of Thio-Azt from 4′-Thiofuranoid 1,2-Glycal.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2003, v. 178, n. 6, p. 1199, doi. 10.1080/10426500307902

By:

Al-Masoudi, Najim A.;
Al-Soud, Yaseen A.;
Khodair, Ahmed I.

Publication type:

Article

Synthesis and anti-HIV activity of new 2-thiolumazine and 2-thiouracil metal complexes.

Published in:

Heteroatom Chemistry, 2011, v. 22, n. 1, p. 44, doi. 10.1002/hc.20654

By:

Al-Masoudi, Najim A.;
Saleh, Basil A.;
Karim, Nesreen Abdul;
Issa, Ahmed Y.;
Pannecouque, Christoph

Publication type:

Article

Nitroimidazoles, part 4: Synthesis and anti-HIV activity of new 5-alkylsulfanyl and 5-(4′-arylsulfonyl)piperazinyl-4-nitroimidazole derivatives.

Published in:

Heteroatom Chemistry, 2007, v. 18, n. 4, p. 333, doi. 10.1002/hc.20301

By:

Al-Soud, Yaseen A.;
Al-Masoudi, Najim A.;
De Clercq, Erik;
Paneccoque, Christoph

Publication type:

Article

Microwave-assisted synthesis and anti-HIV activity of new benzenesulfonamides bearing 2,5-disubstituted-1,3,4-oxadiazole moiety.

Published in:

Heteroatom Chemistry, 2007, v. 18, n. 4, p. 425, doi. 10.1002/hc.20316

By:

Zareef, Muhammad;
Iqbal, Rashid;
Al-Masoudi, Najim A.;
Zaidi, Javid H.;
Arfan, Muhammad

Publication type:

Article

Synthesis and anti-HIV activity of new chiral 1,2,4-triazoles and 1,3,4-thiadiazoles.

Published in:

Heteroatom Chemistry, 2007, v. 18, n. 3, p. 316, doi. 10.1002/hc.20282

By:

Akhtar, Tashfeen;
Hameed, Shahid;
Al-Masoudi, Najim A.;
Khan, Khalid M.

Publication type:

Article

Synthesis, Biological Evaluation and Molecular Docking Study of Novel Benzhydryl Piperazine‐1,2,3‐Triazoline Hybrids.

Published in:

ChemistrySelect, 2024, v. 9, n. 17, p. 1, doi. 10.1002/slct.202400813

By:

Al‐Masoudi, Najim A.;
Jihad, Raad S.;
Abdul‐Rida, Nabeel A.;
Al‐Shamari, Amer M. J.;
Saeed, Bahjat;
Al‐Masoudi, Wasfi A.

Publication type:

Article

Synthesis, anti-HIV and cytotoxicity evaluation of chiral 2,5-disubstituted 1,3,4-thiadiazole derivatives bearing the sulfonamide scaffold.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2024, v. 79, n. 2/3, p. 89, doi. 10.1515/znb-2023-0078

By:

Israr, Anum;
Hameed, Shahid;
Al-Masoudi, Najim A.

Publication type:

Article

Design, synthesis, and in-silico study of new letrozole derivatives as prospective anticancer and antioxidant agents.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2023, v. 78, n. 6, p. 343, doi. 10.1515/znb-2022-0151

By:

Jihad, Raad S.;
Abdul-Rida, Nabeel A.;
Al-Shamari, Amer M. J.;
Al-Masoudi, Najim A.;
Saeed, Bahjat A.

Publication type:

Article

Synthesis, cytotoxicity and in silico study of some novel benzocoumarin-chalcone-bearing aryl ester derivatives and benzocoumarin-derived arylamide analogs.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2021, v. 76, n. 3/4, p. 201, doi. 10.1515/znb-2020-0204

By:

Abdul-Ridha, Nabeel A.;
Salmaan, Afraah D.;
Sabah, Rita;
Saeed, Bahjat;
Al-Masoudi, Najim A.

Publication type:

Article

New cholic acid analogs: synthesis and 17<italic>β</italic>-hydroxydehydrogenase (17<italic>β</italic>-HSD) inhibition activity.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2018, v. 73, n. 3/4, p. 211, doi. 10.1515/znb-2018-0192

By:

Al-Masoudi, Najim A.;
Sami, Abbas;
Abdul-Rida, Nabeel A.;
Fortscher, Martin

Publication type:

Article

New cholic acid analogs: synthesis and 17β-hydroxydehydrogenase (17β-HSD) inhibition activity.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2018, p. 211, doi. 10.1515/znb-2018-0192

By:

Al-Masoudi, Najim A.;
Sami, Abbas;
Abdul-Rida, Nabeel A.;
Fortscher, Martin

Publication type:

Article

Synthesis, anti-HIV activity and molecular modeling study of 3-aryl-6-adamantylmethyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2015, v. 70, n. 8, p. 609, doi. 10.1515/znb-2015-0032

By:

Khan, Mahmood-ul-Hassan;
Hameed, Shahid;
Farman, Muhammad;
Al-Masoudi, Najim A.;
Stoeckli-Evans, Helen

Publication type:

Article

Synthesis, biological activity and modeling study of some thiopyrimidine derivatives and their platinum(II) and ruthenium(III) metal complexes.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2015, v. 70, n. 5, p. 343, doi. 10.1515/znb-2014-0246

By:

Al-Masoudi, Najim A.;
Abbas, Azhar;
Al-Asadi, Mohammed J.B.

Publication type:

Article

New triazolothiadiazole and triazolothiadiazine derivatives as kinesin Eg5 and HIV inhibitors: synthesis, QSAR and modeling studies.

Published in:

Zeitschrift für Naturforschung B: A Journal of Chemical Sciences, 2015, v. 70, n. 1, p. 47, doi. 10.1515/znb-2014-0162

By:

Khan, Imtiaz;
Hameed, Shahid;
Al-Masoudi, Najim A.;
Abdul-Reda, Nabeel A.;
Simpson, Jim

Publication type:

Article

A New Approach to the Synthesis of Benzothiazole, Benzoxazole, and Pyridine Nucleosides as Potential Antitumor Agents.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2003, v. 22, n. 11, p. 2061, doi. 10.1081/NCN-120026407

By:

Khodair, Ahmed I.;
Al-Masoudi, Najim A.;
Gesson, Jean-Pierre

Publication type:

Article

Synthesis of N-Substituted 1-Amino-2,3-dihydro-1H-imidazole-2-thione-N-nucleosides and S-Glycosylated Derivatives.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2003, v. 22, n. 3, p. 299, doi. 10.1081/NCN-120021429

By:

Al-Masoudi, Iman A.;
Khodair, Ahmed I.;
Al-Soud, Yaseen A.;
Al-Masoudi, Najim A.

Publication type:

Article

NEW GLYCOSYL-(CARBOXAMIDE)-1,2,3-TRIAZOLE-N-NUCLEOSIDES: SYNTHESIS AND ANTITUMOR ACTIVITY.

Published in:

Nucleosides, Nucleotides & Nucleic Acids, 2002, v. 21, n. 4/5, p. 361, doi. 10.1081/NCN-120006830

By:

Al-Masoudi, Najim A.;
Al-Soud, Yaseen A.

Publication type:

Article

A ruthenium complexes of monastrol and its pyrimidine analogues: Synthesis and biological properties.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2019, v. 194, n. 11, p. 1020, doi. 10.1080/10426507.2019.1597362

By:

Al-Masoudi, Wasfi A.;
Al-Masoudi, Najim A.

Publication type:

Article

Synthesis, X-ray structure, in vitro HIV and kinesin Eg5 inhibition activities of new arene ruthenium complexes of pyrimidine analogs.

Published in:

Journal of Coordination Chemistry, 2017, v. 70, n. 12, p. 2061, doi. 10.1080/00958972.2017.1334259

By:

Al-Masoudi, Wasfi A.;
Al-Masoudi, Najim A.;
Weibert, Bernhard;
Winter, Rainer

Publication type:

Article

Design, Synthesis, Docking Studies and Molecular Dynamics Simulation of New 1,3,5‐Triazine Derivatives as Anticancer Agents Selectively Targeting Pancreatic Adenocarcinoma (Capan‐1).

Published in:

Chemistry & Biodiversity, 2024, v. 21, n. 5, p. 1, doi. 10.1002/cbdv.202400112

By:

Asghar, Shazia;
Hameed, Shahid;
Al‐Masoudi, Najim A;
Saeed, Bahjat;
Shtaiwi, Amneh

Publication type:

Article

SYNTHESIS OF 1-[4-(1,5-DIALKYL-1 H -1,2,4-TRIAZOL-3-YL)]BENZYL-1 H -INDOLES AND 5,6-DIHALOQUINOLONES.

Published in:

Organic Preparations & Procedures International, 2002, v. 34, n. 6, p. 658, doi. 10.1080/00304940209355790

By:

Al-Soud, Yaseen A.;
Halah, Rana F.;
Al-Masoudi, Najim A.

Publication type:

Article

Amino acid derivatives. Part 6. New analogs of the angiotensin-converting enzyme 'Captopril'. Synthesis and anti-HIV activity.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 242

By:

Al-Masoudi, Najim A.;
Hamad, Nawar S.;
Hameed, Shahid;
Pannecouque, Christophe

Publication type:

Article

Amino acid derivatives. Part 5. Synthesis and anti-HIV activity of new sebacoyl precursor derived thioureido-amino acid and phthalimide derivatives.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2010, p. 185

By:

Al-Masoudi, Najim A.;
Al-Haidery, Nahed;
Faili, Naeem T.;
Pannecouque, C.

Publication type:

Article

Synthesis and in vitro antiproliferative activity of new adamantylthiazolyl-1,3,4-oxadiazoles.

Published in:

ARKIVOC: Online Journal of Organic Chemistry, 2009, p. 85

By:

Zahid, Maryam;
Yasin, Khawaja A.;
Akhtar, Tashfeen;
Rama, Nasim H.;
Hameed, Shahid;
Al-Masoudi, Najim A.;
Loddo, Roberta;
La Colla, Paolo

Publication type:

Article

Synthesis and Biological Evaluation of New Dipyridylpteridines, Lumazines, and Related Analogues.

Published in:

Journal of Heterocyclic Chemistry, 2017, v. 54, n. 2, p. 895, doi. 10.1002/jhet.2651

By:

Abbas, Zina A. A.;
Abu ‐ Mejdad, Najwa M. J.;
Atwan, Zeenah W.;
Al ‐ Masoudi, Najim A.

Publication type:

Article

Antibacterial, antifungal, antiherbicidal, and antifungicidal activity of 4,6-dimethoxyhomophthalic acid and related compounds.

Published in:

Pharmaceutical Chemistry Journal, 2008, v. 42, n. 6, p. 335, doi. 10.1007/s11094-008-0121-y

By:

Qadeer, Ghulam;
Rama, Nasim Hasan;
Zareef, Muhammad;
Al-Masoudi, Najim A.

Publication type:

Article

In vitro anti-HIV activity of diverse substituted nitrosopyrimidine analogues.

Published in:

Chemistry & Biology Interface, 2016, v. 6, n. 2, p. 69

By:

Al-Masoudi, Najim A.;
March, Yossra A.;
Al-Ameri, Jenan J.;
Ali, Dawood S.;
Pannecouque, Christophe

Publication type:

Article

Exploration of the in vitro anti-HIV and cyclin-dependent kinase 2 (CDK2) inhibitory activities of new 6-aryl-pyrimidines and their nitroso analogues.

Published in:

Chemistry & Biology Interface, 2016, v. 6, n. 1, p. 1

By:

Al-Masoudi, Najim A.;
Saeed, Bahjat A.;
Ali, Dawood S.;
Alias, Rita S.;
Jaffer, Nadhir N. A.;
Pannecouque, Christophe

Publication type:

Article

In vitro anti-HIV and HCV activity of new thioureido and thiazole analogues of cholesterol conjugated α-amino acid residues and in silico molecular modeling study.

Published in:

Chemistry & Biology Interface, 2015, v. 5, n. 6, p. 333

By:

Al-Masoudi, Najim A.;
Ali, Dawood S.;
Pannecouque, Christophe

Publication type:

Article

Novel 4-nitroimidazole analogues: synthesis, in vitro biological evaluation, in silico studies, and molecular dynamics simulation.

Published in:

Zeitschrift für Naturforschung. Section C: A Journal of Biosciences, 2024, v. 79, n. 3/4, p. 61, doi. 10.1515/znc-2023-0146

By:

Al-Soud, Yaseen A.;
Al-Sawakhnah, Sondos O.;
Al-Qawasmeh, Raed A.;
Al-Masoudi, Najim A.;
Al-Ahmad, Ala'a H.;
Al-Maliki, Lamiaa;
van Geelen, Lasse;
Kalscheuer, Rainer;
Saeed, Bahjat A.;
Shtaiwi, Amneh;
Stark, Holger

Publication type:

Article

New CYP17 Hydroxylase Inhibitors: Synthesis, Biological Evaluation, QSAR, and Molecular Docking Study of New Pregnenolone Analogs.

Published in:

Archiv der Pharmazie, 2014, v. 347, n. 12, p. 896, doi. 10.1002/ardp.201400255

By:

Al ‐ Masoudi, Najim A.;
Ali, Dawood S.;
Saeed, Bahjat;
Hartmann, Rolf W.;
Engel, Matthias;
Rashid, Sajid;
Saeed, Aamer

Publication type:

Article

Synthesis, QSAR and anti-HIV activity of new 5-benzylthio-1,3,4-oxadiazoles derived from α-amino acids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2011, v. 26, n. 5, p. 668, doi. 10.3109/14756366.2010.546792

By:

Syed, Tayyaba;
Akhtar, Tashfeen;
Al-Masoudi, Najim A.;
Jones, Peter G.;
Hameed, Shahid

Publication type:

Article

Nitroimidazoles, Part 2.

Published in:

Chemistry & Biodiversity, 2006, v. 3, n. 5, p. 515, doi. 10.1002/cbdv.200690055

By:

Al-Masoudi, Najim A.;
Al-Soud, Yaseen A.;
Kalogerakis, Aris;
Pannecouque, Christophe;
De Clercq, Erik

Publication type:

Article

A novel pregnene analogs: synthesis, cytotoxicity on prostate cancer of PC-3 and LNCPa-AI cells and in silico molecular docking study.

Published in:

Molecular Diversity, 2021, v. 25, n. 2, p. 661, doi. 10.1007/s11030-020-10038-w

By:

Abdul-Rida, Nabeel A.;
Farhan, Ali M.;
Al-Masoudi, Najim A.;
Saeed, Bahjat A.;
Miller, Dannah;
Lin, Ming-Fong

Publication type:

Article

Synthesis of new chiral 1,3,4-thiadiazole-based di- and tri-arylsulfonamide residues and evaluation of in vitro anti-HIV activity and cytotoxicity.

Published in:

Molecular Diversity, 2018, v. 22, n. 4, p. 957, doi. 10.1007/s11030-018-9851-2

By:

Shafique, Maria;
Hameed, Shahid;
Naseer, Muhammad Moazzam;
Al-Masoudi, Najim Aboud

Publication type:

Article

Amino acid derivatives, part 3: New peptide and glycopeptide derivatives conjugated naphthalene. Synthesis, antitumor, anti-HIV, and BVDV evaluation.

Published in:

Heteroatom Chemistry, 2005, v. 16, n. 7, p. 576, doi. 10.1002/hc.20149

By:

Al-Masoudi, Najim A.;
Al-Masoudi, Iman A.;
Ali, Ibrahim A. I.;
Saeed, Bahjat;
Colla, Palo La

Publication type:

Article

Amino acid derivatives, part 2: Synthesis, antiviral, and antitumor activity of simple protected amino acids functionalized at N-terminus with naphthalene side chain.

Published in:

Heteroatom Chemistry, 2005, v. 16, n. 2, p. 148, doi. 10.1002/hc.20082

By:

Ali, Ibrahim A. I.;
Al-Masoudi, Iman A.;
Saeed, Bahjat;
Al-Masoudi, Najim A.;
La Colla, Palo

Publication type:

Article

New benzylpiperazine derivatives bearing mono- and bis-dialkyl substituted 1,2,4-triazoles.

Published in:

Heteroatom Chemistry, 2005, v. 16, n. 1, p. 28, doi. 10.1002/hc.20061

By:

Al-Soud, Yaseen A.;
Qalalweh, Mohammed N. A.;
Al-Sa'doni, Haitham H.;
Al-Masoudi, Najim A.

Publication type:

Article

N- and C-acyclic thionuleoside analogues of 1,2,3-triazole.

Published in:

Heteroatom Chemistry, 2004, v. 15, n. 5, p. 380, doi. 10.1002/hc.20030

By:

Al-Masoudi, Najim A.;
Al-Soud, Yaseen A.;
Abdul-Zahra, Asmehan

Publication type:

Article

Synthesis of 3′-1,2,4-triazolo- and 3′-1,3,4-thiadiazoliminothymidines.

Published in:

Heteroatom Chemistry, 2003, v. 14, n. 4, p. 298, doi. 10.1002/hc.10146

By:

Al-Soud, Yaseen A.;
Al-Masoudi, Najim A.

Publication type:

Article

Synthesis, Anticancer Activity, and Molecular Docking Studies of Novel Substituted Isoxazole Derivatives Tethered 4‐Nitroimidazole.

Published in:

ChemistrySelect, 2025, v. 10, n. 24, p. 1, doi. 10.1002/slct.202500932

By:

Saber, Sadeekah O.;
Al‐Masoudi, Najim A.;
Al‐Soud, Yaseen A.;
Abu Qatouseh, Luay;
Saeed, Bahjat A.;
Al‐Qawasmeh, Raed A.

Publication type:

Article

New tamoxifen analogs for breast cancer therapy: synthesis, aromatase inhibition and in silico studies.

Published in:

Journal of Biomolecular Structure & Dynamics, 2023, v. 41, n. 22, p. 12798, doi. 10.1080/07391102.2023.2175375

By:

Al-Kelabi, Hasan;
Al-Duhaidahawi, Dunya;
Al-Khafaji, Khattab;
Al-Masoudi, Najim A.

Publication type:

Article

Synthesis and Antiviral Activity of New Substituted Methyl [2-(arylmethylene-hydrazino)-4-oxo-thiazolidin-5-ylidene]acetates.

Published in:

Archiv der Pharmazie, 2013, v. 346, n. 8, p. 618, doi. 10.1002/ardp.201300057

By:

Saeed, Aamer;
Al ‐ Masoudi, Najim A.;
Latif, Muhammad

Publication type:

Article

Amino Acid Derivatives, Part 4: Synthesis and Anti-HIV Activity of New Naphthalene Derivatives.

Published in:

Archiv der Pharmazie, 2010, v. 343, n. 7, p. 397, doi. 10.1002/ardp.200900293

By:

Hamad, Nawar S.;
Al-Haidery, Nahed H.;
Al-Masoudi, Iman A.;
Sabri, Mey;
Sabri, Luma;
Al-Masoudi, Najim A.

Publication type:

Article

Platinum and Palladium-triazole Complexes as Highly Potential Antitumor Agents.

Published in:

Archiv der Pharmazie, 2010, v. 343, n. 4, p. 222, doi. 10.1002/ardp.200900140

By:

Al-Masoudi, Najim A.;
Abdullah, Bayazeed H.;
Essa, Ali H.;
Loddo, Roberta;
LaColla, Paolo

Publication type:

Article

Synthesis and Antiviral Activity of 1-[(1,5-Dialkyl-1 H-1,2,4-triazol-3-yl)methyl]thymines.

Published in:

Archiv der Pharmazie, 1999, v. 332, n. 4, p. 143, doi. 10.1002/(SICI)1521-4184(19994)332:4<143::AID-ARDP143>3.0.CO;2-C

By:

Al-Soud, Yaseen A.;
Al-Masoudi, Najim A.

Publication type:

Article