Works by Akdemir, Atilla

Results: 35

Synthesis, anti‐TB activities, and molecular docking studies of 4‐(1,2,3‐triazoyl)arylmethanone derivatives.

Published in:

Journal of Biochemical & Molecular Toxicology, 2022, v. 36, n. 4, p. 1, doi. 10.1002/jbt.22998

By:

Turkmen, Yunus;
Yagiz Erdemir, Güler;
Yuksel Mayda, Pelin;
Akdemir, Atilla;
Gunaydin Akyildiz, Aysenur;
Altundas, Aliye

Publication type:

Article

Novel sulfonamide-based compounds as dual inhibitors of hCYP1B1 and hCYP19A1 with anticancer activity against breast cancer cells.

Published in:

Journal of Research in Pharmacy, 2025, v. 29, n. 3, p. 1098, doi. 10.12991/jrespharm.1694239

By:

İNCE-ERGÜÇ, Elif;
ERASLAN-ELMA, Pınar;
AKDEMIR, Atilla;
KARALI, Nilgun;
GURER-ORHAN, Hande

Publication type:

Article

Antiviral Properties of 5‑Sulfamoyl‑1H‑Indole-Linked Spirothiazolidinone Derivatives: A Study on Human Parainfluenza Virus-2.

Published in:

Journal of Research in Pharmacy, 2024, v. 28, n. 1, p. 213, doi. 10.29228/jrp.689

By:

TRAWALLY, Muhammed;
YILMAZ, Fatıma Nur;
ÖZBEK ÇELİK, Berna;
AKDEMİR, Atilla;
GÜZEL AKDEMİR, Özlen

Publication type:

Article

Molecular modelling studies to suggest novel scaffolds against SARS-CoV-2 target enzymes.

Published in:

Journal of Research in Pharmacy, 2021, v. 25, n. 6, p. 1010, doi. 10.29228/jrp.96

By:

ŞAHİN, Ahmet Fatih;
KÜÇÜKGÜZEL, Ş. Güniz;
AKDEMİR, Atilla

Publication type:

Article

Urease inhibitors for the treatment of H. pylori.

Published in:

Expert Opinion on Therapeutic Patents, 2025, v. 35, n. 1, p. 17, doi. 10.1080/13543776.2024.2423004

By:

Güzel-Akdemir, Özlen;
Akdemir, Atilla

Publication type:

Article

A Study On Synthesis, Biological Activities and Molecular Modelling of Some Novel Trisubstituted 1,2,4‐Triazole Derivatives.

Published in:

ChemistrySelect, 2018, v. 3, n. 31, p. 8813, doi. 10.1002/slct.201801578

By:

Gultekin, Ergun;
Kolcuoglu, Yakup;
Akdemir, Atilla;
Sirin, Yakup;
Bektas, Hakan;
Bekircan, Olcay

Publication type:

Article

New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1631, doi. 10.1080/14756366.2021.1954918

By:

Maccallini, Cristina;
Gallorini, Marialucia;
Sisto, Francesca;
Akdemir, Atilla;
Ammazzalorso, Alessandra;
De Filippis, Barbara;
Fantacuzzi, Marialuigia;
Giampietro, Letizia;
Carradori, Simone;
Cataldi, Amelia;
Amoroso, Rosa

Publication type:

Article

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1400, doi. 10.1080/14756366.2019.1651315

By:

Rotondi, Giulia;
Guglielmi, Paolo;
Carradori, Simone;
Secci, Daniela;
De Monte, Celeste;
De Filippis, Barbara;
Maccallini, Cristina;
Amoroso, Rosa;
Cirilli, Roberto;
Akdemir, Atilla;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1051, doi. 10.1080/14756366.2019.1611801

By:

Ammazzalorso, Alessandra;
Carradori, Simone;
Angeli, Andrea;
Akdemir, Atilla;
De Filippis, Barbara;
Fantacuzzi, Marialuigia;
Giampietro, Letizia;
Maccallini, Cristina;
Amoroso, Rosa;
Supuran, Claudiu T.

Publication type:

Article

Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 528, doi. 10.1080/14756366.2018.1564045

By:

Akdemir, Atilla;
Angeli, Andrea;
Göktaş, Füsun;
Eraslan Elma, Pınar;
Karalı, Nilgün;
Supuran, Claudiu T.

Publication type:

Article

Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1299, doi. 10.1080/14756366.2018.1499628

By:

Güzel-Akdemir, Özlen;
Angeli, Andrea;
Demir, Kübra;
Supuran, Claudiu T.;
Akdemir, Atilla

Publication type:

Article

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 51, doi. 10.1080/14756366.2016.1235040

By:

D'Ascenzio, Melissa;
Guglielmi, Paolo;
Carradori, Simone;
Secci, Daniela;
Florio, Rosalba;
Mollica, Adriano;
Ceruso, Mariangela;
Akdemir, Atilla;
Sobolev, Anatoly P.;
Supuran, Claudiu T.

Publication type:

Article

Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2015, v. 30, n. 1, p. 114, doi. 10.3109/14756366.2014.892936

By:

Akdemir, Atilla;
De Monte, Celeste;
Carradori, Simone;
Supuran, Claudiu T.

Publication type:

Article

Azole-Based Compounds That Are Active against Candida Biofilm: In Vitro , In Vivo and In Silico Studies.

Published in:

Antibiotics (2079-6382), 2022, v. 11, n. 10, p. N.PAG, doi. 10.3390/antibiotics11101375

By:

Carradori, Simone;
Ammazzalorso, Alessandra;
De Filippis, Barbara;
Şahin, Ahmet Fatih;
Akdemir, Atilla;
Orekhova, Anastasia;
Bonincontro, Graziana;
Simonetti, Giovanna

Publication type:

Article

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment.

Published in:

Metabolites (2218-1989), 2020, v. 10, n. 10, p. 412, doi. 10.3390/metabo10100412

By:

Angeli, Andrea;
Carta, Fabrizio;
Nocentini, Alessio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Akdemir, Atilla;
Onnis, Valentina;
Eldehna, Wagdy M.;
Capasso, Clemente;
Simone, Giuseppina De;
Monti, Simona Maria;
Carradori, Simone;
Donald, William A.;
Dedhar, Shoukat;
Supuran, Claudiu T.

Publication type:

Article

Synthesis, cytotoxic activities and molecular modeling studies of some 2-aminonaphtho[2,3-d][1,3]thiazole-4,9-dione derivatives.

Published in:

Organic Communications, 2020, v. 13, n. 4, p. 184, doi. 10.25135/acg.oc.91.20.11.1913

By:

Yanık, Hülya;
Ayan, Sümeyra;
Akdemir, Atilla;
Erdoğan, Ömer;
Üstündağ, Cem Bülent;
Çevik, Özge;
Yılmaz, Özgür

Publication type:

Article

Design and synthesis of novel peptidomimetics for cancer immunotherapy.

Published in:

Organic Communications, 2020, v. 13, n. 3, p. 89, doi. 10.25135/acg.oc.86.20.09.1802

By:

Köse, Ceyda;
Uysal, Esra;
Yazıcı, Büşra;
Tuğay, Zeynep;
Dingiş Birgül, Serap İpek;
Yanık, Hamdullah;
Tavukçuoğlu, Ece;
Gülyüz, Sevgi;
Akdemir, Atilla;
Esendağlı, Güneş;
Yılmaz, Özgür;
Alptürk, Onur

Publication type:

Article

Evaluation of new 2-hydroxy-N-(4-oxo-2-substituted phenyl-1,3- thiazolidin-3-yl)-2-phenylacetamide derivatives as potential antimycobacterial agents.

Published in:

Organic Communications, 2020, v. 13, n. 2, p. 33, doi. 10.25135/acg.oc.78.20.05.1655

By:

Güzel-Akdemir, Özlen;
Demir-Yazıcı, Kübra;
Trawally, Muhammed;
Dingiş-Birgü, Serap İpek;
Akdemir, Atilla

Publication type:

Article

Novel Indole-Based Hydrazones as Potent Inhibitors of the α-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae.

Published in:

International Journal of Molecular Sciences, 2020, v. 21, n. 9, p. 3131, doi. 10.3390/ijms21093131

By:

Demir-Yazıcı, Kübra;
Güzel-Akdemir, Özlen;
Angeli, Andrea;
Supuran, Claudiu T.;
Akdemir, Atilla

Publication type:

Article

Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII.

Published in:

International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2354, doi. 10.3390/ijms20092354

By:

Demir-Yazıcı, Kübra;
Bua, Silvia;
Akgüneş, Nurgül Mutlu;
Akdemir, Atilla;
Supuran, Claudiu T.;
Güzel-Akdemir, Özlen

Publication type:

Article

Computer-aided Drug Design on Glioblastoma Multiforme: Investigating Possible Inhibitors Against Factor H.

Published in:

Bezmialem Science, 2022, v. 10, p. S30

By:

ÖNCEL, Muhammed Miran;
KAZANCIOĞLU, Rümeyza;
KHAN, Mohammad Asif;
HATİBOĞLU, Mustafa Aziz;
AKDEMİR, Atilla

Publication type:

Article

YÖRESEL TAVIR BAĞLAMINDA SAHİH TİLAVET KRİTERLERİ.

Published in:

Review of the Faculty of Divinity of Amasya University, 2018, n. 11, p. 9, doi. 10.18498/amauifd.503733

By:

Akdemir, Mustafa Atilla

Publication type:

Article

The Quest for Ligands Against Kinesin Motor Protein Eg5.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 5, p. 1, doi. 10.1002/ardp.70010

By:

Sahin, Ahmet Fatih;
Carradori, Simone;
Ricci, Alessia;
Rashad, Muhammad;
Akdemir, Atilla

Publication type:

Article

Synthesis, In Vitro Evaluation, and Molecular Docking Studies of Novel 3,5‐Diphenyl‐1H‐1,2,4‐Triazole Derivatives as Potential hEGFR Inhibitors.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 5, p. 1, doi. 10.1002/ardp.70007

By:

Kolcuoglu, Yakup;
Bekircan, Olcay;
Ustalar, Narin;
Türe, Aslı;
Akdemir, Atilla;
Sanlier, Senay Hamarat

Publication type:

Article

New 1H‐indole‐2,3‐dione 3‐thiosemicarbazones with 3‐sulfamoylphenyl moiety as selective carbonic anhydrase inhibitors.

Published in:

Archiv der Pharmazie, 2022, v. 355, n. 8, p. 1, doi. 10.1002/ardp.202200023

By:

Eraslan‐Elma, Pınar;
Akdemir, Atilla;
Berrino, Emanuela;
Bozdağ, Murat;
Supuran, Claudiu T.;
Karalı, Nilgün

Publication type:

Article

Synthesis of new 1,2,4‐triazole–(thio)semicarbazide hybrid molecules: Their tyrosinase inhibitor activities and molecular docking analysis.

Published in:

Archiv der Pharmazie, 2021, v. 354, n. 8, p. 1, doi. 10.1002/ardp.202100058

By:

Gultekin, Ergün;
Bekircan, Olcay;
Kolcuoğlu, Yakup;
Akdemir, Atilla

Publication type:

Article

rac‐ and meso‐Cyclohexanoids: Their α‐, β‐glycosidases, antibacterial, antifungal activities, and molecular docking studies.

Published in:

Archiv der Pharmazie, 2020, v. 353, n. 3, p. 1, doi. 10.1002/ardp.201900267

By:

Karakılıç, Emel;
Baran, Şule;
Öğütçü, Hatice;
Akdemir, Atilla;
Baran, Arif

Publication type:

Article

Synthesis and Functional Investigations of Computer Designed Novel Cladribine-Like Compounds for the Treatment of Multiple Sclerosis.

Published in:

Archiv der Pharmazie, 2017, v. 350, n. 11, p. n/a, doi. 10.1002/ardp.201700185

By:

Yavuz, Serkan;
Çetin, Aysu;
Akdemir, Atilla;
Doyduk, Doğukan;
Dişli, Ali;
Çelik Turgut, Gurbet;
Şen, Alaattin;
Yıldırır, Yılmaz

Publication type:

Article

Design, Synthesis, and Investigation of Anticancer and Antioxidant Potential of Novel Indole‐Based Melatonin Analogues in Breast Cancer.

Published in:

ChemistrySelect, 2024, v. 9, n. 25, p. 1, doi. 10.1002/slct.202400817

By:

Ince‐Erguc, Elif;
Durgun, Kubra;
Akdemir, Atilla;
Suzen, Sibel;
Gurer‐Orhan, Hande

Publication type:

Article

İnsan Metilentetrahidrofolat Redüktaz Enziminin Kristal Yapısı İçin Bir Model.

Published in:

Journal of Harran University Medical Faculty / Harran Üniversitesi Tıp Fakültesi Dergisi, 2015, v. 12, n. 1, p. 23

By:

İzmirli, Müzeyyen;
Akdemir, Atilla;
Gögebakan, Bülent;
Alptekin, Davut

Publication type:

Article

Design and synthesis of new heterocyclic compounds containing 5-[(1H-1,2,4-triazol-1-yl)methyl]-3H-1,2,4-triazole-3-thione structure as potent hEGFR inhibitors.

Published in:

Journal of Biomolecular Structure & Dynamics, 2023, v. 41, n. 22, p. 12753, doi. 10.1080/07391102.2023.2167113

By:

Kolcuoglu, Yakup;
Bekircan, Olcay;
Fazli, Hilal;
Sahin, Emine;
Ture, Aslı;
Akdemir, Atilla;
Hamarat Sanlier, Senay

Publication type:

Article

Aromatase inhibition by 2-methyl indole hydrazone derivatives evaluated via molecular docking and in vitro activity studies.

Published in:

Xenobiotica, 2019, v. 49, n. 5, p. 549, doi. 10.1080/00498254.2018.1482029

By:

Ozcan-Sezer, Senem;
Ince, Elif;
Akdemir, Atilla;
Ceylan, €Ozlem €Ozt€urk;
Suzen, Sibel;
Gurer-Orhan, Hande

Publication type:

Article

Thiosemicarbazide-Substituted Coumarins as Selective Inhibitors of the Tumor Associated Human Carbonic Anhydrases IX and XII.

Published in:

Molecules, 2022, v. 27, n. 14, p. N.PAG, doi. 10.3390/molecules27144610

By:

Gumus, Arzu;
Bozdag, Murat;
Akdemir, Atilla;
Angeli, Andrea;
Selleri, Silvia;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Five- and Six-Membered Nitrogen-Containing Compounds as Selective Carbonic Anhydrase Activators.

Published in:

Molecules, 2017, v. 22, n. 12, p. 2178, doi. 10.3390/molecules22122178

By:

Mollica, Adriano;
Macedonio, Giorgia;
Stefanucci, Azzurra;
Carradori, Simone;
Akdemir, Atilla;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Synthesis of flurbiprofen thiadiazole urea derivatives and assessment of biological activities and molecular docking studies.

Published in:

Chemical Biology & Drug Design, 2023, v. 102, n. 6, p. 1458, doi. 10.1111/cbdd.14336

By:

Zengin Kurt, Belma;
Altundağ, Özlem;
Tokgöz, Merve Nur;
Öztürk Civelek, Dilek;
Tuncay, Fulya Oz;
Cakmak, Ummuhan;
Kolcuoğlu, Yakup;
Akdemir, Atilla;
Sönmez, Fatih

Publication type:

Article