Works matching AU Ghorab, Mostafa M.

Results: 47

Chemistry of 2-cyanomethylene-4-thiazolidinone.

Published in:

Journal of Sulfur Chemistry, 2017, v. 38, n. 3, p. 314, doi. 10.1080/17415993.2016.1263304

By:

El-Gaby, Mohamed S. A.;
Ammar, Yousry A.;
El-Hag Ali, Gameel A. M.;
Helal, Mohamed H. M.;
Salem, Mohamed A.;
Ghorab, Mostafa M.

Publication type:

Article

Novel iodoquinazolinones bearing sulfonamide moiety as potential antioxidants and neuroprotectors.

Published in:

Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-42239-2

By:

Soliman, Aiten M.;
Ghorab, Walid M.;
Lotfy, Dina M.;
Karam, Heba M.;
Ghorab, Mostafa M.;
Ramadan, Laila A.

Publication type:

Article

Novel iodoquinazolinones bearing sulfonamide moiety as potential antioxidants and neuroprotectors.

Published in:

Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-42239-2

By:

Soliman, Aiten M.;
Ghorab, Walid M.;
Lotfy, Dina M.;
Karam, Heba M.;
Ghorab, Mostafa M.;
Ramadan, Laila A.

Publication type:

Article

Synthesis, antimicrobial activity and docking study of some novel 4-(4,4-dimethyl-2,6-dioxocyclohexylidene)methylamino derivatives carrying biologically active sulfonamide moiety.

Published in:

Arabian Journal of Chemistry, 2020, v. 13, n. 1, p. 545, doi. 10.1016/j.arabjc.2017.05.022

By:

Ghorab, Mostafa M.;
Soliman, Aiten M.;
Alsaid, Mansour S.;
Askar, Ahmed A.

Publication type:

Article

Novel Quinazoline Derivatives Bearing a Sulfapyridine Moiety as Anticancer and Radiosensitizing Agents.

Published in:

Journal of Heterocyclic Chemistry, 2014, v. 51, p. E255, doi. 10.1002/jhet.1830

By:

Ghorab, Mostafa M.;
Ragab, Fatma A.;
Heiba, Helmi I.;
Bayomi, Ahmad A.

Publication type:

Article

Synthesis and antitumor activity of some novel hydrazide, 1,2-dihydropyridine, chromene, and benzochromene derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2012, v. 49, n. 2, p. 272, doi. 10.1002/jhet.829

By:

Ghorab, Mostafa M.;
Al-Said, Mansour S.

Publication type:

Article

Design and synthesis of some novel quinoline derivatives as anticancer and radiosensitizing agents targeting VEGFR tyrosine kinase.

Published in:

Journal of Heterocyclic Chemistry, 2011, v. 48, n. 6, p. 1269, doi. 10.1002/jhet.749

By:

Ghorab, Mostafa M.;
Ragab, Fatma A.;
Heiba, Helmy I.;
Ghorab, Walid M.

Publication type:

Article

In vitro cytotoxic evaluation of some new heterocyclic sulfonamide derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2011, v. 48, n. 3, p. 563, doi. 10.1002/jhet.619

By:

Ghorab, Mostafa M.;
Al-Said, Mansour S.;
El-Hossary, Ebaa M.

Publication type:

Article

Novel Thiophenes, Thienopyrimidines, and Triazolothienopyrimidines for the Evaluation of Anticancer and Augmentation Effects of γ-Radiation.

Published in:

Archiv der Pharmazie, 2010, v. 343, n. 7, p. 404, doi. 10.1002/ardp.200900150

By:

Shaaban, Mohamed A.;
Ghorab, Mostafa M.;
Heiba, Helmy I.;
Kamel, Mona M.;
Zaher, Nashwa H.;
Mostafa, Mohamed I.

Publication type:

Article

The Antiproliferative and Apoptotic Effects of a Novel Quinazoline Carrying Substituted-Sulfonamides: In Vitro and Molecular Docking Study.

Published in:

Molecules, 2022, v. 27, n. 3, p. 981, doi. 10.3390/molecules27030981

By:

Alqahtani, Ali S.;
Ghorab, Mostafa M.;
Nasr, Fahd A.;
Ahmed, Mohammad Z.;
Al-Mishari, Abdullah A.;
Attia, Sabry M.

Publication type:

Article

In-Vitro Anticancer Evaluation of Some Novel Thioureido-Benzensulfonamide Derivatives.

Published in:

Molecules, 2016, v. 21, n. 4, p. 409, doi. 10.3390/molecules21040409

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Al-Dosari, Mohammed S.;
El-Gazzar, Marwa G.;
Arbab, Ahmed H.

Publication type:

Article

Design, Synthesis and Anticancer Evaluation of Novel Quinazoline-Sulfonamide Hybrids.

Published in:

Molecules, 2016, v. 21, n. 2, p. 189, doi. 10.3390/molecules21020189

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Al-Dosari, Mohammed S.;
El-Gazzar, Marwa G.;
Parvez, Mohammad K.

Publication type:

Article

Crystal Structure of 4-(2-chloroacetamido)pyridinium chloride monohydrate, C7H10Cl2N2O2.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2017, v. 232, n. 1, p. 91, doi. 10.1515/ncrs-2016-0164

By:

Alsaid, Mansour S.;
Ghorab, Mostafa M.;
Ghabbour, Hazem A.

Publication type:

Article

Crystal structure of 4-((4,4-dimethyl-2, 6-dioxocyclohexylidine)methylamino)- N-(3,4-dimethylisoxazol-5-yl)benzenesulfonamide, C20H23N3O5S.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 4, p. 1117, doi. 10.1515/ncrs-2016-0082

By:

Alsaid, Mansour S.;
Ghorab, Mostafa M.;
AlRuqi, Obaid S.;
Ghabbour, Hazem A.;
Al-Mishari, Abdullah A.

Publication type:

Article

Crystal structure of ethyl-5-amino-1-(2,4-dinitrophenyl)-1 H-pyrazole-4-carboxylate, C12H11N5O6.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 699, doi. 10.1515/ncrs-2015-0239

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Ghabbour, Hazem A.

Publication type:

Article

Crystal structure of 2-((2-chloropyridin-3-ylamino)methylene)malononitrile, C9H5ClN4.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 711, doi. 10.1515/ncrs-2015-0242

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Al-Mishari, Abdullah A.;
AlRuqi, Obaid S.;
Ghabbour, Hazem A.

Publication type:

Article

Crystal structure of ( Z)-4-(4-oxopent-2-en-2-ylamino)benzenesulfonamide, C11H14N2O3S.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 867, doi. 10.1515/ncrs-2015-0297

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Ghabbour, Hazem A.;
Al-Mishari, Abdullah A.

Publication type:

Article

Crystal structure of 2-((dimethylamino)methylene)-5,5-Dimethylcyclohexane-1,3-dione, C11H17NO2.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 3, p. 903, doi. 10.1515/ncrs-2016-0002

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Ghabbour, Hazem A.;
Al-Mishari, Abdullah A.

Publication type:

Article

Crystal structure of (E)-1-(3,4-dimethoxyphenyl)-3-(dimethylamino)prop-2-en-1-one, C13H17NO3.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2016, v. 231, n. 2, p. 437, doi. 10.1515/ncrs-2015-0121

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Ghabbour, Hazem A.;
Hoong-Kun Fun

Publication type:

Article

Radioprotective and Antitumor Activity of Some Novel Amino Acids and Imidazoles Containing Thieno[2,3-d]pyrimidine Moiety.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2009, v. 184, n. 12, p. 3241, doi. 10.1080/10426500903126351

By:

Alqasoumi, Saleh I.;
Ragab, Fatma A.;
Alafeefy, Ahmed M.;
Galal, Marwa;
Ghorab, Mostafa M.

Publication type:

Article

Computer-Based Ligand Design and Synthesis of Some New Sulfonamides Bearing Pyrrole or Pyrrolopyrimidine Moieties Having Potential Antitumor and Radioprotective Activities.

Published in:

Phosphorus, Sulfur & Silicon & the Related Elements, 2008, v. 183, n. 1, p. 90, doi. 10.1080/10426500701557104

By:

Ghorab, Mostafa M.;
Heiba, Helmy I.;
Khalil, Amira I.;
Abou El Ella, Dalal A.;
Noaman, Eman

Publication type:

Article

Dapson in heterocyclic chemistry, part VIII: synthesis, molecular docking and anticancer activity of some novel sulfonylbiscompounds carrying biologically active 1,3-dihydropyridine, chromene and chromenopyridine moieties.

Published in:

Chemistry Central Journal, 2012, v. 6, n. 1, p. 64, doi. 10.1186/1752-153X-6-64

By:

Al-Said, Mansour S.;
Ghorab, Mostafa M.;
Nissan, Yassin M.

Publication type:

Article

Novel N-(Substituted) Thioacetamide Quinazolinone Benzenesulfonamides as Antimicrobial Agents.

Published in:

International Journal of Nanomedicine, 2020, v. 15, p. 3161, doi. 10.2147/IJN.S241433

By:

Ghorab, Mostafa M;
Alqahtani, Ali S;
Soliman, Aiten M;
Askar, Ahmed A

Publication type:

Article

Antimicrobial and anticancer activity of some novel fluorinated thiourea derivatives carrying sulfonamide moieties: synthesis, biological evaluation and molecular docking.

Published in:

Chemistry Central Journal, 2017, v. 11, p. 1, doi. 10.1186/s13065-017-0258-4

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
El-Gaby, Mohamed S. A.;
Elaasser, Mahmoud M.;
Nissan, Yassin M.

Publication type:

Article

Crystal structure of the co-crystalline adduct 4-((4,4-dimethyl-2,6-dioxocyclohexylidene) methylamino)-N-(4,6-dimethylpyrimidin-2-yl) benzenesulfonamide - acetic acid (1/1), C21H24N4O4S ⋅ C2H4O2.

Published in:

Zeitschrift für Kristallographie / New Crystal Structures, 2017, v. 232, n. 3, p. 417, doi. 10.1515/ncrs-2016-0295

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Al-Dosari, Mohmmed S.;
Ghabbour, Hazem A.

Publication type:

Article

Synthesis, Antimicrobial, and Antibiofilm Activities of Some Novel 7-Methoxyquinoline Derivatives Bearing Sulfonamide Moiety against Urinary Tract Infection-Causing Pathogenic Microbes.

Published in:

International Journal of Molecular Sciences, 2023, v. 24, n. 10, p. 8933, doi. 10.3390/ijms24108933

By:

Ghorab, Mostafa M.;
M. Soliman, Aiten;
El-Sayyad, Gharieb S.;
Abdel-Kader, Maged S.;
El-Batal, Ahmed I.

Publication type:

Article

Cytotoxicity of Newly Synthesized Quinazoline–Sulfonamide Derivatives in Human Leukemia Cell Lines and Their Effect on Hematopoiesis in Zebrafish Embryos.

Published in:

International Journal of Molecular Sciences, 2022, v. 23, n. 9, p. 4720, doi. 10.3390/ijms23094720

By:

Alqahtani, Ali S.;
Ghorab, Mostafa M.;
Nasr, Fahd A.;
Ahmed, Mohammad Z.;
Al Mishari, Abdullah A.;
Attia, Sabry M.;
Farooq Khan, Muhammad

Publication type:

Article

Synthesis, Characterization and Anti-Breast Cancer Activity of New 4-Aminoantipyrine-Based Heterocycles.

Published in:

International Journal of Molecular Sciences, 2014, v. 15, n. 5, p. 7539, doi. 10.3390/ijms15057539

By:

Ghorab, Mostafa M.;
El-Gazzar, Marwa G.;
Alsaid, Mansour S.

Publication type:

Article

Synthesis and Anti-Breast Cancer Evaluation of Novel N-(Guanidinyl)benzenesulfonamides.

Published in:

International Journal of Molecular Sciences, 2014, v. 15, n. 4, p. 5582, doi. 10.3390/ijms15045582

By:

Ghorab, Mostafa M.;
El-Gazzar, Marwa G.;
Alsaid, Mansour S.

Publication type:

Article

Synthesis, DFT calculations, and anti-proliferative evaluation of pyrimidine and selenadiazolopyrimidine derivatives as dual Topoisomerase II and HSP90 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2198163

By:

El-Kalyoubi, Samar;
El-Sebaey, Samiha A.;
Rashad, A. M.;
AL-Ghulikah, Hanan A.;
Ghorab, Mostafa M.;
Elfeky, Sherin M.

Publication type:

Article

Novel sulphonamide-bearing methoxyquinazolinone derivatives as anticancer and apoptosis inducers: synthesis, biological evaluation and in silico studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 86, doi. 10.1080/14756366.2021.1983807

By:

Alqahtani, Ali S.;
Ghorab, Mostafa M.;
Nasr, Fahd A.;
Ahmed, Mohammad Z.;
Al-Mishari, Abdullah A.;
Attia, Sabry M.

Publication type:

Article

Synthesis of some quinazolinones inspired from the natural alkaloid L-norephedrine as EGFR inhibitors and radiosensitizers.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 218, doi. 10.1080/14756366.2020.1854243

By:

Ghorab, Mostafa M.;
Abdel-Kader, Maged S.;
Alqahtani, Ali S.;
Soliman, Aiten M.

Publication type:

Article

Novel sulfonamide benzoquinazolinones as dual EGFR/HER2 inhibitors, apoptosis inducers and radiosensitizers.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1030, doi. 10.1080/14756366.2019.1609469

By:

Soliman, Aiten M.;
Alqahtani, Ali S.;
Ghorab, Mostafa M.

Publication type:

Article

Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1565, doi. 10.1080/14756366.2018.1513927

By:

El-Gazzar, Marwa G.;
Nafie, Nessma H.;
Nocentini, Alessio;
Ghorab, Mostafa M.;
Heiba, Helmi I.;
Supuran, Claudiu T.

Publication type:

Article

Benzo[g]quinazolin-based scaffold derivatives as dual EGFR/HER2 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 67, doi. 10.1080/14756366.2017.1389922

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Soliman, Aiten M.;
Al-Mishari, Abdullah A.

Publication type:

Article

VEGFR-2 inhibitors and apoptosis inducers: synthesis and molecular design of new benzo [g] quinazolin bearing benzenesulfonamide moiety.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 893, doi. 10.1080/14756366.2017.1334650

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Soliman, Aiten M.;
Ragab, Fatma A.

Publication type:

Article

Synthesis and biological evaluation of novel 2-phenylquinazoline-4-amine derivatives: identification of 6-phenyl-8H-benzo[g]quinazolino[4,3-b]quinazolin-8-one as a highly potent inducer of NAD(P)H quinone oxidoreductase 1.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, p. 34, doi. 10.3109/14756366.2016.1163343

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
El-Gazzar, Marwa G.;
Higgins, Maureen;
Dinkova-Kostova, Albena T.;
Shahat, Abdelaaty A.

Publication type:

Article

Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel 2-phenylquinazolin-4-amine derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1612, doi. 10.3109/14756366.2016.1158714

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Higgins, Maureen;
Dinkova-Kostova, Albena T.;
Shahat, Abdelaaty A.;
Elghazawy, Nehal H.;
Arafa, Reem K.

Publication type:

Article

NAD(P)H: quinone oxidoreductase 1 inducer activity of novel 4-aminoquinazoline derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 6, p. 1369, doi. 10.3109/14756366.2015.1135913

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
El-Gazzar, Marwa G.;
Higgins, Maureen;
Dinkova-Kostova, Albena T.;
Shahat, Abdelaaty A.

Publication type:

Article

Synthesis, molecular modeling and NAD(P)H:quinone oxidoreductase 1 inducer activity of novel cyanoenone and enone benzenesulfonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 6, p. 840, doi. 10.3109/14756366.2013.858146

By:

Ghorab, Mostafa M.;
Higgins, Maureen;
Alsaid, Mansour S.;
Arafa, Reem K.;
Shahat, Abdelaaty A.;
Dinkova-Kostova, Albena T.

Publication type:

Article

Design, synthesis and molecular docking of novel N,N-dimethylbenzenesulfonamide derivatives as potential antiproliferative agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2014, v. 29, n. 5, p. 619, doi. 10.3109/14756366.2013.833197

By:

Bashandy, Mahmoud S.;
Alsaid, Mansour S.;
Arafa, Reem K.;
Ghorab, Mostafa M.

Publication type:

Article

Utility of methyl 2-isothiocyanatobenzoate in the synthesis of some new quinazoline derivatives as potential anticancer and radiosensitizing agents.

Published in:

Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 12, p. 719

By:

Ghorab, Mostafa M.;
Ragab, Fatma A.;
Heiba, Helmi I.;
Bayomi, Ahmad A.

Publication type:

Article

Novel quinolines bearing a biologically active trimethoxyphenyl moiety as a new class of antitumor agents.

Published in:

Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 9, p. 527, doi. 10.1055/s-0031-1296239

By:

Al-Said, Mansour S.;
Bashandy, Mahmoud S.;
Ghorab, Mostafa M.

Publication type:

Article

Design and synthesis of some novel hydrazide, 1,2 - dihydropyridine, chromene derivatives carrying biologically active sulfone moieties with potential anticancer activity.

Published in:

Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2011, v. 61, n. 9, p. 521, doi. 10.1055/s-0031-1296238

By:

Bashandy, Mahmoud S.;
Al-Said, Mansour S.;
Al-Qasoumi, Saleh I.;
Ghorab, Mostafa M.

Publication type:

Article

Synthesis of Certain New Thieno[2,3-d] pyrimidines as Potential Antitumor and Radioprotective Agents.

Published in:

Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2006, v. 56, n. 7, p. 553

By:

Ghorab, Mostafa M.;
Ragab, Fatma A.;
Noaman, Eman;
Heiba, Helmy I.;
Galal, Marwa

Publication type:

Article

Novel Synthesis of Pyrrolo[2,3-d] pyrimidines Bearing Sulfonamide Moieties as Potential Antitumor and Radioprotective Agents.

Published in:

Drug Research / Arzneimittel-Forschung (Editio Cantor Verlag fur Medizin und Naturwissenschaften), 2006, v. 56, n. 4, p. 301

By:

Ismail, Magda M. F.;
Ghorab, Mostafa M.;
Noaman, Eman;
Ammar, Yousry A.;
Heiba, Helmy I.;
Sayed, Marwa Y.

Publication type:

Article

NAD(P)H:quinone oxidoreductase 1 inducer activity of some novel anilinoquinazoline derivatives.

Published in:

Drug Design, Development & Therapy, 2016, v. 10, p. 2515, doi. 10.2147/DDDT.S105423

By:

Ghorab, Mostafa M.;
Alsaid, Mansour S.;
Higgins, Maureen;
Dinkova-Kostova, Albena T.;
Shahat, Abdelaaty A.;
Elghazawy, Nehal H.;
Arafa, Reem K.

Publication type:

Article