Works matching AU Kaczor, Agnieszka A.


Results: 95
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    Synthesis, Docking Studies and Pharmacological Evaluation of Serotoninergic Ligands Containing a 5-Norbornene-2-Carboxamide Nucleus.

    Published in:
    Molecules, 2022, v. 27, n. 19, p. 6492, doi. 10.3390/molecules27196492
    By:
    • Sparaco, Rosa;
    • Kędzierska, Ewa;
    • Kaczor, Agnieszka A.;
    • Bielenica, Anna;
    • Magli, Elisa;
    • Severino, Beatrice;
    • Corvino, Angela;
    • Gibuła-Tarłowska, Ewa;
    • Kotlińska, Jolanta H.;
    • Andreozzi, Giorgia;
    • Luciano, Paolo;
    • Perissutti, Elisa;
    • Frecentese, Francesco;
    • Casertano, Marcello;
    • Leśniak, Anna;
    • Bujalska-Zadrożny, Magdalena;
    • Oziębło, Małgorzata;
    • Capasso, Raffaele;
    • Santagada, Vincenzo;
    • Caliendo, Giuseppe
    Publication type:
    Article
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    Synthesis, docking studies, and pharmacological evaluation of 2‐hydroxypropyl‐4‐arylpiperazine derivatives as serotoninergic ligands.

    Published in:
    Archiv der Pharmazie, 2021, v. 354, n. 5, p. 1, doi. 10.1002/ardp.202000414
    By:
    • Magli, Elisa;
    • Kędzierska, Ewa;
    • Kaczor, Agnieszka A.;
    • Bielenica, Anna;
    • Severino, Beatrice;
    • Gibuła‐Tarłowska, Ewa;
    • Kotlińska, Jolanta H.;
    • Corvino, Angela;
    • Sparaco, Rosa;
    • Esposito, Giovanna;
    • Albrizio, Stefania;
    • Perissutti, Elisa;
    • Frecentese, Francesco;
    • Leśniak, Anna;
    • Bujalska‐Zadrożny, Magdalena;
    • Struga, Marta;
    • Capasso, Raffaele;
    • Santagada, Vincenzo;
    • Caliendo, Giuseppe;
    • Fiorino, Ferdinando
    Publication type:
    Article
    31

    Synthesis, docking studies, and pharmacological evaluation of 5HT<sub>2C</sub> ligands containing the N′‐cyanoisonicotinamidine or N′‐cyanopicolinamidine nucleus.

    Published in:
    Archiv der Pharmazie, 2019, v. 352, n. 5, p. 1, doi. 10.1002/ardp.201800373
    By:
    • Magli, Elisa;
    • Kędzierska, Ewa;
    • Kaczor, Agnieszka A.;
    • Severino, Beatrice;
    • Corvino, Angela;
    • Perissutti, Elisa;
    • Frecentese, Francesco;
    • Saccone, Irene;
    • Massarelli, Paola;
    • Gibuła‐Tarłowska, Ewa;
    • Kotlińska, Jolanta H.;
    • Santagada, Vincenzo;
    • Caliendo, Giuseppe;
    • Fiorino, Ferdinando
    Publication type:
    Article
    32

    Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds–synthesis, biological activity, and structural evaluation.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2209828
    By:
    • Stępnicki, Piotr;
    • Wronikowska-Denysiuk, Olga;
    • Zięba, Agata;
    • Targowska-Duda, Katarzyna M.;
    • Bartyzel, Agata;
    • Wróbel, Martyna Z.;
    • Wróbel, Tomasz M.;
    • Szałaj, Klaudia;
    • Chodkowski, Andrzej;
    • Mirecka, Karolina;
    • Budzyńska, Barbara;
    • Fornal, Emilia;
    • Turło, Jadwiga;
    • Castro, Marián;
    • Kaczor, Agnieszka A.
    Publication type:
    Article
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    Discovery of nitroaryl urea derivatives with antiproliferative properties.

    Published in:
    Journal of Enzyme Inhibition & Medicinal Chemistry, 2016, v. 31, n. 4, p. 608, doi. 10.3109/14756366.2015.1057716
    By:
    • Wróbel, Tomasz M.;
    • Kiełbus, Michał;
    • Kaczor, Agnieszka A.;
    • Kryštof, Vladimír;
    • Karczmarzyk, Zbigniew;
    • Wysocki, Waldemar;
    • Fruziński, Andrzej;
    • Król, Sylwia K.;
    • Grabarska, Aneta;
    • Stepulak, Andrzej;
    • Matosiuk, Dariusz
    Publication type:
    Article
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    Optimization of 1,2,5-Thiadiazole Carbamates as Potent and Selective ABHD6 Inhibitors.

    Published in:
    ChemMedChem, 2015, v. 10, n. 2, p. 253, doi. 10.1002/cmdc.201402453
    By:
    • Patel, Jayendra Z.;
    • Nevalainen, Tapio J.;
    • Savinainen, Juha R.;
    • Adams, Yahaya;
    • Laitinen, Tuomo;
    • Runyon, Robert S.;
    • Vaara, Miia;
    • Ahenkorah, Stephen;
    • Kaczor, Agnieszka A.;
    • Navia‐Paldanius, Dina;
    • Gynther, Mikko;
    • Aaltonen, Niina;
    • Joharapurkar, Amit A.;
    • Jain, Mukul R.;
    • Haka, Abigail S.;
    • Maxfield, Frederick R.;
    • Laitinen, Jarmo T.;
    • Parkkari, Teija
    Publication type:
    Article
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