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Development and radiosynthesis of the first <sup>18</sup>F‐labeled inhibitor of monocarboxylate transporters (MCTs).
- Published in:
- Journal of Labelled Compounds & Radiopharmaceuticals, 2019, v. 62, n. 8, p. 411, doi. 10.1002/jlcr.3739
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- Publication type:
- Article
<sup>18</sup>F‐Labeled benzylpiperazine derivatives as highly selective ligands for imaging σ<sub>1</sub> receptor with positron emission tomography.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2019, v. 62, n. 8, p. 425, doi. 10.1002/jlcr.3738
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- Publication type:
- Article
Radiosynthesis and biological evaluation of the new PDE10A radioligand [<sup>18</sup>F]AQ28A.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2017, v. 60, n. 1, p. 36, doi. 10.1002/jlcr.3471
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- Publication type:
- Article
Synthesis and evaluation of a <sup>18</sup>F-labeled 4-phenylpiperidine-4-carbonitrile radioligand for σ<sub>1</sub> receptor imaging.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2016, v. 59, n. 9, p. 332, doi. 10.1002/jlcr.3408
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- Publication type:
- Article
In vitro binding profile and radiosynthesis of a novel <sup>18</sup>F-labeled azaspirovesamicol analog as potential ligand for imaging of the vesicular acetylcholine transporter.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2011, v. 54, n. 8, p. 426, doi. 10.1002/jlcr.1891
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- Publication type:
- Article
Synthesis and biological evaluation of a radioiodinated spiropiperidine ligand as a potential σ<sub>1</sub> receptor imaging agent.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2010, v. 53, n. 9, p. 569, doi. 10.1002/jlcr.1777
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- Publication type:
- Article
Radiosynthesis of novel <sup>18</sup>F-labelled derivatives of indiplon as potential GABA<sub>A</sub> receptor imaging tracers for PET.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2008, v. 51, n. 3, p. 123, doi. 10.1002/jlcr.1473
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- Publication type:
- Article
Preparation and biological evaluation of <sup>99m</sup>TcN-4-(cyclohexylpiperazin-1-yl)-dithioformate as a potential sigma receptor imaging agent.
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- Journal of Labelled Compounds & Radiopharmaceuticals, 2007, v. 50, n. 13, p. 1200, doi. 10.1002/jlcr.1438
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- Publication type:
- Article
Nemacol is a small molecule inhibitor of C. elegans vesicular acetylcholine transporter with anthelmintic potential.
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- Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-37452-6
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- Article
Imaging of Gα q Proteins in Mouse and Human Organs and Tissues.
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- Pharmaceutics, 2023, v. 15, n. 1, p. 57, doi. 10.3390/pharmaceutics15010057
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- Publication type:
- Article
Amphiphilic Anionic Oligomer-Stabilized Calcium Phosphate Nanoparticles with Prospects in siRNA Delivery via Convection-Enhanced Delivery.
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- Pharmaceutics, 2022, v. 14, n. 2, p. 326, doi. 10.3390/pharmaceutics14020326
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- Publication type:
- Article
Radiosynthesis and Preclinical Evaluation of an 18 F-Labeled Triazolopyridopyrazine-Based Inhibitor for Neuroimaging of the Phosphodiesterase 2A (PDE2A).
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- Pharmaceuticals (14248247), 2022, v. 15, n. 10, p. 1272, doi. 10.3390/ph15101272
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- Publication type:
- Article
Quantitation of the A 2A Adenosine Receptor Density in the Striatum of Mice and Pigs with [ 18 F]FLUDA by Positron Emission Tomography.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 5, p. 516, doi. 10.3390/ph15050516
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- Publication type:
- Article
Development and Biological Evaluation of the First Highly Potent and Specific Benzamide-Based Radiotracer [ 18 F]BA3 for Imaging of Histone Deacetylases 1 and 2 in Brain.
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- Pharmaceuticals (14248247), 2022, v. 15, n. 3, p. 324, doi. 10.3390/ph15030324
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- Publication type:
- Article
Synthesis of Novel Fluorinated Xanthine Derivatives with High Adenosine A 2B Receptor Binding Affinity.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 5, p. 485, doi. 10.3390/ph14050485
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- Publication type:
- Article
Validation of an LC-MS/MS Method to Quantify the New TRPC6 Inhibitor SH045 (Larixyl N -methylcarbamate) and Its Application in an Exploratory Pharmacokinetic Study in Mice.
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- Pharmaceuticals (14248247), 2021, v. 14, n. 3, p. 259, doi. 10.3390/ph14030259
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- Publication type:
- Article
Development of a New Radiofluorinated Quinoline Analog for PET Imaging of Phosphodiesterase 5 (PDE5) in Brain.
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- Pharmaceuticals (14248247), 2016, v. 9, n. 2, p. 22, doi. 10.3390/ph9020022
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- Publication type:
- Article
Asymmetric Synthesis of Spirocyclic 2-Benzopyrans for Positron Emission Tomography of σ1 Receptors in the Brain.
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- Pharmaceuticals (14248247), 2014, v. 7, n. 1, p. 78, doi. 10.3390/ph7010078
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- Publication type:
- Article
Radiosynthesis and Radiotracer Properties of a 7-(2-[<sup>18</sup>F]Fluoroethoxy)-6-methoxypyrrolidinylquinazoline for Imaging of Phosphodiesterase 10A with PET.
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- Pharmaceuticals (14248247), 2012, v. 5, n. 6, p. 169, doi. 10.3390/ph5020169
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- Publication type:
- Article
A novel thermoregulatory role for PDE10A in mouse and human adipocytes.
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- EMBO Molecular Medicine, 2016, v. 8, n. 7, p. 796, doi. 10.15252/emmm.201506085
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- Publication type:
- Article
Development of F-labeled radiotracers for neuroreceptor imaging with positron emission tomography.
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- Neuroscience Bulletin, 2014, v. 30, n. 5, p. 777, doi. 10.1007/s12264-014-1460-6
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- Publication type:
- Article
Non-Invasive Assessment of Locally Overexpressed Human Adenosine 2A Receptors in the Heart of Transgenic Mice.
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- International Journal of Molecular Sciences, 2022, v. 23, n. 3, p. 1025, doi. 10.3390/ijms23031025
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- Publication type:
- Article
Development of [ 18 F]LU14 for PET Imaging of Cannabinoid Receptor Type 2 in the Brain.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 15, p. 8051, doi. 10.3390/ijms22158051
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- Publication type:
- Article
Design, Radiosynthesis and Preliminary Biological Evaluation in Mice of a Brain-Penetrant 18 F-Labelled σ 2 Receptor Ligand.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 11, p. 5447, doi. 10.3390/ijms22115447
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- Publication type:
- Article
Challenges on Cyclic Nucleotide Phosphodiesterases Imaging with Positron Emission Tomography: Novel Radioligands and (Pre-)Clinical Insights since 2016.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 8, p. 3832, doi. 10.3390/ijms22083832
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- Publication type:
- Article
Development of 18 F-Labeled Radiotracers for PET Imaging of the Adenosine A 2A Receptor: Synthesis, Radiolabeling and Preliminary Biological Evaluation.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 5, p. 2285, doi. 10.3390/ijms22052285
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- Publication type:
- Article
Preclinical Evaluation of [ 18 F]FACH in Healthy Mice and Piglets: An 18 F-Labeled Ligand for Imaging of Monocarboxylate Transporters with PET.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 4, p. 1645, doi. 10.3390/ijms22041645
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- Publication type:
- Article
Synthesis and Biological Evaluation of a Novel 18 F-Labeled Radiotracer for PET Imaging of the Adenosine A 2A Receptor.
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- International Journal of Molecular Sciences, 2021, v. 22, n. 3, p. 1182, doi. 10.3390/ijms22031182
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- Publication type:
- Article
In Silico Finding of Key Interaction Mediated α3β4 and α7 Nicotinic Acetylcholine Receptor Ligand Selectivity of Quinuclidine-Triazole Chemotype.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 17, p. 6189, doi. 10.3390/ijms21176189
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- Article
Development of a Radiofluorinated Adenosine A2B Receptor Antagonist as Potential Ligand for PET Imaging.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 9, p. 3197, doi. 10.3390/ijms21093197
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- Publication type:
- Article
Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging.
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- International Journal of Molecular Sciences, 2017, v. 18, n. 4, p. 768, doi. 10.3390/ijms18040768
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- Publication type:
- Article
Early increase of cannabinoid receptor density after experimental traumatic brain injury in the newborn piglet.
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- Acta Neurobiologiae Experimentalis, 2014, v. 74, n. 2, p. 197, doi. 10.55782/ane-2014-1985
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- Publication type:
- Article
Relation between brain tissue pO<sub>2</sub> and dopamine synthesis of basal ganglia - A <sup>18</sup>FDOPA-PET study in newborn piglets.
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- Journal of Perinatal Medicine, 2000, v. 28, n. 1, p. 54
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- Publication type:
- Article
Structure–Affinity Relationships of Fluorinated Spirocyclic σ<sub>2</sub> Receptor Ligands with an Exocyclic Benzylamino Moiety.
- Published in:
- ChemMedChem, 2019, v. 14, n. 15, p. 1392, doi. 10.1002/cmdc.201900284
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- Publication type:
- Article
First in man study to image alpha4beta2 cerebral nicotinic acetylcholine receptors (nAChRs) in early Alzheimer's disease (AD) with the new radioligand (-)-[18F]-norchloro-fluoro-homoepibatidine (NCFHEB) and PET
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- 2011
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- Publication type:
- Abstract
Thyroid hormone status defines brown adipose tissue activity and browning of white adipose tissues in mice.
- Published in:
- Scientific Reports, 2016, p. 38124, doi. 10.1038/srep38124
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- Publication type:
- Article
Enantioselective σ<sub>1</sub> receptor binding and biotransformation of the spirocyclic PET tracer 1′-benzyl-3-(3-fluoropropyl)-3 H-spiro[[2]benzofuran-1,4′-piperidine].
- Published in:
- Chirality, 2011, v. 23, n. 2, p. 148, doi. 10.1002/chir.20893
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- Publication type:
- Article
A 3D-QSAR model for cannabinoid receptor (CB2) ligands derived from aligned pharmacophors.
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- 2013
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- Publication type:
- Conference Paper/Materials
Synergistic approach of structure-based and ligand-based drug design for the development of selective cannabinod receptor ligands.
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- 2012
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- Publication type:
- Abstract
In vivo measurement of nicotinic acetylcholine receptors with [<sup>18</sup>F]norchloro-fluoro-homoepibatidine.
- Published in:
- Synapse, 2008, v. 62, n. 3, p. 205, doi. 10.1002/syn.20480
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- Publication type:
- Article
Autoradiography of 2-[<sup>18</sup>F]F-A-85380 on nicotinic acetylcholine receptors in the porcine brain in vitro.
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- Synapse, 2006, v. 59, n. 4, p. 201, doi. 10.1002/syn.20232
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- Publication type:
- Article
Positron emission tomography imaging of the serotonin transporter in the pig brain using [<sup>11</sup>C](+)-McN5652 and S-([<sup>18</sup>F]fluoromethyl)-(+)-McN5652.
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- Synapse, 2003, v. 47, n. 2, p. 143, doi. 10.1002/syn.10163
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- Publication type:
- Article
S-[<sup>18</sup>F]fluoromethyl-(+)-McN5652, a PET tracer for the serotonin transporter: Evaluation in rats.
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- Synapse, 2003, v. 47, n. 1, p. 45, doi. 10.1002/syn.10150
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- Publication type:
- Article
Quantitative radioluminography of serotonin uptake sites in the porcine brain.
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- Synapse, 2001, v. 39, n. 4, p. 351, doi. 10.1002/1098-2396(20010315)39:4<351::AID-SYN1019>3.0.CO;2-M
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- Publication type:
- Article
Hydroxyalkylation with Cyclic Sulfates: Synthesis of Carbazole Derived CB<sub>2</sub> Ligands with Increased Polarity.
- Published in:
- Archiv der Pharmazie, 2014, v. 347, n. 1, p. 21, doi. 10.1002/ardp.201300255
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- Publication type:
- Article
Automated radiosynthesis of the adenosine A<sub>2A</sub> receptor‐targeting radiotracer [<sup>18</sup>F]FLUDA.
- Published in:
- Journal of Labelled Compounds & Radiopharmaceuticals, 2022, v. 65, n. 6, p. 162, doi. 10.1002/jlcr.3970
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- Publication type:
- Article
One-step radiosynthesis of the MCTs imaging agent [18F]FACH by aliphatic 18F-labelling of a methylsulfonate precursor containing an unprotected carboxylic acid group.
- Published in:
- Scientific Reports, 2019, v. 9, n. 1, p. 1, doi. 10.1038/s41598-019-55354-w
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- Publication type:
- Article
Suppressed Fat Appetite after Roux-en-Y Gastric Bypass Surgery Associates with Reduced Brain μ-opioid Receptor Availability in Diet-Induced Obese Male Rats.
- Published in:
- Frontiers in Neuroscience, 2017, v. 10, p. 1, doi. 10.3389/fnins.2016.00620
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- Publication type:
- Article
Changes in Binding of [I]CLINDE, a High-Affinity Translocator Protein 18 kDa (TSPO) Selective Radioligand in a Rat Model of Traumatic Brain Injury.
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- NeuroMolecular Medicine, 2016, v. 18, n. 2, p. 158, doi. 10.1007/s12017-016-8385-y
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- Publication type:
- Article
Traumatic Brain Injury Elicits Similar Alterations in α7 Nicotinic Receptor Density in Two Different Experimental Models.
- Published in:
- NeuroMolecular Medicine, 2011, v. 13, n. 1, p. 44, doi. 10.1007/s12017-010-8136-4
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- Publication type:
- Article