Works matching AU Bua, Silvia
Results: 40
Carbonic anhydrase inhibitory activity of phthalimide-capped benzene sulphonamide derivatives.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2235089
- By:
- Publication type:
- Article
The three-tails approach as a new strategy to improve selectivity of action of sulphonamide inhibitors against tumour-associated carbonic anhydrase IX and XII.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 930, doi. 10.1080/14756366.2022.2053526
- By:
- Publication type:
- Article
Vanillin enones as selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII. The out of the active site pocket for the design of selective inhibitors?
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 2118, doi. 10.1080/14756366.2021.1982933
- By:
- Publication type:
- Article
Sulphonamide inhibition profile of Staphylococcus aureus β-carbonic anhydrase.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1834, doi. 10.1080/14756366.2020.1826942
- By:
- Publication type:
- Article
Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1765, doi. 10.1080/14756366.2020.1822829
- By:
- Publication type:
- Article
Escherichia coliγ-carbonic anhydrase: characterisation and effects of simple aromatic/heterocyclic sulphonamide inhibitors.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1545, doi. 10.1080/14756366.2020.1800670
- By:
- Publication type:
- Article
S-substituted 2-mercaptoquinazolin-4(3H)-one and 4-ethylbenzensulfonamides act as potent and selective human carbonic anhydrase IX and XII inhibitors.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 733, doi. 10.1080/14756366.2020.1742117
- By:
- Publication type:
- Article
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1697, doi. 10.1080/14756366.2019.1666836
- By:
- Publication type:
- Article
Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamides as carbonic anhydrase isoforms I and II inhibitors.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1457, doi. 10.1080/14756366.2019.1652282
- By:
- Publication type:
- Article
Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2019, v. 34, n. 1, p. 1193, doi. 10.1080/14756366.2019.1630616
- By:
- Publication type:
- Article
Discovery of novel 1,3-diaryltriazene sulfonamides as carbonic anhydrase I, II, VII, and IX inhibitors.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1575, doi. 10.1080/14756366.2018.1515933
- By:
- Publication type:
- Article
Synthesis, X-ray structure, in silico calculation, and carbonic anhydrase inhibitory properties of benzylimidazole metal complexes.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1150, doi. 10.1080/14756366.2018.1481404
- By:
- Publication type:
- Article
Evaluation of sulphonamide derivatives acting as inhibitors of human carbonic anhydrase isoforms I, II and Mycobacterium tuberculosis β-class enzyme Rv3273.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 962, doi. 10.1080/14756366.2018.1471475
- By:
- Publication type:
- Article
Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 1125, doi. 10.1080/14756366.2018.1467901
- By:
- Publication type:
- Article
Mono- and di-thiocarbamate inhibition studies of the δ-carbonic anhydrase TweCAδ from the marine diatom Thalassiosira weissflogii.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 707, doi. 10.1080/14756366.2018.1450400
- By:
- Publication type:
- Article
Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 629, doi. 10.1080/14756366.2018.1446432
- By:
- Publication type:
- Article
Resolution of co-eluting isomers of anti-inflammatory drugs conjugated to carbonic anhydrase inhibitors from plasma in liquid chromatography by energy-resolved tandem mass spectrometry.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2018, v. 33, n. 1, p. 671, doi. 10.1080/14756366.2018.1445737
- By:
- Publication type:
- Article
Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 1187, doi. 10.1080/14756366.2017.1367775
- By:
- Publication type:
- Article
Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 885, doi. 10.1080/14756366.2017.1337759
- By:
- Publication type:
- Article
Advances in new psychoactive substances identification: the U.R.I.To.N. Consortium.
- Published in:
- Journal of Enzyme Inhibition & Medicinal Chemistry, 2017, v. 32, n. 1, p. 841, doi. 10.1080/14756366.2017.1333987
- By:
- Publication type:
- Article
Comparison of the Sulfonamide Inhibition Profiles of the α-Carbonic Anhydrase Isoforms (SpiCA1, SpiCA2 and SpiCA3) Encoded by the Genome of the Scleractinian Coral Stylophora pistillata.
- Published in:
- Marine Drugs, 2019, v. 17, n. 3, p. 146, doi. 10.3390/md17030146
- By:
- Publication type:
- Article
Structural and biochemical characterization of novel carbonic anhydrases from Phaeodactylum tricornutum.
- Published in:
- Acta Crystallographica: Section D, Structural Biology, 2020, v. 76, n. 7, p. 676, doi. 10.1107/S2059798320007202
- By:
- Publication type:
- Article
Natural Polyphenols Selectively Inhibit β‐Carbonic Anhydrase from the Dandruff‐Producing Fungus <italic>Malassezia globosa</italic>: Activity and Modeling Studies.
- Published in:
- ChemMedChem, 2018, v. 13, n. 8, p. 816, doi. 10.1002/cmdc.201800015
- By:
- Publication type:
- Article
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains.
- Published in:
- International Journal of Molecular Sciences, 2024, v. 25, n. 5, p. 2584, doi. 10.3390/ijms25052584
- By:
- Publication type:
- Article
The Effect of Substituted Benzene-Sulfonamides and Clinically Licensed Drugs on the Catalytic Activity of CynT2, a Carbonic Anhydrase Crucial for Escherichia coli Life Cycle.
- Published in:
- International Journal of Molecular Sciences, 2020, v. 21, n. 11, p. 4175, doi. 10.3390/ijms21114175
- By:
- Publication type:
- Article
Novel Diamide-Based Benzenesulfonamides as Selective Carbonic Anhydrase IX Inhibitors Endowed with Antitumor Activity: Synthesis, Biological Evaluation and In Silico Insights.
- Published in:
- International Journal of Molecular Sciences, 2019, v. 20, n. 10, p. 2484, doi. 10.3390/ijms20102484
- By:
- Publication type:
- Article
Indole-Based Hydrazones Containing A Sulfonamide Moiety as Selective Inhibitors of Tumor-Associated Human Carbonic Anhydrase Isoforms IX and XII.
- Published in:
- International Journal of Molecular Sciences, 2019, v. 20, n. 9, p. 2354, doi. 10.3390/ijms20092354
- By:
- Publication type:
- Article
Novel 8-Substituted Coumarins That Selectively Inhibit Human Carbonic Anhydrase IX and XII.
- Published in:
- International Journal of Molecular Sciences, 2019, v. 20, n. 5, p. 1208, doi. 10.3390/ijms20051208
- By:
- Publication type:
- Article
Sulfonamide Inhibition Studies of a New β-Carbonic Anhydrase from the Pathogenic Protozoan Entamoeba histolytica.
- Published in:
- International Journal of Molecular Sciences, 2018, v. 19, n. 12, p. 3946, doi. 10.3390/ijms19123946
- By:
- Publication type:
- Article
Comparison of the Anion Inhibition Profiles of the α-CA Isoforms (SpiCA1, SpiCA2 and SpiCA3) from the Scleractinian Coral Stylophora pistillata.
- Published in:
- International Journal of Molecular Sciences, 2018, v. 19, n. 7, p. 2128, doi. 10.3390/ijms19072128
- By:
- Publication type:
- Article
Carbonic Anhydrase Inhibition Activities of Schiff's Bases Based on Quinazoline-Linked Benzenesulfonamide.
- Published in:
- Molecules, 2022, v. 27, n. 22, p. 7703, doi. 10.3390/molecules27227703
- By:
- Publication type:
- Article
Hypoxia-Activated Prodrug Derivatives of Carbonic Anhydrase Inhibitors in Benzenesulfonamide Series: Synthesis and Biological Evaluation.
- Published in:
- Molecules, 2020, v. 25, n. 10, p. 2347, doi. 10.3390/molecules25102347
- By:
- Publication type:
- Article
Dual P-Glycoprotein and CA XII Inhibitors: A New Strategy to Reverse the P-gp Mediated Multidrug Resistance (MDR) in Cancer Cells †.
- Published in:
- Molecules, 2020, v. 25, n. 7, p. 1748, doi. 10.3390/molecules25071748
- By:
- Publication type:
- Article
Extending the Inhibition Profiles of Coumarin-Based Compounds Against Human Carbonic Anhydrases: Synthesis, Biological, and In Silico Evaluation.
- Published in:
- Molecules, 2019, v. 24, n. 19, p. 3580, doi. 10.3390/molecules24193580
- By:
- Publication type:
- Article
Cloning, Characterization and Anion Inhibition Studies of a β-Carbonic Anhydrase from the Pathogenic Protozoan Entamoeba histolytica.
- Published in:
- Molecules, 2018, v. 23, n. 12, p. 3112, doi. 10.3390/molecules23123112
- By:
- Publication type:
- Article
Novel 6- and 7-Substituted Coumarins with Inhibitory Action against Lipoxygenase and Tumor-Associated Carbonic Anhydrase IX.
- Published in:
- Molecules, 2018, v. 23, n. 1, p. 153, doi. 10.3390/molecules23010153
- By:
- Publication type:
- Article
Novel Sulfamide-Containing Compounds as Selective Carbonic Anhydrase I Inhibitors.
- Published in:
- Molecules, 2017, v. 22, n. 7, p. 1049, doi. 10.3390/molecules22071049
- By:
- Publication type:
- Article
Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.
- Published in:
- Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527
- By:
- Publication type:
- Article
The production and biochemical characterization of α-carbonic anhydrase from Lactobacillus rhamnosus GG.
- Published in:
- Applied Microbiology & Biotechnology, 2022, v. 106, n. 11, p. 4065, doi. 10.1007/s00253-022-11990-3
- By:
- Publication type:
- Article
Activation Studies of the β-Carbonic Anhydrase from the Pathogenic Protozoan Entamoeba histolytica with Amino Acids and Amines.
- Published in:
- Metabolites (2218-1989), 2019, v. 9, n. 2, p. 26, doi. 10.3390/metabo9020026
- By:
- Publication type:
- Article