Works matching DE "PROSTAGLANDIN antagonists"
Results: 64
Optimization of structures, biochemical properties of ketorolac and its degradation products based on computational studies.
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- DARU: Journal of Pharmaceutical Sciences, 2019, v. 27, p. 71, doi. 10.1007/s40199-019-00243-w
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- Publication type:
- Article
THE PROSTAGLANDIN TRANSPORTER: EICOSANOID REUPTAKE, CONTROL OF SIGNALING, AND DEVELOPMENT OF HIGH-AFFINITY INHIBITORS AS DRUG CANDIDATES.
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- Transactions of the American Clinical & Climatological Association, 2015, v. 126, p. 248
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- Publication type:
- Article
Unexamined Endocrine Disruption?
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- Environmental Health Perspectives, 2016, v. 124, n. 4, p. A76, doi. 10.1289/ehp.124-A76
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- Publication type:
- Article
Increased renal sodium absorption by inhibition of prostaglandin synthesis during fasting in healthy man. A possible role of the epithelialsodium channels.
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- BMC Nephrology, 2010, v. 11, p. 28, doi. 10.1186/1471-2369-11-28
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- Publication type:
- Article
Prostaglandins in pathogenesis and treatment of multiple sclerosis.
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- Immunopharmacology & Immunotoxicology, 2010, v. 32, n. 4, p. 543, doi. 10.3109/08923971003667627
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- Publication type:
- Article
A Novel Multi-step Virtual Screening for the Identification of Human and Mouse mPGES-1 Inhibitors.
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- Molecular Informatics, 2016, v. 35, n. 8/9, p. 358, doi. 10.1002/minf.201600024
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- Publication type:
- Article
Piceatannol Inhibits Phorbol Ester-Induced NF-κ B Activation and COX-2 Expression in Cultured Human Mammary Epithelial Cells.
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- Nutrition & Cancer, 2009, v. 61, n. 6, p. 855, doi. 10.1080/01635580903285080
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- Publication type:
- Article
Ionomycin induces prostaglandin E<sub>2</sub> formation in murine osteoblastic MC3T3-E1 cells via mechanisms independent of its ionophoric nature.
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- Biochemistry & Cell Biology, 2016, v. 94, n. 3, p. 236, doi. 10.1139/bcb-2015-0148
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- Publication type:
- Article
Aspirin-exacerbated Respiratory Disease: A Syndrome of Mast Cell-mediated PgD2 Overproduction.
- Published in:
- 2019
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- Publication type:
- journal article
Stress and Poor Cancer Outcomes: It's More Than Psychological.
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- 2012
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- Publication type:
- Opinion
The effect of nitric oxide synthase inhibition with and without inhibition of prostaglandins on blood flow in different human skeletal muscles.
- Published in:
- 2017
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- Publication type:
- journal article
Blood-aqueous barrier in prostaglandin EP2 receptor knockout mice.
- Published in:
- 2002
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- Publication type:
- journal article
Targeting the PGD/CRTH2/DP1 Signaling Pathway in Asthma and Allergic Disease: Current Status and Future Perspectives.
- Published in:
- Drugs, 2017, v. 77, n. 12, p. 1281, doi. 10.1007/s40265-017-0777-2
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- Publication type:
- Article
Cortical hyperostosis as a side-effect of prolonged use of prostaglandins.
- Published in:
- 2016
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- Publication type:
- journal article
CYP2C9 Involvement in ACT-453859 Metabolism.
- Published in:
- 2015
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- Publication type:
- Letter to the Editor
First-in-Man Study of ACT-453859, a Potent CRTH2 Antagonist--Is the Metabolite Formation Influenced by a Polymorphic Enzyme?
- Published in:
- 2015
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- Publication type:
- Letter to the Editor
A novel CRTH2 antagonist: Single- and multiple-dose tolerability, pharmacokinetics, and pharmacodynamics of ACT-453859 in healthy subjects.
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- Journal of Clinical Pharmacology, 2015, v. 55, n. 7, p. 787, doi. 10.1002/jcph.478
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- Publication type:
- Article
Pharmacodynamics, Pharmacokinetics, and Safety of AM211: A Novel and Potent Antagonist of the Prostaglandin D2 Receptor Type 2.
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- Journal of Clinical Pharmacology, 2012, v. 52, n. 10, p. 1482, doi. 10.1177/0091270011421912
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- Publication type:
- Article
Pharmacokinetics of Laropiprant, a Selective Prostaglandin D2 Receptor 1 Antagonist, in Patients With Moderate Hepatic Impairment.
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- Journal of Clinical Pharmacology, 2011, v. 51, n. 3, p. 406, doi. 10.1177/0091270010369240
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- Publication type:
- Article
Single Therapeutic and Supratherapeutic Doses of Laropiprant, a Selective Prostaglandin D 2 Receptor 1 Antagonist, Do Not Prolong the QTcF Interval in Healthy Volunteers.
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- Journal of Clinical Pharmacology, 2010, v. 50, n. 11, p. 1273, doi. 10.1177/0091270009360042
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- Publication type:
- Article
Effects of Laropiprant, a Selective Prostaglandin D<sub>2</sub> Receptor 1 Antagonist, on the Steady-State Pharmacokinetics of Digoxin in Healthy Adult Subjects.
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- Journal of Clinical Pharmacology, 2010, v. 50, n. 7, p. 823, doi. 10.1177/0091270009356571
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- Publication type:
- Article
Celecoxib Improves Host Defense through Prostaglandin Inhibition during Histoplasma capsulatum Infection.
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- Mediators of Inflammation, 2013, v. 2013, p. 1, doi. 10.1155/2013/950981
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- Publication type:
- Article
Nonsteroidal Antiinflammatory Drugs and Acute Renal Failure in Elderly Persons.
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- American Journal of Epidemiology, 2009, v. 151, n. 5, p. 488
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- Publication type:
- Article
Indomethacin inhibits PGE2, regulates inflammatory response, participates in adipogenesis regulation, and improves success rate of fat transplantation in C57/B6 mice.
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- Tropical Journal of Pharmaceutical Research, 2019, v. 18, n. 11, p. 2313, doi. 10.4314/tjpr.v18i11.12
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- Publication type:
- Article
An Algal Metabolite-Based PPAR-γ Agonist Displayed Anti-Inflammatory Effect via Inhibition of the NF-κB Pathway.
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- Marine Drugs, 2019, v. 17, n. 6, p. 321, doi. 10.3390/md17060321
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- Publication type:
- Article
Mir526b and Mir655 Promote Tumour Associated Angiogenesis and Lymphangiogenesis in Breast Cancer.
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- Cancers, 2019, v. 11, n. 7, p. 938, doi. 10.3390/cancers11070938
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- Publication type:
- Article
The role of FGF-2 and BMP-2 in regulation of gene induction, cell proliferation and mineralization.
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- Journal of Orthopaedic Surgery & Research, 2011, v. 6, n. 1, p. 8, doi. 10.1186/1749-799X-6-8
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- Publication type:
- Article
Using human recombinant UDP-glucuronosyltransferase isoforms and a relative activity factor approach to model total body clearance of laropiprant (MK-0524) in humans.
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- Xenobiotica, 2013, v. 43, n. 12, p. 1027, doi. 10.3109/00498254.2013.791761
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- Publication type:
- Article
Prostaglandin E2 and programmed cell death 1 signaling coordinately impair CTL function and survival during chronic viral infection.
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- Nature Medicine, 2015, v. 21, n. 4, p. 327, doi. 10.1038/nm.3831
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- Publication type:
- Article
Synthesis and Intracellular Redox Cycling of Natural Quinones and Their Analogues and Identification of Indoleamine-2,3-dioxygenase (IDO) as Potential Target for Anticancer Activity.
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- Angewandte Chemie, 2015, v. 127, n. 30, p. 8864, doi. 10.1002/ange.201503323
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- Publication type:
- Article
Nonsteroidal Anti-Inflammatory Drugs Alter the Human Mesothelial Pleural Permeability via Ion Cellular Transportation by Inhibiting Prostaglandin Synthesis.
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- Respiration, 2012, v. 84, n. 1, p. 62, doi. 10.1159/000336837
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- Publication type:
- Article
Effect of the Thromboxane Prostaglandin Receptor Antagonist Terutroban on Arterial Thrombogenesis after Repeated Administration in Patients Treated for the Prevention of Ischemic Stroke.
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- Cerebrovascular Diseases, 2009, v. 28, n. 5, p. 505, doi. 10.1159/000236915
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- Publication type:
- Article
Indomethacin-induced inhibition of prostaglandin with hyperkalemia.
- Published in:
- 1979
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- Publication type:
- Case Study
Indomethacin-induced prostaglandin inhibition with hyperkalemia. A reversible cause of hyporeninemic hypoaldosteronism.
- Published in:
- 1979
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- Publication type:
- journal article
A DISCUSSION ON CHEMOPREVENTION OF ORAL CANCER BY SELECTIVE CYCLOOXYGENASE-2 (COX-2) INHIBITORS.
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- Digest Journal of Nanomaterials & Biostructures (DJNB), 2010, v. 5, n. 2, p. 285
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- Publication type:
- Article
Age-related increases in PGD(2) expression impair respiratory DC migration, resulting in diminished T cell responses upon respiratory virus infection in mice.
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- 2011
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- Publication type:
- journal article
Increase in meningeal blood flow by nitric oxide--interaction with calcitonin gene-related peptide receptor and prostaglandin synthesis inhibition.
- Published in:
- 2002
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- Publication type:
- journal article
Indomethacin increases the effect of isosorbide dinitrate on cerebral hemodynamic in migraine patients: pathogenetic and therapeutic implications.
- Published in:
- 1998
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- Publication type:
- journal article
PPARγ as an E3 Ubiquitin-Ligase Impedes Phosphate-Stat6 Stability and Promotes Prostaglandins E<sub>2</sub>-Mediated Inhibition of IgE Production in Asthma.
- Published in:
- Frontiers in Immunology, 2020, v. 11, p. 1, doi. 10.3389/fimmu.2020.01224
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- Publication type:
- Article
Non-steroidal anti-inflammatory treatment in cancer cachexia: A systematic literature review.
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- Acta Oncologica. Supplement, 2013, v. 52, n. 1, p. 6, doi. 10.3109/0284186X.2012.724536
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- Publication type:
- Article
Cancer, cachexia, prostanoids, and NSAIDs.
- Published in:
- 2013
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- Publication type:
- Editorial
Inhibition of Lipopolysaccharide-Induced iNOS, COX- 2, and TNF-α Expression by Aqueous Extract of Orixa Japonica in RAW 264.7 Cells via Suppression of NF-κB Activity.
- Published in:
- Tropical Journal of Pharmaceutical Research, 2011, v. 10, n. 2, p. 161
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- Publication type:
- Article
Do aspirin and acetaminophen affect total menstrual loss?
- Published in:
- 1984
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- Publication type:
- journal article
Fevipiprant, a DP<sub>2</sub> receptor antagonist, inhibits eosinophil migration towards mast cells.
- Published in:
- Clinical & Experimental Allergy, 2019, v. 49, n. 2, p. 255, doi. 10.1111/cea.13304
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- Publication type:
- Article
Intra-Pancreatic Insulin Nourishes Cancer Cells: Do Insulin-Receptor Antagonists such as PGG and EGCG Play a Role?
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- American Journal of Chinese Medicine, 2020, v. 48, n. 4, p. 1005, doi. 10.1142/S0192415X20500482
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- Publication type:
- Article
Global Transcriptomic Analysis of the Canine corpus luteum (CL) During the First Half of Diestrus and Changes Induced by in vivo Inhibition of Prostaglandin Synthase 2 (PTGS2/COX2).
- Published in:
- Frontiers in Endocrinology, 2019, p. 1, doi. 10.3389/fendo.2019.00715
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- Publication type:
- Article
Inhibition of EP4 Signaling Attenuates Aortic Aneurysm Formation.
- Published in:
- PLoS ONE, 2012, v. 7, n. 5, p. 1, doi. 10.1371/journal.pone.0036724
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- Publication type:
- Article
Chronic effects of nitric oxide and prostaglandin inhibition on pressure diuresis and natriuresis in rats.
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- Kidney International Supplement, 1996, n. 55, p. S-141
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- Publication type:
- Article
Repeated application of glucocorticoids exacerbate pruritus via inhibition of prostaglandin D<sub>2</sub> production of mast cells in a murine model of allergic contact dermatitis.
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- Journal of Toxicological Sciences, 2012, v. 37, n. 6, p. 1127, doi. 10.2131/jts.37.1127
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- Publication type:
- Article
Inhibition of secretory phospholipase A2 IIa attenuates prostaglandin E2-induced invasiveness in lung adenocarcinoma.
- Published in:
- Molecular & Cellular Biochemistry, 2019, v. 456, n. 1/2, p. 145, doi. 10.1007/s11010-019-03500-3
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- Publication type:
- Article