Works matching DE "RIMONABANT"

Results: 112

One‐Pot Double Oxidation Synthesis of N‐1‐Piperidonyl Amides From N‐1‐Piperidinyl Amides with meta‐Chloroperbenzoic Acid: Rimonabant Analogue as Model Study.

Published in:

Chemistry - A European Journal, 2023, v. 29, n. 45, p. 1, doi. 10.1002/chem.202300702

By:

Chen, Yu‐Chieh;
Zeng, Wei‐Zheng;
Li, Sin‐Min;
Chou, Jia‐Yu;
Tsai, Shuo‐En;
Fuh Wong, Fung

Publication type:

Article

Rimonabant effects on anxiety induced by simulated public speaking in healthy humans: a preliminary report.

Published in:

Human Psychopharmacology: Clinical & Experimental, 2014, v. 29, n. 1, p. 94, doi. 10.1002/hup.2374

By:

Bergamaschi, Mateus M.;
Queiroz, Regina H. C.;
Chagas, Marcos H. N.;
Linares, Ila M. P.;
Arrais, Kátia C.;
Oliveira, Danielle C. G.;
Queiroz, Maria E.;
Nardi, Antonio E.;
Huestis, Marilyn A.;
Hallak, Jaime E. C.;
Zuardi, Antonio W.;
Moreira, Fabrício A.;
Crippa, José A. S.

Publication type:

Article

Involvement of adipokines in rimonabant-mediated insulin sensitivity in ob/obmice.

Published in:

Journal of Pharmacy & Pharmacology, 2009, v. 61, n. 11, p. 1493, doi. 10.1211/jpp/61.11.0008

By:

Jogeswar Mohapatra;
Manoranjan Sharma;
Satinder Singh;
Gaurav Pandya;
Abhijit Chatterjee;
Ramachandran Balaraman;
Pankaj R. Patel;
Mukul R. Jain

Publication type:

Article

Pyrrole‐Thiazolidin‐4‐one Analogues Exhibit Promising Anti‐Tuberculosis Activity.

Published in:

Asian Journal of Organic Chemistry, 2024, v. 13, n. 6, p. 1, doi. 10.1002/ajoc.202400054

By:

Ahmed, Shujauddin;
Mital, Alka;
Akhir, Abdul;
Saxena, Deepanshi;
Jahan, Kousar;
Dubey, Gurudutt;
Bharatam, P. V.;
Dasgupta, Arunava;
Chopra, Sidharth;
Jain, Rahul

Publication type:

Article

Interfering with reconsolidation by rimonabant results in blockade of heroin-associated memory.

Published in:

Frontiers in Pharmacology, 2024, p. 01, doi. 10.3389/fphar.2024.1361838

By:

Jiang Lin;
Yilin Peng;
Jinlong Zhang;
Junzhe Cheng;
Qianqian Chen;
Binbin Wang;
Yuhang Liu;
Shuliang Niu;
Jie Yan

Publication type:

Article

Rimonabant Kills Colon Cancer Stem Cells without Inducing Toxicity in Normal Colon Organoids.

Published in:

Frontiers in Pharmacology, 2018, p. 1, doi. 10.3389/fphar.2017.00949

By:

Fiore, Donatella;
Ramesh, Prashanthi;
Proto, Maria C.;
Piscopo, Chiara;
Franceschelli, Silvia;
Anzelmo, Serena;
Medema, Jan P.;
Bifulco, Maurizio;
Gazzerro, Patrizia

Publication type:

Article

Comparative effects of cannabinoid CB1 receptor agonist and antagonist on timing impulsivity induced by d-amphetamine in a differential reinforcement of low-rate response task in male rats.

Published in:

Psychopharmacology, 2022, v. 239, n. 5, p. 1459, doi. 10.1007/s00213-021-06018-z

By:

Chen, Shuo-Fu;
Hsu, Wei-Chung;
Lu, Xi-Yun;
Chuang, Chuen-Yu;
Liao, Ruey-Ming

Publication type:

Article

Cannabinoid receptor-1 signaling contributions to sign-tracking and conditioned reinforcement in rats.

Published in:

Psychopharmacology, 2018, v. 235, n. 10, p. 3031, doi. 10.1007/s00213-018-4993-6

By:

Bacharach, Sam Z.;
Nasser, Helen M.;
Zlebnik, Natalie E.;
Dantrassy, Hannah M.;
Kochli, Daniel E.;
Gyawali, Utsav;
Cheer, Joseph F.;
Calu, Donna J.

Publication type:

Article

Δ9 -Tetrahydrocannabinol-like discriminative stimulus effects of five novel synthetic cannabinoids in rats.

Published in:

Psychopharmacology, 2018, v. 235, n. 3, p. 673, doi. 10.1007/s00213-017-4783-6

By:

Gatch, Michael B.;
Forster, Michael J.

Publication type:

Article

Cannabinoid withdrawal in mice: inverse agonist vs neutral antagonist.

Published in:

Psychopharmacology, 2015, v. 232, n. 15, p. 2751, doi. 10.1007/s00213-015-3907-0

By:

Tai, Sherrica;
Nikas, Spyros;
Shukla, Vidyanand;
Vemuri, Kiran;
Makriyannis, Alexandros;
Järbe, Torbjörn

Publication type:

Article

Rimonabant's reductive effects on high densities of food reinforcement, but not palatability, in lean and obese Zucker rats.

Published in:

Psychopharmacology, 2014, v. 231, n. 10, p. 2159, doi. 10.1007/s00213-013-3366-4

By:

Buckley, Jessica;
Rasmussen, Erin

Publication type:

Article

Differentiation between low- and high-efficacy CB receptor agonists using a drug discrimination protocol for rats.

Published in:

Psychopharmacology, 2014, v. 231, n. 3, p. 489, doi. 10.1007/s00213-013-3257-8

By:

Järbe, Torbjörn;
LeMay, Brian;
Halikhedkar, Aneetha;
Wood, JodiAnne;
Vadivel, Subramanian;
Zvonok, Alexander;
Makriyannis, Alexandros

Publication type:

Article

Low dose naloxone attenuates the pruritic but not anorectic response to rimonabant in male rats.

Published in:

Psychopharmacology, 2013, v. 226, n. 2, p. 415, doi. 10.1007/s00213-012-2916-5

By:

Wright, F.;
Rodgers, R.

Publication type:

Article

Erratum to: Sensitization to cocaine is inhibited after intra-accumbal GR103691 or rimonabant, but it is enhanced after co-infusion indicating functional interaction between accumbens D and CB1 receptors.

Published in:

2012

By:

Ramiro-Fuentes, Susana;
Fernandez-Espejo, Emilio

Publication type:

Correction Notice

Tethered agonist activated ADGRF1 structure and signalling analysis reveal basis for G protein coupling.

Published in:

Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-38083-7

By:

Jones, Daniel T. D.;
Dates, Andrew N.;
Rawson, Shaun D.;
Burruss, Maggie M.;
Lipper, Colin H.;
Blacklow, Stephen C.

Publication type:

Article

CORRECTION.

Published in:: 2006
Publication type:: Correction Notice

The effects of weight loss using dietary manipulation and rimonabant therapy on arterial stiffness in type 2 diabetes

Published in:

Artery Research, 2010, v. 4, n. 2, p. 47, doi. 10.1016/j.artres.2010.04.001

By:

Chakera, A.;
Bunce, S.;
Heppenstall, C.;
Smith, J.C.

Publication type:

Article

RP-HPLC Method Development and its Validation for Quantitative Determination of Rimonabant in Human Plasma.

Published in:

Eurasian Journal of Analytical Chemistry, 2012, v. 7, n. 3, p. 115

By:

Bankey, Shravan K.;
Jain, Surendra K.;
Basniwal, Pawan K.;
Jain, Deepti

Publication type:

Article

CB1 receptor antagonist rimonabant protects against chronic intermittent hypoxia-induced renal injury in rats.

Published in:

2021

By:

Zhao, Li;
Liu, Tao;
Dou, Zhan-jun;
Wang, Mei-ting;
Hu, Zi-xuan;
Wang, Bei

Publication type:

journal article

CB1 Receptor-Dependent and Independent Induction of Lipolysis in Primary Rat Adipocytes by the Inverse Agonist Rimonabant (SR141716A).

Published in:

Molecules, 2020, v. 25, n. 4, p. 896, doi. 10.3390/molecules25040896

By:

Müller, Günter A.;
Herling, Andreas W.;
Wied, Susanne;
Müller, Timo D.

Publication type:

Article

Uso terapêutico dos canabinoides em psiquiatria.

Published in:

Brazilian Journal of Psychiatry / Revista Brasileira de Psiquiatria, 2010, v. 32, p. S56

By:

Crippa, José Alexandre S.;
Zuardi, Antonio Waldo;
Hallak, Jaime E. C.

Publication type:

Article

Rimonabant Precipitates Anxiety in Rats Withdrawn from Palatable Food: Role of the Central Amygdala.

Published in:

Neuropsychopharmacology, 2013, v. 38, n. 12, p. 2498, doi. 10.1038/npp.2013.153

By:

Blasio, Angelo;
Iemolo, Attilio;
Sabino, Valentina;
Petrosino, Stefania;
Steardo, Luca;
Rice, Kenner C;
Orlando, Pierangelo;
Iannotti, Fabio Arturo;
Di Marzo, Vincenzo;
Zorrilla, Eric P;
Cottone, Pietro

Publication type:

Article

Genetic Deletion of Fatty Acid Amide Hydrolase Alters Emotional Behavior and Serotonergic Transmission in the Dorsal Raphe, Prefrontal Cortex, and Hippocampus.

Published in:

Neuropsychopharmacology, 2010, v. 35, n. 10, p. 2083, doi. 10.1038/npp.2010.80

By:

Bambico, Francis Rodriguez;
Cassano, Tommaso;
Dominguez-Lopez, Sergio;
Katz, Noam;
Walker, Claire Dominique;
Piomelli, Daniele;
Gobbi, Gabriella

Publication type:

Article

A Common Polymorphism in the Cannabinoid Receptor 1 (CNR1) Gene is Associated with Antipsychotic-Induced Weight Gain in Schizophrenia.

Published in:

Neuropsychopharmacology, 2010, v. 35, n. 6, p. 1315, doi. 10.1038/npp.2009.235

By:

Tiwari, Arun K.;
Zai, Clement C.;
Likhodi, Olga;
Lisker, Annika;
Singh, Deepika;
Souza, Renan P.;
Batra, Poonam;
Zaidi, Syed H. E.;
Sheng Chen;
Fang Liu;
Puls, Imke;
Meltzer, Herbert Y.;
Lieberman, Jeffrey A.;
Kennedy, James L.;
Müller, Daniel J

Publication type:

Article

The Cannabinoid CB1 Antagonist TM38837 With Limited Penetrance to the Brain Shows Reduced Fear-Promoting Effects in Mice.

Published in:

Frontiers in Pharmacology, 2019, p. N.PAG, doi. 10.3389/fphar.2019.00207

By:

Micale, Vincenzo;
Drago, Filippo;
Noerregaard, Pia K.;
Elling, Christian E.;
Wotjak, Carsten T.

Publication type:

Article

Cannabinoid CB1 receptor mediates glucocorticoid effects on hormone secretion induced by volume and osmotic changes.

Published in:

Clinical & Experimental Pharmacology & Physiology, 2012, v. 39, n. 2, p. 151, doi. 10.1111/j.1440-1681.2011.05658.x

By:

Ruginsk, SG;
Uchoa, ET;
Elias, LLK;
Antunes-Rodrigues, J

Publication type:

Article

Gastrointestinal Adverse Events of Cannabinoid 1 Receptor Inverse Agonists suggest their Potential Use in Irritable Bowel Syndrome with Constipation: A Systematic Review and Meta-Analysis.

Published in:

Journal of Gastrointestinal & Liver Diseases, 2019, v. 28, n. 4, p. 473, doi. 10.15403/jgld-265

By:

Fabisiak, Adam;
Włodarczyk, Marcin;
Fabisiak, Natalia;
Storr, Martin;
Fichna, Jakub

Publication type:

Article

Cannabinoid receptor 1 antagonist treatment induces glucagon release and shows an additive therapeutic effect with GLP-1 agonist in diet-induced obese mice.

Published in:

Canadian Journal of Physiology & Pharmacology, 2014, v. 92, n. 12, p. 975, doi. 10.1139/cjpp-2014-0310

By:

Patel, Kartikkumar Navinchandra;
Joharapurkar, Amit Arvind;
Patel, Vishal;
Kshirsagar, Samadhan Govind;
Bahekar, Rajesh;
Srivastava, Brijesh Kumar;
Jain, Mukul R.

Publication type:

Article

Compensatory Activation of Cannabinoid CB2 Receptor Inhibition of GABA Release in the Rostral Ventromedial Medulla in Inflammatory Pain.

Published in:

Journal of Neuroscience, 2017, v. 37, n. 3, p. 626, doi. 10.1523/JNEUROSCI.1310-16.2017

By:

Ming-Hua Li;
Suchland, Katherine L.;
Ingram, Susan L.

Publication type:

Article

Computational investigation on the binding modes of Rimonabant analogs with CB1 and CB2.

Published in:

Chemical Biology & Drug Design, 2018, v. 92, n. 3, p. 1699, doi. 10.1111/cbdd.13337

By:

Liu, Cheng;
Yuan, Congmin;
Wu, Pinwen;
Zhu, Chen;
Fang, Hao;
Wang, Lili;
Fu, Wei

Publication type:

Article

Hypertension and Diabetes: Should We Treat Early Surrogates?

Published in:

Diabetes Care, 2009, v. 32, p. S290, doi. 10.2337/dc09-S329

By:

Nilsson, Peter M.

Publication type:

Article

Rimonabant inhibits TNF-α-induced endothelial IL-6 secretion via CB1 receptor and cAMP-dependent protein kinase pathway.

Published in:

Acta Pharmacologica Sinica, 2010, v. 31, n. 11, p. 1447, doi. 10.1038/aps.2010.126

By:

Nan-lan HUANG;
Jyh-ming JUANG;
Yi-ho WANG;
Chia-hsiang HSUEH;
Yao-jen LIANG;
Jiunn-lee LIN;
Chia-ti TSAI;
Ling-ping LAI

Publication type:

Article

Targeting the Endocannabinoid/CB1 Receptor System For Treating Major Depression Through Antidepressant Activities of Curcumin and Dexanabinol-Loaded Solid Lipid Nanoparticles.

Published in:

Cellular Physiology & Biochemistry (Karger AG), 2017, v. 42, n. 6, p. 2281, doi. 10.1159/000480001

By:

He, Xiaolie;
Yang, Li;
Wang, Mei;
Zhuang, Xizhen;
Huang, Ruiqi;
Zhu, Rongrong;
Wang, Shilong

Publication type:

Article

The CB1 Neutral Antagonist AM4113 Retains the Therapeutic Efficacy of the Inverse Agonist Rimonabant for Nicotine Dependence and Weight Loss with Better Psychiatric Tolerability.

Published in:

International Journal of Neuropsychopharmacology, 2016, v. 19, n. 12, p. 1, doi. 10.1093/ijnp/pyw068

By:

Gueye, Aliou B.;
Pryslawsky, Yaroslaw;
Trigo, Jose M.;
Poulia, Nafsika;
Delis, Foteini;
Antoniou, Katerina;
Loureiro, Michael;
Laviolette, Steve R.;
Vemuri, Kiran;
Makriyannis, Alexandros;
Le Foll, Bernard

Publication type:

Article

The CB1 Neutral Antagonist Tetrahydrocannabivarin Reduces Default Mode Network and Increases Executive Control Network Resting State Functional Connectivity in Healthy Volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2016, v. 19, n. 2, p. 1, doi. 10.1093/ijnp/pyv092

By:

Rzepa, Ewelina;
Tudge, Luke;
McCabe, Ciara

Publication type:

Article

Neural Effects of Cannabinoid CB1 Neutral Antagonist Tetrahydrocannabivarin on Food Reward and Aversion in Healthy Volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2015, v. 18, n. 6, p. 1, doi. 10.1093/ijnp/pyu094

By:

Tudge, Luke;
Williams, Clare;
Cowen, Philip J.;
McCabe, Ciara

Publication type:

Article

Reduced neural response to reward following 7 days treatment with the cannabinoid CB1 antagonist rimonabant in healthy volunteers.

Published in:

International Journal of Neuropsychopharmacology, 2010, v. 13, n. 8, p. 1103, doi. 10.1017/S1461145710000453

By:

Horder, Jamie;
Harmer, Catherine J.;
Cowen, Philip J.;
McCabe, Ciara

Publication type:

Article

Synthesis and Anticancer Activity of 1,2,3-Triazole Fused N-Arylpyrazole Derivatives.

Published in:

Russian Journal of General Chemistry, 2019, v. 89, n. 4, p. 831, doi. 10.1134/S1070363219040315

By:

Lakkakula, R.;
Roy, A.;
Mukkanti, K.;
Sridhar, G.

Publication type:

Article

Context-dependent effects of the CB1 receptor antagonist rimonabant on morphine-induced behavioral sensitization in female mice.

Published in:

Frontiers in Pharmacology, 2023, v. 14, p. 1, doi. 10.3389/fphar.2023.1100527

By:

Marinho, Eduardo A. V.;
Justo Oliveira-Lima, Alexandre;
Reis, Henrique S.;
Santos-Baldaia, Renan;
Wuo-Silva, Raphael;
Hollais, Andre W.;
Yokoyama, Thais S.;
Frussa-Filho, Roberto;
Berro, Lais F.

Publication type:

Article

Endocannabinoids regulate adipokine production and the immune balance of omental adipose tissue in human obesity.

Published in:

International Journal of Obesity, 2013, v. 37, n. 6, p. 874, doi. 10.1038/ijo.2012.123

By:

Ge, Q;
Maury, E;
Rycken, L;
Gérard, J;
Noël, L;
Detry, R;
Navez, B;
Brichard, S M

Publication type:

Article

CB1 blockade-induced weight loss over 48 weeks decreases liver fat in proportion to weight loss in humans.

Published in:

International Journal of Obesity, 2013, v. 37, n. 5, p. 699, doi. 10.1038/ijo.2012.116

By:

Bergholm, R;
Sevastianova, K;
Santos, A;
Kotronen, A;
Urjansson, M;
Hakkarainen, A;
Lundbom, J;
Tiikkainen, M;
Rissanen, A;
Lundbom, N;
Yki-Järvinen, H

Publication type:

Article

Anti-obesity effects of the combined administration of CB1 receptor antagonist rimonabant and melanin-concentrating hormone antagonist SNAP-94847 in diet-induced obese mice.

Published in:

International Journal of Obesity, 2013, v. 37, n. 2, p. 279, doi. 10.1038/ijo.2012.35

By:

Verty, A N A;
Lockie, S H;
Stefanidis, A;
Oldfield, B J

Publication type:

Article

Oral Communication 12, Tuesday Sept. 25th 5.00 pm–6.00 pm; Room: Lecture Hall 3.

Published in:: Alcohol & Alcoholism. Supplement, 2007, v. 42, p. i46, doi. 10.1093/alcalc/agm124
Publication type:: Article

Symposium 17 Monday Sept. 24th 6.30 pm–8.00 pm; Room: Lecture Hall 1.

Published in:: 2007
Publication type:: Proceeding

A systematic review of the effectiveness of smoking relapse prevention interventions for abstinent smokers.

Published in:

Addiction, 2010, v. 105, n. 8, p. 1362, doi. 10.1111/j.1360-0443.2010.02996.x

By:

Agboola, Shade;
McNeill, Ann;
Coleman, Tim;
Leonardi Bee, Jo

Publication type:

Article

CB1 receptor blockade ameliorates hepatic fat infiltration and inflammation and increases Nrf2-AMPK pathway in a rat model of severely uncontrolled diabetes.

Published in:

PLoS ONE, 2018, v. 13, n. 10, p. 1, doi. 10.1371/journal.pone.0206152

By:

Chang, Eugene;
Kim, Dae-Hee;
Yang, Hyekyung;
Lee, Da Hyun;
Bae, Soo Han;
Park, Cheol-Young

Publication type:

Article

Nonopioid placebo analgesia is mediated by CB1 cannabinoid receptors.

Published in:

Nature Medicine, 2011, v. 17, n. 10, p. 1228, doi. 10.1038/nm.2435

By:

Benedetti, Fabrizio;
Amanzio, Martina;
Rosato, Rosalba;
Blanchard, Catherine

Publication type:

Article

Efficacy and Safety of Ezetimibe Plus Orlistat or Rimonabant in Statin-Intolerant Nondiabetic Overweight/Obese Patients With Dyslipidemia.

Published in:

Journal of Cardiovascular Pharmacology & Therapeutics, 2009, v. 14, n. 4, p. 274, doi. 10.1177/1074248409343935

By:

Florentin, Matilda;
Kostapanos, Michael S.;
Nakou, Eleni S.;
Elisaf, Moses;
Liberopoulos, Evangelos N.

Publication type:

Article

Pleiotropic effects of Rimonabant and Simvastatin on obesity associated multiple metabolic risk factors in rats.

Published in:

European Review for Medical & Pharmacological Sciences, 2012, v. 16, n. 6, p. 797

By:

SALEM, N.A.;
ASSAF, N.;
AHMED, H.H.

Publication type:

Article

Seventeen years since rimonabant's downfall: reassessing its suicidality risk profile.

Published in:

Obesity (19307381), 2024, v. 32, n. 7, p. 1235, doi. 10.1002/oby.24019

By:

Cohen, Yuval;
Kolodziej, Andrew;
Morningstar, Marshall

Publication type:

Article