Works matching IS 00071188 AND DT 2012 AND VI 165 AND IP 6

Results: 40

Mandarin Translations.
Published in:
2012
Publication type:
journal article
Modulation of mouse gastrointestinal motility by allyl isothiocyanate, a constituent of cruciferous vegetables (Brassicaceae): evidence for TRPA1-independent effects.
Published in:
2012
By:
- Capasso R;
- Aviello G;
- Romano B;
- Borrelli F;
- De Petrocellis L;
- Di Marzo V;
- Izzo AA;
- Capasso, Raffaele;
- Aviello, Gabriella;
- Romano, Barbara;
- Borrelli, Francesca;
- De Petrocellis, Luciano;
- Di Marzo, Vincenzo;
- Izzo, Angelo A
Publication type:
journal article
TNF-α-induces airway hyperresponsiveness to cholinergic stimulation in guinea pig airways.
Published in:
2012
By:
- Makwana R;
- Gozzard N;
- Spina D;
- Page C;
- Makwana, R;
- Gozzard, N;
- Spina, D;
- Page, C
Publication type:
journal article
Role of 5-HT(1) receptor subtypes in the modulation of pain and synaptic transmission in rat spinal superficial dorsal horn.
Published in:
2012
By:
- Jeong HJ;
- Mitchell VA;
- Vaughan CW;
- Jeong, Hyo-Jin;
- Mitchell, Vanessa A;
- Vaughan, Christopher W
Publication type:
journal article
Different in vitro and in vivo profiles of substituted 3-aminopropylphosphinate and 3-aminopropyl(methyl)phosphinate GABA(B) receptor agonists as inhibitors of transient lower oesophageal sphincter relaxation.
Published in:
2012
By:
- Lehmann A;
- Antonsson M;
- Aurell-Holmberg A;
- Blackshaw LA;
- Brändén L;
- Elebring T;
- Jensen J;
- Kärrberg L;
- Mattsson JP;
- Nilsson K;
- Oja SS;
- Saransaari P;
- von Unge S;
- Lehmann, A;
- Antonsson, M;
- Aurell-Holmberg, A;
- Blackshaw, L A;
- Brändén, L;
- Elebring, T;
- Jensen, J
Publication type:
journal article
Potent anti-inflammatory effect of a novel furan-2,5-dione derivative, BPD, mediated by dual suppression of COX-2 activity and LPS-induced inflammatory gene expression via NF-κB inactivation.
Published in:
2012
By:
- Shin JS;
- Park SJ;
- Ryu S;
- Kang HB;
- Kim TW;
- Choi JH;
- Lee JY;
- Cho YW;
- Lee KT;
- Shin, Ji-Sun;
- Park, Seung-Jae;
- Ryu, Suran;
- Kang, Han Byul;
- Kim, Tae Woo;
- Choi, Jung-Hye;
- Lee, Jae-Yeol;
- Cho, Young-Wuk;
- Lee, Kyung-Tae
Publication type:
journal article
Roflumilast inhibits the release of chemokines and TNF-α from human lung macrophages stimulated with lipopolysaccharide.
Published in:
2012
By:
- Buenestado A;
- Grassin-Delyle S;
- Guitard F;
- Naline E;
- Faisy C;
- Israël-Biet D;
- Sage E;
- Bellamy JF;
- Tenor H;
- Devillier P;
- Buenestado, A;
- Grassin-Delyle, S;
- Guitard, F;
- Naline, E;
- Faisy, C;
- Israël-Biet, D;
- Sage, E;
- Bellamy, J F;
- Tenor, H;
- Devillier, P
Publication type:
journal article
A novel fluorescent histamine H(1) receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands.
Published in:
2012
By:
- Rose RH;
- Briddon SJ;
- Hill SJ;
- Rose, Rachel H;
- Briddon, Stephen J;
- Hill, Stephen J
Publication type:
journal article
The orexin receptor OX(1)R in colon cancer: a promising therapeutic target and a new paradigm in G protein-coupled receptor signalling through ITIMs.
Published in:
2012
By:
- Laburthe M;
- Voisin T;
- Laburthe, Marc;
- Voisin, Thierry
Publication type:
journal article
Hydrogen sulphide-releasing diclofenac derivatives inhibit breast cancer-induced osteoclastogenesis in vitro and prevent osteolysis ex vivo.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1914, doi. 10.1111/j.1476-5381.2011.01704.x
By:
- Frantzias, J;
- Logan, JG;
- Mollat, P;
- Sparatore, A;
- Del Soldato, P;
- Ralston, SH;
- Idris, AI
Publication type:
Article
Potent anti-inflammatory effect of a novel furan-2,5-dione derivative, BPD, mediated by dual suppression of COX-2 activity and LPS-induced inflammatory gene expression via NF-κB inactivation.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1926, doi. 10.1111/j.1476-5381.2011.01670.x
By:
- Shin, Ji-Sun;
- Park, Seung-Jae;
- Ryu, Suran;
- Kang, Han Byul;
- Kim, Tae Woo;
- Choi, Jung-Hye;
- Lee, Jae-Yeol;
- Cho, Young-Wuk;
- Lee, Kyung-Tae
Publication type:
Article
Structure-activity relationships of vanilloid receptor agonists for arteriolar TRPV1.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1801, doi. 10.1111/j.1476-5381.2011.01645.x
By:
- Czikora, Á;
- Lizanecz, E;
- Bakó, P;
- Rutkai, I;
- Ruzsnavszky, F;
- Magyar, J;
- Pórszász, R;
- Kark, T;
- Facskó, A;
- Papp, Z;
- Édes, I;
- Tóth, A
Publication type:
Article
Role of 5-HT1 receptor subtypes in the modulation of pain and synaptic transmission in rat spinal superficial dorsal horn.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1956, doi. 10.1111/j.1476-5381.2011.01685.x
By:
- Jeong, Hyo-Jin;
- Mitchell, Vanessa A;
- Vaughan, Christopher W
Publication type:
Article
Role of endothelin-1 in the hyper-responsiveness to nitrovasodilators following acute NOS inhibition.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1992, doi. 10.1111/j.1476-5381.2011.01696.x
By:
- Bourque, Stephane L;
- Whittingham, Heather A;
- Brien, Susan E;
- Davidge, Sandra T;
- Adams, Michael A
Publication type:
Article
Roflumilast inhibits the release of chemokines and TNF-α from human lung macrophages stimulated with lipopolysaccharide.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1877, doi. 10.1111/j.1476-5381.2011.01667.x
By:
- Buenestado, A;
- Grassin-Delyle, S;
- Guitard, F;
- Naline, E;
- Faisy, C;
- Israël-Biet, D;
- Sage, E;
- Bellamy, JF;
- Tenor, H;
- Devillier, P
Publication type:
Article
Polymorphisms of ADORA2A modulate psychomotor vigilance and the effects of caffeine on neurobehavioural performance and sleep EEG after sleep deprivation.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1904, doi. 10.1111/j.1476-5381.2011.01689.x
By:
- Bodenmann, S;
- Hohoff, C;
- Freitag, C;
- Deckert, J;
- Rétey, J V;
- Bachmann, V;
- Landolt, H-P
Publication type:
Article
Behind the curtain: cellular mechanisms for allosteric modulation of calcium-sensing receptors.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1670, doi. 10.1111/j.1476-5381.2011.01403.x
By:
- Cavanaugh, Alice;
- Huang, Ying;
- Breitwieser, Gerda E
Publication type:
Article
Modulation of mouse gastrointestinal motility by allyl isothiocyanate, a constituent of cruciferous vegetables ( Brassicaceae): evidence for TRPA1-independent effects.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1966, doi. 10.1111/j.1476-5381.2011.01703.x
By:
- Capasso, Raffaele;
- Aviello, Gabriella;
- Romano, Barbara;
- Borrelli, Francesca;
- De Petrocellis, Luciano;
- Di Marzo, Vincenzo;
- Izzo, Angelo A
Publication type:
Article
A novel fluorescent histamine H1 receptor antagonist demonstrates the advantage of using fluorescence correlation spectroscopy to study the binding of lipophilic ligands.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1789, doi. 10.1111/j.1476-5381.2011.01640.x
By:
- Rose, Rachel H;
- Briddon, Stephen J;
- Hill, Stephen J
Publication type:
Article
d-Amino acid oxidase-mediated increase in spinal hydrogen peroxide is mainly responsible for formalin-induced tonic pain.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1941, doi. 10.1111/j.1476-5381.2011.01680.x
By:
- Lu, Jin-Miao;
- Gong, Nian;
- Wang, Yan-Chao;
- Wang, Yong-Xiang
Publication type:
Article
Ursolic acid induces apoptosis in human leukaemia cells and exhibits anti-leukaemic activity in nude mice through the PKB pathway.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1813, doi. 10.1111/j.1476-5381.2011.01684.x
By:
- Gao, Ning;
- Cheng, Senping;
- Budhraja, Amit;
- Gao, Ziyi;
- Chen, Jieping;
- Liu, E-Hu;
- Huang, Cheng;
- Chen, Deying;
- Yang, Zailin;
- Liu, Qun;
- Li, Ping;
- Shi, Xianglin;
- Zhang, Zhuo
Publication type:
Article
Regulation of GPCR activity, trafficking and localization by GPCR-interacting proteins.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1717, doi. 10.1111/j.1476-5381.2011.01552.x
By:
- Magalhaes, Ana C;
- Dunn, Henry;
- Ferguson, Stephen SG
Publication type:
Article
A novel angiopoietin-derived peptide displays anti-angiogenic activity and inhibits tumour-induced and retinal neovascularization.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1891, doi. 10.1111/j.1476-5381.2011.01677.x
By:
- Palmer, GM;
- Tiran, Z;
- Zhou, Z;
- Capozzi, ME;
- Park, W;
- Coletta, C;
- Pyriochou, A;
- Kliger, Y;
- Levy, O;
- Borukhov, I;
- Dewhirst, MW;
- Rotman, G;
- Penn, JS;
- Papapetropoulos, A
Publication type:
Article
Mechanisms of rapid opioid receptor desensitization, resensitization and tolerance in brain neurons.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1704, doi. 10.1111/j.1476-5381.2011.01482.x
By:
- Dang, Vu C;
- Christie, MacDonald J
Publication type:
Article
Identification of drugs and drug metabolites as substrates of multidrug resistance protein 2 (MRP2) using triple-transfected MDCK-OATP1B1-UGT1A1-MRP2 cells.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1836, doi. 10.1111/j.1476-5381.2011.01672.x
By:
- Fahrmayr, C;
- König, J;
- Auge, D;
- Mieth, M;
- Fromm, MF
Publication type:
Article
Pharmacological modulation of chemokine receptor function.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1617, doi. 10.1111/j.1476-5381.2011.01551.x
By:
- Scholten, DJ;
- Canals, M;
- Maussang, D;
- Roumen, L;
- Smit, MJ;
- Wijtmans, M;
- de Graaf, C;
- Vischer, HF;
- Leurs, R
Publication type:
Article
Constitutive formation of an RXFP1-signalosome: a novel paradigm in GPCR function and regulation.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1644, doi. 10.1111/j.1476-5381.2011.01470.x
By:
- Halls, Michelle L
Publication type:
Article
Lifting the lid on GPCRs: the role of extracellular loops.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1688, doi. 10.1111/j.1476-5381.2011.01629.x
By:
- Wheatley, M;
- Wootten, D;
- Conner, MT;
- Simms, J;
- Kendrick, R;
- Logan, RT;
- Poyner, DR;
- Barwell, J
Publication type:
Article
Predicting the emetic liability of novel chemical entities: a comparative study.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1848, doi. 10.1111/j.1476-5381.2011.01669.x
By:
- du Sert, Nathalie Percie;
- Holmes, Anthony M;
- Wallis, Rob;
- Andrews, Paul LR
Publication type:
Article
GPCR expression in tissues and cells: Are the optimal receptors being used as drug targets?
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1613, doi. 10.1111/j.1476-5381.2011.01434.x
By:
- Insel, PA;
- Snead, A;
- Murray, F;
- Zhang, L;
- Yokouchi, H;
- Katakia, T;
- Kwon, O;
- Dimucci, D;
- Wilderman, A
Publication type:
Article
Comparative effects of different modes of renin angiotensin system inhibition on hypercholesterolaemia-induced atherosclerosis.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 2000, doi. 10.1111/j.1476-5381.2011.01712.x
By:
- Lu, Hong;
- Balakrishnan, Anju;
- Howatt, Deborah A;
- Wu, Congqing;
- Charnigo, Richard;
- Liau, Gene;
- Cassis, Lisa A;
- Daugherty, Alan
Publication type:
Article
Corticosteroid-induced gene expression in allergen-challenged asthmatic subjects taking inhaled budesonide.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1737, doi. 10.1111/j.1476-5381.2011.01620.x
By:
- Kelly, MM;
- King, EM;
- Rider, CF;
- Gwozd, C;
- Holden, NS;
- Eddleston, J;
- Zuraw, B;
- Leigh, R;
- O'Byrne, PM;
- Newton, R
Publication type:
Article
Inhibitory effect of bufalin and cinobufagin on steroidogenesis via the activation of ERK in human adrenocortical cells.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1868, doi. 10.1111/j.1476-5381.2011.01671.x
By:
- Kau, Mei-Mei;
- Wang, Jiing-Rong;
- Tsai, Shiow-Chwen;
- Yu, Ching-Han;
- Wang, Paulus S
Publication type:
Article
Different in vitro and in vivo profiles of substituted 3-aminopropylphosphinate and 3-aminopropyl(methyl)phosphinate GABAB receptor agonists as inhibitors of transient lower oesophageal sphincter relaxation.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1757, doi. 10.1111/j.1476-5381.2011.01682.x
By:
- Lehmann, A;
- Antonsson, M;
- Aurell-Holmberg, A;
- Blackshaw, LA;
- Brändén, L;
- Elebring, T;
- Jensen, J;
- Kärrberg, L;
- Mattsson, JP;
- Nilsson, K;
- Oja, SS;
- Saransaari, P;
- von Unge, S
Publication type:
Article
The orexin receptor OX1R in colon cancer: a promising therapeutic target and a new paradigm in G protein-coupled receptor signalling through ITIMs.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1678, doi. 10.1111/j.1476-5381.2011.01510.x
By:
- Laburthe, Marc;
- Voisin, Thierry
Publication type:
Article
Ketamine-induced ventricular structural, sympathetic and electrophysiological remodelling: pathological consequences and protective effects of metoprolol.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1748, doi. 10.1111/j.1476-5381.2011.01635.x
By:
- Li, Y;
- Shi, J;
- Yang, BF;
- Liu, L;
- Han, CL;
- Li, WM;
- Dong, DL;
- Pan, ZW;
- Liu, GZ;
- Geng, JQ;
- Sheng, L;
- Tan, XY;
- Sun, DH;
- Gong, ZH;
- Gong, YT
Publication type:
Article
Biased signalling and allosteric machines: new vistas and challenges for drug discovery.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1659, doi. 10.1111/j.1476-5381.2011.01749.x
By:
- Kenakin, Terry P
Publication type:
Article
TNF-α-induces airway hyperresponsiveness to cholinergic stimulation in guinea pig airways.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1978, doi. 10.1111/j.1476-5381.2011.01675.x
By:
- Makwana, R;
- Gozzard, N;
- Spina, D;
- Page, C
Publication type:
Article
Antiplatelet and antithrombotic effect of F 16618, a new thrombin proteinase-activated receptor-1 (PAR1) antagonist.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1827, doi. 10.1111/j.1476-5381.2011.01668.x
By:
- Dumas, M;
- Nadal-Wollbold, F;
- Gaussem, P;
- Perez, M;
- Mirault, T;
- Létienne, R;
- Bourbon, T;
- Grelac, F;
- Le Grand, B;
- Bachelot-Loza, C
Publication type:
Article
Themed section: molecular pharmacology of GPCRs.
Published in:
British Journal of Pharmacology, 2012, v. 165, n. 6, p. 1609, doi. 10.1111/j.1476-5381.2011.01679.x
By:
- Summers, RJ
Publication type:
Article