Works matching DE "THIAZOLE derivatives"

Results: 391

Catalytic Enantioselective Synthesis of Tertiary Thiols From 5 H-Thiazol-4-ones and Nitroolefins: Bifunctional Ureidopeptide-Based Brønsted Base Catalysis.

Published in:

Angewandte Chemie, 2013, v. 125, n. 45, p. 12062, doi. 10.1002/ange.201305644

By:

Diosdado, Saioa;
Etxabe, Julen;
Izquierdo, Joseba;
Landa, Aitor;
Mielgo, Antonia;
Olaizola, Iurre;
López, Rosa;
Palomo, Claudio

Publication type:

Article

2-Benzamido- N-(1 H-benzo[ d]imidazol-2-yl)thiazole-4-carboxamide derivatives as potent inhibitors of CK1δ/ε.

Published in:

Amino Acids, 2012, v. 43, n. 4, p. 1577, doi. 10.1007/s00726-012-1234-x

By:

Bischof, Joachim;
Leban, Johann;
Zaja, Mirko;
Grothey, Arnhild;
Radunsky, Barbara;
Othersen, Olaf;
Strobl, Stefan;
Vitt, Daniel;
Knippschild, Uwe

Publication type:

Article

Synthesis and antifungal activity of novel piperidinyl thiazole derivatives.

Published in:

Pest Management Science, 2025, v. 81, n. 5, p. 2566, doi. 10.1002/ps.8431

By:

Shanbhag, Gajanan;
Naik, Maruti;
Wagh, Dnyaneshwar;
Autkar, Santosh;
Hagalavadi M, Venkatesh;
Wachendorff, Ulrike;
Pabba, Jagadish;
Klausener, Alexander

Publication type:

Article

Design, synthesis, and fungicidal activities of novel piperazine thiazole derivatives containing oxime ether or oxime ester moieties.

Published in:

Pest Management Science, 2023, v. 79, n. 5, p. 1977, doi. 10.1002/ps.7374

By:

Peng, Xing‐Jie;
Tian, Xue‐Rong;
Yu, Shu‐Jing;
Zhao, Tong‐Tong;
Bian, Qiang;
Zhao, Wei‐Guang

Publication type:

Article

The AMPK Agonist PT1 and mTOR Inhibitor 3HOI-BA-01 Protect Cardiomyocytes After Ischemia Through Induction of Autophagy.

Published in:

2016

By:

Huang, Ling;
Dai, Kai;
Chen, Manhua;
Zhou, Wenping;
Wang, Xiaoling;
Chen, Jing;
Zhou, Wei

Publication type:

journal article

SWFB and GA Strategies for Variable Selection in QSAR Studies for the Validation of Thiazolidine-2,4-Dione Derivatives as Promising Antitumor Candidates.

Published in:

Indian Journal of Pharmaceutical Education & Research, 2017, v. 51, n. 3, p. 436, doi. 10.5530/ijper.51.3.72

By:

Asati, Vivek;
Bharti, Sanjay Kumar;
Rathore, Ankita;
Mahapatra, Debarshi Kar

Publication type:

Article

DEVELOPMENT OF NEW 2-METHYL-4-SALICYLAMIDE THIAZOLE DERIVATIVES: SYNTHESIS, ANTIMICROBIAL ACTIVITY EVALUATION, LIPOPHILICITY AND MOLECULAR DOCKING STUDY.

Published in:

Farmacia, 2021, v. 69, n. 4, p. 724, doi. 10.31925/farmacia.2021.4.13

By:

POP, BIANCA;
IONUȚ, IOANA;
MARC, GABRIEL;
VODNAR, DAN CRISTIAN;
PÎRNĂU, ADRIAN;
VLASE, LAURIAN;
ONIGA, OVIDIU

Publication type:

Article

HETEROCYCLES 42. SYNTHESIS AND CHARACTERIZATION OF NEW THIAZOLO[3,2-B] [1,2,4]TRIAZOLE DERIVATIVES WITH ANTI-INFLAMMATORY POTENTIAL.

Published in:

Farmacia, 2018, v. 66, n. 1, p. 88

By:

CRISTINA, ANAMARIA;
LEONTE, DENISA;
VLASE, LAURIAN;
BENCZE, LÁSZLÓ CSABA;
IMRE, SILVIA;
ZAHARIA, VALENTIN

Publication type:

Article

Synthesis, Cytotoxic, and Antioxidant Activity of Some Benzoquinoline-Based Heterocycles.

Published in:

Polycyclic Aromatic Compounds, 2024, v. 44, n. 9, p. 5938, doi. 10.1080/10406638.2023.2270767

By:

El-Helw, Eman A. E.;
Asran, Mahmoud;
Azab, Mohammad E.;
Helal, Maher H.;
Ramadan, Sayed K.

Publication type:

Article

Synthesis and in-Silico Studies of Some New Thiazole Carboxamide Derivatives with Theoretical Investigation.

Published in:

Polycyclic Aromatic Compounds, 2024, v. 44, n. 6, p. 3990, doi. 10.1080/10406638.2023.2243639

By:

A. Kheder, Nabila;
Ather, Hissana;
R. Emam, Dalia;
S. Mahmoud, Naglaa;
Fahim, Asmaa M.;
M. Farag, Ahmad

Publication type:

Article

Syntheses and Molecular Docking Analysis of Some New Thiazole and Thiazine Derivatives as Three Armed Molecules with a Triazine Ring as a Core Component: A Search for anti-Obesity Agents.

Published in:

Polycyclic Aromatic Compounds, 2024, v. 44, n. 1, p. 275, doi. 10.1080/10406638.2023.2173617

By:

Badrey, Mohamed G.;
Gomha, Sobhi M.;
Abdelmonsef, Aboubakr H.;
El-Reedy, Ahmed A. M.

Publication type:

Article

Synthesis, Molecular Docking, and Antitumor Evaluation of Some New Pyrazole, Pyridine, and Thiazole Derivatives Incorporating Sulfonamide Residue.

Published in:

Polycyclic Aromatic Compounds, 2023, v. 43, n. 9, p. 7769, doi. 10.1080/10406638.2022.2140170

By:

Elgogary, Sameh R.;
El‑Telbani, Emad M.;
Khidre, Rizk E.

Publication type:

Article

Theoretical Insights into the Solvation, Electronic, Chemical Properties and Molecular Docking of Some Thiazole Derivatives.

Published in:

Polycyclic Aromatic Compounds, 2023, v. 43, n. 2, p. 1546, doi. 10.1080/10406638.2022.2030767

By:

Al-Otaibi, Jamelah S.;
Mary, Y. Sheena;
Mary, Y. Shyma

Publication type:

Article

Microwave-Assisted One-Pot Three Component Synthesis of Some Thiazolyl(Hydrazonoethyl)Thiazoles as Potential Anti-Breast Cancer Agents.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 10, p. 7232, doi. 10.1080/10406638.2021.1998146

By:

Mahmoud, Huda K.;
Abdelhady, Hyam A.;
Elaasser, Mahmoud M.;
Hassain, Doaa Z. H.;
Gomha, Sobhi M.

Publication type:

Article

Convenient Synthesis of Some New Thiophene, Pyrazole, and Thiazole Derivatives Bearing Biologically Active Sulfonyl Guanidine Moiety.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 9, p. 6628, doi. 10.1080/10406638.2021.1988999

By:

Fouad, Sawsan A.;
El-Gendey, Marwa S.;
Ahmed, Entsar M.;
Hessein, Sadia A.;
Ammar, Yousry A.;
Zaki, Yasser H.

Publication type:

Article

An Economic Synthesis of New Thiazole Derivative as a Potent Anticancer, Anti-Antibiotic Resistant Bacteria, and Larvicidal Agent.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 9, p. 6537, doi. 10.1080/10406638.2021.1984952

By:

Mabkhot, Yahia N.;
Khaled, Jamal M. A.;
Alharbi, Naiyf S. H. A.;
Mohammed, Fahd Ali Nasr;
Abdo Almekhlafi, Fahd;
Abutaha, Nael Mahmmoud;
Kheder, Nabila A.;
Asiri, Yahya I.;
Bin Muhsinah, Abdullatif;
Alsayari, Abdulrhman

Publication type:

Article

Synthesis of Two Isomeric Thiadiazine and Thiazole Derivatives from a Hydrazonoyl Halide.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 8, p. 5196, doi. 10.1080/10406638.2021.1936085

By:

Al-Faiyz, Yasair S.;
Sayed, Abdelwahed R.

Publication type:

Article

Synthesis, Antimicrobial Capability and Molecular Docking of Heterocyclic Scaffolds Clubbed by 2-Azetidinone, Thiazole and Quinoline Derivatives.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 7, p. 3924, doi. 10.1080/10406638.2021.1877747

By:

Desai, Nisheeth C.;
Harsora, Jalpa P.;
Monapara, Jahnvi D.;
Khedkar, Vijay M.

Publication type:

Article

Synthesis, Antimicrobial and Anticancer Evaluations of Novel Thiazoles Incorporated Diphenyl Sulfone Moiety.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 5, p. 2521, doi. 10.1080/10406638.2020.1837887

By:

Shaaban, Mohamed R.;
Farghaly, Thoraya A.;
Alsaedi, Amani M. R.

Publication type:

Article

Synthesis, Molecular Docking and Antitumor Activity of New Dithiazoles.

Published in:

Polycyclic Aromatic Compounds, 2021, v. 41, n. 8, p. 1591, doi. 10.1080/10406638.2019.1689512

By:

Farghaly, Thoraya A.;
El-Metwaly, Nashwa;
Al-Soliemy, Amerah M.;
Katouah, Hanadi A.;
Muhammad, Zeinab A.;
Sabour, Rehab

Publication type:

Article

Synthesis and Biological Evaluation of Some New Thiophene, Thiazole, Dithiolane Derivatives and Related Compounds.

Published in:

Polycyclic Aromatic Compounds, 2020, v. 40, n. 5, p. 1445, doi. 10.1080/10406638.2018.1555174

By:

Fadda, Ahmed A.;
Tawfik, Eman H.;
Selim, Yasser A.

Publication type:

Article

Iodine Catalysed Oxidative Cross‐Coupling of Thioureas and Amines without Desulfurization.

Published in:

Asian Journal of Organic Chemistry, 2023, v. 12, n. 5, p. 1, doi. 10.1002/ajoc.202300032

By:

Serrao, Lavina Gladis;
Rai P., Vishakha;
Periyasamy, Ganga;
Maddani, Mahagundappa Rachappa

Publication type:

Article

One Pot Catalyst‐free Synthesis of Substituted Di‐amino N‐tosyl Benzoyl Thiazoles byRegioselective C−N Bond Cleavage and Its Anticancer Activity.

Published in:

Asian Journal of Organic Chemistry, 2022, v. 11, n. 1, p. 1, doi. 10.1002/ajoc.202100675

By:

Bangade, Vikas M.;
Dadmal, Tulshiram L.;
Popatkar, Bhushan B.;
Mali, Prakash R.;
Meshram, Harshadas M.

Publication type:

Article

Cascade Nucleophilic Addition/cyclization/C−N Coupling of o‐Iodo‐phenyl Isothiocyanates with Propargylamines: Access to Benzimidazo[2,1‐b]thiazole Derivatives.

Published in:

Asian Journal of Organic Chemistry, 2021, v. 10, n. 12, p. 3253, doi. 10.1002/ajoc.202100545

By:

Zhong, Xianqiang;
He, Feng;
Ran, Qiuye;
Li, Wenjing;
Xiong, Huilan;
Zhou, Wei

Publication type:

Article

[3+2]‐Cycloaddition of Azaoxyallyl Cations with Cyclopropenones and Cyclopropenethiones: Synthesis of Spirocyclic Oxazole and Thiazole Derivatives.

Published in:

Asian Journal of Organic Chemistry, 2019, v. 8, n. 8, p. 1376, doi. 10.1002/ajoc.201900272

By:

Zhou, Shuang‐Jing;
Cheng, Xiao;
Xuan, Jun

Publication type:

Article

A Copper‐Catalyzed Domino Reaction of Alkynyl Bromides and Oxazolidine‐2‐thiones: Synthesis of Thiazol‐2‐ones.

Published in:

Asian Journal of Organic Chemistry, 2018, v. 7, n. 5, p. 888, doi. 10.1002/ajoc.201800154

By:

Xie, Chunsong;
Zhang, Yuhong

Publication type:

Article

Scientific Opinion on Flavouring Group Evaluation 76, Revision 1 (FGE.76Rev1): Consideration of sulphur-containing heterocyclic compounds evaluated by JECFA (59th meeting) structurally related to thiazoles, thiophene, thiazoline and thienyl derivatives from chemical group 29 and miscellaneous substances from chemical group 30 evaluated by EFSA in FGE.21Rev3

Published in:: EFSA Journal, 2013, v. 11, n. 11, p. 1, doi. 10.2903/j.efsa.2013.3455
Publication type:: Article

Novel Thiazole Derivatives of Medicinal Potential: Synthesis and Modeling.

Published in:

Journal of Chemistry, 2017, p. 1, doi. 10.1155/2017/4102796

By:

Abdel-Sattar, Nour E. A.;
El-Naggar, Abeer M.;
Abdel-Mottaleb, M. S. A.

Publication type:

Article

Modification of 4-(4-chlorothiophen-2-yl) thiazol-2-amine derivatives for the treatment of analgesia and inflammation: synthesis and in vitro, in vivo, and in silico studies.

Published in:

Frontiers in Pharmacology, 2024, p. 01, doi. 10.3389/fphar.2024.1366695

By:

Mahnashi, Mater H.;
Rashid, Umer;
Almasoudi, Hassan Hussain;
Nahari, Mohammed H.;
Ahmad, Imran;
Binshaya, Abdulkarim S.;
Abdulaziz, Osama;
Alsuwat, Meshari A.;
Jan, Muhammad Saeed;
Sadiq, Abdul

Publication type:

Article

Exploration of naphthalenone-thiazole hybrids for TNF-α, COX-2 inhibition and anti-oxidant capability.

Published in:

Research on Chemical Intermediates, 2025, v. 51, n. 3, p. 1609, doi. 10.1007/s11164-025-05513-8

By:

Yadav, Jyoti;
Chaudhary, R. P.

Publication type:

Article

Structural, conformational and therapeutic studies on new thiazole complexes: drug-likeness and MOE-simulation assessments.

Published in:

Research on Chemical Intermediates, 2021, v. 47, n. 5, p. 1979, doi. 10.1007/s11164-020-04380-9

By:

Abu-Dief, Ahmed M.;
El-Metwaly, Nashwa M.;
Alzahrani, Seraj Omar;
Alkhatib, Fatmah;
Abumelha, Hana M.;
El-Dabea, Tarek;
Ali El‐Remaily, Mahmoud Abd El Aleem Ali

Publication type:

Article

Biological evaluation and in silico molecular docking study of a new series of thiazol-2-yl-hydrazone conglomerates.

Published in:

Research on Chemical Intermediates, 2018, v. 44, n. 4, p. 2779, doi. 10.1007/s11164-018-3261-z

By:

Bhat, Mahima;
Gurubasavaraja Swamy, P. M.;
Poojary, Boja;
Revanasiddappa, B. C.;
Vijay Kumar, M.;
Kumar, Vasantha

Publication type:

Article

Synthesis and biological evaluation of new 2-aryl-4-((4-aryl-1 H-1,2,3-triazol-1-yl)methyl)thiazole derivatives.

Published in:

Research on Chemical Intermediates, 2018, v. 44, n. 2, p. 1247, doi. 10.1007/s11164-017-3164-4

By:

Shinde, Vikas;
Mahulikar, Pramod;
Mhaske, Pravin C.;
Nawale, Laxman;
Sarkar, Dhiman

Publication type:

Article

Construction of benzo[d]imidazo[2,1-b]thiazole derivatives via a simple multi-component domino cyclization.

Published in:

Research on Chemical Intermediates, 2018, v. 44, n. 1, p. 613, doi. 10.1007/s11164-017-3123-0

By:

Wang, Jianqiang;
Zhang, Wenhui;
Zhao, Zheng;
Mao, Jingpeng;
Guo, Cheng

Publication type:

Article

New tetrazoloquinolinyl methoxyphenyl-4-thiazolidinones: synthesis and antihyperglycemic evaluation.

Published in:

Research on Chemical Intermediates, 2017, v. 43, n. 2, p. 1107, doi. 10.1007/s11164-016-2686-5

By:

Deshmukh, Amarsinh;
Bhosle, Manisha;
Khillare, Lalit;
Dhumal, Sambhaji;
Mishra, Akansha;
Srivastava, Arvind;
Mane, Ramrao

Publication type:

Article

Synthesis and anticancer activity of some new heterocyclic compounds based on 1-cyanoacetyl-3,5-dimethylpyrazole.

Published in:

Research on Chemical Intermediates, 2016, v. 42, n. 2, p. 1071, doi. 10.1007/s11164-015-2074-6

By:

Metwally, Nadia;
Abdelrazek, Fathy;
Eldaly, Salwa

Publication type:

Article

β-Cyclodextrin-SOH-catalyzed facile and highly efficient synthesis of 4-thiazolidinones under solvent free conditions.

Published in:

Research on Chemical Intermediates, 2015, v. 41, n. 12, p. 10027, doi. 10.1007/s11164-015-2010-9

By:

Chaudhari, Mahendra;
Gujar, Jitendra;
Kawade, Deepak;
Shinde, Pravin;
Shingare, Murlidhar

Publication type:

Article

An efficient and facile synthesis of 5-amino-2,3-dihydrobenzo[ b]thiophene-4,6-dicarbonitrile and 5-amino-2,3-dihydrobenzo[ d]thiazole-4,6-dicarbonitrile derivatives.

Published in:

Research on Chemical Intermediates, 2015, v. 41, n. 9, p. 6041, doi. 10.1007/s11164-014-1720-8

By:

Wang, Suhui;
Zha, Yunyun;
Wang, Shilei;
Zhang, Jing;
Sun, Jingyi;
Rong, Liangce;
Cai, Peijun

Publication type:

Article

Electro-generated ortho-quinoide intermediates: templates for feasible construction of a series of novel imidazo[2,1- b]thiazole derivatives through one-pot five-step domino hetero-annulation process.

Published in:

Research on Chemical Intermediates, 2015, v. 41, n. 9, p. 6185, doi. 10.1007/s11164-014-1731-5

By:

Alizadeh, Abdolhamid;
Khodaei, Mohammad;
Kanjouri, Tayyebeh;
Shamsuddin, Mustaffa

Publication type:

Article

Fluorinated azole anticancer drugs: Synthesis, elaborated structure elucidation and docking studies.

Published in:

Arabian Journal of Chemistry, 2022, v. 15, n. 5, p. N.PAG, doi. 10.1016/j.arabjc.2022.103782

By:

Alsaedi, Amani M.R.;
Farghaly, Thoraya A.;
Shaaban, Mohamed R.

Publication type:

Article

Synthesis and In-silico Simulation of Some New Bis-thiazole Derivatives and Their Preliminary Antimicrobial Profile: Investigation of Hydrazonoyl Chloride Addition to Hydroxy-Functionalized Bis-carbazones.

Published in:

Arabian Journal of Chemistry, 2021, v. 14, n. 11, p. N.PAG, doi. 10.1016/j.arabjc.2021.103396

By:

Kassab, Refaie M.;
Gomha, Sobhi M.;
Al-Hussain, Sami A.;
Abo Dena, Ahmed S.;
Abdel-Aziz, Marwa M.;
Zaki, Magdi E.A.;
Muhammad, Zeinab A.

Publication type:

Article

Synthesis and antiproliferative activity studies of new functionalized pyridine linked thiazole derivatives.

Published in:

Arabian Journal of Chemistry, 2021, v. 14, n. 1, p. N.PAG, doi. 10.1016/j.arabjc.2020.11.020

By:

Alqahtani, Alaa M.;
Bayazeed, Abrar A.

Publication type:

Article

Bioactive Fluorenes. Part II. Unprecedented biologically active thiazole derivatives based-2,7-dichlorofluorene as competent DHFR inhibitors: Design, synthesis, and molecular docking approaches.

Published in:

Arabian Journal of Chemistry, 2020, v. 13, n. 5, p. 5451, doi. 10.1016/j.arabjc.2020.03.024

By:

Alsantali, Reem I.;
Hussein, Essam M.;
Obaid, Rami J.;
Morad, Moataz;
Altass, Hatem M.;
Alharbi, Ahmed;
Hameed, Ahmed M.;
Jassas, Rabab.S.;
Abourehab, Mohamed A.S.;
Asghar, Basim H.;
Moussa, Ziad;
Ahmed, Saleh A.

Publication type:

Article

Synthesis and antimicrobial activity of some imidazothiazole derivatives of benzofuran.

Published in:

Arabian Journal of Chemistry, 2017, v. 10, p. S554, doi. 10.1016/j.arabjc.2012.10.018

By:

Shankerrao, Sheelavanth;
Bodke, Yadav D.;
Santoshkumar, S.

Publication type:

Article

Synthesis, characterization and antimicrobial evaluation of 2,5-disubstituted-4-thiazolidinone derivatives.

Published in:

Arabian Journal of Chemistry, 2014, v. 7, n. 3, p. 287, doi. 10.1016/j.arabjc.2010.10.032

By:

Deep, Aakash;
Jain, Sandeep;
Sharma, Prabodh Chander;
Mittal, Sanjeev K.;
Phogat, Priyanka;
Malhotra, Manav

Publication type:

Article

Molecular docking and computational studies investigation on a bioactive anti-cancer drug: Thiazole derivatives.

Published in:

Indian Journal of Chemical Technology, 2022, v. 29, n. 6, p. 616, doi. 10.56042/ijct.v29i6.67406

By:

Viji, A.;
Vijayakumar, R.;
Balachandran, V.;
Vanasundari, K.;
Janaki, M.

Publication type:

Article

Synthesis and in silico ADMET evaluation of new thiazole and thiazolidine-4-one derivatives as non-ulcerog.

Published in:

Journal of the Serbian Chemical Society, 2024, v. 89, n. 11, p. 1411, doi. 10.2298/JSC231029064N

By:

KOOPAEI, MANSUR NASSIRI;
MONAVARI, MAHSHID;
VOUSOOGHI, NASIM;
MOSHIRABADI, SADAF;
ASSARZADEH, MOHAMMAD JAVAD;
AMINI, MOHSEN;
ALMASIRAD, ALI

Publication type:

Article

Synthesis of 2-Arylbenzothiazoles by Copper-Catalyzed One-Pot.

Published in:

Journal of Heterocyclic Chemistry, 2016, v. 53, n. 4, p. 1207, doi. 10.1002/jhet.2385

By:

Xu, Hualong;
Luo, Chun;
Li, Zhengkai;
Xiang, Haifeng;
Zhou, Xiangge

Publication type:

Article

Basic Ionic Liquid as Catalyst and Reaction Media for the One-pot Three-component.

Published in:

Journal of Heterocyclic Chemistry, 2016, v. 53, n. 4, p. 1009, doi. 10.1002/jhet.2406

By:

Shiran, Jafar Abbasi;
Yahyazadeh, Asieh;
Yamin, Bohari M.;
Mamaghani, Manouchehr;
Albadi, Jalal

Publication type:

Article

Synthesis and Antifungal Screening of 2-(2-Aryl-4-methyl-thiazol-5-yl)-5-((2-aryl/benzylthiazol-4-yl)methyl)-1,3,4-oxadiazole Derivatives.

Published in:

Journal of Heterocyclic Chemistry, 2016, v. 53, n. 1, p. 129, doi. 10.1002/jhet.2393

By:

Mhaske, Pravin C.;
Shelke, Shivaji H.;
Gadge, Kisan;
Shinde, Abhijit

Publication type:

Article