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Controlling the Covalent Reactivity of a Kinase Inhibitor with Light.
- Published in:
- Angewandte Chemie, 2021, v. 133, n. 37, p. 20340, doi. 10.1002/ange.202103767
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- Publication type:
- Article
Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway.
- Published in:
- Angewandte Chemie, 2019, v. 131, n. 4, p. 1074, doi. 10.1002/ange.201810312
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- Article
Halogenaromatische π‐Wechselwirkungen modulieren die Verweilzeit von Inhibitoren.
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- Angewandte Chemie, 2018, v. 130, n. 24, p. 7338, doi. 10.1002/ange.201801666
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- Article
Innenrücktitelbild: Das Cysteinom der Proteinkinasen als Zielstruktur in der Arzneistoffentwicklung (Angew. Chem. 16/2018).
- Published in:
- Angewandte Chemie, 2018, v. 130, n. 16, p. 4517, doi. 10.1002/ange.201802502
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- Article
Das Cysteinom der Proteinkinasen als Zielstruktur in der Arzneistoffentwicklung.
- Published in:
- Angewandte Chemie, 2018, v. 130, n. 16, p. 4456, doi. 10.1002/ange.201707875
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- Article
Discovery of a PCAF Bromodomain Chemical Probe.
- Published in:
- Angewandte Chemie, 2017, v. 129, n. 3, p. 845, doi. 10.1002/ange.201610816
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- Article
Rücktitelbild: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. 3/2017).
- Published in:
- Angewandte Chemie, 2017, v. 129, n. 3, p. 928, doi. 10.1002/ange.201612063
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- Publication type:
- Article
Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway.
- Published in:
- Angewandte Chemie International Edition, 2019, v. 58, n. 4, p. 1062, doi. 10.1002/anie.201810312
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- Publication type:
- Article
Discovery of an MLLT1/3 YEATS Domain Chemical Probe.
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- Angewandte Chemie International Edition, 2018, v. 57, n. 50, p. 16302, doi. 10.1002/anie.201810617
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- Article
Halogen–Aromatic π Interactions Modulate Inhibitor Residence Times.
- Published in:
- Angewandte Chemie International Edition, 2018, v. 57, n. 24, p. 7220, doi. 10.1002/anie.201801666
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- Article
Inside Back Cover: The Cysteinome of Protein Kinases as a Target in Drug Development (Angew. Chem. Int. Ed. 16/2018).
- Published in:
- Angewandte Chemie International Edition, 2018, v. 57, n. 16, p. 4429, doi. 10.1002/anie.201802502
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- Publication type:
- Article
The Cysteinome of Protein Kinases as a Target in Drug Development.
- Published in:
- Angewandte Chemie International Edition, 2018, v. 57, n. 16, p. 4372, doi. 10.1002/anie.201707875
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- Publication type:
- Article
Discovery of a PCAF Bromodomain Chemical Probe.
- Published in:
- Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 827, doi. 10.1002/anie.201610816
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- Publication type:
- Article
Back Cover: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. Int. Ed. 3/2017).
- Published in:
- Angewandte Chemie International Edition, 2017, v. 56, n. 3, p. 908, doi. 10.1002/anie.201612063
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- Publication type:
- Article
Discovery of a Novel Class of Covalent Dual Inhibitors Targeting the Protein Kinases BMX and BTK.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 23, p. 9269, doi. 10.3390/ijms21239269
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- Article
Comprehensive Set of Tertiary Complex Structures and Palmitic Acid Binding Provide Molecular Insights into Ligand Design for RXR Isoforms.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 22, p. 8457, doi. 10.3390/ijms21228457
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- Article
Crystal Structure and Inhibitor Identifications Reveal Targeting Opportunity for the Atypical MAPK Kinase ERK3.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 21, p. 7953, doi. 10.3390/ijms21217953
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- Article
Chemical Starting Matter for HNF4α Ligand Discovery and Chemogenomics.
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- International Journal of Molecular Sciences, 2020, v. 21, n. 21, p. 7895, doi. 10.3390/ijms21217895
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- Article
Structure of human aspartyl aminopeptidase complexed with substrate analogue: insight into catalytic mechanism, substrate specificity and M18 peptidase family.
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- BMC Structural Biology, 2012, v. 12, n. 1, p. 14, doi. 10.1186/1472-6807-12-14
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- Article
Lessons from LIMK1 enzymology and their impact on inhibitor design.
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- Biochemical Journal, 2019, v. 476, n. 21, p. 3197, doi. 10.1042/BCJ20190517
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- Article
Conservation of structure, function and inhibitor binding in UNC-51-like kinase 1 and 2 (ULK1/2).
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- Biochemical Journal, 2019, v. 476, n. 5, p. 875, doi. 10.1042/BCJ20190038
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- Article
Structure of cyclin G-associated kinase (GAK) trapped in different conformations using nanobodies.
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- Biochemical Journal, 2014, v. 459, n. 1, p. 59, doi. 10.1042/BJ20131399
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- Article
Co-crystal structures of the protein kinase haspin with bisubstrate inhibitors.
- Published in:
- Acta Crystallographica: Section F, Structural Biology Communications, 2016, v. 72, n. 5, p. 339, doi. 10.1107/S2053230X16004611
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- Article
Modulation of tau tubulin kinases (TTBK1 and TTBK2) impacts ciliogenesis.
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- Scientific Reports, 2023, v. 13, n. 1, p. 1, doi. 10.1038/s41598-023-32854-4
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- Article
Mechanism and consequence of the autoactivation of p38α mitogen-activated protein kinase promoted by TAB1.
- Published in:
- Nature Structural & Molecular Biology, 2013, v. 20, n. 10, p. 1182, doi. 10.1038/nsmb.2668
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- Article
Atad2 is a generalist facilitator of chromatin dynamics in embryonic stem cells.
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- Journal of Molecular Cell Biology, 2016, v. 8, n. 4, p. 349, doi. 10.1093/jmcb/mjv060
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- Article
A New Class of Small Molecule Inhibitor of BMP Signaling.
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- PLoS ONE, 2013, v. 8, n. 4, p. 1, doi. 10.1371/journal.pone.0062721
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- Article
Structural Comparison of Human Mammalian Ste20-Like Kinases.
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- PLoS ONE, 2010, v. 5, n. 8, p. 1, doi. 10.1371/journal.pone.0011905
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- Article
Identification of CLK1 Inhibitors by a Fragment-linking Based Virtual Screening.
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- Molecular Informatics, 2017, v. 36, n. 4, p. n/a, doi. 10.1002/minf.201600123
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- Article
Mutation in the Common Docking Domain Affects MAP Kinase ERK2 Catalysis and Stability.
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- Cancers, 2023, v. 15, n. 11, p. 2938, doi. 10.3390/cancers15112938
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- Article
Discovery of a Potent and Highly Isoform-Selective Inhibitor of the Neglected Ribosomal Protein S6 Kinase Beta 2 (S6K2).
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- Cancers, 2021, v. 13, n. 20, p. 5133, doi. 10.3390/cancers13205133
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- Article
A Consensus Compound/Bioactivity Dataset for Data-Driven Drug Design and Chemogenomics.
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- Molecules, 2022, v. 27, n. 8, p. N.PAG, doi. 10.3390/molecules27082513
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- Article
Image-Based Annotation of Chemogenomic Libraries for Phenotypic Screening.
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- Molecules, 2022, v. 27, n. 4, p. 1439, doi. 10.3390/molecules27041439
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- Article
Structural consequences of BMPR2 kinase domain mutations causing pulmonary arterial hypertension.
- Published in:
- Scientific Reports, 2019, v. 9, n. 1, p. N.PAG, doi. 10.1038/s41598-019-54830-7
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- Article
Kinase Domain Autophosphorylation Rewires the Activity and Substrate Specificity of CK1 Enzymes.
- Published in:
- FASEB Journal, 2022, v. 36, p. N.PAG, doi. 10.1096/fasebj.2022.36.S1.0R463
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- Article
A Specific and Covalent JNK-1 Ligand Selected from an Encoded Self-Assembling Chemical Library.
- Published in:
- Chemistry - A European Journal, 2017, v. 23, n. 34, p. 8152, doi. 10.1002/chem.201701644
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- Article
Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity.
- Published in:
- Angewandte Chemie, 2023, v. 135, n. 11, p. 1, doi. 10.1002/ange.202217532
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- Publication type:
- Article
The orphan nuclear receptor Nurr1 is responsive to non-steroidal anti-inflammatory drugs.
- Published in:
- Communications Chemistry, 2020, v. 3, n. 1, p. 1, doi. 10.1038/s42004-020-0331-0
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- Article
Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity.
- Published in:
- Angewandte Chemie International Edition, 2023, v. 62, n. 11, p. 1, doi. 10.1002/anie.202217532
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- Publication type:
- Article
Controlling the Covalent Reactivity of a Kinase Inhibitor with Light.
- Published in:
- Angewandte Chemie International Edition, 2021, v. 60, n. 37, p. 20178, doi. 10.1002/anie.202103767
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 12, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 11, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 10, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 9, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 7, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 6, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Radiolabeled cCPE Peptides for SPECT Imaging of Claudin-4 Overexpression in Pancreatic Cancer.
- Published in:
- Journal of Nuclear Medicine, 2020, v. 61, n. 5, p. 1, doi. 10.2967/jnumed.120.243113
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- Publication type:
- Article
Comparative structural analyses and nucleotide-binding characterization of the four KH domains of FUBP1.
- Published in:
- Scientific Reports, 2020, v. 10, n. 1, p. 1, doi. 10.1038/s41598-020-69832-z
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- Article
DARPins detect the formation of hetero-tetramers of p63 and p73 in epithelial tissues and in squamous cell carcinoma.
- Published in:
- Cell Death & Disease, 2023, v. 14, n. 10, p. 1, doi. 10.1038/s41419-023-06213-0
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- Article
The ins and outs of selective kinase inhibitor development.
- Published in:
- Nature Chemical Biology, 2015, v. 11, n. 11, p. 818, doi. 10.1038/nchembio.1938
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- Article