Works matching DE "LIPASE inhibitors"

Results: 276

IN-VITRO ANTI LIPASE ACTIVITY OF POLYHERBAL SIDDHA FORMULATION ILAVANGATHI CHOORANAM.

Published in:

Obstetrics & Gynaecology Forum, 2024, v. 34, n. 2, p. 74

By:

Glara, A. F.;
Sureka, A.;
Subhathra, M.;
Girija, N. Sabari;
Ashmi, R.;
Varghese, Thomas Reshmee

Publication type:

Article

Variations of the chemical components and biological activities of Thymus capitatus essential oil from three regions in Palestine.

Published in:

Scientific Reports, 2025, v. 15, n. 1, p. 1, doi. 10.1038/s41598-025-92835-7

By:

Jaradat, Nidal;
Barkat, Alaa;
Khasati, Ahmad;
Abualhasan, Murad

Publication type:

Article

Evaluation of anti-acne activity of selected Sudanese medicinal plants.

Published in:

Journal of Wood Science, 2013, v. 59, n. 1, p. 73, doi. 10.1007/s10086-012-1303-5

By:

Muddathir, Ali;
Mitsunaga, Tohru

Publication type:

Article

Methyl Oleate Modulates LIP2 Expression in the Lipolytic Yeast Yarrowia lipolytica.

Published in:

Biotechnology Letters, 2005, v. 27, n. 22, p. 1751, doi. 10.1007/s10529-005-3547-2

By:

Fickers, Patrick;
Destain, Jacqueline;
Thonart, Philippe

Publication type:

Article

Lipase-catalyzed acylation of l-carnitine with conjugated linoleic acid in [Bmim]PF<sub>6</sub> ionic liquid.

Published in:

European Food Research & Technology, 2009, v. 229, n. 2, p. 357, doi. 10.1007/s00217-009-1063-7

By:

Tian, Jinqiang;
Wang, Qiang;
Zhang, Zhongyuan

Publication type:

Article

Inhibition of lipase from rice ( Oryza sativa ) by diethyl- p -nitrophenyl phosphate.

Published in:

European Food Research & Technology, 2008, v. 227, n. 1, p. 277, doi. 10.1007/s00217-007-0721-x

By:

M. Raghavendra;
Parigi Kumar;
Vishweshwaraiah Prakash

Publication type:

Article

DNA cleavage function of seryl-histidine dipeptide and its application.

Published in:

Amino Acids, 2008, v. 35, n. 2, p. 251, doi. 10.1007/s00726-007-0597-x

By:

Y. Ma;
X. Chen;
M. Sun;
R. Wan;
C. Zhu;
Y. Li

Publication type:

Article

Anti-Atherosclerotic Action of a New Stimulator of Soluble Guanylate Cyclase in an Experiment.

Published in:

Bulletin of Experimental Biology & Medicine, 2023, v. 174, n. 3, p. 333, doi. 10.1007/s10517-023-05703-7

By:

Bykov, V. V.;
Bykova, A. V.;
Dzyuman, A. N.;
Ivanov, V. V.;
Khazanov, V. A.;
Vengerovskii, A. I.;
Udut, V. V.

Publication type:

Article

Poloxamer 407 as a general lipase inhibitor: its implications in lipid metabolism and atheroma formation in C57BL/6 mice.

Published in:

Journal of Pharmacy & Pharmacology, 2010, v. 62, n. 12, p. 1807, doi. 10.1111/j.2042-7158.2010.01138.x

By:

Johnston, Thomas P.

Publication type:

Article

In Vitro Antioxidant, Anti-Inflammatory, and Digestive Enzymes Inhibition Activities of Hydro-Ethanolic Leaf and Bark Extracts of Psychotria densinervia (K. Krause) Verdc.

Published in:

Advances in Pharmacological & Pharmaceutical Sciences, 2022, p. 1, doi. 10.1155/2022/8459943

By:

Mba, Jean Romuald;
Zouheira, Djamila;
Dairou, Hadidjatou;
Yadang, Fanta S. A.;
Gael, Nfor Njini;
Ayong, Lawrence;
Kuiate, Jules-Roger;
Agbor, Gabriel A.

Publication type:

Article

Effect of Flaxseed Mucilage on the Probiotic, Antioxidant, and Structural-Mechanical Properties of the Different Lactobacillus Cells.

Published in:

Fermentation (Basel), 2023, v. 9, n. 5, p. 486, doi. 10.3390/fermentation9050486

By:

Sungatullina, Alya;
Petrova, Tatyana;
Kharina, Maria;
Mikshina, Polina;
Nikitina, Elena

Publication type:

Article

Atglistatin Pretreatment Preserves Remote Myocardium Function Following Myocardial Infarction.

Published in:

2021

By:

Bottermann, Katharina;
Granade, Mitchell E.;
Oenarto, Vici;
Fischer, Jens W.;
Harris, Thurl E.

Publication type:

journal article

EXTRACTION OPTIMIZATION OF Senecio vernalis Waldst. & Kit AND DETERMINATION OF ANTI-α-AMYLASE/α-GLUCOSIDASE, ANTI-LIPASE AND ANTIOXIDANT ACTIVITIES.

Published in:

Trakya University Journal of Natural Sciences, 2021, v. 22, n. 2, p. 245, doi. 10.23902/trkjnat.960073

By:

DOĞAN, Nurcan;
DOĞAN, Cemhan

Publication type:

Article

Discovery of A Novel Synthetic Thiazole-benzimidazole Conjugate that Acts as a Potent Pancreatic Lipase Inhibitor using in silico and in vitro Approaches.

Published in:

Indian Journal of Pharmaceutical Education & Research, 2023, v. 57, n. 1, p. 218, doi. 10.5530/001954642131

By:

Abouzied, Amr Salah;
Bin Break, Mohammed Khaled;
Huwaimel, Bader;
Hussein, Weiam;
Alafnan, Ahmed;
Younes, Kareem Mahmoud

Publication type:

Article

Adjunction of the Lipase Inhibitor Orlistat Improves Grape Seed Extract Neuroprotection against Brain Ischemia/Reperfusion Injury in Rats.

Published in:

Indian Journal of Pharmaceutical Education & Research, 2021, v. 55, n. 2, p. 527, doi. 10.5530/ijper.55.2.91

By:

Ghrir, Slim;
Abbes, Wassim Ben;
Charradi, Kamel;
Elkahoui, Salem;
Limam, Ferid;
Aouani, Ezzedine

Publication type:

Article

Design, Green Synthesis, and Biological Evaluation of New Substituted Tetrahydropyrimidine Derivatives as Acetylcholinesterase Inhibitors.

Published in:

Polycyclic Aromatic Compounds, 2022, v. 42, n. 8, p. 5231, doi. 10.1080/10406638.2021.1933102

By:

Mariki, Ali akbar;
Anaeigoudari, Akbar;
Zahedifar, Mahboobeh;
Pouramiri, Behjat;
Ayati, Adileh;
Lotfi, Safa

Publication type:

Article

Inhibition of Digestive Enzymes and Antioxidant Activity of Extracts from Fruits of Cornus alba, Cornus sanguinea subsp. hungarica and Cornus florida–A Comparative Study.

Published in:

Plants (2223-7747), 2020, v. 9, n. 1, p. 1, doi. 10.3390/plants9010122

By:

Truba, Joanna;
Stanisławska, Iwona;
Walasek, Marta;
Wieczorkowska, Wioleta;
Woliński, Konrad;
Buchholz, Tina;
Melzig, Matthias F.;
Czerwińska, Monika E.

Publication type:

Article

A Histological Study on The Effect of Orlistat Administration on the Liver of the Adult Male Albino Rat and the Possible Protective Effect of Vitamin C.

Published in:

Alexandria Journal of Veterinary Sciences, 2021, v. 70, n. 1, p. 7, doi. 10.5455/ajvs.54417

By:

Fahmi, Maha A.

Publication type:

Article

Synthesis and Biological Significances of New Heterocyclic Compounds Containing 5-(4-Chlorobenzyl)-3-(4-Chlorophenyl)-1H-1,2,4-triazol Ring.

Published in:

Journal of the Chemical Society of Pakistan, 2017, v. 39, n. 6, p. 1055

By:

Ozdemir, Yusuf;
Gultekin, Ergun;
Bekircan, Olcay

Publication type:

Article

Positive effect of Limosilactobacillus plantarum grx16 on nonalcoholic fatty liver disease in rats.

Published in:

International Journal of Dairy Technology, 2023, v. 76, n. 3, p. 710, doi. 10.1111/1471-0307.12956

By:

Qu, Hengxian;
Zhang, Longfei;
Liu, Xiaoxiao;
Liu, Yang;
Mao, Kaidong;
Shen, Guiqi;
Wa, Yunchao;
Chen, Dawei;
Huang, Yujun;
Chen, Xia;
Gu, Ruixia

Publication type:

Article

Effect of selective inhibition of monoacylglycerol lipase (MAGL) on acute nausea, anticipatory nausea, and vomiting in rats and Suncus murinus.

Published in:

Psychopharmacology, 2015, v. 232, n. 3, p. 583, doi. 10.1007/s00213-014-3696-x

By:

Parker, Linda;
Niphakis, Micah;
Downey, Rachel;
Limebeer, Cheryl;
Rock, Erin;
Sticht, Martin;
Morris, Heather;
Abdullah, Rehab;
Lichtman, Aron;
Cravatt, Benjamin

Publication type:

Article

Elucidation of potent mammalian enzymes inhibitors targeting anti-diabetes drug from Castanea mollissima blume, 1851: an edible herbal collected in Vietnam via experimental and computation approaching.

Published in:

Research on Chemical Intermediates, 2024, v. 50, n. 12, p. 6065, doi. 10.1007/s11164-024-05427-x

By:

Le Vu, Thi Thu;
Wang, San-Lang;
Ho, Thi Thanh Thanh;
Luc, Quang Tan;
Phan, Tu Quy;
Phan, Thi Kim Thu;
Dam, Thi Bich Hanh;
Phan, Thi Kim Phung;
Nguyen, Anh Dzung;
Nguyen, Van Bon

Publication type:

Article

Lipase-catalysed one-pot synthesis of thiazole-based Betti bases and their evaluation as potential cholinesterase inhibitors.

Published in:

Research on Chemical Intermediates, 2021, v. 47, n. 7, p. 2731, doi. 10.1007/s11164-021-04441-7

By:

Shaikh, Sarfaraz;
Ramana, M. M. V.

Publication type:

Article

A flavin-monooxygenase catalyzing oxepinone formation and the complete biosynthesis of vibralactone.

Published in:

Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-39108-x

By:

Feng, Ke-Na;
Zhang, Yue;
Zhang, Mingfang;
Yang, Yan-Long;
Liu, Ji-Kai;
Pan, Lifeng;
Zeng, Ying

Publication type:

Article

Structurally diverse brefeldin A derivatives as potent and selective acetylcholinesterase inhibitors from an endophytic fungus Penicillium brefeldianum F4a.

Published in:

Arabian Journal of Chemistry, 2024, v. 17, n. 1, p. N.PAG, doi. 10.1016/j.arabjc.2023.105388

By:

Bai, Yan;
Ren, Duo;
Xue, Xinlei;
Gao, Weixian;
Hu, Jiangchun;
Pan, Huaqi

Publication type:

Article

Extraction and enzymatic modification of dietary fibre from purple aubergine.

Published in:

Czech Journal of Food Sciences, 2023, v. 41, n. 4, p. 304, doi. 10.17221/84/2023-CJFS

By:

SUWALEE FONG-IN;
KAMONLAK WICHARAEW;
PATTARAMON PHALAPAN;
TRAKUL PROMMAJAK

Publication type:

Article

Lemon basil seed-derived peptide: Hydrolysis, purification, and its role as a pancreatic lipase inhibitor that reduces adipogenesis by downregulating SREBP-1c and PPAR-γ in 3T3-L1 adipocytes.

Published in:

PLoS ONE, 2024, v. 19, n. 5, p. 1, doi. 10.1371/journal.pone.0301966

By:

Kuptawach, Kittisak;
Noitung, Sajee;
Buakeaw, Anumart;
Puthong, Songchan;
Sawangkeaw, Ruengwit;
Sangtanoo, Papassara;
Srimongkol, Piroonporn;
Reamtong, Onrapak;
Choowongkomon, Kiattawee;
Karnchanatat, Aphichart

Publication type:

Article

Phillyrin: an adipose triglyceride lipase inhibitor supported by molecular docking, dynamics simulation, and pharmacological validation.

Published in:

Journal of Molecular Modeling, 2024, v. 30, n. 3, p. 1, doi. 10.1007/s00894-024-05875-7

By:

Zhou, Chenyu;
Yan, Lanmeng;
Xu, Jing;
Hamezah, Hamizah Shahirah;
Wang, Tongsheng;
Du, Fangping;
Tong, Xiaohui;
Han, Rongchun

Publication type:

Article

Orlistat for the treatment of antipsychotic-induced weight gain: an eight-week multicenter, randomized, placebo-controlled, double-blind trial.

Published in:

Lipids in Health & Disease, 2024, v. 23, n. 1, p. 1, doi. 10.1186/s12944-024-02214-w

By:

Xie, Peng;
Shao, Tiannan;
Long, Yujun;
Xie, Weiwei;
Liu, Yangjun;
Yang, Ye;
Huang, Yuyan;
Wu, Renrong;
Deng, Qijian;
Tang, Hui

Publication type:

Article

National trends in the use and costs of anti-obesity medications in England 1998-2005.

Published in:

Journal of Public Health, 2007, v. 29, n. 2, p. 199

By:

Janakan Srishanmuganathan;
Hitesh Patel;
Josip Car;
Azeem Majeed

Publication type:

Article

Crystal structure of the thioesterase domain of human fatty acid synthase inhibited by Orlistat.

Published in:

Nature Structural & Molecular Biology, 2007, v. 14, n. 8, p. 704, doi. 10.1038/nsmb1265

By:

Pemble, Charles W.;
Johnson, Lynnette C.;
Kridel, Steven J.;
Lowther, W. Todd

Publication type:

Article

Proteinous pancreatic lipase inhibitor is responsible for the antiobesity effect of young barley (Hordeum vulgare L.) leaf extract.

Published in:

Bioscience, Biotechnology & Biochemistry, 2021, v. 85, n. 8, p. 1885, doi. 10.1093/bbb/zbab096

By:

Kato, Eisuke;
Tsuruma, Ai;
Amishima, Ayaka;
Satoh, Hiroshi

Publication type:

Article

Inhibitory Activity of Chlorogenic Acids in Decaffeinated Green Coffee Beans against Porcine Pancreas Lipase and Effect of a Decaffeinated Green Coffee Bean Extract on an Emulsion of Olive Oil.

Published in:

Bioscience, Biotechnology & Biochemistry, 2012, v. 76, n. 12, p. 2329, doi. 10.1271/bbb.120518

By:

NARITA, Yusaku;
IWAI, Kazuya;
FUKUNAGA, Taiji;
NAKAGIRI, Osamu

Publication type:

Article

Voltammetric lipase activity assay based on dilinolein and a modified carbon paste electrode.

Published in:

Analytical & Bioanalytical Chemistry, 2022, v. 414, n. 17, p. 5033, doi. 10.1007/s00216-022-04135-y

By:

Rogala, Anita;
Rechberger, Julia;
Vasold, Vanessa;
Samphao, Anchalee;
Kalcher, Kurt;
Ortner, Astrid

Publication type:

Article

Evaluation of selected commercial pharmacotherapeutic drugs as potential pancreatic lipase inhibitors and antiproliferative compounds.

Published in:

Drug Development Research, 2019, v. 80, n. 3, p. 310, doi. 10.1002/ddr.21499

By:

Mamdooh, Noor;
Kasabri, Violet;
Al‐Hiari, Yusuf;
Almasri, Ihab;
Al‐Alawi, Sundus;
Bustanji, Yasser

Publication type:

Article

Cholinesterase Inhibitors from an Endophytic Fungus Aspergillus niveus Fv-er401: Metabolomics, Isolation and Molecular Docking.

Published in:

Molecules, 2023, v. 28, n. 6, p. 2559, doi. 10.3390/molecules28062559

By:

Hamed, Ahmed A.;
El-Shiekh, Riham A.;
Mohamed, Osama G.;
Aboutabl, Elsayed A.;
Fathy, Fify I.;
Fawzy, Ghada A.;
Al-Taweel, Areej M.;
Elsayed, Tarek R.;
Tripathi, Ashootosh;
Al-Karmalawy, Ahmed A.

Publication type:

Article

High-Resolution Bioassay Profiling with Complemented Sensitivity and Resolution for Pancreatic Lipase Inhibitor Screening.

Published in:

Molecules, 2022, v. 27, n. 20, p. 6923, doi. 10.3390/molecules27206923

By:

Jian, Jingyi;
Yuan, Jiaming;
Fan, Yu;
Wang, Jincai;
Zhang, Tingting;
Kool, Jeroen;
Jiang, Zhengjin

Publication type:

Article

Multipotent Cholinesterase Inhibitors for the Treatment of Alzheimer's Disease: Synthesis, Biological Analysis and Molecular Docking Study of Benzimidazole-Based Thiazole Derivatives.

Published in:

Molecules, 2022, v. 27, n. 18, p. 6087, doi. 10.3390/molecules27186087

By:

Hussain, Rafaqat;
Ullah, Hayat;
Rahim, Fazal;
Sarfraz, Maliha;
Taha, Muhammad;
Iqbal, Rashid;
Rehman, Wajid;
Khan, Shoaib;
Shah, Syed Adnan Ali;
Hyder, Sajjad;
Alhomrani, Majid;
Alamri, Abdulhakeem S.;
Abdulaziz, Osama;
Abdelaziz, Mahmoud A.

Publication type:

Article

Free Linoleic Acid and Oleic Acid Reduce Fat Digestion and Absorption In Vivo as Potent Pancreatic Lipase Inhibitors Derived from Sesame Meal.

Published in:

Molecules, 2022, v. 27, n. 15, p. 4910, doi. 10.3390/molecules27154910

By:

Li, Xuan;
Morita, Sayo;
Yamada, Hiroaki;
Koga, Keita;
Ota, Wakana;
Furuta, Toma;
Yamatsu, Atsushi;
Kim, Mujo

Publication type:

Article

Rapid Screening of Lipase Inhibitors in Scutellaria baicalensis by Using Porcine Pancreatic Lipase Immobilized on Magnetic Core–Shell Metal–Organic Frameworks.

Published in:

Molecules, 2022, v. 27, n. 11, p. 3475, doi. 10.3390/molecules27113475

By:

Xu, Jinfang;
Cao, Pengkun;
Fan, Zhiyu;
Luo, Xujing;
Yang, Gangqiang;
Qu, Tingli;
Gao, Jianping

Publication type:

Article

The Relationship between the IC 50 Values and the Apparent Inhibition Constant in the Study of Inhibitors of Tyrosinase Diphenolase Activity Helps Confirm the Mechanism of Inhibition.

Published in:

Molecules, 2022, v. 27, n. 10, p. 3141, doi. 10.3390/molecules27103141

By:

Garcia-Molina, Pablo;
Garcia-Molina, Francisco;
Teruel-Puche, Jose Antonio;
Rodriguez-Lopez, Jose Neptuno;
Garcia-Canovas, Francisco;
Muñoz-Muñoz, Jose Luis

Publication type:

Article

In Vitro and In Silico Evaluation of Cholinesterase Inhibition by Alkaloids Obtained from Branches of Abuta panurensis Eichler.

Published in:

Molecules, 2022, v. 27, n. 10, p. 3138, doi. 10.3390/molecules27103138

By:

da Silva Mesquita, Rochelly;
Kyrylchuk, Andrii;
Cherednichenko, Anton;
Costa Sá, Ingrity Suelen;
Macedo Bastos, Lílian;
Moura Araújo da Silva, Felipe;
Saraiva Nunomura, Rita de Cássia;
Grafov, Andriy

Publication type:

Article

Discovery of Novel Epoxyketone Peptides as Lipase Inhibitors.

Published in:

Molecules, 2022, v. 27, n. 7, p. 2261, doi. 10.3390/molecules27072261

By:

Almaliti, Jehad;
Alzweiri, Muhammed;
Alhindy, Momen;
Al-Helo, Tamam;
Daoud, Ibrahim;
Deknash, Raghad;
Naman, C. Benjamin;
Abu-Irmaileh, Bashaer;
Bustanji, Yasser;
Hamad, Islam

Publication type:

Article

Rapid Screening of Lipase Inhibitors from Ophiopogonis Radix Using High-Performance Thin Layer Chromatography by Two Step Gradient Elution Combined with Bioautographic Method.

Published in:

Molecules, 2022, v. 27, n. 4, p. 1155, doi. 10.3390/molecules27041155

By:

Hua, Xue;
Hong, Hui-Jie;
Zhang, Dai-Yan;
Liu, Qiao;
Leong, Fong;
Yang, Qi;
Hu, Yuan-Jia;
Chen, Xiao-Jia

Publication type:

Article

Phytochemical Profile and In Vitro Antioxidant, Antimicrobial, Vital Physiological Enzymes Inhibitory and Cytotoxic Effects of Artemisia jordanica Leaves Essential Oil from Palestine.

Published in:

Molecules, 2021, v. 26, n. 9, p. 2831, doi. 10.3390/molecules26092831

By:

Jaradat, Nidal;
Duarte, Ana Paula;
Luís, Ângelo;
Gallardo, Eugenia

Publication type:

Article

Analgesic and Anticancer Activity of Benzoxazole Clubbed 2-Pyrrolidinones as Novel Inhibitors of Monoacylglycerol Lipase.

Published in:

Molecules, 2021, v. 26, n. 8, p. 2389, doi. 10.3390/molecules26082389

By:

Afzal, Obaid;
Altamimi, Abdulmalik Saleh Alfawaz;
Shahroz, Mir Mohammad;
Sharma, Hemant Kumar;
Riadi, Yassine;
Hassan, Md Quamrul

Publication type:

Article

Bioactivity-Guided Isolation of Phytochemicals from Vaccinium dunalianum Wight and Their Antioxidant and Enzyme Inhibitory Activities.

Published in:

Molecules, 2021, v. 26, n. 7, p. 2075, doi. 10.3390/molecules26072075

By:

Zhao, Tianrui;
Sun, Mengxue;
Kong, Lingpeng;
Xue, Qingwang;
Wang, Yudan;
Wang, Yifen;
Khan, Afsar;
Cao, Jianxin;
Cheng, Guiguang;
Miceli, Natalizia

Publication type:

Article

Exploring Aurone Derivatives as Potential Human Pancreatic Lipase Inhibitors through Molecular Docking and Molecular Dynamics Simulations.

Published in:

Molecules, 2020, v. 25, n. 20, p. 4657, doi. 10.3390/molecules25204657

By:

Nguyen, Phuong Thuy Viet;
Huynh, Han Ai;
Truong, Dat Van;
Tran, Thanh-Dao;
Vo, Cam-Van Thi

Publication type:

Article

Flavonoids in Decorticated Sorghum Grains Exert Antioxidant, Antidiabetic and Antiobesity Activities.

Published in:

Molecules, 2020, v. 25, n. 12, p. 2854, doi. 10.3390/molecules25122854

By:

Ofosu, Fred Kwame;
Elahi, Fazle;
Daliri, Eric Banan-Mwine;
Yeon, Su-Jung;
Ham, Hun Ju;
Kim, Joong-Hark;
Han, Sang-Ik;
Oh, Deog-Hwan

Publication type:

Article

Synthesis and Spectral Identification of Three Schiff Bases with a 2-(Piperazin-1-yl)-N-(thiophen-2-yl methylene)ethanamine Moiety Acting as Novel Pancreatic Lipase Inhibitors: Thermal, DFT, Antioxidant, Antibacterial, and Molecular Docking Investigations

Published in:

Molecules, 2020, v. 25, n. 9, p. 2253, doi. 10.3390/molecules25092253

By:

Warad, Ismail;
Ali, Oraib;
Al Ali, Anas;
Jaradat, Nidal Amin;
Hussein, Fatima;
Abdallah, Lubna;
Al-Zaqri, Nabil;
Alsalme, Ali;
Alharthi, Fahad A.

Publication type:

Article