Works matching IS 18607179 AND DT 2024 AND VI 19 AND IP 24

Results: 27

Cover Feature: Phosphate‐Containing Glycolipids: A Review on Synthesis and Bioactivity (ChemMedChem 24/2024).

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202482402

By:

Pinheiro, Luís;
Freitas, Marisa;
Branco, Paula S.

Publication type:

Article

Front Cover: Cholinesterase Inhibitory Activity and Molecular Docking Studies of Isocryptolepine‐Triazole Adducts (ChemMedChem 24/2024).

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202482401

By:

Tummatorn, Jumreang;
Meewan, Ittipat;
Khunnawutmanotham, Nisachon;
Chimnoi, Nitirat;
Suwanwong, Nutchapong;
Rodphon, Warabhorn;
Thongsornkleeb, Charnsak;
Yang, Jingyue;
Ruchirawat, Somsak

Publication type:

Article

Medicinal Chemistry in Bosnia and Herzegovina ‐ Past, Present and Perspectives**.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400669

By:

Kondža, Martin

Publication type:

Article

Structural Basis for Inhibition of the SARS‐CoV‐2 nsp16 by Substrate‐Based Dual Site Inhibitors.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400618

By:

Kalnins, Gints;
Rudusa, Laura;
Bula, Anna L.;
Zelencova‐Gopejenko, Diana;
Bobileva, Olga;
Sisovs, Mihails;
Tars, Kaspars;
Jirgensons, Aigars;
Jaudzems, Kristaps;
Bobrovs, Raitis

Publication type:

Article

Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400601

By:

Kilbile, Jaydeo T.;
Sapkal, Suryakant B.;
Renzi, Gioele;
D'Agostino, Ilaria;
Boudjelal, Mohamed;
Tamboli, Yasinalli;
Cutarella, Luigi;
Mori, Mattia;
Sgambellone, Silvia;
Villano, Serafina;
Marri, Silvia;
Lucarini, Laura;
Carradori, Simone;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Discovery of Palindrome Dual PPARγ‐GPR40 Agonists for Treating Type 2 Diabetes.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400492

By:

Rodríguez‐Luévano, Ana;
Almanza‐Pérez, Julio C.;
Ortiz‐Andrade, Rolffy;
Lara‐González, Samuel;
Santillán, Rosa;
Navarrete‐Vázquez, Gabriel;
Giacoman‐Martínez, Abraham;
Lazzarini‐Lechuga, Roberto C.;
Bautista, Elihú;
Hidalgo‐Figueroa, Sergio

Publication type:

Article

Two‐Step Synthesis of Enantiomerically Pure Morphans from (R)‐Carvone.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400596

By:

Costanzo, Giuliana;
Cosentino, Giuseppe;
Pasquinucci, Lorella;
Amata, Emanuele;
Schepmann, Dirk;
Wünsch, Bernhard

Publication type:

Article

Serum Circulating mRNA Panel for the Early Detection of Gastric Cancer: A Potential Biomarker Test.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400523

By:

Peng, Xinyu;
Teng, Xiaoyan;
Ma, Qian;
Han, Da

Publication type:

Article

Crystallographic and Selectivity Studies on the Approved HIF Prolyl Hydroxylase Inhibitors Desidustat and Enarodustat.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400504

By:

Corner, Thomas P.;
Salah, Eidarus;
Tumber, Anthony;
Kaur, Samanpreet;
Nakashima, Yu;
Allen, Mark D.;
Schnaubelt, Lara I.;
Fiorini, Giorgia;
Brewitz, Lennart;
Schofield, Christopher J.

Publication type:

Article

Leveraging Natural Product‐Inspired Antifungals to Investigate the Mechanism of Action of Peniciaculin A.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400500

By:

Wilt, Ingrid K.;
Demeritte, Adrian R.;
Kim, Alexander T.;
Wang, Weiwei;
Wuest, William M.

Publication type:

Article

In Vitro and In Vivo Biological Evaluation of Novel 1,4‐Naphthoquinone Derivatives as Potential Anticancer Agents.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400495

By:

Ravichandiran, Palanisamy;
Martyna, Aleksandra;
Kochanowicz, Elżbieta;
Maroli, Nikhil;
Kubiński, Konrad;
Masłyk, Maciej;
Boguszewska‐Czubara, Anna;
Ramesh, Thiyagarajan

Publication type:

Article

Lactam Truncation Yields a Dihydroquinazolinone Scaffold with Potent Antimalarial Activity that Targets PfATP4.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400549

By:

Ashton, Trent D.;
Calic, Petar P. S.;
Dans, Madeline G.;
Kang Ooi, Zi;
Zhou, Qingmiao;
Loi, Katie;
Jarman, Kate E.;
Palandri, Josephine;
Qiu, Deyun;
Lehane, Adele M.;
Maity, Bikash;
De, Nirupam;
Famodimu, Mufuliat T.;
Delves, Michael J.;
Mao, Emma Y.;
Gancheva, Maria R.;
Wilson, Danny W.;
Chowdury, Mrittika;
de Koning‐Ward, Tania F.;
Baud, Delphine

Publication type:

Article

Tumor‐Associated Carbohydrate Antigen 19–9 (CA 19–9), a Promising Target for Antibody‐Based Detection, Diagnosis, and Immunotherapy of Cancer.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400491

By:

Nakisa, Athar;
Sempere, Lorenzo F.;
Chen, Xi;
Qu, Linda T.;
Woldring, Daniel;
Crawford, Howard C.;
Huang, Xuefei

Publication type:

Article

Phenotypic‐Based Discovery and Exploration of a Resorufin Scaffold with Activity against Mycobacterium tuberculosis.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400482

By:

Tran, Eric;
Cheung, Chen‐Yi;
Li, Lucy;
Carter, Glen P.;
Gable, Robert W.;
West, Nicholas P.;
Kaur, Amandeep;
Gee, Yi Sing;
Cook, Gregory M.;
Baell, Jonathan B.;
Jörg, Manuela

Publication type:

Article

Bacterial Secondary Metabolites Embedded in Producer Cell Membranes and Antibiotics Targeting Their Biosynthesis.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400469

By:

Xia, Zhao;
Xiang, Hao;
Shi, Yi‐Ming

Publication type:

Article

Discovery of KW0113 as a First and Effective PROTAC Degrader of DNMT1 Protein.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400467

By:

Wang, Huihui;
Wang, Zhaoliang;
Hu, Linghao;
Yang, Bingjie;
Zong, Liangyi;
Xu, Dounan;
Yu, Bo;
Kong, Xiangqian;
Wang, Mingliang

Publication type:

Article

Substrate‐Based Ligand Design for Phenazine Biosynthesis Enzyme PhzF.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400466

By:

Baumgarten, Janosch;
Schneider, Philipp;
Thiemann, Marie;
Zimmermann, Moritz;
Diederich, Christina;
Blankenfeldt, Wulf;
Kunick, Conrad

Publication type:

Article

Two Step One‐Pot Synthesis of 7‐Azaindole Linked 1,2,3‐Triazole Hybrids: In‐Vitro and In‐Silico Antimicrobial Evaluation.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400451

By:

Sharma, Kanika;
Lal, Bajrang;
Kumar Tittal, Ram;
Lal, Kashmiri;
Vats, Lalit;
Vikas D, Ghule

Publication type:

Article

Cholinesterase Inhibitory Activity and Molecular Docking Studies of Isocryptolepine‐Triazole Adducts.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400447

By:

Tummatorn, Jumreang;
Meewan, Ittipat;
Khunnawutmanotham, Nisachon;
Chimnoi, Nitirat;
Suwanwong, Nutchapong;
Rodphon, Warabhorn;
Thongsornkleeb, Charnsak;
Yang, Jingyue;
Ruchirawat, Somsak

Publication type:

Article

Evaluation of a Radioiodinated G‐Quadruplex Binder in Cervical Cancer Models.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400438

By:

Cristina Oliveira, Maria;
Campello, Maria Paula Cabral;
Gano, Lurdes;
Raposinho, Paula;
Belchior, Ana;
Mendes, Edgar;
Silva, Catarina D.;
Lopes‐Nunes, Jéssica;
Cruz, Carla;
Paulo, António

Publication type:

Article

The Investigation of Hsp90C‐Terminal Inhibitors Containing Amide Bioisosteres.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400418

By:

Amatya, Eva;
Subramanian, Chitra;
Long, Reagan;
McNamara, Kelli;
Cohen, Mark S.;
Blagg, Brian S. J.

Publication type:

Article

Fluorescence‐Based HTS Assays for Ion Channel Modulation in Drug Discovery Pipelines.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400383

By:

Voldřich, Jan;
Matoušová, Marika;
Šmídková, Markéta;
Mertlíková‐Kaiserová, Helena

Publication type:

Article

Cyclodextrin Dimers Functionalized with Biotin as Nanocapsules for Active Doxorubicin Delivery Against MCF‐7 Breast Cell Line.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400368

By:

Bognanni, Noemi;
Scuderi, Chiara;
Giglio, Valentina;
Spiteri, Fabio;
La Piana, Luana;
Condorelli, Daniele;
Barresi, Vincenza;
Vecchio, Graziella

Publication type:

Article

How to Find a Fragment: Methods for Screening and Validation in Fragment‐Based Drug Discovery.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400342

By:

Kirkman, Tim;
dos Santos Silva, Catharina;
Tosin, Manuela;
Bertacine Dias, Marcio Vinicius

Publication type:

Article

Phosphate‐Containing Glycolipids: A Review on Synthesis and Bioactivity.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400315

By:

Pinheiro, Luís;
Freitas, Marisa;
Branco, Paula S.

Publication type:

Article

Flavonol‐Ruthenium Complexes as Antioxidant and Anticancer Agents.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400313

By:

Wu, Ting‐Wei;
Chu, Yi‐Cheng;
Chang, Chuan‐Hsin;
Hsieh, Yu‐Hui;
Tang, Mei‐Hsin;
Hsu, Pei‐Hsuan;
Wu, Hsin‐Ying;
Chen, Jih‐Jung;
Shih, Tzenge‐Lien

Publication type:

Article

Development of Integrin Targeting Chimeras (ITACs) for the Lysosomal Degradation of Extracellular Proteins.

Published in:

ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202300643

By:

Zhou, Yaxian;
Liao, Yaxian;
Zhao, Yuan;
Tang, Weiping

Publication type:

Article